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Compile Data Set for Download or QSAR

Found 148 hits of Enz. Inhib. data with enzyme = 'Dopamine D2 S receptor' and Substrate = 'to-be-curated'   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kcal/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Dopamine D2 S receptor


(Homo sapiens (Human))
BDBM50192233
PNG
(CHEMBL3890178 | US10239870, Example 290)
Show SMILES Cn1c(SCCCN2CC[C@]3(C[C@@H]3c3ccc(cc3)C(F)(F)F)C2)nnc1-c1ccccc1C(N)=O
Show InChI InChI=1/C26H28F3N5OS/c1-33-23(20-6-3-2-5-19(20)22(30)35)31-32-24(33)36-14-4-12-34-13-11-25(16-34)15-21(25)17-7-9-18(10-8-17)26(27,28)29/h2-3,5-10,21H,4,11-16H2,1H3,(H2,30,35)/t21-,25+/s2
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US Patent
39.8n/an/an/an/an/an/an/an/a



Indivior UK Limited

US Patent


Assay Description
CHO cells stably expressing human dopamine receptor type 2, long variant (hD2L), coupled to Gα16 protein (CHO-Gα16-hD2L) were re-suspended ...


US Patent US10239870 (2019)

More data for this
Ligand-Target Pair
Dopamine D2 S receptor


(Homo sapiens (Human))
BDBM371858
PNG
(US10239870, Example 59 | US10239870, Example 60)
Show SMILES Cc1ncoc1-c1nnc(SCCCN2CC[C@]3(CC3c3cc(Cl)cc(Cl)c3)C2)n1C
Show InChI InChI=1/C22H25Cl2N5OS/c1-14-19(30-13-25-14)20-26-27-21(28(20)2)31-7-3-5-29-6-4-22(12-29)11-18(22)15-8-16(23)10-17(24)9-15/h8-10,13,18H,3-7,11-12H2,1-2H3/t18?,22-/s2
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US Patent
61.7n/an/an/an/an/an/an/an/a



Indivior UK Limited

US Patent


Assay Description
CHO cells stably expressing human dopamine receptor type 2, long variant (hD2L), coupled to Gα16 protein (CHO-Gα16-hD2L) were re-suspended ...


US Patent US10239870 (2019)

More data for this
Ligand-Target Pair
Dopamine D2 S receptor


(Homo sapiens (Human))
BDBM50192447
PNG
(CHEMBL3975989 | US10239870, Example 53)
Show SMILES Cc1ncoc1-c1nnc(SCCCN2CC[C@@]3(C[C@@H]3c3ccccc3C(F)(F)F)C2)n1C
Show InChI InChI=1/C23H26F3N5OS/c1-15-19(32-14-27-15)20-28-29-21(30(20)2)33-11-5-9-31-10-8-22(13-31)12-18(22)16-6-3-4-7-17(16)23(24,25)26/h3-4,6-7,14,18H,5,8-13H2,1-2H3/t18-,22-/s2
PDB

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US Patent
63.1n/an/an/an/an/an/an/an/a



Indivior UK Limited

US Patent


Assay Description
CHO cells stably expressing human dopamine receptor type 2, long variant (hD2L), coupled to Gα16 protein (CHO-Gα16-hD2L) were re-suspended ...


US Patent US10239870 (2019)

More data for this
Ligand-Target Pair
Dopamine D2 S receptor


(Homo sapiens (Human))
BDBM371858
PNG
(US10239870, Example 59 | US10239870, Example 60)
Show SMILES Cc1ncoc1-c1nnc(SCCCN2CC[C@]3(CC3c3cc(Cl)cc(Cl)c3)C2)n1C
Show InChI InChI=1/C22H25Cl2N5OS/c1-14-19(30-13-25-14)20-26-27-21(28(20)2)31-7-3-5-29-6-4-22(12-29)11-18(22)15-8-16(23)10-17(24)9-15/h8-10,13,18H,3-7,11-12H2,1-2H3/t18?,22-/s2
PDB

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US Patent
66.1n/an/an/an/an/an/an/an/a



Indivior UK Limited

US Patent


Assay Description
CHO cells stably expressing human dopamine receptor type 2, long variant (hD2L), coupled to Gα16 protein (CHO-Gα16-hD2L) were re-suspended ...


US Patent US10239870 (2019)

More data for this
Ligand-Target Pair
Dopamine D2 S receptor


(Homo sapiens (Human))
BDBM372012
PNG
(US10239870, Example 272)
Show SMILES Cn1c(SCCCN2CC[C@]3(C[C@@H]3c3ccc(cc3)C(F)(F)F)C2)nnc1-c1ccc2[nH]cnc2n1
Show InChI InChI=1/C25H26F3N7S/c1-34-22(20-8-7-19-21(31-20)30-15-29-19)32-33-23(34)36-12-2-10-35-11-9-24(14-35)13-18(24)16-3-5-17(6-4-16)25(26,27)28/h3-8,15,18H,2,9-14H2,1H3,(H,29,30,31)/t18-,24+/s2
PDB

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US Patent
95.5n/an/an/an/an/an/an/an/a



Indivior UK Limited

US Patent


Assay Description
CHO cells stably expressing human dopamine receptor type 2, long variant (hD2L), coupled to Gα16 protein (CHO-Gα16-hD2L) were re-suspended ...


US Patent US10239870 (2019)

More data for this
Ligand-Target Pair
Dopamine D2 S receptor


(Homo sapiens (Human))
BDBM372001
PNG
(US10239870, Example 259 | US10239870, Example 260)
Show SMILES Cn1c(SCCCN2CC[C@]3(CC3c3ccc(cc3)C(F)(F)F)C2)nnc1-c1csnn1
Show InChI InChI=1/C21H23F3N6S2/c1-29-18(17-12-32-28-25-17)26-27-19(29)31-10-2-8-30-9-7-20(13-30)11-16(20)14-3-5-15(6-4-14)21(22,23)24/h3-6,12,16H,2,7-11,13H2,1H3/t16?,20-/s2
PDB

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US Patent
112n/an/an/an/an/an/an/an/a



Indivior UK Limited

US Patent


Assay Description
CHO cells stably expressing human dopamine receptor type 2, long variant (hD2L), coupled to Gα16 protein (CHO-Gα16-hD2L) were re-suspended ...


US Patent US10239870 (2019)

More data for this
Ligand-Target Pair
Dopamine D2 S receptor


(Homo sapiens (Human))
BDBM371850
PNG
(US10239870, Example 49)
Show SMILES Cc1ncoc1-c1nnc(SCCCN2CC[C@]3(CC3c3ccccc3F)C2)n1C
Show InChI InChI=1/C22H26FN5OS/c1-15-19(29-14-24-15)20-25-26-21(27(20)2)30-11-5-9-28-10-8-22(13-28)12-17(22)16-6-3-4-7-18(16)23/h3-4,6-7,14,17H,5,8-13H2,1-2H3/t17?,22-/s2
PDB

UniProtKB/TrEMBL

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US Patent
123n/an/an/an/an/an/an/an/a



Indivior UK Limited

US Patent


Assay Description
CHO cells stably expressing human dopamine receptor type 2, long variant (hD2L), coupled to Gα16 protein (CHO-Gα16-hD2L) were re-suspended ...


US Patent US10239870 (2019)

More data for this
Ligand-Target Pair
Dopamine D2 S receptor


(Homo sapiens (Human))
BDBM372001
PNG
(US10239870, Example 259 | US10239870, Example 260)
Show SMILES Cn1c(SCCCN2CC[C@]3(CC3c3ccc(cc3)C(F)(F)F)C2)nnc1-c1csnn1
Show InChI InChI=1/C21H23F3N6S2/c1-29-18(17-12-32-28-25-17)26-27-19(29)31-10-2-8-30-9-7-20(13-30)11-16(20)14-3-5-15(6-4-14)21(22,23)24/h3-6,12,16H,2,7-11,13H2,1H3/t16?,20-/s2
PDB

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US Patent
129n/an/an/an/an/an/an/an/a



Indivior UK Limited

US Patent


Assay Description
CHO cells stably expressing human dopamine receptor type 2, long variant (hD2L), coupled to Gα16 protein (CHO-Gα16-hD2L) were re-suspended ...


US Patent US10239870 (2019)

More data for this
Ligand-Target Pair
Dopamine D2 S receptor


(Homo sapiens (Human))
BDBM371908
PNG
(US10239870, Example 132)
Show SMILES Cn1c(SCCCN2CC[C@]3(CC3c3ccccc3C(F)(F)F)C2)nnc1-c1ccc(=O)[nH]c1
Show InChI InChI=1/C24H26F3N5OS/c1-31-21(16-7-8-20(33)28-14-16)29-30-22(31)34-12-4-10-32-11-9-23(15-32)13-19(23)17-5-2-3-6-18(17)24(25,26)27/h2-3,5-8,14,19H,4,9-13,15H2,1H3,(H,28,33)/t19?,23-/s2
PDB

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US Patent
135n/an/an/an/an/an/an/an/a



Indivior UK Limited

US Patent


Assay Description
CHO cells stably expressing human dopamine receptor type 2, long variant (hD2L), coupled to Gα16 protein (CHO-Gα16-hD2L) were re-suspended ...


US Patent US10239870 (2019)

More data for this
Ligand-Target Pair
Dopamine D2 S receptor


(Homo sapiens (Human))
BDBM372016
PNG
(US10239870, Example 276)
Show SMILES Cn1c(SCCCN2CC[C@]3(C[C@@H]3c3ccc(cc3)C(F)(F)F)C2)nnc1-c1ccc(cc1)-n1cnnc1
Show InChI InChI=1/C27H28F3N7S/c1-35-24(20-5-9-22(10-6-20)37-17-31-32-18-37)33-34-25(35)38-14-2-12-36-13-11-26(16-36)15-23(26)19-3-7-21(8-4-19)27(28,29)30/h3-10,17-18,23H,2,11-16H2,1H3/t23-,26+/s2
PDB

UniProtKB/TrEMBL

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US Patent
166n/an/an/an/an/an/an/an/a



Indivior UK Limited

US Patent


Assay Description
CHO cells stably expressing human dopamine receptor type 2, long variant (hD2L), coupled to Gα16 protein (CHO-Gα16-hD2L) were re-suspended ...


US Patent US10239870 (2019)

More data for this
Ligand-Target Pair
Dopamine D2 S receptor


(Homo sapiens (Human))
BDBM50192316
PNG
(CHEMBL3985877 | US10239870, Example 57)
Show SMILES Cc1ncoc1-c1nnc(SCCCN2CC[C@]3(C[C@H]3c3ccc(F)cc3C(F)(F)F)C2)n1C
Show InChI InChI=1/C23H25F4N5OS/c1-14-19(33-13-28-14)20-29-30-21(31(20)2)34-9-3-7-32-8-6-22(12-32)11-18(22)16-5-4-15(24)10-17(16)23(25,26)27/h4-5,10,13,18H,3,6-9,11-12H2,1-2H3/t18-,22-/s2
PDB

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US Patent
166n/an/an/an/an/an/an/an/a



Indivior UK Limited

US Patent


Assay Description
CHO cells stably expressing human dopamine receptor type 2, long variant (hD2L), coupled to Gα16 protein (CHO-Gα16-hD2L) were re-suspended ...


US Patent US10239870 (2019)

More data for this
Ligand-Target Pair
Dopamine D2 S receptor


(Homo sapiens (Human))
BDBM371889
PNG
(US10239870, Example 108)
Show SMILES Cn1c(SCCCN2CC[C@]3(CC3c3ccc(cc3)C(F)(F)F)C2)nnc1C1CCC(N)CC1
Show InChI InChI=1/C25H34F3N5S/c1-32-22(18-5-9-20(29)10-6-18)30-31-23(32)34-14-2-12-33-13-11-24(16-33)15-21(24)17-3-7-19(8-4-17)25(26,27)28/h3-4,7-8,18,20-21H,2,5-6,9-16,29H2,1H3/t18?,20?,21?,24-/s2
PDB

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US Patent
191n/an/an/an/an/an/an/an/a



Indivior UK Limited

US Patent


Assay Description
CHO cells stably expressing human dopamine receptor type 2, long variant (hD2L), coupled to Gα16 protein (CHO-Gα16-hD2L) were re-suspended ...


US Patent US10239870 (2019)

More data for this
Ligand-Target Pair
Dopamine D2 S receptor


(Homo sapiens (Human))
BDBM50192454
PNG
(CHEMBL3911264 | US10239870, Example 12)
Show SMILES Cc1ncoc1-c1nnc(SCCCN2CC[C@@]3(C[C@H]3c3ccc(cc3)C(F)(F)F)C2)n1C
Show InChI InChI=1/C23H26F3N5OS/c1-15-19(32-14-27-15)20-28-29-21(30(20)2)33-11-3-9-31-10-8-22(13-31)12-18(22)16-4-6-17(7-5-16)23(24,25)26/h4-7,14,18H,3,8-13H2,1-2H3/t18-,22+/s2
PDB

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US Patent
214n/an/an/an/an/an/an/an/a



Indivior UK Limited

US Patent


Assay Description
CHO cells stably expressing human dopamine receptor type 2, long variant (hD2L), coupled to Gα16 protein (CHO-Gα16-hD2L) were re-suspended ...


US Patent US10239870 (2019)

More data for this
Ligand-Target Pair
Dopamine D2 S receptor


(Homo sapiens (Human))
BDBM50192445
PNG
(CHEMBL3959240 | US10239870, Example 285)
Show SMILES Cn1c(SCCCN2CC[C@]3(C[C@@H]3c3ccc(cc3)C(F)(F)F)C2)nnc1-c1ccc(cc1)S(N)(=O)=O
Show InChI InChI=1/C25H28F3N5O2S2/c1-32-22(18-5-9-20(10-6-18)37(29,34)35)30-31-23(32)36-14-2-12-33-13-11-24(16-33)15-21(24)17-3-7-19(8-4-17)25(26,27)28/h3-10,21H,2,11-16H2,1H3,(H2,29,34,35)/t21-,24+/s2
PDB

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US Patent
219n/an/an/an/an/an/an/an/a



Indivior UK Limited

US Patent


Assay Description
CHO cells stably expressing human dopamine receptor type 2, long variant (hD2L), coupled to Gα16 protein (CHO-Gα16-hD2L) were re-suspended ...


US Patent US10239870 (2019)

More data for this
Ligand-Target Pair
Dopamine D2 S receptor


(Homo sapiens (Human))
BDBM50192248
PNG
(CHEMBL3927895 | US10239870, Example 30)
Show SMILES Cc1ncoc1-c1nnc(SCCCN2CC[C@]3(C[C@@H]3c3ccc(cc3F)C(F)(F)F)C2)n1C
Show InChI InChI=1/C23H25F4N5OS/c1-14-19(33-13-28-14)20-29-30-21(31(20)2)34-9-3-7-32-8-6-22(12-32)11-17(22)16-5-4-15(10-18(16)24)23(25,26)27/h4-5,10,13,17H,3,6-9,11-12H2,1-2H3/t17-,22+/s2
PDB

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US Patent
224n/an/an/an/an/an/an/an/a



Indivior UK Limited

US Patent


Assay Description
CHO cells stably expressing human dopamine receptor type 2, long variant (hD2L), coupled to Gα16 protein (CHO-Gα16-hD2L) were re-suspended ...


US Patent US10239870 (2019)

More data for this
Ligand-Target Pair
Dopamine D2 S receptor


(Homo sapiens (Human))
BDBM50192239
PNG
(CHEMBL3922143 | US10239870, Example 48)
Show SMILES Cc1ncoc1-c1nnc(SCCCN2CC[C@]3(C[C@@H]3c3ccc(F)cc3)C2)n1C
Show InChI InChI=1/C22H26FN5OS/c1-15-19(29-14-24-15)20-25-26-21(27(20)2)30-11-3-9-28-10-8-22(13-28)12-18(22)16-4-6-17(23)7-5-16/h4-7,14,18H,3,8-13H2,1-2H3/t18-,22+/s2
PDB

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US Patent
240n/an/an/an/an/an/an/an/a



Indivior UK Limited

US Patent


Assay Description
CHO cells stably expressing human dopamine receptor type 2, long variant (hD2L), coupled to Gα16 protein (CHO-Gα16-hD2L) were re-suspended ...


US Patent US10239870 (2019)

More data for this
Ligand-Target Pair
Dopamine D2 S receptor


(Homo sapiens (Human))
BDBM50192029
PNG
(CHEMBL3917887 | US10239870, Example 39)
Show SMILES Cc1ncoc1-c1nnc(SCCCN2CC[C@]3(C[C@@H]3c3ccc(F)cc3F)C2)n1C
Show InChI InChI=1/C22H25F2N5OS/c1-14-19(30-13-25-14)20-26-27-21(28(20)2)31-9-3-7-29-8-6-22(12-29)11-17(22)16-5-4-15(23)10-18(16)24/h4-5,10,13,17H,3,6-9,11-12H2,1-2H3/t17-,22+/s2
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US Patent
240n/an/an/an/an/an/an/an/a



Indivior UK Limited

US Patent


Assay Description
CHO cells stably expressing human dopamine receptor type 2, long variant (hD2L), coupled to Gα16 protein (CHO-Gα16-hD2L) were re-suspended ...


US Patent US10239870 (2019)

More data for this
Ligand-Target Pair
Dopamine D2 S receptor


(Homo sapiens (Human))
BDBM50192099
PNG
(CHEMBL3914556 | US10239870, Example 244)
Show SMILES Cn1c(SCCCN2CC[C@]3(C[C@@H]3c3ccc(cc3)C(F)(F)F)C2)nnc1-c1nccs1
Show InChI InChI=1/C22H24F3N5S2/c1-29-18(19-26-8-12-31-19)27-28-20(29)32-11-2-9-30-10-7-21(14-30)13-17(21)15-3-5-16(6-4-15)22(23,24)25/h3-6,8,12,17H,2,7,9-11,13-14H2,1H3/t17-,21+/s2
PDB

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US Patent
251n/an/an/an/an/an/an/an/a



Indivior UK Limited

US Patent


Assay Description
CHO cells stably expressing human dopamine receptor type 2, long variant (hD2L), coupled to Gα16 protein (CHO-Gα16-hD2L) were re-suspended ...


US Patent US10239870 (2019)

More data for this
Ligand-Target Pair
Dopamine D2 S receptor


(Homo sapiens (Human))
BDBM371894
PNG
(US10239870, Example 118)
Show SMILES Cn1c(SCCCN2CC[C@]3(C[C@@H]3c3ccc(cc3)C(F)(F)F)C2)nnc1N1CCOCC1
Show InChI InChI=1/C23H30F3N5OS/c1-29-20(31-10-12-32-13-11-31)27-28-21(29)33-14-2-8-30-9-7-22(16-30)15-19(22)17-3-5-18(6-4-17)23(24,25)26/h3-6,19H,2,7-16H2,1H3/t19-,22+/s2
PDB

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US Patent
251n/an/an/an/an/an/an/an/a



Indivior UK Limited

US Patent


Assay Description
CHO cells stably expressing human dopamine receptor type 2, long variant (hD2L), coupled to Gα16 protein (CHO-Gα16-hD2L) were re-suspended ...


US Patent US10239870 (2019)

More data for this
Ligand-Target Pair
Dopamine D2 S receptor


(Homo sapiens (Human))
BDBM50192255
PNG
(CHEMBL3956758 | US10239870, Example 249)
Show SMILES Cn1cc(cn1)-c1nnc(SCCCN2CC[C@]3(C[C@@H]3c3ccc(cc3)C(F)(F)F)C2)n1C
Show InChI InChI=1/C23H27F3N6S/c1-30-14-17(13-27-30)20-28-29-21(31(20)2)33-11-3-9-32-10-8-22(15-32)12-19(22)16-4-6-18(7-5-16)23(24,25)26/h4-7,13-14,19H,3,8-12,15H2,1-2H3/t19-,22+/s2
PDB

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US Patent
269n/an/an/an/an/an/an/an/a



Indivior UK Limited

US Patent


Assay Description
CHO cells stably expressing human dopamine receptor type 2, long variant (hD2L), coupled to Gα16 protein (CHO-Gα16-hD2L) were re-suspended ...


US Patent US10239870 (2019)

More data for this
Ligand-Target Pair
Dopamine D2 S receptor


(Homo sapiens (Human))
BDBM371953
PNG
(US10239870, Example 190)
Show SMILES Cn1c(SCCCN2CC[C@]3(C[C@@H]3c3ccc(cc3F)C(F)(F)F)C2)nnc1-c1ccc(cn1)C(N)=O
Show InChI InChI=1/C25H26F4N6OS/c1-34-22(20-6-3-15(13-31-20)21(30)36)32-33-23(34)37-10-2-8-35-9-7-24(14-35)12-18(24)17-5-4-16(11-19(17)26)25(27,28)29/h3-6,11,13,18H,2,7-10,12,14H2,1H3,(H2,30,36)/t18-,24+/s2
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275n/an/an/an/an/an/an/an/a



Indivior UK Limited

US Patent


Assay Description
CHO cells stably expressing human dopamine receptor type 2, long variant (hD2L), coupled to Gα16 protein (CHO-Gα16-hD2L) were re-suspended ...


US Patent US10239870 (2019)

More data for this
Ligand-Target Pair
Dopamine D2 S receptor


(Homo sapiens (Human))
BDBM371911
PNG
(US10239870, Example 135)
Show SMILES Cn1c(SCCCN2CC[C@]3(CC3c3ccccc3C(F)(F)F)C2)nnc1-c1cc[nH]c(=O)c1
Show InChI InChI=1/C24H26F3N5OS/c1-31-21(16-7-9-28-20(33)13-16)29-30-22(31)34-12-4-10-32-11-8-23(15-32)14-19(23)17-5-2-3-6-18(17)24(25,26)27/h2-3,5-7,9,13,19H,4,8,10-12,14-15H2,1H3,(H,28,33)/t19?,23-/s2
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288n/an/an/an/an/an/an/an/a



Indivior UK Limited

US Patent


Assay Description
CHO cells stably expressing human dopamine receptor type 2, long variant (hD2L), coupled to Gα16 protein (CHO-Gα16-hD2L) were re-suspended ...


US Patent US10239870 (2019)

More data for this
Ligand-Target Pair
Dopamine D2 S receptor


(Homo sapiens (Human))
BDBM371969
PNG
(US10239870, Example 213)
Show SMILES Cn1c(SCCCN2CC[C@]3(CC3c3ccc(cc3F)C(F)(F)F)C2)nnc1-c1ccncn1
Show InChI InChI=1/C23H24F4N6S/c1-32-20(19-5-7-28-14-29-19)30-31-21(32)34-10-2-8-33-9-6-22(13-33)12-17(22)16-4-3-15(11-18(16)24)23(25,26)27/h3-5,7,11,14,17H,2,6,8-10,12-13H2,1H3/t17?,22-/s2
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295n/an/an/an/an/an/an/an/a



Indivior UK Limited

US Patent


Assay Description
CHO cells stably expressing human dopamine receptor type 2, long variant (hD2L), coupled to Gα16 protein (CHO-Gα16-hD2L) were re-suspended ...


US Patent US10239870 (2019)

More data for this
Ligand-Target Pair
Dopamine D2 S receptor


(Homo sapiens (Human))
BDBM372014
PNG
(US10239870, Example 274)
Show SMILES Cn1c(SCCCN2CC[C@]3(C[C@@H]3c3ccc(cc3)C(F)(F)F)C2)nnc1-c1ccc(cc1)-c1nnco1
Show InChI InChI=1/C27H27F3N6OS/c1-35-23(19-3-5-20(6-4-19)24-33-31-17-37-24)32-34-25(35)38-14-2-12-36-13-11-26(16-36)15-22(26)18-7-9-21(10-8-18)27(28,29)30/h3-10,17,22H,2,11-16H2,1H3/t22-,26+/s2
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302n/an/an/an/an/an/an/an/a



Indivior UK Limited

US Patent


Assay Description
CHO cells stably expressing human dopamine receptor type 2, long variant (hD2L), coupled to Gα16 protein (CHO-Gα16-hD2L) were re-suspended ...


US Patent US10239870 (2019)

More data for this
Ligand-Target Pair
Dopamine D2 S receptor


(Homo sapiens (Human))
BDBM371998
PNG
(US10239870, Example 256)
Show SMILES Cn1c(SCCCN2CC[C@]3(CC3c3ccc(cc3)C(F)(F)F)C2)nnc1-c1cccs1
Show InChI InChI=1/C23H25F3N4S2/c1-29-20(19-4-2-12-31-19)27-28-21(29)32-13-3-10-30-11-9-22(15-30)14-18(22)16-5-7-17(8-6-16)23(24,25)26/h2,4-8,12,18H,3,9-11,13-15H2,1H3/t18?,22-/s2
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331n/an/an/an/an/an/an/an/a



Indivior UK Limited

US Patent


Assay Description
CHO cells stably expressing human dopamine receptor type 2, long variant (hD2L), coupled to Gα16 protein (CHO-Gα16-hD2L) were re-suspended ...


US Patent US10239870 (2019)

More data for this
Ligand-Target Pair
Dopamine D2 S receptor


(Homo sapiens (Human))
BDBM371904
PNG
(US10239870, Example 128)
Show SMILES Cn1c(SCCCN2CC[C@]3(C[C@@H]3c3ccc(cc3)C(F)(F)F)C2)nnc1-c1ccc(=O)[nH]c1
Show InChI InChI=1/C24H26F3N5OS/c1-31-21(17-5-8-20(33)28-14-17)29-30-22(31)34-12-2-10-32-11-9-23(15-32)13-19(23)16-3-6-18(7-4-16)24(25,26)27/h3-8,14,19H,2,9-13,15H2,1H3,(H,28,33)/t19-,23+/s2
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339n/an/an/an/an/an/an/an/a



Indivior UK Limited

US Patent


Assay Description
CHO cells stably expressing human dopamine receptor type 2, long variant (hD2L), coupled to Gα16 protein (CHO-Gα16-hD2L) were re-suspended ...


US Patent US10239870 (2019)

More data for this
Ligand-Target Pair
Dopamine D2 S receptor


(Homo sapiens (Human))
BDBM371999
PNG
(US10239870, Example 257)
Show SMILES Cn1c(SCCCN2CC[C@]3(CC3c3ccc(cc3)C(F)(F)F)C2)nnc1-c1ccsc1
Show InChI InChI=1/C23H25F3N4S2/c1-29-20(17-7-12-31-14-17)27-28-21(29)32-11-2-9-30-10-8-22(15-30)13-19(22)16-3-5-18(6-4-16)23(24,25)26/h3-7,12,14,19H,2,8-11,13,15H2,1H3/t19?,22-/s2
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347n/an/an/an/an/an/an/an/a



Indivior UK Limited

US Patent


Assay Description
CHO cells stably expressing human dopamine receptor type 2, long variant (hD2L), coupled to Gα16 protein (CHO-Gα16-hD2L) were re-suspended ...


US Patent US10239870 (2019)

More data for this
Ligand-Target Pair
Dopamine D2 S receptor


(Homo sapiens (Human))
BDBM50192318
PNG
(CHEMBL3979523 | US10239870, Example 284)
Show SMILES CC(=O)c1ccc(cc1)-c1nnc(SCCCN2CC[C@]3(C[C@@H]3c3ccc(cc3)C(F)(F)F)C2)n1C
Show InChI InChI=1/C27H29F3N4OS/c1-18(35)19-4-6-21(7-5-19)24-31-32-25(33(24)2)36-15-3-13-34-14-12-26(17-34)16-23(26)20-8-10-22(11-9-20)27(28,29)30/h4-11,23H,3,12-17H2,1-2H3/t23-,26+/s2
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347n/an/an/an/an/an/an/an/a



Indivior UK Limited

US Patent


Assay Description
CHO cells stably expressing human dopamine receptor type 2, long variant (hD2L), coupled to Gα16 protein (CHO-Gα16-hD2L) were re-suspended ...


US Patent US10239870 (2019)

More data for this
Ligand-Target Pair
Dopamine D2 S receptor


(Homo sapiens (Human))
BDBM50192449
PNG
(CHEMBL3950540 | US10239870, Example 283)
Show SMILES Cn1c(SCCCN2CC[C@]3(C[C@@H]3c3ccc(cc3)C(F)(F)F)C2)nnc1-c1ccc(cc1)C#N
Show InChI InChI=1/C26H26F3N5S/c1-33-23(20-5-3-18(16-30)4-6-20)31-32-24(33)35-14-2-12-34-13-11-25(17-34)15-22(25)19-7-9-21(10-8-19)26(27,28)29/h3-10,22H,2,11-15,17H2,1H3/t22-,25+/s2
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347n/an/an/an/an/an/an/an/a



Indivior UK Limited

US Patent


Assay Description
CHO cells stably expressing human dopamine receptor type 2, long variant (hD2L), coupled to Gα16 protein (CHO-Gα16-hD2L) were re-suspended ...


US Patent US10239870 (2019)

More data for this
Ligand-Target Pair
Dopamine D2 S receptor


(Homo sapiens (Human))
BDBM50192317
PNG
(CHEMBL3899125 | US10239870, Example 281)
Show SMILES Cn1c(SCCCN2CC[C@]3(C[C@@H]3c3ccc(cc3)C(F)(F)F)C2)nnc1-c1ccc(cc1)C(N)=O
Show InChI InChI=1/C26H28F3N5OS/c1-33-23(19-5-3-18(4-6-19)22(30)35)31-32-24(33)36-14-2-12-34-13-11-25(16-34)15-21(25)17-7-9-20(10-8-17)26(27,28)29/h3-10,21H,2,11-16H2,1H3,(H2,30,35)/t21-,25+/s2
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355n/an/an/an/an/an/an/an/a



Indivior UK Limited

US Patent


Assay Description
CHO cells stably expressing human dopamine receptor type 2, long variant (hD2L), coupled to Gα16 protein (CHO-Gα16-hD2L) were re-suspended ...


US Patent US10239870 (2019)

More data for this
Ligand-Target Pair
Dopamine D2 S receptor


(Homo sapiens (Human))
BDBM371933
PNG
(US10239870, Example 168)
Show SMILES Cc1ncccc1-c1nnc(SCCCN2CC[C@]3(CC3c3ccccc3C(F)(F)F)C2)n1C
Show InChI InChI=1/C25H28F3N5S/c1-17-18(8-5-11-29-17)22-30-31-23(32(22)2)34-14-6-12-33-13-10-24(16-33)15-21(24)19-7-3-4-9-20(19)25(26,27)28/h3-5,7-9,11,21H,6,10,12-16H2,1-2H3/t21?,24-/s2
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363n/an/an/an/an/an/an/an/a



Indivior UK Limited

US Patent


Assay Description
CHO cells stably expressing human dopamine receptor type 2, long variant (hD2L), coupled to Gα16 protein (CHO-Gα16-hD2L) were re-suspended ...


US Patent US10239870 (2019)

More data for this
Ligand-Target Pair
Dopamine D2 S receptor


(Homo sapiens (Human))
BDBM50192243
PNG
(CHEMBL3978613 | US10239870, Example 234)
Show SMILES Cc1cc(on1)-c1nnc(SCCCN2CC[C@]3(C[C@@H]3c3ccc(cc3)C(F)(F)F)C2)n1C
Show InChI InChI=1/C23H26F3N5OS/c1-15-12-19(32-29-15)20-27-28-21(30(20)2)33-11-3-9-31-10-8-22(14-31)13-18(22)16-4-6-17(7-5-16)23(24,25)26/h4-7,12,18H,3,8-11,13-14H2,1-2H3/t18-,22+/s2
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380n/an/an/an/an/an/an/an/a



Indivior UK Limited

US Patent


Assay Description
CHO cells stably expressing human dopamine receptor type 2, long variant (hD2L), coupled to Gα16 protein (CHO-Gα16-hD2L) were re-suspended ...


US Patent US10239870 (2019)

More data for this
Ligand-Target Pair
Dopamine D2 S receptor


(Homo sapiens (Human))
BDBM50192240
PNG
(CHEMBL3941818 | US10239870, Example 278)
Show SMILES Cn1c(SCCCN2CC[C@]3(C[C@@H]3c3ccc(cc3)C(F)(F)F)C2)nnc1-c1ccc(cc1)-c1ncco1
Show InChI InChI=1/C28H28F3N5OS/c1-35-24(20-3-5-21(6-4-20)25-32-12-15-37-25)33-34-26(35)38-16-2-13-36-14-11-27(18-36)17-23(27)19-7-9-22(10-8-19)28(29,30)31/h3-10,12,15,23H,2,11,13-14,16-18H2,1H3/t23-,27+/s2
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389n/an/an/an/an/an/an/an/a



Indivior UK Limited

US Patent


Assay Description
CHO cells stably expressing human dopamine receptor type 2, long variant (hD2L), coupled to Gα16 protein (CHO-Gα16-hD2L) were re-suspended ...


US Patent US10239870 (2019)

More data for this
Ligand-Target Pair
Dopamine D2 S receptor


(Homo sapiens (Human))
BDBM50192033
PNG
(CHEMBL3905582 | US10239870, Example 261)
Show SMILES Cn1c(SCCCN2CC[C@]3(C[C@@H]3c3ccc(cc3)C(F)(F)F)C2)nnc1-c1csnn1
Show InChI InChI=1/C21H23F3N6S2/c1-29-18(17-12-32-28-25-17)26-27-19(29)31-10-2-8-30-9-7-20(13-30)11-16(20)14-3-5-15(6-4-14)21(22,23)24/h3-6,12,16H,2,7-11,13H2,1H3/t16-,20+/s2
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398n/an/an/an/an/an/an/an/a



Indivior UK Limited

US Patent


Assay Description
CHO cells stably expressing human dopamine receptor type 2, long variant (hD2L), coupled to Gα16 protein (CHO-Gα16-hD2L) were re-suspended ...


US Patent US10239870 (2019)

More data for this
Ligand-Target Pair
Dopamine D2 S receptor


(Homo sapiens (Human))
BDBM371975
PNG
(US10239870, Example 221)
Show SMILES Cn1c(SCCCN2CC[C@]3(CC3c3ccc(cc3F)C(F)(F)F)C2)nnc1-c1cnccn1
Show InChI InChI=1/C23H24F4N6S/c1-32-20(19-13-28-6-7-29-19)30-31-21(32)34-10-2-8-33-9-5-22(14-33)12-17(22)16-4-3-15(11-18(16)24)23(25,26)27/h3-4,6-7,11,13,17H,2,5,8-10,12,14H2,1H3/t17?,22-/s2
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427n/an/an/an/an/an/an/an/a



Indivior UK Limited

US Patent


Assay Description
CHO cells stably expressing human dopamine receptor type 2, long variant (hD2L), coupled to Gα16 protein (CHO-Gα16-hD2L) were re-suspended ...


US Patent US10239870 (2019)

More data for this
Ligand-Target Pair
Dopamine D2 S receptor


(Homo sapiens (Human))
BDBM50192099
PNG
(CHEMBL3914556 | US10239870, Example 244)
Show SMILES Cn1c(SCCCN2CC[C@]3(C[C@@H]3c3ccc(cc3)C(F)(F)F)C2)nnc1-c1nccs1
Show InChI InChI=1/C22H24F3N5S2/c1-29-18(19-26-8-12-31-19)27-28-20(29)32-11-2-9-30-10-7-21(14-30)13-17(21)15-3-5-16(6-4-15)22(23,24)25/h3-6,8,12,17H,2,7,9-11,13-14H2,1H3/t17-,21+/s2
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427n/an/an/an/an/an/an/an/a



Indivior UK Limited

US Patent


Assay Description
CHO cells stably expressing human dopamine receptor type 2, long variant (hD2L), coupled to Gα16 protein (CHO-Gα16-hD2L) were re-suspended ...


US Patent US10239870 (2019)

More data for this
Ligand-Target Pair
Dopamine D2 S receptor


(Homo sapiens (Human))
BDBM371952
PNG
(US10239870, Example 189)
Show SMILES Cn1c(SCCCN2CC[C@]3(C[C@@H]3c3ccc(cc3)C(F)(F)F)C2)nnc1-c1ccc(cn1)C(N)=O
Show InChI InChI=1/C25H27F3N6OS/c1-33-22(20-8-5-17(14-30-20)21(29)35)31-32-23(33)36-12-2-10-34-11-9-24(15-34)13-19(24)16-3-6-18(7-4-16)25(26,27)28/h3-8,14,19H,2,9-13,15H2,1H3,(H2,29,35)/t19-,24+/s2
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437n/an/an/an/an/an/an/an/a



Indivior UK Limited

US Patent


Assay Description
CHO cells stably expressing human dopamine receptor type 2, long variant (hD2L), coupled to Gα16 protein (CHO-Gα16-hD2L) were re-suspended ...


US Patent US10239870 (2019)

More data for this
Ligand-Target Pair
Dopamine D2 S receptor


(Homo sapiens (Human))
BDBM371956
PNG
(US10239870, Example 193)
Show SMILES Cn1c(SCCCN2CC[C@]3(C[C@@H]3c3ccc(cc3)C(F)(F)F)C2)nnc1-c1cccc(n1)C(N)=O
Show InChI InChI=1/C25H27F3N6OS/c1-33-22(20-5-2-4-19(30-20)21(29)35)31-32-23(33)36-13-3-11-34-12-10-24(15-34)14-18(24)16-6-8-17(9-7-16)25(26,27)28/h2,4-9,18H,3,10-15H2,1H3,(H2,29,35)/t18-,24+/s2
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437n/an/an/an/an/an/an/an/a



Indivior UK Limited

US Patent


Assay Description
CHO cells stably expressing human dopamine receptor type 2, long variant (hD2L), coupled to Gα16 protein (CHO-Gα16-hD2L) were re-suspended ...


US Patent US10239870 (2019)

More data for this
Ligand-Target Pair
Dopamine D2 S receptor


(Homo sapiens (Human))
BDBM371955
PNG
(US10239870, Example 192)
Show SMILES Cn1c(SCCCN2CC[C@]3(C[C@@H]3c3ccc(cc3)C(F)(F)F)C2)nnc1-c1cncc(c1)C(N)=O
Show InChI InChI=1/C25H27F3N6OS/c1-33-22(18-11-17(21(29)35)13-30-14-18)31-32-23(33)36-10-2-8-34-9-7-24(15-34)12-20(24)16-3-5-19(6-4-16)25(26,27)28/h3-6,11,13-14,20H,2,7-10,12,15H2,1H3,(H2,29,35)/t20-,24+/s2
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437n/an/an/an/an/an/an/an/a



Indivior UK Limited

US Patent


Assay Description
CHO cells stably expressing human dopamine receptor type 2, long variant (hD2L), coupled to Gα16 protein (CHO-Gα16-hD2L) were re-suspended ...


US Patent US10239870 (2019)

More data for this
Ligand-Target Pair
Dopamine D2 S receptor


(Homo sapiens (Human))
BDBM371905
PNG
(US10239870, Example 129)
Show SMILES Cn1c(SCCCN2CC[C@]3(CC3c3ccc(cc3F)C(F)(F)F)C2)nnc1-c1ccc(=O)[nH]c1
Show InChI InChI=1/C24H25F4N5OS/c1-32-21(15-3-6-20(34)29-13-15)30-31-22(32)35-10-2-8-33-9-7-23(14-33)12-18(23)17-5-4-16(11-19(17)25)24(26,27)28/h3-6,11,13,18H,2,7-10,12,14H2,1H3,(H,29,34)/t18?,23-/s2
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447n/an/an/an/an/an/an/an/a



Indivior UK Limited

US Patent


Assay Description
CHO cells stably expressing human dopamine receptor type 2, long variant (hD2L), coupled to Gα16 protein (CHO-Gα16-hD2L) were re-suspended ...


US Patent US10239870 (2019)

More data for this
Ligand-Target Pair
Dopamine D2 S receptor


(Homo sapiens (Human))
BDBM371898
PNG
(US10239870, Example 122)
Show SMILES Cn1c(SCCCN2CC[C@]3(CC3c3ccc(cc3)C(F)(F)F)C2)nnc1-c1cccc(=O)[nH]1
Show InChI InChI=1/C24H26F3N5OS/c1-31-21(19-4-2-5-20(33)28-19)29-30-22(31)34-13-3-11-32-12-10-23(15-32)14-18(23)16-6-8-17(9-7-16)24(25,26)27/h2,4-9,18H,3,10-15H2,1H3,(H,28,33)/t18?,23-/s2
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457n/an/an/an/an/an/an/an/a



Indivior UK Limited

US Patent


Assay Description
CHO cells stably expressing human dopamine receptor type 2, long variant (hD2L), coupled to Gα16 protein (CHO-Gα16-hD2L) were re-suspended ...


US Patent US10239870 (2019)

More data for this
Ligand-Target Pair
Dopamine D2 S receptor


(Homo sapiens (Human))
BDBM50192315
PNG
(CHEMBL3981856 | US10239870, Example 287)
Show SMILES Cn1c(SCCCN2CC[C@]3(C[C@@H]3c3ccc(cc3)C(F)(F)F)C2)nnc1-c1ccc(CC(N)=O)cc1
Show InChI InChI=1/C27H30F3N5OS/c1-34-24(20-5-3-18(4-6-20)15-23(31)36)32-33-25(34)37-14-2-12-35-13-11-26(17-35)16-22(26)19-7-9-21(10-8-19)27(28,29)30/h3-10,22H,2,11-17H2,1H3,(H2,31,36)/t22-,26+/s2
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468n/an/an/an/an/an/an/an/a



Indivior UK Limited

US Patent


Assay Description
CHO cells stably expressing human dopamine receptor type 2, long variant (hD2L), coupled to Gα16 protein (CHO-Gα16-hD2L) were re-suspended ...


US Patent US10239870 (2019)

More data for this
Ligand-Target Pair
Dopamine D2 S receptor


(Homo sapiens (Human))
BDBM371980
PNG
(US10239870, Example 228)
Show SMILES Cn1c(SCCCN2CC[C@]3(C[C@@H]3c3ccc(cc3)C(F)(F)F)C2)nnc1-c1cnc(cn1)C(N)=O
Show InChI InChI=1/C24H26F3N7OS/c1-33-21(19-13-29-18(12-30-19)20(28)35)31-32-22(33)36-10-2-8-34-9-7-23(14-34)11-17(23)15-3-5-16(6-4-15)24(25,26)27/h3-6,12-13,17H,2,7-11,14H2,1H3,(H2,28,35)/t17-,23+/s2
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468n/an/an/an/an/an/an/an/a



Indivior UK Limited

US Patent


Assay Description
CHO cells stably expressing human dopamine receptor type 2, long variant (hD2L), coupled to Gα16 protein (CHO-Gα16-hD2L) were re-suspended ...


US Patent US10239870 (2019)

More data for this
Ligand-Target Pair
Dopamine D2 S receptor


(Homo sapiens (Human))
BDBM50192250
PNG
(CHEMBL3895585 | US10239870, Example 240)
Show SMILES Cn1c(SCCCN2CC[C@]3(C[C@H]3c3ccc(cc3)C(F)(F)F)C2)nnc1-c1nccs1
Show InChI InChI=1/C22H24F3N5S2/c1-29-18(19-26-8-12-31-19)27-28-20(29)32-11-2-9-30-10-7-21(14-30)13-17(21)15-3-5-16(6-4-15)22(23,24)25/h3-6,8,12,17H,2,7,9-11,13-14H2,1H3/t17-,21-/s2
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468n/an/an/an/an/an/an/an/a



Indivior UK Limited

US Patent


Assay Description
CHO cells stably expressing human dopamine receptor type 2, long variant (hD2L), coupled to Gα16 protein (CHO-Gα16-hD2L) were re-suspended ...


US Patent US10239870 (2019)

More data for this
Ligand-Target Pair
Dopamine D2 S receptor


(Homo sapiens (Human))
BDBM372023
PNG
(US10239870, Example 286)
Show SMILES Cn1c(SCCCN2CC[C@]3(C[C@@H]3c3ccc(cc3)C(F)(F)F)C2)nnc1-c1ccc(CC#N)cc1
Show InChI InChI=1/C27H28F3N5S/c1-34-24(21-5-3-19(4-6-21)11-13-31)32-33-25(34)36-16-2-14-35-15-12-26(18-35)17-23(26)20-7-9-22(10-8-20)27(28,29)30/h3-10,23H,2,11-12,14-18H2,1H3/t23-,26+/s2
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468n/an/an/an/an/an/an/an/a



Indivior UK Limited

US Patent


Assay Description
CHO cells stably expressing human dopamine receptor type 2, long variant (hD2L), coupled to Gα16 protein (CHO-Gα16-hD2L) were re-suspended ...


US Patent US10239870 (2019)

More data for this
Ligand-Target Pair
Dopamine D2 S receptor


(Homo sapiens (Human))
BDBM371996
PNG
(US10239870, Example 254)
Show SMILES Cn1c(SCCCN2CC[C@]3(CC3c3ccc(cc3)C(F)(F)F)C2)nnc1-c1ccco1
Show InChI InChI=1/C23H25F3N4OS/c1-29-20(19-4-2-12-31-19)27-28-21(29)32-13-3-10-30-11-9-22(15-30)14-18(22)16-5-7-17(8-6-16)23(24,25)26/h2,4-8,12,18H,3,9-11,13-15H2,1H3/t18?,22-/s2
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479n/an/an/an/an/an/an/an/a



Indivior UK Limited

US Patent


Assay Description
CHO cells stably expressing human dopamine receptor type 2, long variant (hD2L), coupled to Gα16 protein (CHO-Gα16-hD2L) were re-suspended ...


US Patent US10239870 (2019)

More data for this
Ligand-Target Pair
Dopamine D2 S receptor


(Homo sapiens (Human))
BDBM372015
PNG
(US10239870, Example 275)
Show SMILES Cc1nc(no1)-c1ccc(cc1)-c1nnc(SCCCN2CC[C@]3(C[C@@H]3c3ccc(cc3)C(F)(F)F)C2)n1C
Show InChI InChI=1/C28H29F3N6OS/c1-18-32-24(35-38-18)20-4-6-21(7-5-20)25-33-34-26(36(25)2)39-15-3-13-37-14-12-27(17-37)16-23(27)19-8-10-22(11-9-19)28(29,30)31/h4-11,23H,3,12-17H2,1-2H3/t23-,27+/s2
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479n/an/an/an/an/an/an/an/a



Indivior UK Limited

US Patent


Assay Description
CHO cells stably expressing human dopamine receptor type 2, long variant (hD2L), coupled to Gα16 protein (CHO-Gα16-hD2L) were re-suspended ...


US Patent US10239870 (2019)

More data for this
Ligand-Target Pair
Dopamine D2 S receptor


(Homo sapiens (Human))
BDBM50192326
PNG
(CHEMBL3955608 | US10239870, Example 220)
Show SMILES Cn1c(SCCCN2CC[C@]3(C[C@@H]3c3ccc(cc3)C(F)(F)F)C2)nnc1-c1cnccn1
Show InChI InChI=1/C23H25F3N6S/c1-31-20(19-14-27-8-9-28-19)29-30-21(31)33-12-2-10-32-11-7-22(15-32)13-18(22)16-3-5-17(6-4-16)23(24,25)26/h3-6,8-9,14,18H,2,7,10-13,15H2,1H3/t18-,22+/s2
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479n/an/an/an/an/an/an/an/a



Indivior UK Limited

US Patent


Assay Description
CHO cells stably expressing human dopamine receptor type 2, long variant (hD2L), coupled to Gα16 protein (CHO-Gα16-hD2L) were re-suspended ...


US Patent US10239870 (2019)

More data for this
Ligand-Target Pair
Dopamine D2 S receptor


(Homo sapiens (Human))
BDBM50192319
PNG
(CHEMBL3920167 | US10239870, Example 279)
Show SMILES Cn1c(SCCCN2CC[C@]3(C[C@@H]3c3ccc(cc3)C(F)(F)F)C2)nnc1-c1cccc(c1)-c1ncco1
Show InChI InChI=1/C28H28F3N5OS/c1-35-24(20-4-2-5-21(16-20)25-32-11-14-37-25)33-34-26(35)38-15-3-12-36-13-10-27(18-36)17-23(27)19-6-8-22(9-7-19)28(29,30)31/h2,4-9,11,14,16,23H,3,10,12-13,15,17-18H2,1H3/t23-,27+/s2
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501n/an/an/an/an/an/an/an/a



Indivior UK Limited

US Patent


Assay Description
CHO cells stably expressing human dopamine receptor type 2, long variant (hD2L), coupled to Gα16 protein (CHO-Gα16-hD2L) were re-suspended ...


US Patent US10239870 (2019)

More data for this
Ligand-Target Pair
Dopamine D2 S receptor


(Homo sapiens (Human))
BDBM371997
PNG
(US10239870, Example 255)
Show SMILES Cn1c(SCCCN2CC[C@]3(CC3c3ccc(cc3)C(F)(F)F)C2)nnc1-c1ccoc1
Show InChI InChI=1/C23H25F3N4OS/c1-29-20(17-7-11-31-14-17)27-28-21(29)32-12-2-9-30-10-8-22(15-30)13-19(22)16-3-5-18(6-4-16)23(24,25)26/h3-7,11,14,19H,2,8-10,12-13,15H2,1H3/t19?,22-/s2
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501n/an/an/an/an/an/an/an/a



Indivior UK Limited

US Patent


Assay Description
CHO cells stably expressing human dopamine receptor type 2, long variant (hD2L), coupled to Gα16 protein (CHO-Gα16-hD2L) were re-suspended ...


US Patent US10239870 (2019)

More data for this
Ligand-Target Pair
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