Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Scavenger mRNA-decapping enzyme (DcpS) (Homo sapiens (Human)) | BDBM50232538![]() (5-((1-(2-fluorobenzyl)piperidin-4-yl)methoxy)quina...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt UniProtKB/TrEMBL B.MOAD DrugBank antibodypedia GoogleScholar | CHEMBL DrugBank MMDB PC cid PC sid PDB UniChem Similars | DrugBank MMDB PDB Article PubMed | n/a | n/a | 7.62 | n/a | 4 | n/a | n/a | n/a | n/a |
deCODE Chemistry Inc | Assay Description In vitro biochemical assay using scavenger decapping enzyme (DcpS) as a target and cell based assay using SMN2 b-lactamase NSC-34 cell reporter gene. | ACS Chem Biol 3: 711-22 (2008) Article DOI: 10.1021/cb800120t BindingDB Entry DOI: 10.7270/Q2Z036HN | |||||||||||
More data for this Ligand-Target Pair | ![]() 3D Structure (crystal) | ||||||||||||
Scavenger mRNA-decapping enzyme (DcpS) (Homo sapiens (Human)) | BDBM36533![]() (D157555) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt UniProtKB/TrEMBL B.MOAD DrugBank antibodypedia GoogleScholar | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 9.38 | n/a | 108 | n/a | n/a | n/a | n/a |
deCODE Chemistry Inc | Assay Description In vitro biochemical assay using scavenger decapping enzyme (DcpS) as a target and cell based assay using SMN2 b-lactamase NSC-34 cell reporter gene. | ACS Chem Biol 3: 711-22 (2008) Article DOI: 10.1021/cb800120t BindingDB Entry DOI: 10.7270/Q2Z036HN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Scavenger mRNA-decapping enzyme (DcpS) (Homo sapiens (Human)) | BDBM36531![]() (D158963) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt UniProtKB/TrEMBL B.MOAD DrugBank antibodypedia GoogleScholar | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 23.4 | n/a | 223 | n/a | n/a | n/a | n/a |
deCODE Chemistry Inc | Assay Description In vitro biochemical assay using scavenger decapping enzyme (DcpS) as a target and cell based assay using SMN2 b-lactamase NSC-34 cell reporter gene. | ACS Chem Biol 3: 711-22 (2008) Article DOI: 10.1021/cb800120t BindingDB Entry DOI: 10.7270/Q2Z036HN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ACT1 (R335K) (Baker's yeast) | BDBM65515![]() (76343-93-6 | LAT-A | LatA | Latrunculin A) | PDB GoogleScholar | PC cid PC sid PDB UniChem | PDB Article PubMed | n/a | n/a | 40 | n/a | n/a | n/a | n/a | n/a | 30 |
Novartis Pharma AG | Assay Description Saturated ACT1 wild type (WT) as well as engineered ACT1 R183K (R183K) and ACT1 R335K (R335K) cultures were adjusted to 10 OD600 and 3 uL of serial 1... | ACS Chem Biol 12: 2264-2269 (2017) Article DOI: 10.1021/acschembio.7b00385 BindingDB Entry DOI: 10.7270/Q25B00MP | |||||||||||
More data for this Ligand-Target Pair | ![]() 3D Structure (crystal) | ||||||||||||
Scavenger mRNA-decapping enzyme (DcpS) (Homo sapiens (Human)) | BDBM36530![]() (D157493) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt UniProtKB/TrEMBL B.MOAD DrugBank antibodypedia GoogleScholar | DrugBank MMDB PC cid PC sid PDB UniChem Similars | DrugBank MMDB PDB Article PubMed | n/a | n/a | 43.9 | n/a | 67 | n/a | n/a | n/a | n/a |
deCODE Chemistry Inc | Assay Description In vitro biochemical assay using scavenger decapping enzyme (DcpS) as a target and cell based assay using SMN2 b-lactamase NSC-34 cell reporter gene. | ACS Chem Biol 3: 711-22 (2008) Article DOI: 10.1021/cb800120t BindingDB Entry DOI: 10.7270/Q2Z036HN | |||||||||||
More data for this Ligand-Target Pair | ![]() 3D Structure (crystal) | ||||||||||||
ACT1 (Baker's yeast) | BDBM65515![]() (76343-93-6 | LAT-A | LatA | Latrunculin A) | PDB MMDB UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | PC cid PC sid PDB UniChem | PDB Article PubMed | n/a | n/a | 70 | n/a | n/a | n/a | n/a | n/a | 30 |
Novartis Pharma AG | Assay Description Saturated ACT1 wild type (WT) as well as engineered ACT1 R183K (R183K) and ACT1 R335K (R335K) cultures were adjusted to 10 OD600 and 3 uL of serial 1... | ACS Chem Biol 12: 2264-2269 (2017) Article DOI: 10.1021/acschembio.7b00385 BindingDB Entry DOI: 10.7270/Q25B00MP | |||||||||||
More data for this Ligand-Target Pair | ![]() 3D Structure (crystal) | ||||||||||||
Scavenger mRNA-decapping enzyme (DcpS) (Homo sapiens (Human)) | BDBM36532![]() (D158885) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt UniProtKB/TrEMBL B.MOAD DrugBank antibodypedia GoogleScholar | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 101 | n/a | 795 | n/a | n/a | n/a | n/a |
deCODE Chemistry Inc | Assay Description In vitro biochemical assay using scavenger decapping enzyme (DcpS) as a target and cell based assay using SMN2 b-lactamase NSC-34 cell reporter gene. | ACS Chem Biol 3: 711-22 (2008) Article DOI: 10.1021/cb800120t BindingDB Entry DOI: 10.7270/Q2Z036HN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ACT1 (R183K) (Baker's yeast) | BDBM65515![]() (76343-93-6 | LAT-A | LatA | Latrunculin A) | PDB GoogleScholar | PC cid PC sid PDB UniChem | PDB Article PubMed | n/a | n/a | 110 | n/a | n/a | n/a | n/a | n/a | 30 |
Novartis Pharma AG | Assay Description Saturated ACT1 wild type (WT) as well as engineered ACT1 R183K (R183K) and ACT1 R335K (R335K) cultures were adjusted to 10 OD600 and 3 uL of serial 1... | ACS Chem Biol 12: 2264-2269 (2017) Article DOI: 10.1021/acschembio.7b00385 BindingDB Entry DOI: 10.7270/Q25B00MP | |||||||||||
More data for this Ligand-Target Pair | ![]() 3D Structure (crystal) | ||||||||||||
ACT1 (Baker's yeast) | BDBM65506![]() (CHEBI:80062 | Chivosazole F | SCHEMBL1889389) | PDB MMDB UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 140 | n/a | n/a | n/a | n/a | n/a | 30 |
Novartis Pharma AG | Assay Description Saturated ACT1 wild type (WT) as well as engineered ACT1 R183K (R183K) and ACT1 R335K (R335K) cultures were adjusted to 10 OD600 and 3 uL of serial 1... | ACS Chem Biol 12: 2264-2269 (2017) Article DOI: 10.1021/acschembio.7b00385 BindingDB Entry DOI: 10.7270/Q25B00MP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ACT1 (R335K) (Baker's yeast) | BDBM65506![]() (CHEBI:80062 | Chivosazole F | SCHEMBL1889389) | PDB GoogleScholar | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 270 | n/a | n/a | n/a | n/a | n/a | 30 |
Novartis Pharma AG | Assay Description Saturated ACT1 wild type (WT) as well as engineered ACT1 R183K (R183K) and ACT1 R335K (R335K) cultures were adjusted to 10 OD600 and 3 uL of serial 1... | ACS Chem Biol 12: 2264-2269 (2017) Article DOI: 10.1021/acschembio.7b00385 BindingDB Entry DOI: 10.7270/Q25B00MP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Scavenger mRNA-decapping enzyme (DcpS) (Homo sapiens (Human)) | BDBM36529![]() (D156676) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt UniProtKB/TrEMBL B.MOAD DrugBank antibodypedia GoogleScholar | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 339 | n/a | 2.54E+3 | n/a | n/a | n/a | n/a |
deCODE Chemistry Inc | Assay Description In vitro biochemical assay using scavenger decapping enzyme (DcpS) as a target and cell based assay using SMN2 b-lactamase NSC-34 cell reporter gene. | ACS Chem Biol 3: 711-22 (2008) Article DOI: 10.1021/cb800120t BindingDB Entry DOI: 10.7270/Q2Z036HN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ACT1 (R183K) (Baker's yeast) | BDBM65506![]() (CHEBI:80062 | Chivosazole F | SCHEMBL1889389) | PDB GoogleScholar | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 380 | n/a | n/a | n/a | n/a | n/a | 30 |
Novartis Pharma AG | Assay Description Saturated ACT1 wild type (WT) as well as engineered ACT1 R183K (R183K) and ACT1 R335K (R335K) cultures were adjusted to 10 OD600 and 3 uL of serial 1... | ACS Chem Biol 12: 2264-2269 (2017) Article DOI: 10.1021/acschembio.7b00385 BindingDB Entry DOI: 10.7270/Q25B00MP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ACT1 (R183K) (Baker's yeast) | BDBM65516![]() (CHEBI:84382 | CHEMBL2426321 | Chondramide C | SCHE...) | PDB GoogleScholar | CHEBI CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.19E+4 | n/a | n/a | n/a | n/a | n/a | 30 |
Novartis Pharma AG | Assay Description Saturated ACT1 wild type (WT) as well as engineered ACT1 R183K (R183K) and ACT1 R335K (R335K) cultures were adjusted to 10 OD600 and 3 uL of serial 1... | ACS Chem Biol 12: 2264-2269 (2017) Article DOI: 10.1021/acschembio.7b00385 BindingDB Entry DOI: 10.7270/Q25B00MP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ACT1 (R335K) (Baker's yeast) | BDBM65516![]() (CHEBI:84382 | CHEMBL2426321 | Chondramide C | SCHE...) | PDB GoogleScholar | CHEBI CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.51E+4 | n/a | n/a | n/a | n/a | n/a | 30 |
Novartis Pharma AG | Assay Description Saturated ACT1 wild type (WT) as well as engineered ACT1 R183K (R183K) and ACT1 R335K (R335K) cultures were adjusted to 10 OD600 and 3 uL of serial 1... | ACS Chem Biol 12: 2264-2269 (2017) Article DOI: 10.1021/acschembio.7b00385 BindingDB Entry DOI: 10.7270/Q25B00MP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ACT1 (Baker's yeast) | BDBM65516![]() (CHEBI:84382 | CHEMBL2426321 | Chondramide C | SCHE...) | PDB MMDB UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | CHEBI CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.67E+4 | n/a | n/a | n/a | n/a | n/a | 30 |
Novartis Pharma AG | Assay Description Saturated ACT1 wild type (WT) as well as engineered ACT1 R183K (R183K) and ACT1 R335K (R335K) cultures were adjusted to 10 OD600 and 3 uL of serial 1... | ACS Chem Biol 12: 2264-2269 (2017) Article DOI: 10.1021/acschembio.7b00385 BindingDB Entry DOI: 10.7270/Q25B00MP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Scavenger mRNA-decapping enzyme (DcpS) (Homo sapiens (Human)) | BDBM36535![]() (D157554) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt UniProtKB/TrEMBL B.MOAD DrugBank antibodypedia GoogleScholar | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 921 | n/a | n/a | n/a | n/a |
deCODE Chemistry Inc | Assay Description In vitro biochemical assay using scavenger decapping enzyme (DcpS) as a target and cell based assay using SMN2 b-lactamase NSC-34 cell reporter gene. | ACS Chem Biol 3: 711-22 (2008) Article DOI: 10.1021/cb800120t BindingDB Entry DOI: 10.7270/Q2Z036HN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Scavenger mRNA-decapping enzyme (DcpS) (Homo sapiens (Human)) | BDBM36534![]() (D156095) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt UniProtKB/TrEMBL B.MOAD DrugBank antibodypedia GoogleScholar | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 104 | n/a | n/a | n/a | n/a |
deCODE Chemistry Inc | Assay Description In vitro biochemical assay using scavenger decapping enzyme (DcpS) as a target and cell based assay using SMN2 b-lactamase NSC-34 cell reporter gene. | ACS Chem Biol 3: 711-22 (2008) Article DOI: 10.1021/cb800120t BindingDB Entry DOI: 10.7270/Q2Z036HN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Scavenger mRNA-decapping enzyme (DcpS) (Homo sapiens (Human)) | BDBM36536![]() (D153215) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt UniProtKB/TrEMBL B.MOAD DrugBank antibodypedia GoogleScholar | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 243 | n/a | n/a | n/a | n/a |
deCODE Chemistry Inc | Assay Description In vitro biochemical assay using scavenger decapping enzyme (DcpS) as a target and cell based assay using SMN2 b-lactamase NSC-34 cell reporter gene. | ACS Chem Biol 3: 711-22 (2008) Article DOI: 10.1021/cb800120t BindingDB Entry DOI: 10.7270/Q2Z036HN | |||||||||||
More data for this Ligand-Target Pair |