TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Catania
Curated by ChEMBL
University Of Catania
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-pentazocine from sigma1 receptor in guinea pig brain membranes by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 3.63E+5nMAssay Description:Inhibition of human CES1More data for this Ligand-Target Pair
Affinity DataKi: 5.64E+5nMAssay Description:Inhibition of HDAC in human Hela cells nuclear extracts by fluorimetric assayMore data for this Ligand-Target Pair
TargetUDP-glucuronosyltransferase 2B7(Homo sapiens (Human))
The University Of British Columbia
Curated by ChEMBL
The University Of British Columbia
Curated by ChEMBL
Affinity DataKi: 1.60E+6nMAssay Description:Inhibition of AZT glucuronidation by human recombinant UGT2B7More data for this Ligand-Target Pair
Affinity DataKi: 7.90E+6nMAssay Description:Inhibition of human CES2More data for this Ligand-Target Pair
Affinity DataKi: 9.15E+6nMAssay Description:Mechanism based inhibition of human cytochrome P450 2A6 measured by coumarin 7-hydroxylationMore data for this Ligand-Target Pair