TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))
Universita Degli Studi Di Torino
Curated by ChEMBL
Universita Degli Studi Di Torino
Curated by ChEMBL
Affinity DataEC50: 2.85E+3nMAssay Description:Inhibition of MRP1 expressed in MDCK cells assessed as calcein AM accumulation by fluorescence assayMore data for this Ligand-Target Pair
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))
Universita Degli Studi Di Torino
Curated by ChEMBL
Universita Degli Studi Di Torino
Curated by ChEMBL
Affinity DataEC50: 1.90E+4nMAssay Description:Inhibition of MRP1 in human 2008/MRP1 cells assessed as potentiation of doxorubicin-induced cytotoxicity by measuring reduction in cell survival afte...More data for this Ligand-Target Pair
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))
Universita Degli Studi Di Torino
Curated by ChEMBL
Universita Degli Studi Di Torino
Curated by ChEMBL
Affinity DataEC50: 1.24E+4nMAssay Description:Modulation of MRP1 mediated drug efflux in doxorubicin-resistant human H69 cells assessed as accumulation of calcein AM incubated for 15 mins prior t...More data for this Ligand-Target Pair