Affinity DataEC50: 1.80nMAssay Description:Effective concentration which increases intracellular c-AMP production in human Prostanoid IP receptorMore data for this Ligand-Target Pair
TargetProstaglandin E2 receptor EP4 subtype(Mus musculus (Mouse))
Minase Research Institute
Curated by ChEMBL
Minase Research Institute
Curated by ChEMBL
Affinity DataEC50: 2.5nMAssay Description:Effective concentration which increases intracellular c-AMP production in mouse Prostanoid EP4 receptorMore data for this Ligand-Target Pair
TargetProstaglandin E2 receptor EP4 subtype(Mus musculus (Mouse))
Minase Research Institute
Curated by ChEMBL
Minase Research Institute
Curated by ChEMBL
Affinity DataEC50: 2.5nMAssay Description:Affinity for mouse Prostanoid EP1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetProstaglandin E2 receptor EP4 subtype(Mus musculus (Mouse))
Minase Research Institute
Curated by ChEMBL
Minase Research Institute
Curated by ChEMBL
Affinity DataEC50: 2.5nMAssay Description:Affinity for mouse Prostanoid EP4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetProstaglandin E2 receptor EP2 subtype(Mus musculus (Mouse))
Minase Research Institute
Curated by ChEMBL
Minase Research Institute
Curated by ChEMBL
Affinity DataEC50: 2.60nMAssay Description:Effective concentration which increases intracellular c-AMP production in mouse Prostanoid EP2 receptorMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 4 group A member 2(Rattus norvegicus)
Goethe University Frankfurt
Curated by ChEMBL
Goethe University Frankfurt
Curated by ChEMBL
Affinity DataEC50: 3.00E+3nMAssay Description:Agonist activity at Nurr1 in rat N27-A cells measured by NBRE-based luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 4 group A member 2(Mus musculus)
Goethe University Frankfurt
Curated by ChEMBL
Goethe University Frankfurt
Curated by ChEMBL
Affinity DataEC50: 3.00E+3nMAssay Description:Agonist activity at Nurr1 in mouse MN9D cells measured by Gal4-based luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 4 group A member 2(Mus musculus)
Goethe University Frankfurt
Curated by ChEMBL
Goethe University Frankfurt
Curated by ChEMBL
Affinity DataEC50: 3.00E+3nMAssay Description:Agonist activity at Nurr1 in mouse MN9D cells measured by NBRE-based luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 4 group A member 2(Homo sapiens (Human))
Goethe University Frankfurt
Curated by ChEMBL
Goethe University Frankfurt
Curated by ChEMBL
Affinity DataEC50: 3.00E+3nMAssay Description:Agonist activity at Nurr1 in human SK-N-BE(2)-C cells measured by Gal4-based luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 4 group A member 2(Rattus norvegicus)
Goethe University Frankfurt
Curated by ChEMBL
Goethe University Frankfurt
Curated by ChEMBL
Affinity DataEC50: 3.00E+3nMAssay Description:Agonist activity at Nurr1 in rat N27-A cells measured by Gal4-based luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 4 group A member 2(Homo sapiens (Human))
Goethe University Frankfurt
Curated by ChEMBL
Goethe University Frankfurt
Curated by ChEMBL
Affinity DataEC50: 3.00E+3nMAssay Description:Agonist activity at Nurr1 in human SK-N-BE(2)-C cells measured by NBRE-based luciferase reporter gene assayMore data for this Ligand-Target Pair