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Found 29 of ec50 for UniProtKB: P10980
TargetMuscarinic acetylcholine receptor M2(RAT)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50423968(CHEMBL2313377)
Affinity DataEC50:  640nMAssay Description:Positive allosteric modulation of rat muscarinic M2 receptor assessed as acetylcholine responseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50258723(7-chloro-1-(4-(trifluoromethyl)benzyl)indoline-2,3...)
Affinity DataEC50:  2.80E+3nMAssay Description:Agonist activity at rat muscarinic M2 expressed in CHO cells assessed as stimulation of calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50258723(7-chloro-1-(4-(trifluoromethyl)benzyl)indoline-2,3...)
Affinity DataEC50:  2.84E+3nMAssay Description:Activation of rat muscarinic M2 receptor expressed in CHO cells coexpressing chimeric Gqi5 protein assessed as potentiation of acetylcholine-induced ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50356972(CHEMBL1916234)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at rat muscarinic M2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50356969(CHEMBL1916226)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at rat muscarinic M2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50356970(CHEMBL1916227)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at rat muscarinic M2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50356968(CHEMBL1916225)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at rat muscarinic M2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50356978(CHEMBL1916233)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at rat muscarinic M2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50356977(CHEMBL1916232)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at rat muscarinic M2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50356976(CHEMBL1916231)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at rat muscarinic M2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50356975(CHEMBL1916230)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at rat muscarinic M2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50356974(CHEMBL1916229)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at rat muscarinic M2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50356973(CHEMBL1916235)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at rat muscarinic M2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50356971(CHEMBL1916228)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at rat muscarinic M2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50207517(CHEMBL3915634)
Affinity DataEC50: >3.00E+4nMAssay Description:Binding affinity to rat M2 receptor by radio-ligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50207516(CHEMBL3942511)
Affinity DataEC50: >3.00E+4nMAssay Description:Binding affinity to rat M2 receptor by radio-ligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50207463(CHEMBL3963788)
Affinity DataEC50: >3.00E+4nMAssay Description:Binding affinity to rat M2 receptor by radio-ligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM43821(4-(2-benzamidoethylamino)-1-piperidinecarboxylic a...)
Affinity DataEC50: >3.00E+4nMAssay Description:Partial agonist activity at rat muscarinic M2 receptor expressed in CHO cells calcium responseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50356969(CHEMBL1916226)
Affinity DataEC50: >3.00E+4nMAssay Description:Partial agonist activity at rat muscarinic M2 receptor expressed in CHO cells calcium responseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50423967(CHEMBL2057417)
Affinity DataEC50: >3.00E+4nMAssay Description:Positive allosteric modulation of rat muscarinic M2 receptor assessed as acetylcholine responseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50356966(CHEMBL1916224)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at rat muscarinic M2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM43822(4-[2-(o-toluoylamino)ethylamino]piperidine-1-carbo...)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at rat muscarinic M2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50356966(CHEMBL1916224)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at rat recombinant muscarinic M2 receptor by HTS cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM43822(4-[2-(o-toluoylamino)ethylamino]piperidine-1-carbo...)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at rat recombinant muscarinic M2 receptor by HTS cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50258656(1-(4-methoxybenzyl)-5-(trifluoromethoxy)indoline-2...)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at rat muscarinic M2 expressed in CHO cells assessed as stimulation of calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50258439(1-(4-bromobenzyl)indoline-2,3-dione | CHEMBL523685...)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at rat muscarinic M2 expressed in CHO cells assessed as stimulation of calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50249403(CHEMBL4091821)
Affinity DataEC50: >3.00E+4nMAssay Description:Activity at rat M2 receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50263887(1-(1'-(2-methylbenzyl)-1,4'-bipiperidin-4-yl)-1H-b...)
Affinity DataEC50: >3.00E+4nMAssay Description:Partial agonist activity at rat muscarinic M2 receptor expressed in CHO cells calcium responseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50023229(CHEMBL3329755)
Affinity DataEC50: >3.00E+4nMAssay Description:Activity at rat muscarinic acetylcholine receptor subtype 2 expressed in CHO cells co-transfected with chimeric Gqi5 by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed