Affinity DataKi: 1.20nMAssay Description:Binding affinity against Dopamine receptor D1 in rat striatal membranes using [3H]SCH-23390More data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Displacement of [3H]fenoldopam from Dopamine receptor D1 of rat striatum membranesMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Binding affinity against Dopamine receptor D2 in rat striatal membranes using [3H]spiperoneMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University Of Nebraska
Curated by PDSP Ki Database
University Of Nebraska
Curated by PDSP Ki Database
Affinity DataKi: 35nMAssay Description:Compound was tested for its binding affinity against Alpha-2 adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:Affinity towards Dopamine receptor D1More data for this Ligand-Target Pair
Affinity DataKi: 151nMAssay Description:Compound was tested for its binding affinity against Alpha-1 adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 790nMAssay Description:Compound was tested for inhibition of [3H]spiroperidol binding against Dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: 810nMAssay Description:Affinity towards Dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: 1.92E+3nMAssay Description:Non-competitive inhibition of JMJD2E relative to alpha-ketoglutarateMore data for this Ligand-Target Pair