Affinity DataKd: 1.50E+4nMAssay Description:Binding affinity to RXRalpha-LBD (unknown origin) measured up to 120 sec by surface plasma resonance methodMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Eindhoven University Of Technology
Curated by ChEMBL
Eindhoven University Of Technology
Curated by ChEMBL
Affinity DataKd: 3.30E+3nMAssay Description:Binding affinity to PPARgamma LBD (unknown origin) assessed as dissociation constant followed by heating for 3 mins by Bradford assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Eindhoven University Of Technology
Curated by ChEMBL
Eindhoven University Of Technology
Curated by ChEMBL
Affinity DataKd: 48nMAssay Description:Binding affinity to PPARg (unknown origin) by SPR assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Eindhoven University Of Technology
Curated by ChEMBL
Eindhoven University Of Technology
Curated by ChEMBL
Affinity DataKd: 1.20nMAssay Description:Inhibition of FTase-catalyzed incorporation of [3H]- FPP radioligand into recombinant Ha-Ras by 50% at an enzyme concentration of 1 nM.More data for this Ligand-Target Pair