TargetPhenylethanolamine N-methyltransferase(Homo sapiens (Human))
Astex Therapeutics
Curated by ChEMBL
Astex Therapeutics
Curated by ChEMBL
TargetPhenylethanolamine N-methyltransferase(Homo sapiens (Human))
Astex Therapeutics
Curated by ChEMBL
Astex Therapeutics
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of rabbit adrenal phenylethanolamine N-methyl-transferaseMore data for this Ligand-Target Pair
TargetPhenylethanolamine N-methyltransferase(Homo sapiens (Human))
Astex Therapeutics
Curated by ChEMBL
Astex Therapeutics
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Dissociation constant(Ki) of compound was determined to measure PNMT-inhibitory potencyMore data for this Ligand-Target Pair
Affinity DataIC50: 24nMAssay Description:Inhibition of Mer in mouse BaF3 cellsMore data for this Ligand-Target Pair
TargetPhenylethanolamine N-methyltransferase(Homo sapiens (Human))
Astex Therapeutics
Curated by ChEMBL
Astex Therapeutics
Curated by ChEMBL
Affinity DataIC50: 34nMAssay Description:Inhibition of Mer in mouse BaF3 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 34nMAssay Description:Inhibition of Mer in mouse BaF3 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 39nMAssay Description:Inhibition of Mer in mouse BaF3 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 51nMAssay Description:Inhibition of Mer in mouse BaF3 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 55nMAssay Description:Inhibition of Mer in mouse BaF3 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 61nMAssay Description:Inhibition of Mer in mouse BaF3 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 78nMAssay Description:Inhibition of Mer in mouse BaF3 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 79nMAssay Description:Inhibition of Mer in mouse BaF3 cellsMore data for this Ligand-Target Pair
TargetPhenylethanolamine N-methyltransferase(Homo sapiens (Human))
Astex Therapeutics
Curated by ChEMBL
Astex Therapeutics
Curated by ChEMBL
Affinity DataIC50: 80nMAssay Description:Inhibition of rabbit adrenal phenylethanolamine N-methyl-transferaseMore data for this Ligand-Target Pair
Affinity DataIC50: 80nMAssay Description:Inhibition of Mer in mouse BaF3 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 92nMAssay Description:Inhibition of Mer in mouse BaF3 cellsMore data for this Ligand-Target Pair
TargetPhenylethanolamine N-methyltransferase(Homo sapiens (Human))
Astex Therapeutics
Curated by ChEMBL
Astex Therapeutics
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of rabbit adrenal phenylethanolamine N-methyl-transferaseMore data for this Ligand-Target Pair
TargetPhenylethanolamine N-methyltransferase(Homo sapiens (Human))
Astex Therapeutics
Curated by ChEMBL
Astex Therapeutics
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:In vitro inhibitory potency of the compound was measured against phenylethanolamine N-methyltransferaseMore data for this Ligand-Target Pair
Affinity DataIC50: 110nMAssay Description:Inhibition of Mer in mouse BaF3 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 110nMAssay Description:Inhibition of Mer in mouse BaF3 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 130nMAssay Description:Inhibition of Mer in mouse BaF3 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 130nMAssay Description:Inhibition of Mer in mouse BaF3 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 150nMAssay Description:Inhibition of Mer in mouse BaF3 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 180nMAssay Description:Inhibition of Mer in mouse BaF3 cellsMore data for this Ligand-Target Pair
TargetPhenylethanolamine N-methyltransferase(Homo sapiens (Human))
Astex Therapeutics
Curated by ChEMBL
Astex Therapeutics
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:In vitro inhibitory potency of the compound was measured against phenylethanolamine N-methyltransferaseMore data for this Ligand-Target Pair
TargetPhenylethanolamine N-methyltransferase(Homo sapiens (Human))
Astex Therapeutics
Curated by ChEMBL
Astex Therapeutics
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Dissociation constant(Ki) of compound was determined to measure Phenylethanolamine N-methyltransferase inhibitory potencyMore data for this Ligand-Target Pair
TargetPhenylethanolamine N-methyltransferase(Homo sapiens (Human))
Astex Therapeutics
Curated by ChEMBL
Astex Therapeutics
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:In vitro inhibitory potency of the compound was measured against phenylethanolamine N-methyltransferaseMore data for this Ligand-Target Pair
Affinity DataIC50: 210nMAssay Description:Inhibition of Mer in mouse BaF3 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 240nMAssay Description:Inhibition of Mer in mouse BaF3 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 280nMAssay Description:Inhibition of Mer in mouse BaF3 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 280nMAssay Description:Inhibition of Mer in mouse BaF3 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 290nMAssay Description:Inhibition of Mer in mouse BaF3 cellsMore data for this Ligand-Target Pair
TargetPhenylethanolamine N-methyltransferase(Homo sapiens (Human))
Astex Therapeutics
Curated by ChEMBL
Astex Therapeutics
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:Inhibition of rabbit adrenal phenylethanolamine N-methyl-transferaseMore data for this Ligand-Target Pair
TargetPhenylethanolamine N-methyltransferase(Homo sapiens (Human))
Astex Therapeutics
Curated by ChEMBL
Astex Therapeutics
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:Dissociation constant(Ki) of compound was determined to measure Phenylethanolamine N-methyltransferase inhibitory potencyMore data for this Ligand-Target Pair
Affinity DataIC50: 370nMAssay Description:Inhibition of Mer in mouse BaF3 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 370nMAssay Description:Inhibition of Mer in mouse BaF3 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 440nMAssay Description:Inhibition of Mer in mouse BaF3 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 570nMAssay Description:Inhibition of Mer in mouse BaF3 cellsMore data for this Ligand-Target Pair
TargetPhenylethanolamine N-methyltransferase(Homo sapiens (Human))
Astex Therapeutics
Curated by ChEMBL
Astex Therapeutics
Curated by ChEMBL
Affinity DataIC50: 600nMAssay Description:Invitro inhibitory potency of the compound was measured against phenylethanolamine N-methyltransferaseMore data for this Ligand-Target Pair
Affinity DataIC50: 630nMAssay Description:Inhibition of Mer in mouse BaF3 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 730nMAssay Description:Inhibition of Mer in mouse BaF3 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 810nMAssay Description:Inhibition of Mer in mouse BaF3 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 910nMAssay Description:Inhibition of Mer in mouse BaF3 cellsMore data for this Ligand-Target Pair
TargetPhenylethanolamine N-methyltransferase(Homo sapiens (Human))
Astex Therapeutics
Curated by ChEMBL
Astex Therapeutics
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of rabbit adrenal phenylethanolamine N-methyl-transferaseMore data for this Ligand-Target Pair
TargetPhenylethanolamine N-methyltransferase(Homo sapiens (Human))
Astex Therapeutics
Curated by ChEMBL
Astex Therapeutics
Curated by ChEMBL
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of rabbit adrenal phenylethanolamine N-methyl-transferaseMore data for this Ligand-Target Pair
TargetPhenylethanolamine N-methyltransferase(Homo sapiens (Human))
Astex Therapeutics
Curated by ChEMBL
Astex Therapeutics
Curated by ChEMBL
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of rabbit adrenal phenylethanolamine N-methyl-transferaseMore data for this Ligand-Target Pair
TargetPhenylethanolamine N-methyltransferase(Homo sapiens (Human))
Astex Therapeutics
Curated by ChEMBL
Astex Therapeutics
Curated by ChEMBL
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of rabbit adrenal phenylethanolamine N-methyl-transferaseMore data for this Ligand-Target Pair
TargetPhenylethanolamine N-methyltransferase(Homo sapiens (Human))
Astex Therapeutics
Curated by ChEMBL
Astex Therapeutics
Curated by ChEMBL
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of rabbit adrenal phenylethanolamine N-methyl-transferaseMore data for this Ligand-Target Pair
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of Mer in mouse BaF3 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 4.11E+3nMAssay Description:Inhibition of Mer in mouse BaF3 cellsMore data for this Ligand-Target Pair