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Compile Data Set for Download or QSAR

Found 180 hits with Last Name = 'ringgenberg' and Initial = 'jd'   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Progesterone receptor


(Homo sapiens (Human))
BDBM18627
PNG
((10S,11S,14S,15S,17R)-17-[4-(dimethylamino)phenyl]...)
Show SMILES CC#C[C@]1(O)CC[C@H]2[C@@H]3CCC4=CC(=O)CCC4=C3[C@H](C[C@]12C)c1ccc(cc1)N(C)C
Show InChI InChI=1/C29H35NO2/c1-5-15-29(32)16-14-26-24-12-8-20-17-22(31)11-13-23(20)27(24)25(18-28(26,29)2)19-6-9-21(10-7-19)30(3)4/h6-7,9-10,17,24-26,32H,8,11-14,16,18H2,1-4H3/t24-,25+,26-,28-,29-/s2
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1.10n/an/an/an/an/an/an/an/a



Ligand Pharmaceuticals

Curated by ChEMBL


Assay Description
Binding affinity at human progesterone receptor.


Bioorg Med Chem Lett 13: 2075-8 (2003)


Article DOI: 10.1016/s0960-894x(03)00256-7
BindingDB Entry DOI: 10.7270/Q2P55P2M
More data for this
Ligand-Target Pair
3D
3D Structure (crystal)
Androgen Receptor


(Homo sapiens (Human))
BDBM18161
PNG
((1S,2S,7S,10R,11S,14S,15S)-14-hydroxy-2,15-dimethy...)
Show SMILES C[C@]12CC[C@H]3[C@@H](CC[C@H]4CC(=O)CC[C@]34C)[C@@H]1CC[C@@H]2O
Show InChI InChI=1/C19H30O2/c1-18-9-7-13(20)11-12(18)3-4-14-15-5-6-17(21)19(15,2)10-8-16(14)18/h12,14-17,21H,3-11H2,1-2H3/t12-,14-,15-,16-,17-,18-,19-/s2
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2n/an/an/an/an/an/an/an/a



Ligand Pharmaceuticals, Inc.

Curated by ChEMBL


Assay Description
Agonist activity to the human androgen receptor (hAR) in CV-1 cells


Bioorg Med Chem Lett 9: 1335-40 (1999)


Article DOI: 10.1016/s0960-894x(99)00186-9
BindingDB Entry DOI: 10.7270/Q2JM2B4G
More data for this
Ligand-Target Pair
3D
3D Structure (crystal)
Androgen Receptor


(Homo sapiens (Human))
BDBM50077104
PNG
(CHEMBL431493 | Cis-(4aR,12bS)-11-Trifluoromethyl-2...)
Show SMILES FC(F)(F)c1cc(=O)[nH]c2cc3NC[C@@H]4CCCC[C@@H]4c3cc12
Show InChI InChI=1S/C17H17F3N2O/c18-17(19,20)13-6-16(23)22-15-7-14-11(5-12(13)15)10-4-2-1-3-9(10)8-21-14/h5-7,9-10,21H,1-4,8H2,(H,22,23)/t9-,10-/m0/s1
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2n/an/an/an/an/an/an/an/a



Ligand Pharmaceuticals, Inc.

Curated by ChEMBL


Assay Description
Binding affinity to the human androgen receptor (hAR), using [3H]DHT as radioligand in a competitive binding assay


Bioorg Med Chem Lett 9: 1335-40 (1999)


Article DOI: 10.1016/s0960-894x(99)00186-9
BindingDB Entry DOI: 10.7270/Q2JM2B4G
More data for this
Ligand-Target Pair
Androgen Receptor


(Homo sapiens (Human))
BDBM50077095
PNG
(CHEMBL281945 | Trans-7-Methyl-4-trifluoromethyl-6-...)
Show SMILES C[C@H]1CNc2cc3[nH]c(=O)cc(c3cc2C1CCC(F)(F)F)C(F)(F)F
Show InChI InChI=1S/C17H16F6N2O/c1-8-7-24-13-6-14-11(12(17(21,22)23)5-15(26)25-14)4-10(13)9(8)2-3-16(18,19)20/h4-6,8-9,24H,2-3,7H2,1H3,(H,25,26)/t8-,9?/m0/s1
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2n/an/an/an/an/an/an/an/a



Ligand Pharmaceuticals, Inc.

Curated by ChEMBL


Assay Description
Binding affinity to the human androgen receptor (hAR), using [3H]DHT as radioligand in a competitive binding assay


Bioorg Med Chem Lett 9: 1335-40 (1999)


Article DOI: 10.1016/s0960-894x(99)00186-9
BindingDB Entry DOI: 10.7270/Q2JM2B4G
More data for this
Ligand-Target Pair
Progesterone receptor


(Homo sapiens (Human))
BDBM50129168
PNG
(7-Fluoro-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-az...)
Show SMILES CC1=CC(C)(C)Nc2ccc-3c(COc4c(F)cc(cc-34)C#N)c12
Show InChI InChI=1S/C20H17FN2O/c1-11-8-20(2,3)23-17-5-4-13-14-6-12(9-22)7-16(21)19(14)24-10-15(13)18(11)17/h4-8,23H,10H2,1-3H3
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4.5n/an/an/an/an/an/an/an/a



Ligand Pharmaceuticals

Curated by ChEMBL


Assay Description
Binding affinity at human progesterone receptor.


Bioorg Med Chem Lett 13: 2075-8 (2003)


Article DOI: 10.1016/s0960-894x(03)00256-7
BindingDB Entry DOI: 10.7270/Q2P55P2M
More data for this
Ligand-Target Pair
Progesterone receptor


(Homo sapiens (Human))
BDBM50129166
PNG
(9-Chloro-7-fluoro-2,2,4-trimethyl-2,5-dihydro-1H-6...)
Show SMILES CC1=CC(C)(C)Nc2ccc-3c(COc4c(F)cc(Cl)cc-34)c12
Show InChI InChI=1S/C19H17ClFNO/c1-10-8-19(2,3)22-16-5-4-12-13-6-11(20)7-15(21)18(13)23-9-14(12)17(10)16/h4-8,22H,9H2,1-3H3
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5.60n/an/an/an/an/an/an/an/a



Ligand Pharmaceuticals

Curated by ChEMBL


Assay Description
Binding towards human progesterone receptor


Bioorg Med Chem Lett 13: 2075-8 (2003)


Article DOI: 10.1016/s0960-894x(03)00256-7
BindingDB Entry DOI: 10.7270/Q2P55P2M
More data for this
Ligand-Target Pair
Progesterone receptor


(Homo sapiens (Human))
BDBM50129165
PNG
(2,2,4-Trimethyl-9-nitro-2,5-dihydro-1H-6-oxa-1-aza...)
Show SMILES CC1=CC(C)(C)Nc2ccc-3c(COc4ccc(cc-34)[N+]([O-])=O)c12
Show InChI InChI=1S/C19H18N2O3/c1-11-9-19(2,3)20-16-6-5-13-14-8-12(21(22)23)4-7-17(14)24-10-15(13)18(11)16/h4-9,20H,10H2,1-3H3
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6.80n/an/an/an/an/an/an/an/a



Ligand Pharmaceuticals

Curated by ChEMBL


Assay Description
Binding affinity at human progesterone receptor.


Bioorg Med Chem Lett 13: 2075-8 (2003)


Article DOI: 10.1016/s0960-894x(03)00256-7
BindingDB Entry DOI: 10.7270/Q2P55P2M
More data for this
Ligand-Target Pair
Androgen Receptor


(Homo sapiens (Human))
BDBM18190
PNG
(6-ethyl-4-(trifluoromethyl)-1H,2H,6H,7H,8H,9H-pyri...)
Show SMILES CCC1CCNc2cc3[nH]c(=O)cc(c3cc12)C(F)(F)F
Show InChI InChI=1/C15H15F3N2O/c1-2-8-3-4-19-12-7-13-10(5-9(8)12)11(15(16,17)18)6-14(21)20-13/h5-8,19H,2-4H2,1H3,(H,20,21)
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7n/an/an/an/an/an/an/an/a



Ligand Pharmaceuticals, Inc.

Curated by ChEMBL


Assay Description
Binding affinity to the human androgen receptor (hAR), using [3H]DHT as radioligand in a competitive binding assay


Bioorg Med Chem Lett 9: 1335-40 (1999)


Article DOI: 10.1016/s0960-894x(99)00186-9
BindingDB Entry DOI: 10.7270/Q2JM2B4G
More data for this
Ligand-Target Pair
Androgen Receptor


(Homo sapiens (Human))
BDBM50077105
PNG
(CHEMBL418198 | Trans-6-Ethyl-7-methyl-4-trifluorom...)
Show SMILES CCC1[C@@H](C)CNc2cc3[nH]c(=O)cc(c3cc12)C(F)(F)F
Show InChI InChI=1S/C16H17F3N2O/c1-3-9-8(2)7-20-13-6-14-11(4-10(9)13)12(16(17,18)19)5-15(22)21-14/h4-6,8-9,20H,3,7H2,1-2H3,(H,21,22)/t8-,9?/m0/s1
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8n/an/an/an/an/an/an/an/a



Ligand Pharmaceuticals, Inc.

Curated by ChEMBL


Assay Description
Binding affinity to the human androgen receptor (hAR), using [3H]DHT as radioligand in a competitive binding assay


Bioorg Med Chem Lett 9: 1335-40 (1999)


Article DOI: 10.1016/s0960-894x(99)00186-9
BindingDB Entry DOI: 10.7270/Q2JM2B4G
More data for this
Ligand-Target Pair
Androgen Receptor


(Homo sapiens (Human))
BDBM50077115
PNG
(CHEMBL282204 | Cis-6,7-Dimethyl-4-trifluoromethyl-...)
Show SMILES C[C@@H]1CNc2cc3[nH]c(=O)cc(c3cc2C1C)C(F)(F)F
Show InChI InChI=1S/C15H15F3N2O/c1-7-6-19-12-5-13-10(3-9(12)8(7)2)11(15(16,17)18)4-14(21)20-13/h3-5,7-8,19H,6H2,1-2H3,(H,20,21)/t7-,8?/m1/s1
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8n/an/an/an/an/an/an/an/a



Ligand Pharmaceuticals, Inc.

Curated by ChEMBL


Assay Description
Binding affinity to the human androgen receptor (hAR), using [3H]DHT as radioligand in a competitive binding assay


Bioorg Med Chem Lett 9: 1335-40 (1999)


Article DOI: 10.1016/s0960-894x(99)00186-9
BindingDB Entry DOI: 10.7270/Q2JM2B4G
More data for this
Ligand-Target Pair
Androgen Receptor


(Homo sapiens (Human))
BDBM50077112
PNG
(CHEMBL27812 | Cis-(3aR,11bS)-10-Trifluoromethyl-1,...)
Show SMILES FC(F)(F)c1cc(=O)[nH]c2cc3NC[C@@H]4CCC[C@@H]4c3cc12
Show InChI InChI=1S/C16H15F3N2O/c17-16(18,19)12-5-15(22)21-14-6-13-10(4-11(12)14)9-3-1-2-8(9)7-20-13/h4-6,8-9,20H,1-3,7H2,(H,21,22)/t8-,9-/m0/s1
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8n/an/an/an/an/an/an/an/a



Ligand Pharmaceuticals, Inc.

Curated by ChEMBL


Assay Description
Agonist activity to the human androgen receptor (hAR) in CV-1 cells


Bioorg Med Chem Lett 9: 1335-40 (1999)


Article DOI: 10.1016/s0960-894x(99)00186-9
BindingDB Entry DOI: 10.7270/Q2JM2B4G
More data for this
Ligand-Target Pair
Androgen Receptor


(Homo sapiens (Human))
BDBM50077111
PNG
(6-Ethyl-1-methyl-4-trifluoromethyl-6,7,8,9-tetrahy...)
Show SMILES CCC1CCNc2cc3n(C)c(=O)cc(c3cc12)C(F)(F)F
Show InChI InChI=1/C16H17F3N2O/c1-3-9-4-5-20-13-8-14-11(6-10(9)13)12(16(17,18)19)7-15(22)21(14)2/h6-9,20H,3-5H2,1-2H3
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9n/an/an/an/an/an/an/an/a



Ligand Pharmaceuticals, Inc.

Curated by ChEMBL


Assay Description
Binding affinity to the human androgen receptor (hAR), using [3H]DHT as radioligand in a competitive binding assay


Bioorg Med Chem Lett 9: 1335-40 (1999)


Article DOI: 10.1016/s0960-894x(99)00186-9
BindingDB Entry DOI: 10.7270/Q2JM2B4G
More data for this
Ligand-Target Pair
Androgen Receptor


(Homo sapiens (Human))
BDBM50077097
PNG
(6-Methyl-4-trifluoromethyl-6,7,8,9-tetrahydro-1H-p...)
Show SMILES CC1CCNc2cc3[nH]c(=O)cc(c3cc12)C(F)(F)F
Show InChI InChI=1/C14H13F3N2O/c1-7-2-3-18-11-6-12-9(4-8(7)11)10(14(15,16)17)5-13(20)19-12/h4-7,18H,2-3H2,1H3,(H,19,20)
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9n/an/an/an/an/an/an/an/a



Ligand Pharmaceuticals, Inc.

Curated by ChEMBL


Assay Description
Antagonistic activity against human androgen receptor (hAR) in CV-1 cells was determined as a function of maximal inhibition of dihydrotestosterone u...


Bioorg Med Chem Lett 9: 1335-40 (1999)


Article DOI: 10.1016/s0960-894x(99)00186-9
BindingDB Entry DOI: 10.7270/Q2JM2B4G
More data for this
Ligand-Target Pair
Androgen Receptor


(Homo sapiens (Human))
BDBM50077108
PNG
(6,6-Dimethyl-4-trifluoromethyl-6,7,8,9-tetrahydro-...)
Show SMILES CC1(C)CCNc2cc3[nH]c(=O)cc(c3cc12)C(F)(F)F
Show InChI InChI=1S/C15H15F3N2O/c1-14(2)3-4-19-12-7-11-8(5-10(12)14)9(15(16,17)18)6-13(21)20-11/h5-7,19H,3-4H2,1-2H3,(H,20,21)
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12n/an/an/an/an/an/an/an/a



Ligand Pharmaceuticals, Inc.

Curated by ChEMBL


Assay Description
Binding affinity to the human androgen receptor (hAR), using [3H]DHT as radioligand in a competitive binding assay


Bioorg Med Chem Lett 9: 1335-40 (1999)


Article DOI: 10.1016/s0960-894x(99)00186-9
BindingDB Entry DOI: 10.7270/Q2JM2B4G
More data for this
Ligand-Target Pair
Progesterone receptor


(Homo sapiens (Human))
BDBM50129171
PNG
(9-Bromo-7-fluoro-2,2,4-trimethyl-2,5-dihydro-1H-6-...)
Show SMILES CC1=CC(C)(C)Nc2ccc-3c(COc4c(F)cc(Br)cc-34)c12
Show InChI InChI=1S/C19H17BrFNO/c1-10-8-19(2,3)22-16-5-4-12-13-6-11(20)7-15(21)18(13)23-9-14(12)17(10)16/h4-8,22H,9H2,1-3H3
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12n/an/an/an/an/an/an/an/a



Ligand Pharmaceuticals

Curated by ChEMBL


Assay Description
Binding affinity at human progesterone receptor.


Bioorg Med Chem Lett 13: 2075-8 (2003)


Article DOI: 10.1016/s0960-894x(03)00256-7
BindingDB Entry DOI: 10.7270/Q2P55P2M
More data for this
Ligand-Target Pair
Androgen Receptor


(Homo sapiens (Human))
BDBM50077109
PNG
(6-Isopropyl-4-trifluoromethyl-6,7,8,9-tetrahydro-1...)
Show SMILES CC(C)C1CCNc2cc3[nH]c(=O)cc(c3cc12)C(F)(F)F
Show InChI InChI=1/C16H17F3N2O/c1-8(2)9-3-4-20-13-7-14-11(5-10(9)13)12(16(17,18)19)6-15(22)21-14/h5-9,20H,3-4H2,1-2H3,(H,21,22)
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13n/an/an/an/an/an/an/an/a



Ligand Pharmaceuticals, Inc.

Curated by ChEMBL


Assay Description
Binding affinity to the human androgen receptor (hAR), using [3H]DHT as radioligand in a competitive binding assay


Bioorg Med Chem Lett 9: 1335-40 (1999)


Article DOI: 10.1016/s0960-894x(99)00186-9
BindingDB Entry DOI: 10.7270/Q2JM2B4G
More data for this
Ligand-Target Pair
Progesterone receptor


(Homo sapiens (Human))
BDBM50072702
PNG
(9-Chloro-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-az...)
Show SMILES CC1=CC(C)(C)Nc2ccc-3c(COc4ccc(Cl)cc-34)c12
Show InChI InChI=1S/C19H18ClNO/c1-11-9-19(2,3)21-16-6-5-13-14-8-12(20)4-7-17(14)22-10-15(13)18(11)16/h4-9,21H,10H2,1-3H3
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13n/an/an/an/an/an/an/an/a



Ligand Pharmaceuticals

Curated by ChEMBL


Assay Description
Binding affinity at human progesterone receptor.


Bioorg Med Chem Lett 13: 2075-8 (2003)


Article DOI: 10.1016/s0960-894x(03)00256-7
BindingDB Entry DOI: 10.7270/Q2P55P2M
More data for this
Ligand-Target Pair
Progesterone receptor


(Homo sapiens (Human))
BDBM50129163
PNG
(7,9-Difluoro-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-...)
Show SMILES CC1=CC(C)(C)Nc2ccc-3c(COc4c(F)cc(F)cc-34)c12
Show InChI InChI=1S/C19H17F2NO/c1-10-8-19(2,3)22-16-5-4-12-13-6-11(20)7-15(21)18(13)23-9-14(12)17(10)16/h4-8,22H,9H2,1-3H3
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14n/an/an/an/an/an/an/an/a



Ligand Pharmaceuticals

Curated by ChEMBL


Assay Description
Binding towards human progesterone receptor


Bioorg Med Chem Lett 13: 2075-8 (2003)


Article DOI: 10.1016/s0960-894x(03)00256-7
BindingDB Entry DOI: 10.7270/Q2P55P2M
More data for this
Ligand-Target Pair
Progesterone receptor


(Homo sapiens (Human))
BDBM50129159
PNG
(9-Bromo-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza...)
Show SMILES CC1=CC(C)(C)Nc2ccc-3c(COc4ccc(Br)cc-34)c12
Show InChI InChI=1S/C19H18BrNO/c1-11-9-19(2,3)21-16-6-5-13-14-8-12(20)4-7-17(14)22-10-15(13)18(11)16/h4-9,21H,10H2,1-3H3
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15n/an/an/an/an/an/an/an/a



Ligand Pharmaceuticals

Curated by ChEMBL


Assay Description
Binding affinity at human progesterone receptor.


Bioorg Med Chem Lett 13: 2075-8 (2003)


Article DOI: 10.1016/s0960-894x(03)00256-7
BindingDB Entry DOI: 10.7270/Q2P55P2M
More data for this
Ligand-Target Pair
Androgen Receptor


(Homo sapiens (Human))
BDBM50077096
PNG
(CHEMBL25802 | Trans-11-Trifluoromethyl-2,3,4,4a,5,...)
Show SMILES FC(F)(F)c1cc(=O)[nH]c2cc3NC[C@H]4CCCC[C@@H]4c3cc12
Show InChI InChI=1S/C17H17F3N2O/c18-17(19,20)13-6-16(23)22-15-7-14-11(5-12(13)15)10-4-2-1-3-9(10)8-21-14/h5-7,9-10,21H,1-4,8H2,(H,22,23)/t9-,10+/m1/s1
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15n/an/an/an/an/an/an/an/a



Ligand Pharmaceuticals, Inc.

Curated by ChEMBL


Assay Description
Agonist activity to the human androgen receptor (hAR) in CV-1 cells


Bioorg Med Chem Lett 9: 1335-40 (1999)


Article DOI: 10.1016/s0960-894x(99)00186-9
BindingDB Entry DOI: 10.7270/Q2JM2B4G
More data for this
Ligand-Target Pair
Androgen Receptor


(Homo sapiens (Human))
BDBM50077099
PNG
(CHEMBL436344 | Trans-6,7-Dimethyl-4-trifluoromethy...)
Show SMILES C[C@H]1CNc2cc3[nH]c(=O)cc(c3cc2C1C)C(F)(F)F
Show InChI InChI=1S/C15H15F3N2O/c1-7-6-19-12-5-13-10(3-9(12)8(7)2)11(15(16,17)18)4-14(21)20-13/h3-5,7-8,19H,6H2,1-2H3,(H,20,21)/t7-,8?/m0/s1
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16n/an/an/an/an/an/an/an/a



Ligand Pharmaceuticals, Inc.

Curated by ChEMBL


Assay Description
Binding affinity to the human androgen receptor (hAR), using [3H]DHT as radioligand in a competitive binding assay


Bioorg Med Chem Lett 9: 1335-40 (1999)


Article DOI: 10.1016/s0960-894x(99)00186-9
BindingDB Entry DOI: 10.7270/Q2JM2B4G
More data for this
Ligand-Target Pair
Progesterone receptor


(Homo sapiens (Human))
BDBM50366558
PNG
(ONAPRISTONE | ZK-98299)
Show SMILES CN(C)c1ccc(cc1)[C@H]1C[C@]2(C)[C@@H](CC[C@]2(O)CCCO)[C@@H]2CCC3=CC(=O)CCC3=C12
Show InChI InChI=1S/C29H39NO3/c1-28-18-25(19-5-8-21(9-6-19)30(2)3)27-23-12-10-22(32)17-20(23)7-11-24(27)26(28)13-15-29(28,33)14-4-16-31/h5-6,8-9,17,24-26,31,33H,4,7,10-16,18H2,1-3H3/t24-,25+,26-,28+,29+/m0/s1
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18n/an/an/an/an/an/an/an/a



Ligand Pharmaceuticals

Curated by ChEMBL


Assay Description
Binding affinity at human progesterone receptor.


Bioorg Med Chem Lett 13: 2075-8 (2003)


Article DOI: 10.1016/s0960-894x(03)00256-7
BindingDB Entry DOI: 10.7270/Q2P55P2M
More data for this
Ligand-Target Pair
Androgen Receptor


(Homo sapiens (Human))
BDBM50077114
PNG
(4-Trifluoromethyl-6,7,8,9-tetrahydro-1H-pyrido[3,2...)
Show SMILES FC(F)(F)c1cc(=O)[nH]c2cc3NCCCc3cc12
Show InChI InChI=1S/C13H11F3N2O/c14-13(15,16)9-5-12(19)18-11-6-10-7(4-8(9)11)2-1-3-17-10/h4-6,17H,1-3H2,(H,18,19)
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19n/an/an/an/an/an/an/an/a



Ligand Pharmaceuticals, Inc.

Curated by ChEMBL


Assay Description
Agonist activity to the human androgen receptor (hAR) in CV-1 cells


Bioorg Med Chem Lett 9: 1335-40 (1999)


Article DOI: 10.1016/s0960-894x(99)00186-9
BindingDB Entry DOI: 10.7270/Q2JM2B4G
More data for this
Ligand-Target Pair
Progesterone receptor


(Homo sapiens (Human))
BDBM50072715
PNG
(9-Fluoro-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-az...)
Show SMILES CC1=CC(C)(C)Nc2ccc-3c(COc4ccc(F)cc-34)c12
Show InChI InChI=1S/C19H18FNO/c1-11-9-19(2,3)21-16-6-5-13-14-8-12(20)4-7-17(14)22-10-15(13)18(11)16/h4-9,21H,10H2,1-3H3
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19n/an/an/an/an/an/an/an/a



Ligand Pharmaceuticals

Curated by ChEMBL


Assay Description
Binding affinity at human progesterone receptor.


Bioorg Med Chem Lett 13: 2075-8 (2003)


Article DOI: 10.1016/s0960-894x(03)00256-7
BindingDB Entry DOI: 10.7270/Q2P55P2M
More data for this
Ligand-Target Pair
Androgen Receptor


(Homo sapiens (Human))
BDBM50077100
PNG
(6-Isobutyl-4-trifluoromethyl-6,7,8,9-tetrahydro-1H...)
Show SMILES CC(C)CC1CCNc2cc3[nH]c(=O)cc(c3cc12)C(F)(F)F
Show InChI InChI=1/C17H19F3N2O/c1-9(2)5-10-3-4-21-14-8-15-12(6-11(10)14)13(17(18,19)20)7-16(23)22-15/h6-10,21H,3-5H2,1-2H3,(H,22,23)
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22n/an/an/an/an/an/an/an/a



Ligand Pharmaceuticals, Inc.

Curated by ChEMBL


Assay Description
Binding affinity to the human androgen receptor (hAR), using [3H]DHT as radioligand in a competitive binding assay


Bioorg Med Chem Lett 9: 1335-40 (1999)


Article DOI: 10.1016/s0960-894x(99)00186-9
BindingDB Entry DOI: 10.7270/Q2JM2B4G
More data for this
Ligand-Target Pair
Androgen Receptor


(Homo sapiens (Human))
BDBM50403736
PNG
(CHEMBL2113261)
Show SMILES CC[C@@H]1[C@H](C)CNc2cc3[nH]c(=O)cc(c3cc12)C(F)(F)F
Show InChI InChI=1S/C16H17F3N2O/c1-3-9-8(2)7-20-13-6-14-11(4-10(9)13)12(16(17,18)19)5-15(22)21-14/h4-6,8-9,20H,3,7H2,1-2H3,(H,21,22)/t8-,9-/m1/s1
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27n/an/an/an/an/an/an/an/a



Ligand Pharmaceuticals, Inc.

Curated by ChEMBL


Assay Description
Binding affinity to the human androgen receptor (hAR), using [3H]DHT as radioligand in a competitive binding assay


Bioorg Med Chem Lett 9: 1335-40 (1999)


Article DOI: 10.1016/s0960-894x(99)00186-9
BindingDB Entry DOI: 10.7270/Q2JM2B4G
More data for this
Ligand-Target Pair
Androgen Receptor


(Homo sapiens (Human))
BDBM50077113
PNG
(6-Propyl-4-trifluoromethyl-6,7,8,9-tetrahydro-1H-p...)
Show SMILES CCCC1CCNc2cc3[nH]c(=O)cc(c3cc12)C(F)(F)F
Show InChI InChI=1/C16H17F3N2O/c1-2-3-9-4-5-20-13-8-14-11(6-10(9)13)12(16(17,18)19)7-15(22)21-14/h6-9,20H,2-5H2,1H3,(H,21,22)
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29n/an/an/an/an/an/an/an/a



Ligand Pharmaceuticals, Inc.

Curated by ChEMBL


Assay Description
Binding affinity to the human androgen receptor (hAR), using [3H]DHT as radioligand in a competitive binding assay


Bioorg Med Chem Lett 9: 1335-40 (1999)


Article DOI: 10.1016/s0960-894x(99)00186-9
BindingDB Entry DOI: 10.7270/Q2JM2B4G
More data for this
Ligand-Target Pair
Progesterone receptor


(Homo sapiens (Human))
BDBM50129173
PNG
(7,9-Difluoro-2,2,4-trimethyl-2,3,4,5-tetrahydro-1H...)
Show SMILES CC1CC(C)(C)Nc2ccc-3c(COc4c(F)cc(F)cc-34)c12
Show InChI InChI=1/C19H19F2NO/c1-10-8-19(2,3)22-16-5-4-12-13-6-11(20)7-15(21)18(13)23-9-14(12)17(10)16/h4-7,10,22H,8-9H2,1-3H3
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45n/an/an/an/an/an/an/an/a



Ligand Pharmaceuticals

Curated by ChEMBL


Assay Description
Inhibition of human progesterone receptor activation in T47D human breast cancer cell.


Bioorg Med Chem Lett 13: 2075-8 (2003)


Article DOI: 10.1016/s0960-894x(03)00256-7
BindingDB Entry DOI: 10.7270/Q2P55P2M
More data for this
Ligand-Target Pair
Progesterone receptor


(Homo sapiens (Human))
BDBM50072721
PNG
(2,2,4,9-Tetramethyl-2,5-dihydro-1H-6-oxa-1-aza-chr...)
Show SMILES CC1=CC(C)(C)Nc2ccc-3c(COc4ccc(C)cc-34)c12
Show InChI InChI=1S/C20H21NO/c1-12-5-8-18-15(9-12)14-6-7-17-19(16(14)11-22-18)13(2)10-20(3,4)21-17/h5-10,21H,11H2,1-4H3
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45n/an/an/an/an/an/an/an/a



Ligand Pharmaceuticals

Curated by ChEMBL


Assay Description
Binding affinity at human progesterone receptor.


Bioorg Med Chem Lett 13: 2075-8 (2003)


Article DOI: 10.1016/s0960-894x(03)00256-7
BindingDB Entry DOI: 10.7270/Q2P55P2M
More data for this
Ligand-Target Pair
Androgen Receptor


(Homo sapiens (Human))
BDBM50077110
PNG
(6,6-Diethyl-4-trifluoromethyl-6,7,8,9-tetrahydro-1...)
Show SMILES CCC1(CC)CCNc2cc3[nH]c(=O)cc(c3cc12)C(F)(F)F
Show InChI InChI=1S/C17H19F3N2O/c1-3-16(4-2)5-6-21-14-9-13-10(7-12(14)16)11(17(18,19)20)8-15(23)22-13/h7-9,21H,3-6H2,1-2H3,(H,22,23)
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58n/an/an/an/an/an/an/an/a



Ligand Pharmaceuticals, Inc.

Curated by ChEMBL


Assay Description
Antagonistic activity against human androgen receptor (hAR) in CV-1 cells was determined as a function of maximal inhibition of dihydrotestosterone u...


Bioorg Med Chem Lett 9: 1335-40 (1999)


Article DOI: 10.1016/s0960-894x(99)00186-9
BindingDB Entry DOI: 10.7270/Q2JM2B4G
More data for this
Ligand-Target Pair
Androgen Receptor


(Homo sapiens (Human))
BDBM50403735
PNG
(CHEMBL2113248)
Show SMILES CC(C)C[C@@H]1[C@@H](C)CNc2cc3[nH]c(=O)cc(c3cc12)C(F)(F)F
Show InChI InChI=1S/C18H21F3N2O/c1-9(2)4-11-10(3)8-22-15-7-16-13(5-12(11)15)14(18(19,20)21)6-17(24)23-16/h5-7,9-11,22H,4,8H2,1-3H3,(H,23,24)/t10-,11+/m0/s1
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72n/an/an/an/an/an/an/an/a



Ligand Pharmaceuticals, Inc.

Curated by ChEMBL


Assay Description
Binding affinity to the human androgen receptor (hAR), using [3H]DHT as radioligand in a competitive binding assay


Bioorg Med Chem Lett 9: 1335-40 (1999)


Article DOI: 10.1016/s0960-894x(99)00186-9
BindingDB Entry DOI: 10.7270/Q2JM2B4G
More data for this
Ligand-Target Pair
Progesterone receptor


(Homo sapiens (Human))
BDBM50072700
PNG
(2,2,4-Trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysen...)
Show SMILES CC1=CC(C)(C)Nc2ccc-3c(COc4ccccc-34)c12
Show InChI InChI=1S/C19H19NO/c1-12-10-19(2,3)20-16-9-8-13-14-6-4-5-7-17(14)21-11-15(13)18(12)16/h4-10,20H,11H2,1-3H3
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84n/an/an/an/an/an/an/an/a



Ligand Pharmaceuticals

Curated by ChEMBL


Assay Description
Inhibition of human progesterone receptor activation in T47D human breast cancer cell.


Bioorg Med Chem Lett 13: 2075-8 (2003)


Article DOI: 10.1016/s0960-894x(03)00256-7
BindingDB Entry DOI: 10.7270/Q2P55P2M
More data for this
Ligand-Target Pair
Progesterone receptor


(Homo sapiens (Human))
BDBM50129160
PNG
(9-Methoxy-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-a...)
Show SMILES COc1ccc2OCc3c(ccc4NC(C)(C)C=C(C)c34)-c2c1
Show InChI InChI=1S/C20H21NO2/c1-12-10-20(2,3)21-17-7-6-14-15-9-13(22-4)5-8-18(15)23-11-16(14)19(12)17/h5-10,21H,11H2,1-4H3
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86n/an/an/an/an/an/an/an/a



Ligand Pharmaceuticals

Curated by ChEMBL


Assay Description
Binding affinity at human progesterone receptor.


Bioorg Med Chem Lett 13: 2075-8 (2003)


Article DOI: 10.1016/s0960-894x(03)00256-7
BindingDB Entry DOI: 10.7270/Q2P55P2M
More data for this
Ligand-Target Pair
Progesterone receptor


(Homo sapiens (Human))
BDBM50129167
PNG
(2,2,4-Trimethyl-9-nitro-2,3,4,5-tetrahydro-1H-6-ox...)
Show SMILES CC1CC(C)(C)Nc2ccc-3c(COc4ccc(cc-34)[N+]([O-])=O)c12
Show InChI InChI=1/C19H20N2O3/c1-11-9-19(2,3)20-16-6-5-13-14-8-12(21(22)23)4-7-17(14)24-10-15(13)18(11)16/h4-8,11,20H,9-10H2,1-3H3
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144n/an/an/an/an/an/an/an/a



Ligand Pharmaceuticals

Curated by ChEMBL


Assay Description
Antagonistic activity at human progesterone receptor in CV-1 cells.


Bioorg Med Chem Lett 13: 2075-8 (2003)


Article DOI: 10.1016/s0960-894x(03)00256-7
BindingDB Entry DOI: 10.7270/Q2P55P2M
More data for this
Ligand-Target Pair
Progesterone receptor


(Homo sapiens (Human))
BDBM50129161
PNG
(9-Chloro-2,2,4,7-tetramethyl-2,5-dihydro-1H-6-oxa-...)
Show SMILES CC1=CC(C)(C)Nc2ccc-3c(COc4c(C)cc(Cl)cc-34)c12
Show InChI InChI=1S/C20H20ClNO/c1-11-7-13(21)8-15-14-5-6-17-18(16(14)10-23-19(11)15)12(2)9-20(3,4)22-17/h5-9,22H,10H2,1-4H3
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205n/an/an/an/an/an/an/an/a



Ligand Pharmaceuticals

Curated by ChEMBL


Assay Description
Binding affinity at human progesterone receptor.


Bioorg Med Chem Lett 13: 2075-8 (2003)


Article DOI: 10.1016/s0960-894x(03)00256-7
BindingDB Entry DOI: 10.7270/Q2P55P2M
More data for this
Ligand-Target Pair
Progesterone receptor


(Homo sapiens (Human))
BDBM50129158
PNG
(7-Fluoro-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-az...)
Show SMILES CC1=CC(C)(C)Nc2ccc-3c(COc4c(F)cccc-34)c12
Show InChI InChI=1S/C19H18FNO/c1-11-9-19(2,3)21-16-8-7-12-13-5-4-6-15(20)18(13)22-10-14(12)17(11)16/h4-9,21H,10H2,1-3H3
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248n/an/an/an/an/an/an/an/a



Ligand Pharmaceuticals

Curated by ChEMBL


Assay Description
Binding affinity at human progesterone receptor.


Bioorg Med Chem Lett 13: 2075-8 (2003)


Article DOI: 10.1016/s0960-894x(03)00256-7
BindingDB Entry DOI: 10.7270/Q2P55P2M
More data for this
Ligand-Target Pair
Androgen Receptor


(Homo sapiens (Human))
BDBM50077094
PNG
(6-Ethyl-1,9-dimethyl-4-trifluoromethyl-6,7,8,9-tet...)
Show SMILES CCC1CCN(C)c2cc3n(C)c(=O)cc(c3cc12)C(F)(F)F
Show InChI InChI=1/C17H19F3N2O/c1-4-10-5-6-21(2)14-9-15-12(7-11(10)14)13(17(18,19)20)8-16(23)22(15)3/h7-10H,4-6H2,1-3H3
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263n/an/an/an/an/an/an/an/a



Ligand Pharmaceuticals, Inc.

Curated by ChEMBL


Assay Description
Antagonistic activity against human androgen receptor (hAR) in CV-1 cells was determined as a function of maximal inhibition of dihydrotestosterone u...


Bioorg Med Chem Lett 9: 1335-40 (1999)


Article DOI: 10.1016/s0960-894x(99)00186-9
BindingDB Entry DOI: 10.7270/Q2JM2B4G
More data for this
Ligand-Target Pair
Progesterone receptor


(Homo sapiens (Human))
BDBM50129170
PNG
(7-Chloro-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-az...)
Show SMILES CC1=CC(C)(C)Nc2ccc-3c(COc4c(Cl)cccc-34)c12
Show InChI InChI=1S/C19H18ClNO/c1-11-9-19(2,3)21-16-8-7-12-13-5-4-6-15(20)18(13)22-10-14(12)17(11)16/h4-9,21H,10H2,1-3H3
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273n/an/an/an/an/an/an/an/a



Ligand Pharmaceuticals

Curated by ChEMBL


Assay Description
Binding affinity at human progesterone receptor.


Bioorg Med Chem Lett 13: 2075-8 (2003)


Article DOI: 10.1016/s0960-894x(03)00256-7
BindingDB Entry DOI: 10.7270/Q2P55P2M
More data for this
Ligand-Target Pair
Progesterone receptor


(Homo sapiens (Human))
BDBM50129164
PNG
(9-Bromo-7-fluoro-2,2,4-trimethyl-2,5-dihydro-1H-6-...)
Show SMILES CC1=CC(C)(C)Nc2ccc-3c(COc4c(F)c(C=O)c(Br)cc-34)c12
Show InChI InChI=1S/C20H17BrFNO2/c1-10-7-20(2,3)23-16-5-4-11-12-6-15(21)13(8-24)18(22)19(12)25-9-14(11)17(10)16/h4-8,23H,9H2,1-3H3
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290n/an/an/an/an/an/an/an/a



Ligand Pharmaceuticals

Curated by ChEMBL


Assay Description
Binding towards human progesterone receptor; Not tested


Bioorg Med Chem Lett 13: 2075-8 (2003)


Article DOI: 10.1016/s0960-894x(03)00256-7
BindingDB Entry DOI: 10.7270/Q2P55P2M
More data for this
Ligand-Target Pair
Progesterone receptor


(Homo sapiens (Human))
BDBM50129162
PNG
(8-Methoxy-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-a...)
Show SMILES COc1ccc-2c(OCc3c-2ccc2NC(C)(C)C=C(C)c32)c1
Show InChI InChI=1S/C20H21NO2/c1-12-10-20(2,3)21-17-8-7-14-15-6-5-13(22-4)9-18(15)23-11-16(14)19(12)17/h5-10,21H,11H2,1-4H3
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357n/an/an/an/an/an/an/an/a



Ligand Pharmaceuticals

Curated by ChEMBL


Assay Description
Antagonistic activity at human progesterone receptor in CV-1 cells.


Bioorg Med Chem Lett 13: 2075-8 (2003)


Article DOI: 10.1016/s0960-894x(03)00256-7
BindingDB Entry DOI: 10.7270/Q2P55P2M
More data for this
Ligand-Target Pair
Progesterone receptor


(Homo sapiens (Human))
BDBM50129175
PNG
(9-Fluoro-2,2,4-trimethyl-7-nitro-2,3,4,5-tetrahydr...)
Show SMILES CC1CC(C)(C)Nc2ccc-3c(COc4c-3cc(F)cc4[N+]([O-])=O)c12
Show InChI InChI=1/C19H19FN2O3/c1-10-8-19(2,3)21-15-5-4-12-13-6-11(20)7-16(22(23)24)18(13)25-9-14(12)17(10)15/h4-7,10,21H,8-9H2,1-3H3
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370n/an/an/an/an/an/an/an/a



Ligand Pharmaceuticals

Curated by ChEMBL


Assay Description
Inhibition of human progesterone receptor activation in T47D human breast cancer cell.


Bioorg Med Chem Lett 13: 2075-8 (2003)


Article DOI: 10.1016/s0960-894x(03)00256-7
BindingDB Entry DOI: 10.7270/Q2P55P2M
More data for this
Ligand-Target Pair
Progesterone receptor


(Homo sapiens (Human))
BDBM50129176
PNG
(9-Fluoro-2,2,4,7-tetramethyl-2,3,4,5-tetrahydro-1H...)
Show SMILES CC1CC(C)(C)Nc2ccc-3c(COc4c(C)cc(F)cc-34)c12
Show InChI InChI=1/C20H22FNO/c1-11-7-13(21)8-15-14-5-6-17-18(16(14)10-23-19(11)15)12(2)9-20(3,4)22-17/h5-8,12,22H,9-10H2,1-4H3
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391n/an/an/an/an/an/an/an/a



Ligand Pharmaceuticals

Curated by ChEMBL


Assay Description
Binding affinity at human progesterone receptor.


Bioorg Med Chem Lett 13: 2075-8 (2003)


Article DOI: 10.1016/s0960-894x(03)00256-7
BindingDB Entry DOI: 10.7270/Q2P55P2M
More data for this
Ligand-Target Pair
Progesterone receptor


(Homo sapiens (Human))
BDBM50129169
PNG
(9-Bromo-7-methoxy-2,2,4-trimethyl-2,5-dihydro-1H-6...)
Show SMILES COc1cc(Br)cc-2c1OCc1c-2ccc2NC(C)(C)C=C(C)c12
Show InChI InChI=1S/C20H20BrNO2/c1-11-9-20(2,3)22-16-6-5-13-14-7-12(21)8-17(23-4)19(14)24-10-15(13)18(11)16/h5-9,22H,10H2,1-4H3
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476n/an/an/an/an/an/an/an/a



Ligand Pharmaceuticals

Curated by ChEMBL


Assay Description
Binding affinity at human progesterone receptor.


Bioorg Med Chem Lett 13: 2075-8 (2003)


Article DOI: 10.1016/s0960-894x(03)00256-7
BindingDB Entry DOI: 10.7270/Q2P55P2M
More data for this
Ligand-Target Pair
Androgen Receptor


(Homo sapiens (Human))
BDBM50077107
PNG
(6-Ethyl-9-methyl-4-trifluoromethyl-6,7,8,9-tetrahy...)
Show SMILES CCC1CCN(C)c2cc3[nH]c(=O)cc(c3cc12)C(F)(F)F
Show InChI InChI=1/C16H17F3N2O/c1-3-9-4-5-21(2)14-8-13-11(6-10(9)14)12(16(17,18)19)7-15(22)20-13/h6-9H,3-5H2,1-2H3,(H,20,22)
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630n/an/an/an/an/an/an/an/a



Ligand Pharmaceuticals, Inc.

Curated by ChEMBL


Assay Description
Binding affinity to the human androgen receptor (hAR), using [3H]DHT as radioligand in a competitive binding assay


Bioorg Med Chem Lett 9: 1335-40 (1999)


Article DOI: 10.1016/s0960-894x(99)00186-9
BindingDB Entry DOI: 10.7270/Q2JM2B4G
More data for this
Ligand-Target Pair
Progesterone receptor


(Homo sapiens (Human))
BDBM50129177
PNG
(2,2,4-Trimethyl-8-trifluoromethyl-2,5-dihydro-1H-6...)
Show SMILES CC1=CC(C)(C)Nc2ccc-3c(COc4cc(ccc-34)C(F)(F)F)c12
Show InChI InChI=1S/C20H18F3NO/c1-11-9-19(2,3)24-16-7-6-13-14-5-4-12(20(21,22)23)8-17(14)25-10-15(13)18(11)16/h4-9,24H,10H2,1-3H3
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>1.00E+3n/an/an/an/an/an/an/an/a



Ligand Pharmaceuticals

Curated by ChEMBL


Assay Description
Binding affinity at human progesterone receptor.


Bioorg Med Chem Lett 13: 2075-8 (2003)


Article DOI: 10.1016/s0960-894x(03)00256-7
BindingDB Entry DOI: 10.7270/Q2P55P2M
More data for this
Ligand-Target Pair
Androgen Receptor


(Homo sapiens (Human))
BDBM50077102
PNG
(6-(3,5-Bis-trifluoromethyl-phenyl)-4-trifluorometh...)
Show SMILES FC(F)(F)c1cc(cc(c1)C(F)(F)F)C1CCNc2cc3[nH]c(=O)cc(c3cc12)C(F)(F)F
Show InChI InChI=1/C21H13F9N2O/c22-19(23,24)10-3-9(4-11(5-10)20(25,26)27)12-1-2-31-16-8-17-14(6-13(12)16)15(21(28,29)30)7-18(33)32-17/h3-8,12,31H,1-2H2,(H,32,33)
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>1.00E+3n/an/an/an/an/an/an/an/a



Ligand Pharmaceuticals, Inc.

Curated by ChEMBL


Assay Description
Agonist activity to the human androgen receptor (hAR) in CV-1 cells


Bioorg Med Chem Lett 9: 1335-40 (1999)


Article DOI: 10.1016/s0960-894x(99)00186-9
BindingDB Entry DOI: 10.7270/Q2JM2B4G
More data for this
Ligand-Target Pair
Progesterone receptor


(Homo sapiens (Human))
BDBM50129174
PNG
(7,9-Dibromo-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1...)
Show SMILES CC1=CC(C)(C)Nc2ccc-3c(COc4c(Br)cc(Br)cc-34)c12
Show InChI InChI=1S/C19H17Br2NO/c1-10-8-19(2,3)22-16-5-4-12-13-6-11(20)7-15(21)18(13)23-9-14(12)17(10)16/h4-8,22H,9H2,1-3H3
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>1.00E+3n/an/an/an/an/an/an/an/a



Ligand Pharmaceuticals

Curated by ChEMBL


Assay Description
Binding towards human progesterone receptor


Bioorg Med Chem Lett 13: 2075-8 (2003)


Article DOI: 10.1016/s0960-894x(03)00256-7
BindingDB Entry DOI: 10.7270/Q2P55P2M
More data for this
Ligand-Target Pair
Androgen Receptor


(Homo sapiens (Human))
BDBM50403734
PNG
(CHEMBL2113247)
Show SMILES C[C@@H]1CNc2cc3[nH]c(=O)cc(c3cc2[C@@H]1CCC(F)(F)F)C(F)(F)F
Show InChI InChI=1S/C17H16F6N2O/c1-8-7-24-13-6-14-11(12(17(21,22)23)5-15(26)25-14)4-10(13)9(8)2-3-16(18,19)20/h4-6,8-9,24H,2-3,7H2,1H3,(H,25,26)/t8-,9-/m1/s1
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>1.00E+3n/an/an/an/an/an/an/an/a



Ligand Pharmaceuticals, Inc.

Curated by ChEMBL


Assay Description
Agonist activity to the human androgen receptor (hAR) in CV-1 cells


Bioorg Med Chem Lett 9: 1335-40 (1999)


Article DOI: 10.1016/s0960-894x(99)00186-9
BindingDB Entry DOI: 10.7270/Q2JM2B4G
More data for this
Ligand-Target Pair
Progesterone receptor


(Homo sapiens (Human))
BDBM50129172
PNG
(2,2,4-Trimethyl-9-phenyl-2,5-dihydro-1H-6-oxa-1-az...)
Show SMILES CC1=CC(C)(C)Nc2ccc-3c(COc4ccc(cc-34)-c3ccccc3)c12
Show InChI InChI=1S/C25H23NO/c1-16-14-25(2,3)26-22-11-10-19-20-13-18(17-7-5-4-6-8-17)9-12-23(20)27-15-21(19)24(16)22/h4-14,26H,15H2,1-3H3
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>1.00E+3n/an/an/an/an/an/an/an/a



Ligand Pharmaceuticals

Curated by ChEMBL


Assay Description
Binding affinity at human progesterone receptor.


Bioorg Med Chem Lett 13: 2075-8 (2003)


Article DOI: 10.1016/s0960-894x(03)00256-7
BindingDB Entry DOI: 10.7270/Q2P55P2M
More data for this
Ligand-Target Pair
Androgen Receptor


(Homo sapiens (Human))
BDBM50077101
PNG
(4-Ethyl-8-oxo-6-trifluoromethyl-3,4,8,9-tetrahydro...)
Show SMILES CCC1CCN(C=O)c2cc3[nH]c(=O)cc(c3cc12)C(F)(F)F
Show InChI InChI=1/C16H15F3N2O2/c1-2-9-3-4-21(8-22)14-7-13-11(5-10(9)14)12(16(17,18)19)6-15(23)20-13/h5-9H,2-4H2,1H3,(H,20,23)
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>1.00E+3n/an/an/an/an/an/an/an/a



Ligand Pharmaceuticals, Inc.

Curated by ChEMBL


Assay Description
Agonist activity to the human androgen receptor (hAR) in CV-1 cells


Bioorg Med Chem Lett 9: 1335-40 (1999)


Article DOI: 10.1016/s0960-894x(99)00186-9
BindingDB Entry DOI: 10.7270/Q2JM2B4G
More data for this
Ligand-Target Pair
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