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1,25-dihydroxyvitamin D(3) 24-hydroxylase, mitochondrial(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL

BDBM50200182((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...)

EC50: 3nMAssay Description:Induction of CYP24A1 (unknown orgin) transcriptional activity trasfected in human MCF7 cells incuabted for 48 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair

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Vitamin D3 receptor(Homo sapiens (Human))
National Institute Of Health Sciences

Curated by ChEMBL

BDBM50200182((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...)

EC50: 1nMAssay Description:Transactivation of GAL4-fused VDR ligand binding domain expressed in human HeLa cells after 16 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
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Vitamin D3 receptor(Homo sapiens (Human))
National Institute Of Health Sciences

Curated by ChEMBL

BDBM50200182((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...)

EC50: 7.70nMAssay Description:Inhibition of human VDR-cofactor interaction by EnBio receptor cofactor assay systemMore data for this Ligand-Target Pair

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Vitamin D3 receptor(Homo sapiens (Human))
National Institute Of Health Sciences

Curated by ChEMBL

BDBM50200182((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...)

EC50: 322nMAssay Description:Transactivation of VDR in human HaCaT cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair

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Vitamin D3 receptor(Homo sapiens (Human))
National Institute Of Health Sciences

Curated by ChEMBL

BDBM50200182((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...)

EC50: 515nMAssay Description:Transactivation of VDR in human Caco2 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair

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Vitamin D3 receptor(Homo sapiens (Human))
National Institute Of Health Sciences

Curated by ChEMBL

BDBM50200182((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...)

EC50: 0.120nMAssay Description:Agonist activity at VDR in human HEK293 cells assessed as transcriptional activity after 16 to 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair

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Vitamin D3 receptor(Homo sapiens (Human))
National Institute Of Health Sciences

Curated by ChEMBL

BDBM50200182((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...)

EC50: 0.600nMAssay Description:Agonist activity at VDR (unknown origin) expressed in HEK293 cells cotransfected with RXRalpha assessed as RXRalpha recruitment by two-hybrid assayMore data for this Ligand-Target Pair

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Vitamin D3 receptor(Rattus norvegicus)
University Of Wisconsin-Madison

Curated by ChEMBL

BDBM50200182((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...)

EC50: 0.200nMAssay Description:Activity at VDR in rat ROS 17/2.8 cells assessed as transcriptional activation of 24-hydroxylase gene promoter after 16 hrs by luciferase reporter ge...More data for this Ligand-Target Pair

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Vitamin D3 receptor(Homo sapiens (Human))
National Institute Of Health Sciences

Curated by ChEMBL

BDBM50200182((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...)

EC50: 10nMAssay Description:Activation of VDR in human THP1 cells assessed as increase in 25-hydroxyvitamin D-24-hydroxylase mRNA expression by RT-PCRMore data for this Ligand-Target Pair

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Vitamin D3 receptor(Homo sapiens (Human))
National Institute Of Health Sciences

Curated by ChEMBL

BDBM50200182((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...)

EC50: 10nMAssay Description:Activation of VDR in human THP1 cells assessed as increase in cathelicidin antimicrobial peptide mRNA expression by RT-PCRMore data for this Ligand-Target Pair

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Vitamin D3 receptor(Homo sapiens (Human))
National Institute Of Health Sciences

Curated by ChEMBL

BDBM50200182((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...)

EC50: 0.300nMAssay Description:Agonist activity at VDR expressed in human HuH7 cells after 24 hrs by pDR3-luciferase reporter gene assayMore data for this Ligand-Target Pair

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Vitamin D3 receptor(Rattus norvegicus)
University Of Wisconsin-Madison

Curated by ChEMBL

BDBM50200182((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...)

EC50: 0.200nMAssay Description:Activity at rat recombinant full length VDR expressed in rat ROS 17/2.8 cells transfected with 24-hydroxylase gene promoter assessed as transcription...More data for this Ligand-Target Pair

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Vitamin D3 receptor(Homo sapiens (Human))
National Institute Of Health Sciences

Curated by ChEMBL

BDBM50200182((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...)

EC50: 3.90nMAssay Description:Activation of VDR in human Jurkat cells expressing lentiviral VDRE-luciferase vector assessed as VDRE-mediated transcriptional activity measured afte...More data for this Ligand-Target Pair

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Vitamin D3 receptor(Homo sapiens (Human))
National Institute Of Health Sciences

Curated by ChEMBL

BDBM50200182((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...)

EC50: 223nMAssay Description:Activation of VDR in human Caco2 cells expressing lentiviral VDRE-luciferase vector assessed as VDRE-mediated transcriptional activity measured after...More data for this Ligand-Target Pair

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Vitamin D3 receptor(Homo sapiens (Human))
National Institute Of Health Sciences

Curated by ChEMBL

BDBM50200182((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...)

EC50: 250nMAssay Description:Activation of VDR in human HaCaT cells expressing lentiviral VDRE-luciferase vector assessed as VDRE-mediated transcriptional activity measured after...More data for this Ligand-Target Pair

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Vitamin D3 receptor(Bos taurus)
Showa Pharmaceutical University

Curated by ChEMBL

BDBM50200182((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...)

EC50: 0.0500nMAssay Description:Displacement of [3H]1,25-(OH)2D3 from bovine thymus vitamin D receptorMore data for this Ligand-Target Pair

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Vitamin D3 receptor(Rattus norvegicus)
University Of Wisconsin-Madison

Curated by ChEMBL

BDBM50200182((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...)

EC50: 0.300nMAssay Description:Activity at VDR in rat osteosarcoma cells assessed as induction of 24-hydroxylase reporter gene transcription by luciferase reporter gene assayMore data for this Ligand-Target Pair

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Vitamin D3 receptor(Homo sapiens (Human))
National Institute Of Health Sciences

Curated by ChEMBL

BDBM50200182((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...)

EC50: 0.0100nMAssay Description:Activity at human VDR expressed in human HOS cells transfected with pGL3-hOc, pCDNA-hVDR and phRL-TK assessed as assessed as transcriptional activati...More data for this Ligand-Target Pair

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Vitamin D3 receptor(Rattus norvegicus)
University Of Wisconsin-Madison

Curated by ChEMBL

BDBM50200182((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...)

EC50: 0.200nMAssay Description:Agonist activity at rat VDR in ROS 17/2.8 cells transfected with Cyp24a1 reporter plasmid assessed as increase in Cyp24a1 transcription after 16 hrs ...More data for this Ligand-Target Pair

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Vitamin D3 receptor(Homo sapiens (Human))
National Institute Of Health Sciences

Curated by ChEMBL

BDBM50200182((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...)

EC50: 2.5nMAssay Description:Transactivation of full length human VDR expressed in human HeLa cells assessed as increase in CYP24 transcription after 18 hrs by luciferase reporte...More data for this Ligand-Target Pair

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Vitamin D3 receptor(Homo sapiens (Human))
National Institute Of Health Sciences

Curated by ChEMBL

BDBM50200182((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...)

EC50: 3.28nMAssay Description:Agonist activity at VDR in human MCF7 cells assessed as transcription of CYP24A1 gene after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair

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Vitamin D3 receptor(Rattus norvegicus)
University Of Wisconsin-Madison

Curated by ChEMBL

BDBM50200182((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...)

EC50: 0.200nMAssay Description:Activity at VDR in rat osteosarcoma cells assessed as 24-hydroxylase transcription by reporter gene assayMore data for this Ligand-Target Pair

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Vitamin D3 receptor(Rattus norvegicus)
University Of Wisconsin-Madison

Curated by ChEMBL

BDBM50200182((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...)

EC50: 0.0500nMAssay Description:Displacement of 1-alpha,25-dihydroxyvitamin from rat recombinant VDRMore data for this Ligand-Target Pair

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Vitamin D3 receptor(Bos taurus)
Showa Pharmaceutical University

Curated by ChEMBL

BDBM50200182((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...)

EC50: 0.0710nMAssay Description:Displacement of [3H]1,25-(OH)2D3 from vitamin D receptor in bovine thymusMore data for this Ligand-Target Pair

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Vitamin D3 receptor(Homo sapiens (Human))
National Institute Of Health Sciences

Curated by ChEMBL

BDBM50200182((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...)

EC50: 0.5nMAssay Description:Induction of transactivation of human VDR responsive gene in COS7 cells by rat osteopontin luciferase reporter gene assayMore data for this Ligand-Target Pair

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Vitamin D3 receptor(Homo sapiens (Human))
National Institute Of Health Sciences

Curated by ChEMBL

BDBM50200182((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...)

EC50: 15nMAssay Description:Agonist activity at VDR ligand binding domain (unknown origin) by reporter gene assayMore data for this Ligand-Target Pair

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Vitamin D3 receptor(Homo sapiens (Human))
National Institute Of Health Sciences

Curated by ChEMBL

BDBM50200182((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...)

EC50: 3nMAssay Description:Agonist activity at CMX-GAL4 tagged human VDR expressed in HEK293 cells assessed as increase in transcriptional activity by luciferase reporter gene ...More data for this Ligand-Target Pair

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Vitamin D3 receptor(Homo sapiens (Human))
National Institute Of Health Sciences

Curated by ChEMBL

BDBM50200182((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...)

EC50: 0.555nMAssay Description:Effect on VDR transcriptional activity in human osteosarcoma cells in presence of 5% fetal calf serumMore data for this Ligand-Target Pair

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Vitamin D3 receptor(Homo sapiens (Human))
National Institute Of Health Sciences

Curated by ChEMBL

BDBM50200182((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...)

EC50: 0.0106nMAssay Description:Effect on VDR transcriptional activity in human osteosarcoma cellsMore data for this Ligand-Target Pair

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Vitamin D3 receptor(Homo sapiens (Human))
National Institute Of Health Sciences

Curated by ChEMBL

BDBM50200182((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...)

EC50: 3.52nMAssay Description:Effect on VDR transcriptional activity in human Caco-2 cells in presence of 5% fetal calf serumMore data for this Ligand-Target Pair

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Vitamin D3 receptor(Homo sapiens (Human))
National Institute Of Health Sciences

Curated by ChEMBL

BDBM50200182((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...)

EC50: 1nMAssay Description:Agonist activity at human VDR in HEK293 cells assessed as induction of transcriptional transactivation after 24 hrs by mouse osteopontin luciferase r...More data for this Ligand-Target Pair

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Vitamin D3 receptor(Rattus norvegicus)
University Of Wisconsin-Madison

Curated by ChEMBL

BDBM50200182((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...)

EC50: 0.100nMAssay Description:Displacement of [3H]1,25-(OH)2D3 from rat recombinant His-tagged VDR ligand-binding domain expressed in Escherichia coli BL21More data for this Ligand-Target Pair

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Vitamin D3 receptor(Homo sapiens (Human))
National Institute Of Health Sciences

Curated by ChEMBL

BDBM50200182((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...)

EC50: 0.5nMAssay Description:Agonist activity at human VDR in COS7 cells assessed as induction of transcriptional transactivation after 24 hrs by mouse osteopontin luciferase rep...More data for this Ligand-Target Pair

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Vitamin D3 receptor(Homo sapiens (Human))
National Institute Of Health Sciences

Curated by ChEMBL

BDBM50200182((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...)

EC50: 9nMAssay Description:Agonist activity at VDR in human HL60 cells assessed as induction of cell differentiation after 96 hrs by NBT assayMore data for this Ligand-Target Pair

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Vitamin D3 receptor(Homo sapiens (Human))
National Institute Of Health Sciences

Curated by ChEMBL

BDBM50200182((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...)

EC50: >0.900nMAssay Description:Transactivation of VP16-tagged VDR (unknown origin) expressed in HEK293 cells harboring pCMX-GAL4-SRC-1 and MH100(UAS) X 4tk-LUC reporter plasmid ass...More data for this Ligand-Target Pair

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Vitamin D3 receptor(Homo sapiens (Human))
National Institute Of Health Sciences

Curated by ChEMBL

BDBM50200182((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...)

EC50: 0.0700nMAssay Description:Transactivation of VP16-tagged VDR (unknown origin) expressed in HEK293 cells harboring pCMX-GAL4-RXRalpha and MH100(UAS) X 4tk-LUC reporter plasmid ...More data for this Ligand-Target Pair

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Vitamin D3 receptor(Homo sapiens (Human))
National Institute Of Health Sciences

Curated by ChEMBL

BDBM50200182((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...)

EC50: 1.60nMAssay Description:Agonist activity at VDR in human MCF7 cells assessed as increase in transcription of CYP24A1 gene after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair

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Vitamin D3 receptor A(Danio rerio)
Centre National De La Recherche Scientifique

Curated by ChEMBL

BDBM50200182((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...)

EC50: 5.5nMAssay Description:Agonist activity at zebrafish gal4-VDR LBD expressed in human MCF7 cells by luciferase reporter gene based transactivation assayMore data for this Ligand-Target Pair

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Retinoic acid receptor RXR-alpha/Vitamin D3 receptor(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL

BDBM50200182((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...)

EC50: 1.60nMAssay Description:Transactivation of recombinant human VDR/RXRalpha expressed in HEK293 cells after 24 hrs by Dual-luciferase reporter gene assayMore data for this Ligand-Target Pair

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Vitamin D3 receptor(Homo sapiens (Human))
National Institute Of Health Sciences

Curated by ChEMBL

BDBM50200182((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...)

EC50: 9nMAssay Description:Agonist activity at vitamin D3 receptor in human HL-60 cells assessed as induction of cell differentiation after 96 hrs by NBT dye-based microscopic ...More data for this Ligand-Target Pair

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Vitamin D3 receptor(Homo sapiens (Human))
National Institute Of Health Sciences

Curated by ChEMBL

BDBM50200182((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...)

EC50: 0.0110nMAssay Description:Agonist activity at human VDR expressed in HOS cells co-expressing human RXR by Dual-Glo luciferase reporter gene assayMore data for this Ligand-Target Pair

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Vitamin D3 receptor(Mus musculus)
University Of Connecticut

Curated by ChEMBL

BDBM50200182((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...)

EC50: 100nMAssay Description:Activation of VDR in mouse ASZ001 cells assessed as change in Cyp24A1 mRNA expression after 48 hrs by q-PCR analysisMore data for this Ligand-Target Pair

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Vitamin D3 receptor(Homo sapiens (Human))
National Institute Of Health Sciences

Curated by ChEMBL

BDBM50200182((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...)

EC50: 1.60nMAssay Description:Agonist activity at VDR in human HL-60 cells assessed as induction of cell differentiation of promyelocytes to monocytes after 4 days by NBT reductio...More data for this Ligand-Target Pair

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CHEMBL DrugBank MCE
KEGG MMDB PC cid PC sid PDB Patents Similars

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Vitamin D3 receptor(Homo sapiens (Human))
National Institute Of Health Sciences

Curated by ChEMBL

BDBM50200182((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...)

EC50: 7nMAssay Description:Agonist activity at human VDR expressed in African green monkey COS7 cells expressing mouse osteopontin VDRE assessed as induction of receptor transa...More data for this Ligand-Target Pair

Purchase ChEBI
CHEMBL DrugBank MCE
KEGG MMDB PC cid PC sid PDB Patents Similars

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Vitamin D3 receptor(Homo sapiens (Human))
National Institute Of Health Sciences

Curated by ChEMBL

BDBM50200182((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...)

EC50: 4.90nMAssay Description:Agonist activity at human VDR expressed in HEK293 cells expressing mouse osteopontin VDRE assessed as induction of receptor transactivation incubated...More data for this Ligand-Target Pair

Purchase ChEBI
CHEMBL DrugBank MCE
KEGG MMDB PC cid PC sid PDB Patents Similars

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Vitamin D3 receptor(Homo sapiens (Human))
National Institute Of Health Sciences

Curated by ChEMBL

BDBM50200182((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...)

EC50: 0.100nMAssay Description:Agonist activity at human VDRMore data for this Ligand-Target Pair

Purchase ChEBI
CHEMBL DrugBank MCE
KEGG MMDB PC cid PC sid PDB Patents Similars

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Vitamin D3 receptor(Homo sapiens (Human))
National Institute Of Health Sciences

Curated by ChEMBL

BDBM50200182((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...)

EC50: 0.0260nMAssay Description:Transactivation of VDR-mediated osteocalcin promoter in human HOS/SF cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair

Purchase ChEBI
CHEMBL DrugBank MCE
KEGG MMDB PC cid PC sid PDB Patents Similars