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Found 64 of ki for monomerid = 84994
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM84994(CAS_163091 | NSC_163091 | ORG-5222)
Affinity DataKi:  0.130nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM84994(CAS_163091 | NSC_163091 | ORG-5222)
Affinity DataKi:  0.160nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

Target5-hydroxytryptamine receptor 2C(PIG)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM84994(CAS_163091 | NSC_163091 | ORG-5222)
Affinity DataKi:  0.170nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Eli Lilly

Curated by PDSP Ki Database
LigandPNGBDBM84994(CAS_163091 | NSC_163091 | ORG-5222)
Affinity DataKi:  0.200nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM84994(CAS_163091 | NSC_163091 | ORG-5222)
Affinity DataKi:  0.260nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Eli Lilly

Curated by PDSP Ki Database
LigandPNGBDBM84994(CAS_163091 | NSC_163091 | ORG-5222)
Affinity DataKi:  0.270nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM84994(CAS_163091 | NSC_163091 | ORG-5222)
Affinity DataKi:  0.400nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM84994(CAS_163091 | NSC_163091 | ORG-5222)
Affinity DataKi:  0.490nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Mus musculus (Mouse))
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM84994(CAS_163091 | NSC_163091 | ORG-5222)
Affinity DataKi:  0.720nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM84994(CAS_163091 | NSC_163091 | ORG-5222)
Affinity DataKi:  0.770nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM84994(CAS_163091 | NSC_163091 | ORG-5222)
Affinity DataKi:  0.900nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Eli Lilly

Curated by PDSP Ki Database
LigandPNGBDBM84994(CAS_163091 | NSC_163091 | ORG-5222)
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Eli Lilly

Curated by PDSP Ki Database
LigandPNGBDBM84994(CAS_163091 | NSC_163091 | ORG-5222)
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Mayo Foundation

Curated by PDSP Ki Database
LigandPNGBDBM84994(CAS_163091 | NSC_163091 | ORG-5222)
Affinity DataKi:  1.10nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetD(3) dopamine receptor(Homo sapiens (Human))
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM84994(CAS_163091 | NSC_163091 | ORG-5222)
Affinity DataKi:  1.80nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM84994(CAS_163091 | NSC_163091 | ORG-5222)
Affinity DataKi:  1.87nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetHistamine H1 receptor(RAT)
Eli Lilly

Curated by PDSP Ki Database
LigandPNGBDBM84994(CAS_163091 | NSC_163091 | ORG-5222)
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM84994(CAS_163091 | NSC_163091 | ORG-5222)
In DepthDetails ArticlePubMedDrugBank

TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Eli Lilly

Curated by PDSP Ki Database
LigandPNGBDBM84994(CAS_163091 | NSC_163091 | ORG-5222)
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM84994(CAS_163091 | NSC_163091 | ORG-5222)
Affinity DataKi:  2.60nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Eli Lilly

Curated by PDSP Ki Database
LigandPNGBDBM84994(CAS_163091 | NSC_163091 | ORG-5222)
Affinity DataKi:  2.70nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2C adrenergic receptor(RAT)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM84994(CAS_163091 | NSC_163091 | ORG-5222)
Affinity DataKi:  3.70nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM84994(CAS_163091 | NSC_163091 | ORG-5222)
Affinity DataKi:  3.80nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

Target5-hydroxytryptamine receptor 1B(Homo sapiens (Human))
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM84994(CAS_163091 | NSC_163091 | ORG-5222)
Affinity DataKi:  3.90nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetAlpha-2C adrenergic receptor(RAT)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM84994(CAS_163091 | NSC_163091 | ORG-5222)
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM84994(CAS_163091 | NSC_163091 | ORG-5222)
Affinity DataKi:  4.20nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Eli Lilly

Curated by PDSP Ki Database
LigandPNGBDBM84994(CAS_163091 | NSC_163091 | ORG-5222)
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM84994(CAS_163091 | NSC_163091 | ORG-5222)
Affinity DataKi:  6.5nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1D(Homo sapiens (Human))
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM84994(CAS_163091 | NSC_163091 | ORG-5222)
Affinity DataKi:  7.30nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM84994(CAS_163091 | NSC_163091 | ORG-5222)
Affinity DataKi:  9.30nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM84994(CAS_163091 | NSC_163091 | ORG-5222)
Affinity DataKi:  10nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1D(Homo sapiens (Human))
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM84994(CAS_163091 | NSC_163091 | ORG-5222)
Affinity DataKi:  10.2nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1E(Homo sapiens (Human))
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM84994(CAS_163091 | NSC_163091 | ORG-5222)
Affinity DataKi:  11nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM84994(CAS_163091 | NSC_163091 | ORG-5222)
Affinity DataKi:  13nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM84994(CAS_163091 | NSC_163091 | ORG-5222)
Affinity DataKi:  15nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM84994(CAS_163091 | NSC_163091 | ORG-5222)
Affinity DataKi:  16nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine 1D receptor(Bos taurus (Bovine))
Eli Lilly

Curated by PDSP Ki Database
LigandPNGBDBM84994(CAS_163091 | NSC_163091 | ORG-5222)
Affinity DataKi:  18nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Eli Lilly

Curated by PDSP Ki Database
LigandPNGBDBM84994(CAS_163091 | NSC_163091 | ORG-5222)
Affinity DataKi:  19nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Eli Lilly

Curated by PDSP Ki Database
LigandPNGBDBM84994(CAS_163091 | NSC_163091 | ORG-5222)
Affinity DataKi:  24nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1B(Rattus norvegicus (Rat))
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM84994(CAS_163091 | NSC_163091 | ORG-5222)
Affinity DataKi:  55nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1B(Rattus norvegicus (Rat))
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM84994(CAS_163091 | NSC_163091 | ORG-5222)
Affinity DataKi:  68nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 10 subunit alpha(Rattus norvegicus (Rat))
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM84994(CAS_163091 | NSC_163091 | ORG-5222)
Affinity DataKi:  630nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Mus musculus (house mouse))
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM84994(CAS_163091 | NSC_163091 | ORG-5222)
Affinity DataKi:  800nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM84994(CAS_163091 | NSC_163091 | ORG-5222)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtachykinin-1(Homo sapiens (Human))
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM84994(CAS_163091 | NSC_163091 | ORG-5222)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-arrestin-1(RABBIT)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM84994(CAS_163091 | NSC_163091 | ORG-5222)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM84994(CAS_163091 | NSC_163091 | ORG-5222)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM84994(CAS_163091 | NSC_163091 | ORG-5222)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin(GUINEA PIG)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM84994(CAS_163091 | NSC_163091 | ORG-5222)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNorepinephrine transporter(RAT)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM84994(CAS_163091 | NSC_163091 | ORG-5222)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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