TargetGlutamate receptor ionotropic, NMDA 1(RAT)
The Johns Hopkins University
Curated by PDSP Ki Database
The Johns Hopkins University
Curated by PDSP Ki Database
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
The Johns Hopkins University
Curated by PDSP Ki Database
The Johns Hopkins University
Curated by PDSP Ki Database
Affinity DataKi: 53nMAssay Description:Binding affinity of the compound was determined by displacement of [3H]-TCP from PCP N-methyl-D-aspartate glutamate receptor of tissue homogenate pre...More data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, NMDA 2C(Rattus norvegicus (Rat))
National Institute Of Diabetes
Curated by ChEMBL
National Institute Of Diabetes
Curated by ChEMBL
Affinity DataKi: 60nMAssay Description:Binding affinity against phencyclidine receptor was determined by the displacement of [3H]-TCP of whole rat brain minus cerebellum.More data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
The Johns Hopkins University
Curated by PDSP Ki Database
The Johns Hopkins University
Curated by PDSP Ki Database
Affinity DataKi: 65nMAssay Description:Compound was evaluated for its ability to displace [3H]-TCP from PCP N-methyl-D-aspartate glutamate receptor in rat brainMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
The Johns Hopkins University
Curated by PDSP Ki Database
The Johns Hopkins University
Curated by PDSP Ki Database
TargetGlutamate receptor ionotropic, NMDA 2C(Rattus norvegicus (Rat))
National Institute Of Diabetes
Curated by ChEMBL
National Institute Of Diabetes
Curated by ChEMBL
Affinity DataKi: 91nMAssay Description:Binding affinity to sigma site of Phencyclidine receptor by displacement of [3H]-(+)-SKF- 10,047More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 3A(GUINEA PIG)
Syntex Discovery Research
Curated by PDSP Ki Database
Syntex Discovery Research
Curated by PDSP Ki Database
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
The Johns Hopkins University
Curated by PDSP Ki Database
The Johns Hopkins University
Curated by PDSP Ki Database
Affinity DataKi: 520nMAssay Description:Displacement of [3H]5-HT binding to serotonin receptor of rat fundus membranesMore data for this Ligand-Target Pair
Affinity DataKi: 525nMAssay Description:-Log (Ki) value for butyrylcholinesterase by inhibiting DFPMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, NMDA 2C(Rattus norvegicus (Rat))
National Institute Of Diabetes
Curated by ChEMBL
National Institute Of Diabetes
Curated by ChEMBL
Affinity DataKi: 530nMAssay Description:Binding affinity to sigma site of Phencyclidine receptor by displacement of [3H]-(+)-SKF- 10,047More data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
The Johns Hopkins University
Curated by PDSP Ki Database
The Johns Hopkins University
Curated by PDSP Ki Database
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
The Johns Hopkins University
Curated by PDSP Ki Database
The Johns Hopkins University
Curated by PDSP Ki Database
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
TBA
Curated by PDSP Ki Database
TBA
Curated by PDSP Ki Database
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
TBA
Curated by PDSP Ki Database
TBA
Curated by PDSP Ki Database
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
Affinity DataKi: 1.09E+3nMAssay Description:Compound was evaluated for its ability to displace [3H]-(+)-pentazocine from sigma receptor in Guinea pig brainMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
Affinity DataKi: 1.77E+3nMAssay Description:Inhibition of [3H](+)-pentazocine binding to sigma receptor of guinea pig brain homogenatesMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 3A(GUINEA PIG)
Syntex Discovery Research
Curated by PDSP Ki Database
Syntex Discovery Research
Curated by PDSP Ki Database
Affinity DataKi: 1.00E+4nMAssay Description:Mechanism based inhibition of human cytochrome P450 2B6More data for this Ligand-Target Pair