Compile Data Set for Download or QSAR
maximum 50k data
Found 423 of ic50 data for polymerid = 4762
TargetNeuropeptides B/W receptor type 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50362414(CHEMBL1940537)
Affinity DataIC50:  4.20nMAssay Description:Displacement of [125]-hNPW23 from human NPBWR1 expressed in CHO-K1 cells membrane by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptides B/W receptor type 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50362412(CHEMBL1940539)
Affinity DataIC50:  5.90nMAssay Description:Displacement of [125]-hNPW23 from human NPBWR1 expressed in CHO-K1 cells membrane by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptides B/W receptor type 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50362409(CHEMBL1940543)
Affinity DataIC50:  6nMAssay Description:Displacement of [125]-hNPW23 from human NPBWR1 expressed in CHO-K1 cells membrane by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptides B/W receptor type 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50362412(CHEMBL1940539)
Affinity DataIC50:  11nMAssay Description:Antagonist activity at human NPBWR1 expressed in CHO-K1 cells assessed as inhibition of hNPW23 and forskolin-stimulated cAMP production after 1 hr by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptides B/W receptor type 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50362410(CHEMBL1940542)
Affinity DataIC50:  18nMAssay Description:Displacement of [125]-hNPW23 from human NPBWR1 expressed in CHO-K1 cells membrane by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptides B/W receptor type 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50362415(CHEMBL1940536)
Affinity DataIC50:  21nMAssay Description:Displacement of [125]-hNPW23 from human NPBWR1 expressed in CHO-K1 cells membrane by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptides B/W receptor type 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50553728(CHEMBL4757321)
Affinity DataIC50:  30nMAssay Description:Negative allosteric modulation activity at NPBWR1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNeuropeptides B/W receptor type 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50553728(CHEMBL4757321)
Affinity DataIC50:  30nMAssay Description:Antagonist activity at human NPBWR1 assessed as inhibition of agonist-induced cAMP accumulation by cAMP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuropeptides B/W receptor type 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50362413(CHEMBL1940538)
Affinity DataIC50:  35nMAssay Description:Displacement of [125]-hNPW23 from human NPBWR1 expressed in CHO-K1 cells membrane by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptides B/W receptor type 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50362413(CHEMBL1940538)
Affinity DataIC50:  39nMAssay Description:Antagonist activity at human NPBWR1 expressed in CHO-K1 cells assessed as inhibition of hNPW23 and forskolin-stimulated cAMP production after 1 hr by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptides B/W receptor type 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50362414(CHEMBL1940537)
Affinity DataIC50:  40nMAssay Description:Antagonist activity at human NPBWR1 expressed in CHO-K1 cells assessed as inhibition of hNPW23 and forskolin-stimulated cAMP production after 1 hr by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptides B/W receptor type 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50553729(CHEMBL4796786)
Affinity DataIC50:  53nMAssay Description:Antagonist activity at human NPBWR1 assessed as inhibition of agonist-induced cAMP accumulation by cAMP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuropeptides B/W receptor type 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50362409(CHEMBL1940543)
Affinity DataIC50:  70nMAssay Description:Antagonist activity at human NPBWR1 expressed in CHO-K1 cells assessed as inhibition of hNPW23 and forskolin-stimulated cAMP production after 1 hr by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptides B/W receptor type 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50553730(CHEMBL4779758)
Affinity DataIC50:  70nMAssay Description:Antagonist activity at human NPBWR1 assessed as inhibition of agonist-induced cAMP accumulation by cAMP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuropeptides B/W receptor type 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50603458(CHEMBL5196275)
Affinity DataIC50:  71nMAssay Description:Antagonist activity at human NPBWR1 expressed in CHO-RD-HGA16 cells measured by calcium mobilization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNeuropeptides B/W receptor type 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50362411(CHEMBL1940541)
Affinity DataIC50:  95nMAssay Description:Displacement of [125]-hNPW23 from human NPBWR1 expressed in CHO-K1 cells membrane by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptides B/W receptor type 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50425599(CHEMBL2314291)
Affinity DataIC50:  100nMAssay Description:Antagonist activity against human NPBWR1 expressed in HEK293 cells co-expressing Gqi3 assessed as inhibition of agonist-induced response by FLIPR ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptides B/W receptor type 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50362415(CHEMBL1940536)
Affinity DataIC50:  110nMAssay Description:Antagonist activity at human NPBWR1 expressed in CHO-K1 cells assessed as inhibition of hNPW23 and forskolin-stimulated cAMP production after 1 hr by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptides B/W receptor type 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50603462(CHEMBL5198182)
Affinity DataIC50:  113nMAssay Description:Antagonist activity at human NPBWR1 expressed in CHO-RD-HGA16 cells measured by calcium mobilization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNeuropeptides B/W receptor type 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50425598(CHEMBL1972527)
Affinity DataIC50:  120nMAssay Description:Antagonist activity against human NPBWR1 expressed in HEK293 cells co-expressing Gqi3 assessed as inhibition of agonist-induced response by FLIPR ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptides B/W receptor type 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50425597(CHEMBL2314320)
Affinity DataIC50:  140nMAssay Description:Antagonist activity against human NPBWR1 expressed in HEK293 cells co-expressing Gqi3 assessed as inhibition of agonist-induced response by FLIPR ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptides B/W receptor type 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50401576(CHEMBL2207117)
Affinity DataIC50:  160nMAssay Description:Antagonist activity at human NPBWR1 expressed in HEK293T cells co-expressing Galphaqi3 assessed as calcium release after 15 mins by FLIPR assay assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptides B/W receptor type 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50362410(CHEMBL1940542)
Affinity DataIC50:  197nMAssay Description:Antagonist activity at human NPBWR1 expressed in CHO-K1 cells assessed as inhibition of hNPW23 and forskolin-stimulated cAMP production after 1 hr by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptides B/W receptor type 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50553719(CHEMBL4744579)
Affinity DataIC50:  205nMAssay Description:Antagonist activity at human NPBWR1 assessed as inhibition of agonist-induced cAMP accumulation by cAMP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuropeptides B/W receptor type 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50401572(CHEMBL2207121)
Affinity DataIC50:  210nMAssay Description:Antagonist activity at human NPBWR1 expressed in HEK293T cells co-expressing Galphaqi3 assessed as calcium release after 15 mins by FLIPR assay assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptides B/W receptor type 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50425595(CHEMBL2314323)
Affinity DataIC50:  220nMAssay Description:Antagonist activity against human NPBWR1 expressed in HEK293 cells co-expressing Gqi3 assessed as inhibition of agonist-induced response by FLIPR ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptides B/W receptor type 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50425596(CHEMBL1981304)
Affinity DataIC50:  220nMAssay Description:Antagonist activity against human NPBWR1 expressed in HEK293 cells co-expressing Gqi3 assessed as inhibition of agonist-induced response by FLIPR ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptides B/W receptor type 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50401577(CHEMBL2207531)
Affinity DataIC50:  230nMAssay Description:Antagonist activity at human NPBWR1 expressed in HEK293T cells co-expressing Galphaqi3 assessed as calcium release after 15 mins by FLIPR assay assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptides B/W receptor type 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50425594(CHEMBL1987422)
Affinity DataIC50:  240nMAssay Description:Antagonist activity against human NPBWR1 expressed in HEK293 cells co-expressing Gqi3 assessed as inhibition of agonist-induced response by FLIPR ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptides B/W receptor type 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50425593(CHEMBL2314301)
Affinity DataIC50:  240nMAssay Description:Antagonist activity against human NPBWR1 expressed in HEK293 cells co-expressing Gqi3 assessed as inhibition of agonist-induced response by FLIPR ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptides B/W receptor type 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50425591(CHEMBL2314300)
Affinity DataIC50:  250nMAssay Description:Antagonist activity against human NPBWR1 expressed in HEK293 cells co-expressing Gqi3 assessed as inhibition of agonist-induced response by FLIPR ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptides B/W receptor type 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50425592(CHEMBL2314293)
Affinity DataIC50:  250nMAssay Description:Antagonist activity against human NPBWR1 expressed in HEK293 cells co-expressing Gqi3 assessed as inhibition of agonist-induced response by FLIPR ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptides B/W receptor type 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50425590(CHEMBL1964671)
Affinity DataIC50:  260nMAssay Description:Antagonist activity against human NPBWR1 expressed in HEK293 cells co-expressing Gqi3 assessed as inhibition of agonist-induced response by FLIPR ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptides B/W receptor type 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM75901(5-chloranyl-2-(3,5-dimethylphenyl)-4-(4-methoxyphe...)
Affinity DataIC50:  270nMAssay Description:Antagonist activity at human NPBWR1 expressed in HEK293T cells co-expressing Galphaqi3 assessed as calcium release after 15 mins by FLIPR assay assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptides B/W receptor type 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM75938(5-chloranyl-4-(4-methoxyphenoxy)-2-(4-propan-2-ylp...)
Affinity DataIC50:  270nMAssay Description:Antagonist activity at human NPBWR1 expressed in HEK293T cells co-expressing Galphaqi3 assessed as calcium release after 15 mins by FLIPR assay assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptides B/W receptor type 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM75901(5-chloranyl-2-(3,5-dimethylphenyl)-4-(4-methoxyphe...)
Affinity DataIC50:  270nMAssay Description:Antagonist activity against human NPBWR1 expressed in HEK293 cells co-expressing Gqi3 assessed as inhibition of agonist-induced response by FLIPR ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptides B/W receptor type 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM75938(5-chloranyl-4-(4-methoxyphenoxy)-2-(4-propan-2-ylp...)
Affinity DataIC50:  270nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Affiliation: The Scripps Research Institute, TSRI Assa...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetNeuropeptides B/W receptor type 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM75901(5-chloranyl-2-(3,5-dimethylphenyl)-4-(4-methoxyphe...)
Affinity DataIC50:  272nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Affiliation: The Scripps Research Institute, TSRI Assa...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetNeuropeptides B/W receptor type 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50425589(CHEMBL1969065)
Affinity DataIC50:  280nMAssay Description:Antagonist activity against human NPBWR1 expressed in HEK293 cells co-expressing Gqi3 assessed as inhibition of agonist-induced response by FLIPR ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptides B/W receptor type 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM75900(5-chloranyl-4-(4-methoxyphenoxy)-2-(3-propan-2-ylp...)
Affinity DataIC50:  280nMAssay Description:Antagonist activity at human NPBWR1 expressed in HEK293T cells co-expressing Galphaqi3 assessed as calcium release after 15 mins by FLIPR assay assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptides B/W receptor type 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM75900(5-chloranyl-4-(4-methoxyphenoxy)-2-(3-propan-2-ylp...)
Affinity DataIC50:  280nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Affiliation: The Scripps Research Institute, TSRI Assa...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetNeuropeptides B/W receptor type 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM75901(5-chloranyl-2-(3,5-dimethylphenyl)-4-(4-methoxyphe...)
Affinity DataIC50:  281nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Affiliation: The Scripps Research Institute, TSRI Assa...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetNeuropeptides B/W receptor type 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50553720(CHEMBL4754194)
Affinity DataIC50:  282nMAssay Description:Antagonist activity at human NPBWR1 assessed as inhibition of agonist-induced cAMP accumulation by cAMP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuropeptides B/W receptor type 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM75946(2-[3,5-bis(chloranyl)phenyl]-5-chloranyl-4-(4-meth...)
Affinity DataIC50:  287nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Affiliation: The Scripps Research Institute, TSRI Assa...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetNeuropeptides B/W receptor type 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50425588(CHEMBL1965488)
Affinity DataIC50:  290nMAssay Description:Antagonist activity against human NPBWR1 expressed in HEK293 cells co-expressing Gqi3 assessed as inhibition of agonist-induced response by FLIPR ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptides B/W receptor type 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM75918(5-chloranyl-4-(4-methoxyphenoxy)-2-(3-methyl-4-pro...)
Affinity DataIC50:  299nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Affiliation: The Scripps Research Institute, TSRI Assa...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetNeuropeptides B/W receptor type 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM75918(5-chloranyl-4-(4-methoxyphenoxy)-2-(3-methyl-4-pro...)
Affinity DataIC50:  300nMAssay Description:Antagonist activity at human NPBWR1 expressed in HEK293T cells co-expressing Galphaqi3 assessed as calcium release after 15 mins by FLIPR assay assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptides B/W receptor type 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50425587(CHEMBL2314318)
Affinity DataIC50:  320nMAssay Description:Antagonist activity against human NPBWR1 expressed in HEK293 cells co-expressing Gqi3 assessed as inhibition of agonist-induced response by FLIPR ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptides B/W receptor type 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50362416(CHEMBL1940354)
Affinity DataIC50:  324nMAssay Description:Displacement of [125]-hNPW23 from human NPBWR1 expressed in CHO-K1 cells membrane by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptides B/W receptor type 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50362411(CHEMBL1940541)
Affinity DataIC50:  342nMAssay Description:Antagonist activity at human NPBWR1 expressed in CHO-K1 cells assessed as inhibition of hNPW23 and forskolin-stimulated cAMP production after 1 hr by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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