Compile Data Set for Download or QSAR
maximum 50k data
Found 384 of ec50 data for polymerid = 325
TargetVasopressin V1a receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50044777(Arginine Vasopressin | Beta-Hypophamine | CHEBI:34...)
Affinity DataEC50:  0.00400nMAssay Description:Agonist activity at recombinant human V1a receptor expressed in HEK293 cells assessed as increase in intracellular calcium level measured at 3 secs i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50240628(CHEMBL4094454)
Affinity DataEC50:  0.0340nMAssay Description:Agonist activity at human V1b receptor expressed in CHO cells assessed as calcium mobilization measured after 30 mins by Fluo-4-AM dye based FLIPR as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50240628(CHEMBL4094454)
Affinity DataEC50:  0.120nMAssay Description:Agonist activity at human V1a receptor expressed in CHO cells assessed as calcium mobilization measured after 30 mins by Fluo-4-AM dye based FLIPR as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50032908(CHEMBL3342789)
Affinity DataEC50:  0.126nMAssay Description:Compound was evaluated for in vitro potency against angiotensin II receptor, type 1 in isolated rabbit aorta; value ranges from 8.27-8.70More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50282232(CHEMBL4165132)
Affinity DataEC50:  0.126nMAssay Description:Compound was evaluated for in vitro potency against AT1 receptor in isolated rabbit aorta; value ranges from 7.91-7.97More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50350874(CHEMBL1819540)
Affinity DataEC50:  0.140nMAssay Description:Agonist activity at recombinant human vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50350866(CHEMBL1819441)
Affinity DataEC50:  0.155nMAssay Description:Agonist activity at recombinant human vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50282233(CHEMBL4173036)
Affinity DataEC50:  0.158nMAssay Description:Compound was evaluated for in vitro potency against angiotensin II receptor, type 1 in isolated rabbit aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50032907(CHEMBL3342790)
Affinity DataEC50:  0.158nMAssay Description:In vitro for histamine H1 receptor antagonist activity against histamine-induced contractions on isolated guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50240673(CHEMBL4096848)
Affinity DataEC50:  0.170nMAssay Description:Agonist activity at human V1b receptor expressed in CHO cells assessed as calcium mobilization measured after 30 mins by Fluo-4-AM dye based FLIPR as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50205990(CHEMBL395429 | OXYTOCIN)
Affinity DataEC50:  0.180nMAssay Description:Agonist activity at human V1A receptor expressed in HEK293 cells assessed as intracellular calcium level measured at 3 secs interval for 5 mins by fu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50205990(CHEMBL395429 | OXYTOCIN)
Affinity DataEC50:  0.190nMAssay Description:Agonist activity at recombinant human V1a receptor expressed in HEK293 cells assessed as increase in intracellular calcium level measured at 3 secs i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50350852(CHEMBL1817706)
Affinity DataEC50:  0.210nMAssay Description:Agonist activity at recombinant human vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50350875(CHEMBL1819541)
Affinity DataEC50:  0.234nMAssay Description:Agonist activity at recombinant human vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50044777(Arginine Vasopressin | Beta-Hypophamine | CHEBI:34...)
Affinity DataEC50:  0.240nMAssay Description:Agonist activity at human vasopressin V1a expressed in HEK293 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50350868(CHEMBL1819555)
Affinity DataEC50:  0.25nMAssay Description:Agonist activity at recombinant human vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50350851(CHEMBL1817705)
Affinity DataEC50:  0.260nMAssay Description:Agonist activity at recombinant human vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50350876(CHEMBL1819542)
Affinity DataEC50:  0.270nMAssay Description:Agonist activity at recombinant human vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50350869(CHEMBL1817704)
Affinity DataEC50:  0.380nMAssay Description:Agonist activity at recombinant human vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50240595(CHEMBL4070577)
Affinity DataEC50:  0.430nMAssay Description:Agonist activity at human V1b receptor expressed in CHO cells assessed as calcium mobilization measured after 30 mins by Fluo-4-AM dye based FLIPR as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50350877(CHEMBL1819543)
Affinity DataEC50:  0.490nMAssay Description:Agonist activity at recombinant human vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50240663(CHEMBL4078856)
Affinity DataEC50:  0.5nMAssay Description:In vitro inhibitory activity against [3H]DTG binding to Sigma opioid receptor in guinea pig brain membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50350882(CHEMBL1819548)
Affinity DataEC50:  0.540nMAssay Description:Agonist activity at recombinant human vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50240631(CHEMBL4065273)
Affinity DataEC50:  0.550nMAssay Description:Agonist activity at human V1b receptor expressed in CHO cells assessed as calcium mobilization measured after 30 mins by Fluo-4-AM dye based FLIPR as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50240675(CHEMBL4101771)
Affinity DataEC50:  0.550nMAssay Description:Agonist activity at human V1b receptor expressed in CHO cells assessed as calcium mobilization measured after 30 mins by Fluo-4-AM dye based FLIPR as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50350853(CHEMBL1817707)
Affinity DataEC50:  0.570nMAssay Description:Agonist activity at recombinant human vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50350906(CHEMBL1819549)
Affinity DataEC50:  0.617nMAssay Description:Agonist activity at recombinant human vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50240649(CHEMBL4063150)
Affinity DataEC50:  0.650nMAssay Description:Agonist activity at human V1b receptor expressed in CHO cells assessed as calcium mobilization measured after 30 mins by Fluo-4-AM dye based FLIPR as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50350872(CHEMBL1817761)
Affinity DataEC50:  0.690nMAssay Description:Agonist activity at recombinant human vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50350865(CHEMBL1819440)
Affinity DataEC50:  0.690nMAssay Description:Agonist activity at recombinant human vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50350867(CHEMBL1819554)
Affinity DataEC50:  0.800nMAssay Description:Agonist activity at recombinant human vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50350854(CHEMBL1817708)
Affinity DataEC50:  0.820nMAssay Description:Agonist activity at recombinant human vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50350849(CHEMBL1817702)
Affinity DataEC50:  0.891nMAssay Description:Agonist activity at recombinant human vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50350887(CHEMBL1819556)
Affinity DataEC50:  0.940nMAssay Description:Agonist activity at recombinant human vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50350861(CHEMBL1817754)
Affinity DataEC50:  1nMAssay Description:Agonist activity at recombinant human vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50350891(CHEMBL1819560)
Affinity DataEC50:  1.20nMAssay Description:Agonist activity at recombinant human vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50240629(CHEMBL4084223)
Affinity DataEC50:  1.30nMAssay Description:Agonist activity at human V1b receptor expressed in CHO cells assessed as calcium mobilization measured after 30 mins by Fluo-4-AM dye based FLIPR as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50350873(CHEMBL1817770)
Affinity DataEC50:  1.40nMAssay Description:Agonist activity at recombinant human vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50240630(CHEMBL4102192)
Affinity DataEC50:  1.40nMAssay Description:Agonist activity at human V1b receptor expressed in CHO cells assessed as calcium mobilization measured after 30 mins by Fluo-4-AM dye based FLIPR as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50350859(CHEMBL1817752)
Affinity DataEC50:  1.40nMAssay Description:Agonist activity at recombinant human vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50350839(CHEMBL1817692)
Affinity DataEC50:  1.5nMAssay Description:Agonist activity at recombinant human vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50205990(CHEMBL395429 | OXYTOCIN)
Affinity DataEC50:  1.5nMAssay Description:Agonist activity at human V1a receptor expressed in CHO cells assessed as calcium mobilization measured after 30 mins by Fluo-4-AM dye based FLIPR as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50350862(CHEMBL1817755)
Affinity DataEC50:  1.5nMAssay Description:Agonist activity at recombinant human vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50350905(CHEMBL1817772)
Affinity DataEC50:  1.60nMAssay Description:Agonist activity at recombinant human vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50350842(CHEMBL1817695)
Affinity DataEC50:  1.70nMAssay Description:Agonist activity at recombinant human vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50350845(CHEMBL1817698)
Affinity DataEC50:  2.10nMAssay Description:Agonist activity at recombinant human vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50350883(CHEMBL1819550)
Affinity DataEC50:  2.20nMAssay Description:Agonist activity at recombinant human vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50523555(CHEMBL4474284)
Affinity DataEC50:  2.20nMAssay Description:Agonist activity at recombinant human V1a receptor expressed in HEK293 cells assessed as increase in intracellular calcium level measured at 3 secs i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50044677(CHEBI:59204 | Carbetocin)
Affinity DataEC50:  2.30nMAssay Description:Agonist activity at recombinant human V1a receptor expressed in HEK293 cells assessed as increase in intracellular calcium level measured at 3 secs i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50350860(CHEMBL1817753)
Affinity DataEC50:  2.40nMAssay Description:Agonist activity at recombinant human vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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