Affinity DataKd: 19nMAssay Description:In vitro Erk5 binding assay: Ambit Kd values in nanomolar. Kd values generated by Ambit binding assay over a concentration range of the compound.More data for this Ligand-Target Pair
Affinity DataKd: 42nMAssay Description:Binding constant for ERK5 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 48nMAssay Description:Binding constant for ERK5 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 50nMAssay Description:In vitro Erk5 binding assay: Ambit Kd values in nanomolar. Kd values generated by Ambit binding assay over a concentration range of the compound.More data for this Ligand-Target Pair
Affinity DataKd: 57nMAssay Description:In vitro Erk5 binding assay: Ambit Kd values in nanomolar. Kd values generated by Ambit binding assay over a concentration range of the compound.More data for this Ligand-Target Pair
Affinity DataKd: 66nMAssay Description:Binding constant for ERK5 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 80nMAssay Description:In vitro biochemical assays were performed in parallel to determine the most potent tool compound.More data for this Ligand-Target Pair
Affinity DataKd: 80nMAssay Description:In vitro Erk5 binding assay: Ambit Kd values in nanomolar. Kd values generated by Ambit binding assay over a concentration range of the compound.More data for this Ligand-Target Pair
Affinity DataKd: 110nMAssay Description:Binding constant for ERK5 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 130nMAssay Description:In vitro kinase assay profiled against a panel of different kinase binding assay using Ambit kinomeScan technology. Biochemical IC50 values were det...More data for this Ligand-Target Pair
Affinity DataKd: 160nMAssay Description:In vitro kinase assay profiled against a panel of different kinase binding assay using Ambit kinomeScan technology. Biochemical IC50 values were det...More data for this Ligand-Target Pair
Affinity DataKd: 180nMAssay Description:Binding affinity to wild-type human partial length MAPK7 (M1 to A409 residues) expressed in bacterial expression system by Kinomescan assayMore data for this Ligand-Target Pair
Affinity DataKd: 320nMAssay Description:In vitro Erk5 binding assay: Ambit Kd values in nanomolar. Kd values generated by Ambit binding assay over a concentration range of the compound.More data for this Ligand-Target Pair
Affinity DataKd: 510nMAssay Description:Binding constant for ERK5 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 520nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
Affinity DataKd: 520nMAssay Description:Binding constant for ERK5 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 550nMAssay Description:In vitro Erk5 binding assay: Ambit Kd values in nanomolar. Kd values generated by Ambit binding assay over a concentration range of the compound.More data for this Ligand-Target Pair
Affinity DataKd: 620nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
Affinity DataKd: 620nMAssay Description:Binding constant for ERK5 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 620nMAssay Description:Binding constant for ERK5 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 620nMAssay Description:Binding constant for ERK5 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 650nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
Affinity DataKd: 650nMAssay Description:Binding constant for ERK5 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 650nMAssay Description:Binding constant for ERK5 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 670nMAssay Description:In vitro Erk5 binding assay: Ambit Kd values in nanomolar. Kd values generated by Ambit binding assay over a concentration range of the compound.More data for this Ligand-Target Pair
Affinity DataKd: >670nMAssay Description:Binding affinity to ERK5 by immobilized ligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKd: 1.10E+3nMAssay Description:Binding affinity to ERK5More data for this Ligand-Target Pair
Affinity DataKd: 1.10E+3nMAssay Description:Binding constant for ERK5 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 1.50E+3nMAssay Description:Binding affinity to ERK5 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKd: 1.60E+3nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
Affinity DataKd: 1.60E+3nMAssay Description:Binding constant for ERK5 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 1.60E+3nMAssay Description:Binding constant for ERK5 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 1.70E+3nMAssay Description:Binding constant for ERK5 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 2.30E+3nMAssay Description:Binding constant for ERK5 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 2.50E+3nMAssay Description:Binding constant for ERK5 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 2.70E+3nMAssay Description:Binding constant for ERK5 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 3.20E+3nMAssay Description:Binding constant for ERK5 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 5.32E+3nMAssay Description:Binding affinity to wild-type human partial length ERK5 (M1 to A409 residues) expressed in bacterial expression system measured after 1 hr by kinomes...More data for this Ligand-Target Pair
Affinity DataKd: 6.80E+3nMAssay Description:Binding constant for ERK5 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 9.90E+3nMAssay Description:Binding constant for ERK5 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for ERK5 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for ERK5 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for ERK5 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for ERK5 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for ERK5 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for ERK5 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for ERK5 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for ERK5 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for ERK5 kinase domainMore data for this Ligand-Target Pair