Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
alpha-Glucosidase (alpha-Glu) (Homo sapiens) | BDBM18351![]() ((2R,3R,4R,5S)-2-(Hydroxymethyl)piperidine-3,4,5-tr...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | Purchase CHEMBL KEGG MMDB PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 1.00E+3 | n/a | n/a | n/a | n/a | 4.5 | 37 |
Hokuriku University | Assay Description Enzyme activity was determined as the production of fluorescent 4-MU from the substrate. The fluorescence was measured (excitation 362 nm, emission 4... | Bioorg Med Chem 14: 7736-44 (2006) Article DOI: 10.1016/j.bmc.2006.08.003 BindingDB Entry DOI: 10.7270/Q2BZ649B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
alpha-Glucosidase (alpha-Glu) (Homo sapiens) | BDBM18366![]() ((2R,3R,5S,6R)-2,6-bis(hydroxymethyl)piperidine-3,4...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | Purchase PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 1.00E+3 | n/a | n/a | n/a | n/a | 4.5 | 37 |
Hokuriku University | Assay Description Enzyme activity was determined as the production of fluorescent 4-MU from the substrate. The fluorescence was measured (excitation 362 nm, emission 4... | Bioorg Med Chem 14: 7736-44 (2006) Article DOI: 10.1016/j.bmc.2006.08.003 BindingDB Entry DOI: 10.7270/Q2BZ649B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
alpha-Glucosidase (alpha-Glu) (Homo sapiens) | BDBM18353![]() ((2R,3R,4R,5S)-2-(hydroxymethyl)-1-methylpiperidine...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | Purchase CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 1.00E+3 | n/a | n/a | n/a | n/a | 4.5 | 37 |
Hokuriku University | Assay Description Enzyme activity was determined as the production of fluorescent 4-MU from the substrate. The fluorescence was measured (excitation 362 nm, emission 4... | Bioorg Med Chem 14: 7736-44 (2006) Article DOI: 10.1016/j.bmc.2006.08.003 BindingDB Entry DOI: 10.7270/Q2BZ649B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
alpha-Glucosidase (alpha-Glu) (Homo sapiens) | BDBM18358![]() ((2R,3R,4R,5S)-2-(hydroxymethyl)-1-nonylpiperidine-...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | Purchase DrugBank MMDB PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | 1.50E+3 | n/a | n/a | n/a | n/a | 4.5 | 37 |
Hokuriku University | Assay Description Enzyme activity was determined as the production of fluorescent 4-MU from the substrate. The fluorescence was measured (excitation 362 nm, emission 4... | Bioorg Med Chem 14: 7736-44 (2006) Article DOI: 10.1016/j.bmc.2006.08.003 BindingDB Entry DOI: 10.7270/Q2BZ649B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
alpha-Glucosidase (alpha-Glu) (Homo sapiens) | BDBM18357![]() ((2R,3R,4R,5S)-2-(hydroxymethyl)-1-octylpiperidine-...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 2.10E+3 | n/a | n/a | n/a | n/a | 4.5 | 37 |
Hokuriku University | Assay Description Enzyme activity was determined as the production of fluorescent 4-MU from the substrate. The fluorescence was measured (excitation 362 nm, emission 4... | Bioorg Med Chem 14: 7736-44 (2006) Article DOI: 10.1016/j.bmc.2006.08.003 BindingDB Entry DOI: 10.7270/Q2BZ649B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
alpha-Glucosidase (alpha-Glu) (Homo sapiens) | BDBM18356![]() ((2R,3R,4R,5S)-1-hexyl-2-(hydroxymethyl)piperidine-...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 4.00E+3 | n/a | n/a | n/a | n/a | 4.5 | 37 |
Hokuriku University | Assay Description Enzyme activity was determined as the production of fluorescent 4-MU from the substrate. The fluorescence was measured (excitation 362 nm, emission 4... | Bioorg Med Chem 14: 7736-44 (2006) Article DOI: 10.1016/j.bmc.2006.08.003 BindingDB Entry DOI: 10.7270/Q2BZ649B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
alpha-Glucosidase (alpha-Glu) (Homo sapiens) | BDBM18364![]() ((2R,3R,4R,5S,6R)-2-(hydroxymethyl)-6-nonylpiperidi...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 4.80E+3 | n/a | n/a | n/a | n/a | 4.5 | 37 |
Hokuriku University | Assay Description Enzyme activity was determined as the production of fluorescent 4-MU from the substrate. The fluorescence was measured (excitation 362 nm, emission 4... | Bioorg Med Chem 14: 7736-44 (2006) Article DOI: 10.1016/j.bmc.2006.08.003 BindingDB Entry DOI: 10.7270/Q2BZ649B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
alpha-Glucosidase (alpha-Glu) (Homo sapiens) | BDBM18355![]() ((2R,3R,4R,5S)-1-butyl-2-(hydroxymethyl)piperidine-...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | Purchase CHEMBL DrugBank MMDB PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | 5.00E+3 | n/a | n/a | n/a | n/a | 4.5 | 37 |
Hokuriku University | Assay Description Enzyme activity was determined as the production of fluorescent 4-MU from the substrate. The fluorescence was measured (excitation 362 nm, emission 4... | Bioorg Med Chem 14: 7736-44 (2006) Article DOI: 10.1016/j.bmc.2006.08.003 BindingDB Entry DOI: 10.7270/Q2BZ649B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
alpha-Glucosidase (alpha-Glu) (Homo sapiens) | BDBM18363![]() ((2R,3R,4R,5S,6R)-2-(hydroxymethyl)-6-octylpiperidi...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5.00E+3 | n/a | n/a | n/a | n/a | 4.5 | 37 |
Hokuriku University | Assay Description Enzyme activity was determined as the production of fluorescent 4-MU from the substrate. The fluorescence was measured (excitation 362 nm, emission 4... | Bioorg Med Chem 14: 7736-44 (2006) Article DOI: 10.1016/j.bmc.2006.08.003 BindingDB Entry DOI: 10.7270/Q2BZ649B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
alpha-Glucosidase (alpha-Glu) (Homo sapiens) | BDBM18362![]() ((2R,3S,4R,5R,6R)-2-hexyl-6-(hydroxymethyl)piperidi...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.20E+4 | n/a | n/a | n/a | n/a | 4.5 | 37 |
Hokuriku University | Assay Description Enzyme activity was determined as the production of fluorescent 4-MU from the substrate. The fluorescence was measured (excitation 362 nm, emission 4... | Bioorg Med Chem 14: 7736-44 (2006) Article DOI: 10.1016/j.bmc.2006.08.003 BindingDB Entry DOI: 10.7270/Q2BZ649B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
alpha-Glucosidase (alpha-Glu) (Homo sapiens) | BDBM18359![]() ((2R,3R,4R,5S,6R)-2-(hydroxymethyl)-6-methylpiperid...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 2.80E+4 | n/a | n/a | n/a | n/a | 4.5 | 37 |
Hokuriku University | Assay Description Enzyme activity was determined as the production of fluorescent 4-MU from the substrate. The fluorescence was measured (excitation 362 nm, emission 4... | Bioorg Med Chem 14: 7736-44 (2006) Article DOI: 10.1016/j.bmc.2006.08.003 BindingDB Entry DOI: 10.7270/Q2BZ649B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
alpha-Glucosidase (alpha-Glu) (Homo sapiens) | BDBM18361![]() ((2R,3S,4R,5R,6R)-2-butyl-6-(hydroxymethyl)piperidi...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 3.10E+4 | n/a | n/a | n/a | n/a | 4.5 | 37 |
Hokuriku University | Assay Description Enzyme activity was determined as the production of fluorescent 4-MU from the substrate. The fluorescence was measured (excitation 362 nm, emission 4... | Bioorg Med Chem 14: 7736-44 (2006) Article DOI: 10.1016/j.bmc.2006.08.003 BindingDB Entry DOI: 10.7270/Q2BZ649B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
alpha-Glucosidase (alpha-Glu) (Homo sapiens) | BDBM18354![]() ((2R,3R,4R,5S)-2-(hydroxymethyl)-1-propylpiperidine...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 5.60E+4 | n/a | n/a | n/a | n/a | 4.5 | 37 |
Hokuriku University | Assay Description Enzyme activity was determined as the production of fluorescent 4-MU from the substrate. The fluorescence was measured (excitation 362 nm, emission 4... | Bioorg Med Chem 14: 7736-44 (2006) Article DOI: 10.1016/j.bmc.2006.08.003 BindingDB Entry DOI: 10.7270/Q2BZ649B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
alpha-Glucosidase (alpha-Glu) (Homo sapiens) | BDBM18360![]() ((2R,3R,4R,5S,6R)-2-(hydroxymethyl)-6-propylpiperid...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.70E+5 | n/a | n/a | n/a | n/a | 4.5 | 37 |
Hokuriku University | Assay Description Enzyme activity was determined as the production of fluorescent 4-MU from the substrate. The fluorescence was measured (excitation 362 nm, emission 4... | Bioorg Med Chem 14: 7736-44 (2006) Article DOI: 10.1016/j.bmc.2006.08.003 BindingDB Entry DOI: 10.7270/Q2BZ649B | |||||||||||
More data for this Ligand-Target Pair |