Found 174 of ic50 data for polymerid = 2421 
Affinity DataIC50: 1.40nMAssay Description:Displacement of SAENTA-fluorescein from human ENT1 in HL60 cells by flow cytometryMore data for this Ligand-Target Pair
Affinity DataIC50: 2.75nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
Affinity DataIC50: 2.80nMAssay Description:Inhibition of human ENT1 expressed in porcine PK15NTD cells by cell-based [3H]5-uridine uptake assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.20nMAssay Description:Inhibition of human ENT1 expressed in porcine PK15NTD cells by cell-based [3H]5-uridine uptake assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4.60nMAssay Description:Inhibition of human ENT1 expressed in porcine PK15NTD cells by cell-based [3H]5-uridine uptake assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4.79nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
Affinity DataIC50: 5.10nMAssay Description:Displacement of SAENTA-fluorescein from human ENT1 in HL60 cells by flow cytometryMore data for this Ligand-Target Pair
Affinity DataIC50: 5.5nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
Affinity DataKi: 0.430nM ΔG°: -12.6kcal/mole IC50: 7.60nMpH: 7.4 T: 2°CAssay Description:The compounds were tested to determine their ENT1 nucleoside transporter binding ability by a flow cytometric assay using human leukemia K562 cells i...More data for this Ligand-Target Pair
3D Structure (crystal)Affinity DataIC50: 8.51nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
Affinity DataKi: 0.490nM ΔG°: -12.6kcal/mole IC50: 8.67nMpH: 7.4 T: 2°CAssay Description:The compounds were tested to determine their ENT1 nucleoside transporter binding ability by a flow cytometric assay using human leukemia K562 cells i...More data for this Ligand-Target Pair
Affinity DataKi: 0.770nM ΔG°: -12.3kcal/mole IC50: 13.6nMpH: 7.4 T: 2°CAssay Description:The compounds were tested to determine their ENT1 nucleoside transporter binding ability by a flow cytometric assay using human leukemia K562 cells i...More data for this Ligand-Target Pair
Affinity DataKi: 0.860nM ΔG°: -12.2kcal/mole IC50: 15.2nMpH: 7.4 T: 2°CAssay Description:The compounds were tested to determine their ENT1 nucleoside transporter binding ability by a flow cytometric assay using human leukemia K562 cells i...More data for this Ligand-Target Pair
Affinity DataIC50: 15.8nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
Affinity DataIC50: 18nMAssay Description:Inhibition of human ENT1 expressed in porcine PK15NTD cells by cell-based [3H]5-uridine uptake assayMore data for this Ligand-Target Pair
Affinity DataIC50: 18nMAssay Description:Inhibition of human ENT1 expressed in porcine PK15NTD cells by cell-based [3H]5-uridine uptake assayMore data for this Ligand-Target Pair
Affinity DataIC50: 21.4nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
Affinity DataIC50: 21.9nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
Affinity DataIC50: 27.5nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
Affinity DataIC50: 31nMAssay Description:Inhibition of human ENT1 expressed in porcine PK15NTD cells by cell-based [3H]5-uridine uptake assayMore data for this Ligand-Target Pair
Affinity DataIC50: 31.6nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
Affinity DataIC50: 33.1nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
Affinity DataIC50: 66nMAssay Description:Inhibition of human ENT1 expressed in porcine PK15NTD cells by cell-based [3H]5-uridine uptake assayMore data for this Ligand-Target Pair
Affinity DataIC50: 69.2nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
Affinity DataKi: 4.30nM IC50: 76nMAssay Description:The compounds were tested to determine their ENT1 nucleoside transporter binding ability by a flow cytometric assay using human leukemia K562 cells i...More data for this Ligand-Target Pair
Affinity DataIC50: 77.6nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
Affinity DataIC50: 81.3nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
Affinity DataIC50: 87.1nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
Affinity DataIC50: 94nMAssay Description:Inhibition of human ENT1 expressed in porcine PK15NTD cells by cell-based [3H]5-uridine uptake assayMore data for this Ligand-Target Pair
Affinity DataIC50: 107nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
Affinity DataIC50: 123nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
Affinity DataKi: 8.18nM ΔG°: -10.9kcal/mole IC50: 145nMpH: 7.4 T: 2°CAssay Description:The compounds were tested to determine their ENT1 nucleoside transporter binding ability by a flow cytometric assay using human leukemia K562 cells i...More data for this Ligand-Target Pair
Affinity DataKi: 8.20nM IC50: 145nMAssay Description:The compounds were tested to determine their ENT1 nucleoside transporter binding ability by a flow cytometric assay using human leukemia K562 cells i...More data for this Ligand-Target Pair
Affinity DataIC50: 158nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
Affinity DataIC50: 178nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
Affinity DataIC50: 178nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
Affinity DataIC50: 182nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
Affinity DataIC50: 182nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
Affinity DataIC50: 190nMAssay Description:Substrate activity at ENT1 in human BXPC-3 cells assessed as inhibition of cell growth pretreated with ENT1 inhibitor nitrobenzylthioinosine for 5 mi...More data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
Affinity DataIC50: 217nMAssay Description:Inhibition of human ENT1 expressed in porcine PK15NTD cells by cell-based [3H]5-uridine uptake assayMore data for this Ligand-Target Pair
Affinity DataIC50: 224nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
Affinity DataIC50: 245nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
Affinity DataIC50: 251nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
Affinity DataKi: 14.7nM IC50: 260nMAssay Description:The compounds were tested to determine their ENT1 nucleoside transporter binding ability by a flow cytometric assay using human leukemia K562 cells i...More data for this Ligand-Target Pair
Affinity DataKi: 15.8nM IC50: 280nMAssay Description:The compounds were tested to determine their ENT1 nucleoside transporter binding ability by a flow cytometric assay using human leukemia K562 cells i...More data for this Ligand-Target Pair
Affinity DataIC50: 282nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
Affinity DataIC50: 282nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
Affinity DataKi: 16.8nM IC50: 297nMAssay Description:The compounds were tested to determine their ENT1 nucleoside transporter binding ability by a flow cytometric assay using human leukemia K562 cells i...More data for this Ligand-Target Pair
Affinity DataKi: 17.1nM IC50: 302nMAssay Description:The compounds were tested to determine their ENT1 nucleoside transporter binding ability by a flow cytometric assay using human leukemia K562 cells i...More data for this Ligand-Target Pair
