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Found 4 of ec50 for monomerid = 50016017
TargetD(2) dopamine receptor(Homo sapiens (Human))
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50016017((5aR,9aR)-6-Propyl-5,5a,6,7,8,9,9a,10-octahydro-py...)
Affinity DataEC50:  45nMAssay Description:Agonist activity at human dopamine D2L receptor expressed in CHO cell membranes incubated for 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50016017((5aR,9aR)-6-Propyl-5,5a,6,7,8,9,9a,10-octahydro-py...)
Affinity DataEC50:  1nMAssay Description:Agonist activity at human recombinant dopamine D3 receptor expressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50016017((5aR,9aR)-6-Propyl-5,5a,6,7,8,9,9a,10-octahydro-py...)
Affinity DataEC50:  2nMAssay Description:Agonist activity at human recombinant dopamine D2 receptor expressed in rat pituitary cells assessed as inhibition of forskolin-stimulated cAMP accum...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50016017((5aR,9aR)-6-Propyl-5,5a,6,7,8,9,9a,10-octahydro-py...)
Affinity DataEC50:  45nMAssay Description:Agonist activity at human dopamine D2L receptor expressed in CHO cell membranes incubated for 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed