Compile Data Set for Download or QSAR
maximum 50k data
Found 26 of ki for UniProtKB: Q15139
TargetSerine/threonine-protein kinase D1(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50502745(CHEMBL4444206)
Affinity DataKi: <0.200nMAssay Description:Inhibition of full length GST-tagged human PRKD1 expressed in Baculovirus expression system using ATP as substrate incubated for 1 to 2 hrs by transc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase D1(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM159183(US9034866, 660)
Affinity DataKi: <0.200nMAssay Description:Inhibition of full length GST-tagged human PRKD1 expressed in Baculovirus expression system using ATP as substrate incubated for 1 to 2 hrs by transc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase D1(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM158743(US9034866, 218)
Affinity DataKi: <0.200nMAssay Description:Inhibition of full length GST-tagged human PRKD1 expressed in Baculovirus expression system using ATP as substrate incubated for 1 to 2 hrs by transc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase D1(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50502741(CHEMBL4517096)
Affinity DataKi: <0.200nMAssay Description:Inhibition of full length GST-tagged human PRKD1 expressed in Baculovirus expression system using ATP as substrate incubated for 1 to 2 hrs by transc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase D1(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50502746(CHEMBL3941082)
Affinity DataKi: <0.200nMAssay Description:Inhibition of full length GST-tagged human PRKD1 expressed in Baculovirus expression system using ATP as substrate incubated for 1 to 2 hrs by transc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase D1(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM158675(US9034866, 150)
Affinity DataKi:  0.900nMAssay Description:Inhibition of full length GST-tagged human PRKD1 expressed in Baculovirus expression system using ATP as substrate incubated for 1 to 2 hrs by transc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase D1(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50502744(CHEMBL4524153)
Affinity DataKi:  3.60nMAssay Description:Inhibition of full length GST-tagged human PRKD1 expressed in Baculovirus expression system using ATP as substrate incubated for 1 to 2 hrs by transc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase D1(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM159182(US9034866, 659)
Affinity DataKi:  4.20nMAssay Description:Inhibition of full length GST-tagged human PRKD1 expressed in Baculovirus expression system using ATP as substrate incubated for 1 to 2 hrs by transc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase D1(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM158533(US9034866, 8)
Affinity DataKi:  4.90nMAssay Description:Inhibition of full length GST-tagged human PRKD1 expressed in Baculovirus expression system using ATP as substrate incubated for 1 to 2 hrs by transc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase D1(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM158654(US9034866, 129)
Affinity DataKi:  5.90nMAssay Description:Inhibition of full length GST-tagged human PRKD1 expressed in Baculovirus expression system using ATP as substrate incubated for 1 to 2 hrs by transc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase D1(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM158645(US9034866, 120)
Affinity DataKi:  14nMAssay Description:Inhibition of full length GST-tagged human PRKD1 expressed in Baculovirus expression system using ATP as substrate incubated for 1 to 2 hrs by transc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase D1(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM158562(US9034866, 37)
Affinity DataKi:  25nMAssay Description:Inhibition of full length GST-tagged human PRKD1 expressed in Baculovirus expression system using ATP as substrate incubated for 1 to 2 hrs by transc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase D1(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50502743(CHEMBL4461552)
Affinity DataKi:  44nMAssay Description:Inhibition of full length GST-tagged human PRKD1 expressed in Baculovirus expression system using ATP as substrate incubated for 1 to 2 hrs by transc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase D1(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50502747(CHEMBL4546659)
Affinity DataKi:  62nMAssay Description:Inhibition of full length GST-tagged human PRKD1 expressed in Baculovirus expression system using ATP as substrate incubated for 1 to 2 hrs by transc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase D1(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50502742(CHEMBL3978002)
Affinity DataKi:  65nMAssay Description:Inhibition of full length GST-tagged human PRKD1 expressed in Baculovirus expression system using ATP as substrate incubated for 1 to 2 hrs by transc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha/beta/gamma/delta/epsilon/eta/theta type/Serine/threonine-protein kinase D1/D3(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50368315(PROSTRATIN)
Affinity DataKi:  190nMAssay Description:Displacement of [3H]PDBu binding to Protein kinase C of CEM cells with 10% fetal calf serumMore data for this Ligand-Target Pair
TargetProtein kinase C alpha/beta/gamma/delta/epsilon/eta/theta type/Serine/threonine-protein kinase D1/D3(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50281846((2R,3R)-2-Hydroxymethyl-5-oxo-4-tridec-(E)-ylidene...)
Affinity DataKi:  200nMAssay Description:Inhibition of [20-3H]phorbol-12,13-dibutyrate (PDBU) binding to protein kinase CMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C alpha/beta/gamma/delta/epsilon/eta/theta type/Serine/threonine-protein kinase D1/D3(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50281845((2R,3R)-2-Hydroxymethyl-5-oxo-4-tridec-(E)-ylidene...)
Affinity DataKi:  600nMAssay Description:Inhibition of [20-3H]phorbol-12,13-dibutyrate (PDBU) binding to protein kinase CMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C alpha/beta/gamma/delta/epsilon/eta/theta type/Serine/threonine-protein kinase D1/D3(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50041403((2R,3R,4R)-2-Hydroxymethyl-5-oxo-4-tetradecyl-tetr...)
Affinity DataKi:  600nMAssay Description:Inhibition of [20-3H]phorbol-12,13-dibutyrate (PDBU) binding to protein kinase CMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSerine/threonine-protein kinase D1(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50463483(CHEMBL4245242)
Affinity DataKi: >2.00E+3nMAssay Description:Inhibition of PRKD1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase D1(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50463479(CHEMBL4249925)
Affinity DataKi: >2.00E+3nMAssay Description:Inhibition of PRKD1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase D1(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50427363(CHEMBL2326002)
Affinity DataKi:  2.42E+3nMAssay Description:Inhibition of PKC mu (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50216682(1-(5-Isoquinolinesulfonyl)-2-methylpiperazine | 1-...)
Affinity DataKi:  6.00E+3nMAssay Description:Displacement of ATP from protein kinase C (PKC)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed