Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Histone acetyltransferase KAT6A (Homo sapiens) | BDBM50518833![]() (CHEMBL4528993) | PDB UniProtKB/SwissProt GoogleScholar | UniChem | Article PubMed | n/a | n/a | 2 | n/a | n/a | n/a | n/a | n/a | n/a |
Cancer Therapeutics CRC Curated by ChEMBL | Assay Description Inhibition of N-terminal NusA-fused His6-tagged human KAT6A (507 to 778 residues) expressed in Escherichia coli BL21 (DE3) cells using 0.4 uM acetyl ... | J Med Chem 62: 7146-7159 (2019) Article DOI: null | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT6A (Homo sapiens) | BDBM50527224![]() (CHEMBL4468833) | PDB UniProtKB/SwissProt GoogleScholar | UniChem | Article PubMed | n/a | n/a | 5 | n/a | n/a | n/a | n/a | n/a | n/a |
Monash University (Parkville Campus) Curated by ChEMBL | Assay Description Inhibition of N-terminal NusA-fused His6-tagged human KAT6A (507 to 778 residues) expressed in Escherichia coli BL21 (DE3) cells using 0.4 uM acetyl ... | J Med Chem 63: 4655-4684 (2020) Article DOI: null | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT6A (Homo sapiens) | BDBM50527244![]() (CHEMBL4437798) | PDB UniProtKB/SwissProt GoogleScholar | UniChem | Article PubMed | n/a | n/a | 5.5 | n/a | n/a | n/a | n/a | n/a | n/a |
Monash University (Parkville Campus) Curated by ChEMBL | Assay Description Inhibition of N-terminal NusA-fused His6-tagged human KAT6A (507 to 778 residues) expressed in Escherichia coli BL21 (DE3) cells using 0.4 uM acetyl ... | J Med Chem 63: 4655-4684 (2020) Article DOI: null | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT6A (Homo sapiens) | BDBM50527381![]() (CHEMBL4466823) | PDB UniProtKB/SwissProt GoogleScholar | UniChem | Article PubMed | n/a | n/a | 6 | n/a | n/a | n/a | n/a | n/a | n/a |
Monash University (Parkville Campus) Curated by ChEMBL | Assay Description Inhibition of N-terminal NusA-fused His6-tagged human KAT6A (507 to 778 residues) expressed in Escherichia coli BL21 (DE3) cells using 0.4 uM acetyl ... | J Med Chem 63: 4655-4684 (2020) Article DOI: null | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT6A (Homo sapiens) | BDBM50527355![]() (CHEMBL4456585) | PDB UniProtKB/SwissProt GoogleScholar | PDB UniChem | Article PubMed | n/a | n/a | 6.30 | n/a | n/a | n/a | n/a | n/a | n/a |
Monash University (Parkville Campus) Curated by ChEMBL | Assay Description Inhibition of N-terminal NusA-fused His6-tagged human KAT6A (507 to 778 residues) expressed in Escherichia coli BL21 (DE3) cells using 0.4 uM acetyl ... | J Med Chem 63: 4655-4684 (2020) Article DOI: null | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT6A (Homo sapiens) | BDBM50527250![]() (CHEMBL4475883) | PDB UniProtKB/SwissProt GoogleScholar | UniChem | Article PubMed | n/a | n/a | 7 | n/a | n/a | n/a | n/a | n/a | n/a |
Monash University (Parkville Campus) Curated by ChEMBL | Assay Description Inhibition of N-terminal NusA-fused His6-tagged human KAT6A (507 to 778 residues) expressed in Escherichia coli BL21 (DE3) cells using 0.4 uM acetyl ... | J Med Chem 63: 4655-4684 (2020) Article DOI: null | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT6A (Homo sapiens) | BDBM50527238![]() (CHEMBL4539384) | PDB UniProtKB/SwissProt GoogleScholar | UniChem | Article PubMed | n/a | n/a | 8 | n/a | n/a | n/a | n/a | n/a | n/a |
Monash University (Parkville Campus) Curated by ChEMBL | Assay Description Inhibition of N-terminal NusA-fused His6-tagged human KAT6A (507 to 778 residues) expressed in Escherichia coli BL21 (DE3) cells using 0.4 uM acetyl ... | J Med Chem 63: 4655-4684 (2020) Article DOI: null | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT6A (Homo sapiens) | BDBM50518832![]() (CHEMBL4455897) | PDB UniProtKB/SwissProt GoogleScholar | PDB UniChem | Article PubMed | n/a | n/a | 8 | n/a | n/a | n/a | n/a | n/a | n/a |
Cancer Therapeutics CRC Curated by ChEMBL | Assay Description Inhibition of N-terminal NusA-fused His6-tagged human KAT6A (507 to 778 residues) expressed in Escherichia coli BL21 (DE3) cells using 0.4 uM acetyl ... | J Med Chem 62: 7146-7159 (2019) Article DOI: null | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT6A (Homo sapiens) | BDBM50527245![]() (CHEMBL4521125) | PDB UniProtKB/SwissProt GoogleScholar | UniChem | Article PubMed | n/a | n/a | 9 | n/a | n/a | n/a | n/a | n/a | n/a |
Monash University (Parkville Campus) Curated by ChEMBL | Assay Description Inhibition of N-terminal NusA-fused His6-tagged human KAT6A (507 to 778 residues) expressed in Escherichia coli BL21 (DE3) cells using 0.4 uM acetyl ... | J Med Chem 63: 4655-4684 (2020) Article DOI: null | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT6A (Homo sapiens) | BDBM50527328![]() (CHEMBL4441439) | PDB UniProtKB/SwissProt GoogleScholar | UniChem | Article PubMed | n/a | n/a | 9 | n/a | n/a | n/a | n/a | n/a | n/a |
Monash University (Parkville Campus) Curated by ChEMBL | Assay Description Inhibition of N-terminal NusA-fused His6-tagged human KAT6A (507 to 778 residues) expressed in Escherichia coli BL21 (DE3) cells using 0.4 uM acetyl ... | J Med Chem 63: 4655-4684 (2020) Article DOI: null | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT6A (Homo sapiens) | BDBM50527225![]() (CHEMBL4565790) | PDB UniProtKB/SwissProt GoogleScholar | UniChem | Article PubMed | n/a | n/a | 9.40 | n/a | n/a | n/a | n/a | n/a | n/a |
Monash University (Parkville Campus) Curated by ChEMBL | Assay Description Inhibition of N-terminal NusA-fused His6-tagged human KAT6A (507 to 778 residues) expressed in Escherichia coli BL21 (DE3) cells using 0.4 uM acetyl ... | J Med Chem 63: 4655-4684 (2020) Article DOI: null | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT6A (Homo sapiens) | BDBM50518831![]() (CHEMBL4464835) | PDB UniProtKB/SwissProt GoogleScholar | UniChem | Article PubMed | n/a | n/a | 10 | n/a | n/a | n/a | n/a | n/a | n/a |
Cancer Therapeutics CRC Curated by ChEMBL | Assay Description Inhibition of N-terminal NusA-fused His6-tagged human KAT6A (507 to 778 residues) expressed in Escherichia coli BL21 (DE3) cells using 0.4 uM acetyl ... | J Med Chem 62: 7146-7159 (2019) Article DOI: null | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT6A (Homo sapiens) | BDBM50527243![]() (CHEMBL4458272) | PDB UniProtKB/SwissProt GoogleScholar | UniChem | Article PubMed | n/a | n/a | 11 | n/a | n/a | n/a | n/a | n/a | n/a |
Monash University (Parkville Campus) Curated by ChEMBL | Assay Description Inhibition of N-terminal NusA-fused His6-tagged human KAT6A (507 to 778 residues) expressed in Escherichia coli BL21 (DE3) cells using 0.4 uM acetyl ... | J Med Chem 63: 4655-4684 (2020) Article DOI: null | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT6A (Homo sapiens) | BDBM50527263![]() (CHEMBL4465716) | PDB UniProtKB/SwissProt GoogleScholar | UniChem | Article PubMed | n/a | n/a | 13 | n/a | n/a | n/a | n/a | n/a | n/a |
Monash University (Parkville Campus) Curated by ChEMBL | Assay Description Inhibition of N-terminal NusA-fused His6-tagged human KAT6A (507 to 778 residues) expressed in Escherichia coli BL21 (DE3) cells using 0.4 uM acetyl ... | J Med Chem 63: 4655-4684 (2020) Article DOI: null | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT6A (Homo sapiens) | BDBM50527246![]() (CHEMBL4445473) | PDB UniProtKB/SwissProt GoogleScholar | UniChem | Article PubMed | n/a | n/a | 13 | n/a | n/a | n/a | n/a | n/a | n/a |
Monash University (Parkville Campus) Curated by ChEMBL | Assay Description Inhibition of N-terminal NusA-fused His6-tagged human KAT6A (507 to 778 residues) expressed in Escherichia coli BL21 (DE3) cells using 0.4 uM acetyl ... | J Med Chem 63: 4655-4684 (2020) Article DOI: null | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT6A (Homo sapiens) | BDBM50527232![]() (CHEMBL4436877) | PDB UniProtKB/SwissProt GoogleScholar | UniChem | Article PubMed | n/a | n/a | 14 | n/a | n/a | n/a | n/a | n/a | n/a |
Monash University (Parkville Campus) Curated by ChEMBL | Assay Description Inhibition of N-terminal NusA-fused His6-tagged human KAT6A (507 to 778 residues) expressed in Escherichia coli BL21 (DE3) cells using 0.4 uM acetyl ... | J Med Chem 63: 4655-4684 (2020) Article DOI: null | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT6A (Homo sapiens) | BDBM50527240![]() (CHEMBL4541948) | PDB UniProtKB/SwissProt GoogleScholar | UniChem | Article PubMed | n/a | n/a | 14 | n/a | n/a | n/a | n/a | n/a | n/a |
Monash University (Parkville Campus) Curated by ChEMBL | Assay Description Inhibition of N-terminal NusA-fused His6-tagged human KAT6A (507 to 778 residues) expressed in Escherichia coli BL21 (DE3) cells using 0.4 uM acetyl ... | J Med Chem 63: 4655-4684 (2020) Article DOI: null | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT6A (Homo sapiens) | BDBM50527235![]() (CHEMBL4516984) | PDB UniProtKB/SwissProt GoogleScholar | UniChem | Article PubMed | n/a | n/a | 14 | n/a | n/a | n/a | n/a | n/a | n/a |
Monash University (Parkville Campus) Curated by ChEMBL | Assay Description Inhibition of N-terminal NusA-fused His6-tagged human KAT6A (507 to 778 residues) expressed in Escherichia coli BL21 (DE3) cells using 0.4 uM acetyl ... | J Med Chem 63: 4655-4684 (2020) Article DOI: null | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT6A (Homo sapiens) | BDBM50527366![]() (CHEMBL4449163) | PDB UniProtKB/SwissProt GoogleScholar | UniChem | Article PubMed | n/a | n/a | 15 | n/a | n/a | n/a | n/a | n/a | n/a |
Monash University (Parkville Campus) Curated by ChEMBL | Assay Description Inhibition of N-terminal NusA-fused His6-tagged human KAT6A (507 to 778 residues) expressed in Escherichia coli BL21 (DE3) cells using 0.4 uM acetyl ... | J Med Chem 63: 4655-4684 (2020) Article DOI: null | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT6A (Homo sapiens) | BDBM50527382![]() (CHEMBL4518462) | PDB UniProtKB/SwissProt GoogleScholar | UniChem | Article PubMed | n/a | n/a | 16 | n/a | n/a | n/a | n/a | n/a | n/a |
Monash University (Parkville Campus) Curated by ChEMBL | Assay Description Inhibition of N-terminal NusA-fused His6-tagged human KAT6A (507 to 778 residues) expressed in Escherichia coli BL21 (DE3) cells using 0.4 uM acetyl ... | J Med Chem 63: 4655-4684 (2020) Article DOI: null | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT6A (Homo sapiens) | BDBM50527313![]() (CHEMBL4446917) | PDB UniProtKB/SwissProt GoogleScholar | UniChem | Article PubMed | n/a | n/a | 16 | n/a | n/a | n/a | n/a | n/a | n/a |
Monash University (Parkville Campus) Curated by ChEMBL | Assay Description Inhibition of N-terminal NusA-fused His6-tagged human KAT6A (507 to 778 residues) expressed in Escherichia coli BL21 (DE3) cells using 0.4 uM acetyl ... | J Med Chem 63: 4655-4684 (2020) Article DOI: null | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT6A (Homo sapiens) | BDBM50518867![]() (CHEMBL4460509) | PDB UniProtKB/SwissProt GoogleScholar | PDB UniChem | Article PubMed | n/a | n/a | 17 | n/a | n/a | n/a | n/a | n/a | n/a |
Cancer Therapeutics CRC Curated by ChEMBL | Assay Description Inhibition of N-terminal NusA-fused His6-tagged human KAT6A (507 to 778 residues) expressed in Escherichia coli BL21 (DE3) cells using 0.4 uM acetyl ... | J Med Chem 62: 7146-7159 (2019) Article DOI: null | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT6A (Homo sapiens) | BDBM50527302![]() (CHEMBL4573736) | PDB UniProtKB/SwissProt GoogleScholar | UniChem | Article PubMed | n/a | n/a | 17 | n/a | n/a | n/a | n/a | n/a | n/a |
Monash University (Parkville Campus) Curated by ChEMBL | Assay Description Inhibition of N-terminal NusA-fused His6-tagged human KAT6A (507 to 778 residues) expressed in Escherichia coli BL21 (DE3) cells using 0.4 uM acetyl ... | J Med Chem 63: 4655-4684 (2020) Article DOI: null | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT6A (Homo sapiens) | BDBM50527277![]() (CHEMBL4593500) | PDB UniProtKB/SwissProt GoogleScholar | UniChem | Article PubMed | n/a | n/a | 17 | n/a | n/a | n/a | n/a | n/a | n/a |
Monash University (Parkville Campus) Curated by ChEMBL | Assay Description Inhibition of N-terminal NusA-fused His6-tagged human KAT6A (507 to 778 residues) expressed in Escherichia coli BL21 (DE3) cells using 0.4 uM acetyl ... | J Med Chem 63: 4655-4684 (2020) Article DOI: null | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT6A (Homo sapiens) | BDBM50527346![]() (CHEMBL4566403) | PDB UniProtKB/SwissProt GoogleScholar | UniChem | Article PubMed | n/a | n/a | 18 | n/a | n/a | n/a | n/a | n/a | n/a |
Monash University (Parkville Campus) Curated by ChEMBL | Assay Description Inhibition of N-terminal NusA-fused His6-tagged human KAT6A (507 to 778 residues) expressed in Escherichia coli BL21 (DE3) cells using 0.4 uM acetyl ... | J Med Chem 63: 4655-4684 (2020) Article DOI: null | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT6A (Homo sapiens) | BDBM50527251![]() (CHEMBL4588945) | PDB UniProtKB/SwissProt GoogleScholar | UniChem | Article PubMed | n/a | n/a | 18 | n/a | n/a | n/a | n/a | n/a | n/a |
Monash University (Parkville Campus) Curated by ChEMBL | Assay Description Inhibition of N-terminal NusA-fused His6-tagged human KAT6A (507 to 778 residues) expressed in Escherichia coli BL21 (DE3) cells using 0.4 uM acetyl ... | J Med Chem 63: 4655-4684 (2020) Article DOI: null | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT6A (Homo sapiens) | BDBM50527365![]() (CHEMBL4455027) | PDB UniProtKB/SwissProt GoogleScholar | UniChem | Article PubMed | n/a | n/a | 20 | n/a | n/a | n/a | n/a | n/a | n/a |
Monash University (Parkville Campus) Curated by ChEMBL | Assay Description Inhibition of N-terminal NusA-fused His6-tagged human KAT6A (507 to 778 residues) expressed in Escherichia coli BL21 (DE3) cells using 0.4 uM acetyl ... | J Med Chem 63: 4655-4684 (2020) Article DOI: null | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT6A (Homo sapiens) | BDBM50527358![]() (CHEMBL4572653) | PDB UniProtKB/SwissProt GoogleScholar | UniChem | Article PubMed | n/a | n/a | 20 | n/a | n/a | n/a | n/a | n/a | n/a |
Monash University (Parkville Campus) Curated by ChEMBL | Assay Description Inhibition of N-terminal NusA-fused His6-tagged human KAT6A (507 to 778 residues) expressed in Escherichia coli BL21 (DE3) cells using 0.4 uM acetyl ... | J Med Chem 63: 4655-4684 (2020) Article DOI: null | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT6A (Homo sapiens) | BDBM50527221![]() (CHEMBL4464911) | PDB UniProtKB/SwissProt GoogleScholar | UniChem | Article PubMed | n/a | n/a | 23 | n/a | n/a | n/a | n/a | n/a | n/a |
Monash University (Parkville Campus) Curated by ChEMBL | Assay Description Inhibition of N-terminal NusA-fused His6-tagged human KAT6A (507 to 778 residues) expressed in Escherichia coli BL21 (DE3) cells using 0.4 uM acetyl ... | J Med Chem 63: 4655-4684 (2020) Article DOI: null | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT6A (Homo sapiens) | BDBM50527360![]() (CHEMBL4456874) | PDB UniProtKB/SwissProt GoogleScholar | UniChem | Article PubMed | n/a | n/a | 23 | n/a | n/a | n/a | n/a | n/a | n/a |
Monash University (Parkville Campus) Curated by ChEMBL | Assay Description Inhibition of N-terminal NusA-fused His6-tagged human KAT6A (507 to 778 residues) expressed in Escherichia coli BL21 (DE3) cells using 0.4 uM acetyl ... | J Med Chem 63: 4655-4684 (2020) Article DOI: null | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT6A (Homo sapiens) | BDBM50527241![]() (CHEMBL4593937) | PDB UniProtKB/SwissProt GoogleScholar | UniChem | Article PubMed | n/a | n/a | 24 | n/a | n/a | n/a | n/a | n/a | n/a |
Monash University (Parkville Campus) Curated by ChEMBL | Assay Description Inhibition of N-terminal NusA-fused His6-tagged human KAT6A (507 to 778 residues) expressed in Escherichia coli BL21 (DE3) cells using 0.4 uM acetyl ... | J Med Chem 63: 4655-4684 (2020) Article DOI: null | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT6A (Homo sapiens) | BDBM50527327![]() (CHEMBL4453559) | PDB UniProtKB/SwissProt GoogleScholar | UniChem | Article PubMed | n/a | n/a | 24 | n/a | n/a | n/a | n/a | n/a | n/a |
Monash University (Parkville Campus) Curated by ChEMBL | Assay Description Inhibition of N-terminal NusA-fused His6-tagged human KAT6A (507 to 778 residues) expressed in Escherichia coli BL21 (DE3) cells using 0.4 uM acetyl ... | J Med Chem 63: 4655-4684 (2020) Article DOI: null | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT6A (Homo sapiens) | BDBM50527264![]() (CHEMBL4530056) | PDB UniProtKB/SwissProt GoogleScholar | UniChem | Article PubMed | n/a | n/a | 24 | n/a | n/a | n/a | n/a | n/a | n/a |
Monash University (Parkville Campus) Curated by ChEMBL | Assay Description Inhibition of N-terminal NusA-fused His6-tagged human KAT6A (507 to 778 residues) expressed in Escherichia coli BL21 (DE3) cells using 0.4 uM acetyl ... | J Med Chem 63: 4655-4684 (2020) Article DOI: null | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT6A (Homo sapiens) | BDBM50527242![]() (CHEMBL4454163) | PDB UniProtKB/SwissProt GoogleScholar | UniChem | Article PubMed | n/a | n/a | 25 | n/a | n/a | n/a | n/a | n/a | n/a |
Monash University (Parkville Campus) Curated by ChEMBL | Assay Description Inhibition of N-terminal NusA-fused His6-tagged human KAT6A (507 to 778 residues) expressed in Escherichia coli BL21 (DE3) cells using 0.4 uM acetyl ... | J Med Chem 63: 4655-4684 (2020) Article DOI: null | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT6A (Homo sapiens) | BDBM50527364![]() (CHEMBL4445456) | PDB UniProtKB/SwissProt GoogleScholar | UniChem | Article PubMed | n/a | n/a | 26 | n/a | n/a | n/a | n/a | n/a | n/a |
Monash University (Parkville Campus) Curated by ChEMBL | Assay Description Inhibition of N-terminal NusA-fused His6-tagged human KAT6A (507 to 778 residues) expressed in Escherichia coli BL21 (DE3) cells using 0.4 uM acetyl ... | J Med Chem 63: 4655-4684 (2020) Article DOI: null | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT6A (Homo sapiens) | BDBM50527348![]() (CHEMBL4454507) | PDB UniProtKB/SwissProt GoogleScholar | UniChem | Article PubMed | n/a | n/a | 27 | n/a | n/a | n/a | n/a | n/a | n/a |
Monash University (Parkville Campus) Curated by ChEMBL | Assay Description Inhibition of N-terminal NusA-fused His6-tagged human KAT6A (507 to 778 residues) expressed in Escherichia coli BL21 (DE3) cells using 0.4 uM acetyl ... | J Med Chem 63: 4655-4684 (2020) Article DOI: null | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT6A (Homo sapiens) | BDBM50527265![]() (CHEMBL4559662) | PDB UniProtKB/SwissProt GoogleScholar | UniChem | Article PubMed | n/a | n/a | 27 | n/a | n/a | n/a | n/a | n/a | n/a |
Monash University (Parkville Campus) Curated by ChEMBL | Assay Description Inhibition of N-terminal NusA-fused His6-tagged human KAT6A (507 to 778 residues) expressed in Escherichia coli BL21 (DE3) cells using 0.4 uM acetyl ... | J Med Chem 63: 4655-4684 (2020) Article DOI: null | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT6B (Homo sapiens) | BDBM50518832![]() (CHEMBL4455897) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PDB UniChem | Article PubMed | n/a | n/a | 28 | n/a | n/a | n/a | n/a | n/a | n/a |
Cancer Therapeutics CRC Curated by ChEMBL | Assay Description Inhibition of N-terminal GST-tagged recombinant human KAT6B (431 to end residues) expressed in baculovirus infected Sf9 insect cells using acetyl coe... | J Med Chem 62: 7146-7159 (2019) Article DOI: null | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT6A (Homo sapiens) | BDBM50527347![]() (CHEMBL4526110) | PDB UniProtKB/SwissProt GoogleScholar | UniChem | Article PubMed | n/a | n/a | 29 | n/a | n/a | n/a | n/a | n/a | n/a |
Monash University (Parkville Campus) Curated by ChEMBL | Assay Description Inhibition of N-terminal NusA-fused His6-tagged human KAT6A (507 to 778 residues) expressed in Escherichia coli BL21 (DE3) cells using 0.4 uM acetyl ... | J Med Chem 63: 4655-4684 (2020) Article DOI: null | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT6A (Homo sapiens) | BDBM50527375![]() (CHEMBL4554392) | PDB UniProtKB/SwissProt GoogleScholar | UniChem | Article PubMed | n/a | n/a | 29 | n/a | n/a | n/a | n/a | n/a | n/a |
Monash University (Parkville Campus) Curated by ChEMBL | Assay Description Inhibition of N-terminal NusA-fused His6-tagged human KAT6A (507 to 778 residues) expressed in Escherichia coli BL21 (DE3) cells using 0.4 uM acetyl ... | J Med Chem 63: 4655-4684 (2020) Article DOI: null | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT6A (Homo sapiens) | BDBM50527227![]() (CHEMBL4450971) | PDB UniProtKB/SwissProt GoogleScholar | UniChem | Article PubMed | n/a | n/a | 30 | n/a | n/a | n/a | n/a | n/a | n/a |
Monash University (Parkville Campus) Curated by ChEMBL | Assay Description Inhibition of N-terminal NusA-fused His6-tagged human KAT6A (507 to 778 residues) expressed in Escherichia coli BL21 (DE3) cells using 0.4 uM acetyl ... | J Med Chem 63: 4655-4684 (2020) Article DOI: null | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT6A (Homo sapiens) | BDBM50527247![]() (CHEMBL4446616) | PDB UniProtKB/SwissProt GoogleScholar | UniChem | Article PubMed | n/a | n/a | 31 | n/a | n/a | n/a | n/a | n/a | n/a |
Monash University (Parkville Campus) Curated by ChEMBL | Assay Description Inhibition of N-terminal NusA-fused His6-tagged human KAT6A (507 to 778 residues) expressed in Escherichia coli BL21 (DE3) cells using 0.4 uM acetyl ... | J Med Chem 63: 4655-4684 (2020) Article DOI: null | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT6A (Homo sapiens) | BDBM50527359![]() (CHEMBL4441001) | PDB UniProtKB/SwissProt GoogleScholar | UniChem | Article PubMed | n/a | n/a | 32 | n/a | n/a | n/a | n/a | n/a | n/a |
Monash University (Parkville Campus) Curated by ChEMBL | Assay Description Inhibition of N-terminal NusA-fused His6-tagged human KAT6A (507 to 778 residues) expressed in Escherichia coli BL21 (DE3) cells using 0.4 uM acetyl ... | J Med Chem 63: 4655-4684 (2020) Article DOI: null | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT6A (Homo sapiens) | BDBM50527325![]() (CHEMBL4461380) | PDB UniProtKB/SwissProt GoogleScholar | UniChem | Article PubMed | n/a | n/a | 38 | n/a | n/a | n/a | n/a | n/a | n/a |
Monash University (Parkville Campus) Curated by ChEMBL | Assay Description Inhibition of N-terminal NusA-fused His6-tagged human KAT6A (507 to 778 residues) expressed in Escherichia coli BL21 (DE3) cells using 0.4 uM acetyl ... | J Med Chem 63: 4655-4684 (2020) Article DOI: null | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT6A (Homo sapiens) | BDBM50518845![]() (CHEMBL4473722) | PDB UniProtKB/SwissProt GoogleScholar | UniChem | Article PubMed | n/a | n/a | 43 | n/a | n/a | n/a | n/a | n/a | n/a |
Cancer Therapeutics CRC Curated by ChEMBL | Assay Description Inhibition of N-terminal NusA-fused His6-tagged human KAT6A (507 to 778 residues) expressed in Escherichia coli BL21 (DE3) cells using 0.4 uM acetyl ... | J Med Chem 62: 7146-7159 (2019) Article DOI: null | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT6A (Homo sapiens) | BDBM50527220![]() (CHEMBL4451170) | PDB UniProtKB/SwissProt GoogleScholar | UniChem | Article PubMed | n/a | n/a | 43 | n/a | n/a | n/a | n/a | n/a | n/a |
Monash University (Parkville Campus) Curated by ChEMBL | Assay Description Inhibition of N-terminal NusA-fused His6-tagged human KAT6A (507 to 778 residues) expressed in Escherichia coli BL21 (DE3) cells using 0.4 uM acetyl ... | J Med Chem 63: 4655-4684 (2020) Article DOI: null | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT6A (Homo sapiens) | BDBM50527237![]() (CHEMBL4464974) | PDB UniProtKB/SwissProt GoogleScholar | UniChem | Article PubMed | n/a | n/a | 44 | n/a | n/a | n/a | n/a | n/a | n/a |
Monash University (Parkville Campus) Curated by ChEMBL | Assay Description Inhibition of N-terminal NusA-fused His6-tagged human KAT6A (507 to 778 residues) expressed in Escherichia coli BL21 (DE3) cells using 0.4 uM acetyl ... | J Med Chem 63: 4655-4684 (2020) Article DOI: null | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT6A (Homo sapiens) | BDBM50527276![]() (CHEMBL4444077) | PDB UniProtKB/SwissProt GoogleScholar | UniChem | Article PubMed | n/a | n/a | 48 | n/a | n/a | n/a | n/a | n/a | n/a |
Monash University (Parkville Campus) Curated by ChEMBL | Assay Description Inhibition of N-terminal NusA-fused His6-tagged human KAT6A (507 to 778 residues) expressed in Escherichia coli BL21 (DE3) cells using 0.4 uM acetyl ... | J Med Chem 63: 4655-4684 (2020) Article DOI: null | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT6A (Homo sapiens) | BDBM50527304![]() (CHEMBL4560554) | PDB UniProtKB/SwissProt GoogleScholar | UniChem | Article PubMed | n/a | n/a | 52 | n/a | n/a | n/a | n/a | n/a | n/a |
Monash University (Parkville Campus) Curated by ChEMBL | Assay Description Inhibition of N-terminal NusA-fused His6-tagged human KAT6A (507 to 778 residues) expressed in Escherichia coli BL21 (DE3) cells using 0.4 uM acetyl ... | J Med Chem 63: 4655-4684 (2020) Article DOI: null | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone acetyltransferase KAT6A (Homo sapiens) | BDBM50527371![]() (CHEMBL4475866) | PDB UniProtKB/SwissProt GoogleScholar | UniChem | Article PubMed | n/a | n/a | 52 | n/a | n/a | n/a | n/a | n/a | n/a |
Monash University (Parkville Campus) Curated by ChEMBL | Assay Description Inhibition of N-terminal NusA-fused His6-tagged human KAT6A (507 to 778 residues) expressed in Escherichia coli BL21 (DE3) cells using 0.4 uM acetyl ... | J Med Chem 63: 4655-4684 (2020) Article DOI: null | |||||||||||
More data for this Ligand-Target Pair |
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