Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
cholinergic receptor, muscarinic 4 (RAT) | BDBM48044![]() (3-amino-4,6-dimethyl-N-piperonyl-thieno[2,3-b]pyri...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar | Purchase PC cid PC sid UniChem Similars | PCBioAssay | 4.68E-14 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt Screening Center for GPCRs, Ion Channels and Transporters Curated by PubChem BioAssay | Assay Description Assay Provider: Colleen Niswender Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of a Highly Selective in vitro and in vivo... | PubChem Bioassay (2009) BindingDB Entry DOI: 10.7270/Q2NV9GNV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
cholinergic receptor, muscarinic 4 (RAT) | BDBM48043![]() (3-amino-4,6-dimethyl-N-p-anisyl-thieno[2,3-b]pyrid...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar | Purchase PC cid PC sid UniChem Similars | PCBioAssay | 0.0000288 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt Screening Center for GPCRs, Ion Channels and Transporters Curated by PubChem BioAssay | Assay Description Assay Provider: Colleen Niswender Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of a Highly Selective in vitro and in vivo... | PubChem Bioassay (2009) BindingDB Entry DOI: 10.7270/Q2NV9GNV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscarinic acetylcholine receptor M1 (RAT) | BDBM43819![]() (4-[2-(2-thenoylamino)ethylamino]piperidine-1-carbo...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar | Purchase PC cid PC sid UniChem Similars | PCBioAssay | 8.39 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt Screening Center for GPCRs, Ion Channels and Transporters Curated by PubChem BioAssay | Assay Description Assay Provider: P. Jeffrey Conn Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of novel allosteric modulators of the M1 mus... | PubChem Bioassay (2009) BindingDB Entry DOI: 10.7270/Q2FJ2F7F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
cell division cycle 42 (GTP binding protein, 25kDa) (Homo sapiens (Human)) | BDBM54607![]() (4-(2,5-diphenyl-3,4-dihydropyrazol-3-yl)-N,N-dimet...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt UniProtKB/TrEMBL B.MOAD antibodypedia GoogleScholar | Purchase PC cid PC sid UniChem Patents Similars | Article PCBioAssay | 10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
NMMLSC Curated by PubChem BioAssay | Assay Description University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela... | PubChem Bioassay (2009) Article DOI: 10.1021/cb400468c BindingDB Entry DOI: 10.7270/Q2B856J1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ras-related C3 botulinum toxin substrate 1 (Mus musculus) | BDBM54623![]() (1-(2,5-dichlorophenyl)-3-(4-fluorophenyl)-5-(4-met...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt UniProtKB/TrEMBL B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem Similars | PCBioAssay | 10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
NMMLSC Curated by PubChem BioAssay | Assay Description University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela... | PubChem Bioassay (2009) BindingDB Entry DOI: 10.7270/Q25D8Q8M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
cell division cycle 42 (GTP binding protein, 25kDa) (Homo sapiens (Human)) | BDBM50218889![]() (7-chloroindirubin | CHEMBL243777 | cid_11847137) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt UniProtKB/TrEMBL B.MOAD antibodypedia GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | PCBioAssay | 10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
NMMLSC Curated by PubChem BioAssay | Assay Description University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela... | PubChem Bioassay (2009) BindingDB Entry DOI: 10.7270/Q2TB15BF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ras protein (Homo sapiens (Human)) | BDBM54606![]() (4-[3-(4-chlorophenyl)-5-phenyl-2-pyrazolin-1-yl]be...) | GoogleScholar | Purchase PC cid PC sid UniChem Similars | PCBioAssay | 10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
NMMLSC Curated by PubChem BioAssay | Assay Description University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela... | PubChem Bioassay (2009) BindingDB Entry DOI: 10.7270/Q2XW4H7T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ras protein (Homo sapiens (Human)) | BDBM54578![]() (1-[4-(2-fluorophenyl)-1-piperazinyl]-3-[3-(4-metho...) | GoogleScholar | PC cid PC sid UniChem Similars | Article PCBioAssay | 10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
NMMLSC Curated by PubChem BioAssay | Assay Description University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela... | PubChem Bioassay (2009) Article DOI: 10.1111/cbdd.12157 BindingDB Entry DOI: 10.7270/Q2DZ06RB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ras protein (Homo sapiens (Human)) | BDBM54575![]() (3-[3-(2-bromophenyl)-1,2,4-oxadiazol-5-yl]-1-[4-(2...) | GoogleScholar | PC cid PC sid UniChem Similars | Article PCBioAssay | 10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
NMMLSC Curated by PubChem BioAssay | Assay Description University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela... | PubChem Bioassay (2009) Article DOI: 10.1111/cbdd.12157 BindingDB Entry DOI: 10.7270/Q2DZ06RB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ras-related C3 botulinum toxin substrate 1 (Mus musculus) | BDBM54661![]() (4-[3-(4-methoxyphenyl)-5-methyl-3,4-dihydropyrazol...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt UniProtKB/TrEMBL B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem Similars | PCBioAssay | 10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
NMMLSC Curated by PubChem BioAssay | Assay Description University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela... | PubChem Bioassay (2009) BindingDB Entry DOI: 10.7270/Q26D5RFF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ras-related C3 botulinum toxin substrate 1 (Mus musculus) | BDBM54619![]() (3-(4-chlorophenyl)-5-(3,4-dimethoxyphenyl)-1-pheny...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt UniProtKB/TrEMBL B.MOAD DrugBank GoogleScholar | Purchase PC cid PC sid UniChem Similars | PCBioAssay | 10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
NMMLSC Curated by PubChem BioAssay | Assay Description University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela... | PubChem Bioassay (2009) BindingDB Entry DOI: 10.7270/Q26D5RFF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ras protein (Homo sapiens (Human)) | BDBM54606![]() (4-[3-(4-chlorophenyl)-5-phenyl-2-pyrazolin-1-yl]be...) | GoogleScholar | Purchase PC cid PC sid UniChem Similars | PCBioAssay | 10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
NMMLSC Curated by PubChem BioAssay | Assay Description University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela... | PubChem Bioassay (2009) BindingDB Entry DOI: 10.7270/Q2FX77VQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
GTP-binding protein (rab7) (Canis lupus familiaris) | BDBM54642![]() (4-[3-(3-chlorophenyl)-5-(4-methoxyphenyl)-2-pyrazo...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar | PC cid PC sid UniChem Similars | PCBioAssay | 10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
NMMLSC Curated by PubChem BioAssay | Assay Description University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela... | PubChem Bioassay (2009) BindingDB Entry DOI: 10.7270/Q2GT5KM7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
GTP-binding protein (rab7) (Canis lupus familiaris) | BDBM54590![]() (1-(3-fluorophenyl)-3,5-bis(4-methoxyphenyl)-2-pyra...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar | Purchase PC cid PC sid UniChem Similars | PCBioAssay | 10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
NMMLSC Curated by PubChem BioAssay | Assay Description University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela... | PubChem Bioassay (2009) BindingDB Entry DOI: 10.7270/Q2GT5KM7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
cell division cycle 42 (GTP binding protein, 25kDa) (Homo sapiens (Human)) | BDBM54674![]() (3-[3-(4-methoxyphenyl)-5-phenyl-3,4-dihydropyrazol...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt UniProtKB/TrEMBL B.MOAD antibodypedia GoogleScholar | PC cid PC sid UniChem Similars | Article PCBioAssay | 10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
NMMLSC Curated by PubChem BioAssay | Assay Description University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela... | PubChem Bioassay (2009) Article DOI: 10.1021/cb400468c BindingDB Entry DOI: 10.7270/Q2B856J1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G protein signalling regulator 19 (Homo sapiens (Human)) | BDBM33097![]() (3-[[7-(1,3-benzothiazol-2-ylsulfanyl)-4-nitro-2,1,...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar | Purchase PC cid PC sid UniChem Similars | PCBioAssay | 10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
NMMLSC Curated by PubChem BioAssay | Assay Description University of New Mexico Assay Overview: Assay Support: NIH R21NS057014 HTS to identify small molecule regulators of RGS family protein interaction... | PubChem Bioassay (2010) BindingDB Entry DOI: 10.7270/Q26T0K2P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ras protein (Homo sapiens (Human)) | BDBM54619![]() (3-(4-chlorophenyl)-5-(3,4-dimethoxyphenyl)-1-pheny...) | GoogleScholar | Purchase PC cid PC sid UniChem Similars | PCBioAssay | 10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
NMMLSC Curated by PubChem BioAssay | Assay Description University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela... | PubChem Bioassay (2009) BindingDB Entry DOI: 10.7270/Q2FX77VQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ras protein (Homo sapiens (Human)) | BDBM54607![]() (4-(2,5-diphenyl-3,4-dihydropyrazol-3-yl)-N,N-dimet...) | GoogleScholar | Purchase PC cid PC sid UniChem Patents Similars | PCBioAssay | 10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
NMMLSC Curated by PubChem BioAssay | Assay Description University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela... | PubChem Bioassay (2009) BindingDB Entry DOI: 10.7270/Q2FX77VQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscarinic acetylcholine receptor M1 (RAT) | BDBM43822![]() (4-[2-(o-toluoylamino)ethylamino]piperidine-1-carbo...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar | Purchase CHEMBL PC cid PC sid UniChem Similars | PCBioAssay | 14.6 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt Screening Center for GPCRs, Ion Channels and Transporters Curated by PubChem BioAssay | Assay Description Assay Provider: P. Jeffrey Conn Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of novel allosteric modulators of the M1 mus... | PubChem Bioassay (2009) BindingDB Entry DOI: 10.7270/Q2FJ2F7F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscarinic acetylcholine receptor M1 (RAT) | BDBM43820![]() (4-[2-(2-Chloro-benzoylamino)-ethylamino]-piperidin...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar | PC cid PC sid UniChem Similars | PCBioAssay | 17.0 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt Screening Center for GPCRs, Ion Channels and Transporters Curated by PubChem BioAssay | Assay Description Assay Provider: P. Jeffrey Conn Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of novel allosteric modulators of the M1 mus... | PubChem Bioassay (2009) BindingDB Entry DOI: 10.7270/Q2FJ2F7F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ras-related protein Rab-2A. (Canis lupus familiaris) | BDBM54553![]() (1-[4-(2,5-dimethylphenyl)-1-piperazinyl]-3-[3-(4-f...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar | PC cid PC sid UniChem Similars | PCBioAssay | 20 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
NMMLSC Curated by PubChem BioAssay | Assay Description University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela... | PubChem Bioassay (2009) BindingDB Entry DOI: 10.7270/Q21V5CCX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Regulator of G-protein signaling 8 (Homo sapiens (Human)) | BDBM38361![]() (2-(4-pyrrolidin-1-ylsulfonylphenyl)-1,2-benzothiaz...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar | Purchase PC cid PC sid UniChem Similars | PCBioAssay | 20 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
NMMLSC Curated by PubChem BioAssay | Assay Description University of New Mexico Assay Overview: Assay Support: NIH R21NS057014 HTS to identify small molecule regulators of RGS family protein interaction... | PubChem Bioassay (2010) BindingDB Entry DOI: 10.7270/Q2G73C4V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Regulator of G-protein signaling 8 (Homo sapiens (Human)) | BDBM46590![]() (4-[2-[(E)-(2,3-dihydroxy-4-oxocyclohexa-2,5-dien-1...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar | PC cid PC sid UniChem Similars | PCBioAssay | 20 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
NMMLSC Curated by PubChem BioAssay | Assay Description University of New Mexico Assay Overview: Assay Support: NIH R21NS057014 HTS to identify small molecule regulators of RGS family protein interaction... | PubChem Bioassay (2010) BindingDB Entry DOI: 10.7270/Q2G73C4V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Regulator of G-protein signaling 8 (Homo sapiens (Human)) | BDBM32274![]() (2,5-bis(chloranyl)-3-(4-methylpiperazin-1-yl)-6-(2...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar | PC cid PC sid UniChem Similars | PCBioAssay | 20 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
NMMLSC Curated by PubChem BioAssay | Assay Description University of New Mexico Assay Overview: Assay Support: NIH R21NS057014 HTS to identify small molecule regulators of RGS family protein interaction... | PubChem Bioassay (2010) BindingDB Entry DOI: 10.7270/Q2G73C4V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
regulator of G-protein signalling 16 (Homo sapiens (Human)) | BDBM38361![]() (2-(4-pyrrolidin-1-ylsulfonylphenyl)-1,2-benzothiaz...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar | Purchase PC cid PC sid UniChem Similars | PCBioAssay | 20 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
NMMLSC Curated by PubChem BioAssay | Assay Description University of New Mexico Assay Overview: Assay Support: NIH R21NS057014 HTS to identify small molecule regulators of RGS family protein interaction... | PubChem Bioassay (2010) BindingDB Entry DOI: 10.7270/Q2QR4VJR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
regulator of G-protein signalling 16 (Homo sapiens (Human)) | BDBM46590![]() (4-[2-[(E)-(2,3-dihydroxy-4-oxocyclohexa-2,5-dien-1...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar | PC cid PC sid UniChem Similars | PCBioAssay | 20 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
NMMLSC Curated by PubChem BioAssay | Assay Description University of New Mexico Assay Overview: Assay Support: NIH R21NS057014 HTS to identify small molecule regulators of RGS family protein interaction... | PubChem Bioassay (2010) BindingDB Entry DOI: 10.7270/Q2QR4VJR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
regulator of G-protein signalling 16 (Homo sapiens (Human)) | BDBM32274![]() (2,5-bis(chloranyl)-3-(4-methylpiperazin-1-yl)-6-(2...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar | PC cid PC sid UniChem Similars | PCBioAssay | 20 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
NMMLSC Curated by PubChem BioAssay | Assay Description University of New Mexico Assay Overview: Assay Support: NIH R21NS057014 HTS to identify small molecule regulators of RGS family protein interaction... | PubChem Bioassay (2010) BindingDB Entry DOI: 10.7270/Q2QR4VJR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
GTP-binding protein (rab7) (Canis lupus familiaris) | BDBM54583![]() (1-[4-(2,5-dimethylphenyl)-1-piperazinyl]-3-[3-(4-m...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar | PC cid PC sid UniChem Similars | PCBioAssay | 20 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
NMMLSC Curated by PubChem BioAssay | Assay Description University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela... | PubChem Bioassay (2009) BindingDB Entry DOI: 10.7270/Q29885F3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
cell division cycle 42 (GTP binding protein, 25kDa) (Homo sapiens (Human)) | BDBM54577![]() (1-[4-(4-chlorophenyl)-1-piperazinyl]-3-[3-(4-metho...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt UniProtKB/TrEMBL B.MOAD antibodypedia GoogleScholar | PC cid PC sid UniChem Similars | Article PCBioAssay | 20 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
NMMLSC Curated by PubChem BioAssay | Assay Description University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela... | PubChem Bioassay (2009) Article DOI: 10.1021/cb400542w BindingDB Entry DOI: 10.7270/Q20000HB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ras-related C3 botulinum toxin substrate 1 (Mus musculus) | BDBM54709![]() (1-[4-(4-bromophenyl)-1-piperazinyl]-3-[3-(4-methox...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt UniProtKB/TrEMBL B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem Similars | PCBioAssay | 20 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
NMMLSC Curated by PubChem BioAssay | Assay Description University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela... | PubChem Bioassay (2009) BindingDB Entry DOI: 10.7270/Q2JS9NV0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscarinic acetylcholine receptor M1 (RAT) | BDBM43821![]() (4-(2-benzamidoethylamino)-1-piperidinecarboxylic a...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | PCBioAssay | 21.3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt Screening Center for GPCRs, Ion Channels and Transporters Curated by PubChem BioAssay | Assay Description Assay Provider: P. Jeffrey Conn Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of novel allosteric modulators of the M1 mus... | PubChem Bioassay (2009) BindingDB Entry DOI: 10.7270/Q2FJ2F7F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G protein signalling regulator 19 (Homo sapiens (Human)) | BDBM32274![]() (2,5-bis(chloranyl)-3-(4-methylpiperazin-1-yl)-6-(2...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar | PC cid PC sid UniChem Similars | PCBioAssay | 30 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
NMMLSC Curated by PubChem BioAssay | Assay Description University of New Mexico Assay Overview: Assay Support: NIH R21NS057014 HTS to identify small molecule regulators of RGS family protein interaction... | PubChem Bioassay (2010) BindingDB Entry DOI: 10.7270/Q26T0K2P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ras protein (Homo sapiens (Human)) | BDBM50022271![]() (2-(3-Benzoylphenyl)propionic acid | 2-(3-benzoylph...) | GoogleScholar | Purchase CHEBI CHEMBL DrugBank KEGG PC cid PC sid PDB UniChem Patents Similars | PCBioAssay | 30 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
NMMLSC Curated by PubChem BioAssay | Assay Description University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela... | PubChem Bioassay (2009) BindingDB Entry DOI: 10.7270/Q23N21VG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
GTP-binding protein (rab7) (Canis lupus familiaris) | BDBM54605![]() (1-[4-(difluoromethylsulfonyl)phenyl]-3,5-diphenyl-...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar | Purchase PC cid PC sid UniChem Similars | PCBioAssay | 30 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
NMMLSC Curated by PubChem BioAssay | Assay Description University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela... | PubChem Bioassay (2009) BindingDB Entry DOI: 10.7270/Q2GT5KM7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ras-related C3 botulinum toxin substrate 1 (Mus musculus) | BDBM54638![]() (4-[3-(2-bromophenyl)-5-(4-methoxyphenyl)-2-pyrazol...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt UniProtKB/TrEMBL B.MOAD DrugBank GoogleScholar | PC cid PC sid UniChem Similars | PCBioAssay | 40 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
NMMLSC Curated by PubChem BioAssay | Assay Description University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela... | PubChem Bioassay (2009) BindingDB Entry DOI: 10.7270/Q26D5RFF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
GTP-binding protein (rab7) (Canis lupus familiaris) | BDBM54553![]() (1-[4-(2,5-dimethylphenyl)-1-piperazinyl]-3-[3-(4-f...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar | PC cid PC sid UniChem Similars | PCBioAssay | 40 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
NMMLSC Curated by PubChem BioAssay | Assay Description University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela... | PubChem Bioassay (2009) BindingDB Entry DOI: 10.7270/Q29885F3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
GTP-binding protein (rab7) (Canis lupus familiaris) | BDBM54578![]() (1-[4-(2-fluorophenyl)-1-piperazinyl]-3-[3-(4-metho...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar | PC cid PC sid UniChem Similars | PCBioAssay | 40 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
NMMLSC Curated by PubChem BioAssay | Assay Description University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela... | PubChem Bioassay (2009) BindingDB Entry DOI: 10.7270/Q29885F3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
regulator of G-protein signalling 16 (Homo sapiens (Human)) | BDBM47719![]() ((4-chlorodithiazol-5-ylidene)-(4-chloro-2-methyl-p...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar | PC cid PC sid UniChem Similars | PCBioAssay | 40 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
NMMLSC Curated by PubChem BioAssay | Assay Description University of New Mexico Assay Overview: Assay Support: NIH R21NS057014 HTS to identify small molecule regulators of RGS family protein interaction... | PubChem Bioassay (2010) BindingDB Entry DOI: 10.7270/Q2QR4VJR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
regulator of G-protein signalling 16 (Homo sapiens (Human)) | BDBM46608![]() ((4E)-5-methyl-4-[(3-nitroanilino)methylene]-2-phen...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar | PC cid PC sid UniChem Similars | PCBioAssay | 40 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
NMMLSC Curated by PubChem BioAssay | Assay Description University of New Mexico Assay Overview: Assay Support: NIH R21NS057014 HTS to identify small molecule regulators of RGS family protein interaction... | PubChem Bioassay (2010) BindingDB Entry DOI: 10.7270/Q2QR4VJR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
GTP-binding protein (rab7) (Canis lupus familiaris) | BDBM54595![]() (3-(4-chlorophenyl)-5-(4-methoxyphenyl)-2-phenyl-3,...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar | Purchase PC cid PC sid UniChem Similars | PCBioAssay | 40 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
NMMLSC Curated by PubChem BioAssay | Assay Description University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela... | PubChem Bioassay (2009) BindingDB Entry DOI: 10.7270/Q2GT5KM7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
cell division cycle 42 (GTP binding protein, 25kDa) (Homo sapiens (Human)) | BDBM54605![]() (1-[4-(difluoromethylsulfonyl)phenyl]-3,5-diphenyl-...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt UniProtKB/TrEMBL B.MOAD antibodypedia GoogleScholar | Purchase PC cid PC sid UniChem Similars | Article PCBioAssay | 50 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
NMMLSC Curated by PubChem BioAssay | Assay Description University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela... | PubChem Bioassay (2009) Article DOI: 10.1021/cb4007562 BindingDB Entry DOI: 10.7270/Q2KS6Q0S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ras-related protein Rab-2A. (Canis lupus familiaris) | BDBM54578![]() (1-[4-(2-fluorophenyl)-1-piperazinyl]-3-[3-(4-metho...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar | PC cid PC sid UniChem Similars | PCBioAssay | 50 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
NMMLSC Curated by PubChem BioAssay | Assay Description University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela... | PubChem Bioassay (2009) BindingDB Entry DOI: 10.7270/Q21V5CCX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ras-related C3 botulinum toxin substrate 1 (Mus musculus) | BDBM54570![]() (3-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]-1-[4-...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt UniProtKB/TrEMBL B.MOAD DrugBank GoogleScholar | Purchase PC cid PC sid UniChem Similars | PCBioAssay | 50 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
NMMLSC Curated by PubChem BioAssay | Assay Description University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela... | PubChem Bioassay (2009) BindingDB Entry DOI: 10.7270/Q2JS9NV0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
G protein signalling regulator 19 (Homo sapiens (Human)) | BDBM47764![]() ((4E)-5-methyl-4-[[3-[[(Z)-(3-methyl-1-phenyl-5-sul...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar | PC cid PC sid UniChem Similars | PCBioAssay | 50 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
NMMLSC Curated by PubChem BioAssay | Assay Description University of New Mexico Assay Overview: Assay Support: NIH R21NS057014 HTS to identify small molecule regulators of RGS family protein interaction... | PubChem Bioassay (2010) BindingDB Entry DOI: 10.7270/Q26T0K2P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
GTP-binding protein (rab7) (Canis lupus familiaris) | BDBM54567![]() (1-[4-(2,5-dimethylphenyl)-1-piperazinyl]-3-[3-[3-(...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar | PC cid PC sid UniChem Similars | PCBioAssay | 50 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
NMMLSC Curated by PubChem BioAssay | Assay Description University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela... | PubChem Bioassay (2009) BindingDB Entry DOI: 10.7270/Q29885F3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ras-related protein Rab-2A. (Canis lupus familiaris) | BDBM54548![]() (3-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]-1-[4-...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar | PC cid PC sid UniChem Similars | PCBioAssay | 50 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
NMMLSC Curated by PubChem BioAssay | Assay Description University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela... | PubChem Bioassay (2009) BindingDB Entry DOI: 10.7270/Q21V5CCX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ras-related protein Rab-2A. (Canis lupus familiaris) | BDBM54549![]() (1-[4-(2,5-dimethylphenyl)-1-piperazinyl]-3-(3-phen...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar | PC cid PC sid UniChem Similars | PCBioAssay | 50 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
NMMLSC Curated by PubChem BioAssay | Assay Description University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela... | PubChem Bioassay (2009) BindingDB Entry DOI: 10.7270/Q21V5CCX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ras-related protein Rab-2A. (Canis lupus familiaris) | BDBM54590![]() (1-(3-fluorophenyl)-3,5-bis(4-methoxyphenyl)-2-pyra...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar | Purchase PC cid PC sid UniChem Similars | PCBioAssay | 60 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
NMMLSC Curated by PubChem BioAssay | Assay Description University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela... | PubChem Bioassay (2016) BindingDB Entry DOI: 10.7270/Q2ZW1JC6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Regulator of G-protein signaling 8 (Homo sapiens (Human)) | BDBM43363![]() (2,5-bis(chloranyl)-3-piperidin-1-yl-6-(2-piperidin...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar | Purchase PC cid PC sid UniChem Similars | PCBioAssay | 60 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
NMMLSC Curated by PubChem BioAssay | Assay Description University of New Mexico Assay Overview: Assay Support: NIH R21NS057014 HTS to identify small molecule regulators of RGS family protein interaction... | PubChem Bioassay (2010) BindingDB Entry DOI: 10.7270/Q2G73C4V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ras-related C3 botulinum toxin substrate 1 (Mus musculus) | BDBM54570![]() (3-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]-1-[4-...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt UniProtKB/TrEMBL B.MOAD DrugBank GoogleScholar | Purchase PC cid PC sid UniChem Similars | Article PCBioAssay | 60 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
NMMLSC Curated by PubChem BioAssay | Assay Description University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela... | PubChem Bioassay (2009) Article DOI: 10.1111/cbdd.12142 BindingDB Entry DOI: 10.7270/Q2PC30TH | |||||||||||
More data for this Ligand-Target Pair |
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