Compile Data Set for Download or QSAR
maximum 50k data
Found 142 of ic50 data for polymerid = 49000597,49000598
TargetGalanin receptor type 2(Homo sapiens (Human))
Phenex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM392076(US10301272, Example 7/9)
Affinity DataIC50:  0.190nMAssay Description:Displacement of [125I]-endothelin-1 from human recombinant GAL2 receptor after 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGalanin receptor type 2(Homo sapiens (Human))
Phenex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50378616(GALANIN)
Affinity DataIC50:  0.800nMAssay Description:Binding affinity to human GAL2 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 2(Homo sapiens (Human))
Phenex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50378616(GALANIN)
Affinity DataIC50:  2.60nMAssay Description:Binding affinity to human GAL2 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 2(Homo sapiens (Human))
Phenex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50208989(CHEMBL506553)
Affinity DataIC50:  2.60nMAssay Description:Displacement of [125I]galanin from human recombinant GAL2 receptor expressed in CHO cells measured after 120 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 2(RAT)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50256745((2S)-2-amino-3-((2-(benzyloxy)phenyl)(3-fluorophen...)
Affinity DataIC50:  21.1nMAssay Description:Inhibition of [3H]glycine uptake at rat glycine transporter 2 expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 2(RAT)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50256746((3S,6S,9S,15aR)-9-sec-butyl-6-((1-methoxy-1H-indol...)
Affinity DataIC50:  87.7nMAssay Description:Inhibition of [3H]glycine uptake at rat glycine transporter 2 expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 2(RAT)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50256706((3S,6S,9S,12S)-3-benzyl-6,9,12-tri-sec-butyl-1,4,7...)
Affinity DataIC50:  226nMAssay Description:Inhibition of [3H]glycine uptake at rat glycine transporter 2 expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 2(RAT)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50256665((3S,6S,9S,12S)-3-benzyl-9,12-di-sec-butyl-6-((2S,3...)
Affinity DataIC50:  278nMAssay Description:Inhibition of [3H]glycine uptake at rat glycine transporter 2 expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 2(Homo sapiens (Human))
Phenex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50358677(CHEMBL1922007)
Affinity DataIC50:  330nMAssay Description:Displacement of [125I]galanin from GalR2 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 2(Homo sapiens (Human))
Phenex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50358683(CHEMBL1922013)
Affinity DataIC50:  380nMAssay Description:Displacement of [125I]galanin from GalR2 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 2(Homo sapiens (Human))
Phenex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50358676(CHEMBL1922006)
Affinity DataIC50:  380nMAssay Description:Displacement of [125I]galanin from GalR2 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 2(Homo sapiens (Human))
Phenex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50358680(CHEMBL1922010)
Affinity DataIC50:  430nMAssay Description:Displacement of [125I]galanin from GalR2 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 2(Homo sapiens (Human))
Phenex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50358675(CHEMBL1922005)
Affinity DataIC50:  440nMAssay Description:Displacement of [125I]galanin from GalR2 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 2(RAT)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50256704((3S,6S,9S,12S)-3-benzyl-9-sec-butyl-6-((2S,3R)-3-h...)
Affinity DataIC50:  450nMAssay Description:Inhibition of [3H]glycine uptake at rat glycine transporter 2 expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 2(Homo sapiens (Human))
Phenex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50358679(CHEMBL1922009)
Affinity DataIC50:  540nMAssay Description:Displacement of [125I]galanin from GalR2 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 2(RAT)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50256705((3S,6S,9S,12S)-3-benzyl-6-((2S,3R)-3-hydroxybutan-...)
Affinity DataIC50:  542nMAssay Description:Inhibition of [3H]glycine uptake at rat glycine transporter 2 expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 2(Homo sapiens (Human))
Phenex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50358658(CHEMBL1921999)
Affinity DataIC50:  550nMAssay Description:Displacement of [125I]galanin from GalR2 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 2(Homo sapiens (Human))
Phenex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50358662(CHEMBL1922003)
Affinity DataIC50:  560nMAssay Description:Displacement of [125I]galanin from GalR2 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 2(RAT)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50256666((3S,6S,9S,12S)-3-benzyl-12-sec-butyl-6-((2S,3R)-3-...)
Affinity DataIC50:  574nMAssay Description:Inhibition of [3H]glycine uptake at rat glycine transporter 2 expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 2(Homo sapiens (Human))
Phenex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50358667(CHEMBL1922016)
Affinity DataIC50:  770nMAssay Description:Displacement of [125I]galanin from GalR2 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 2(Homo sapiens (Human))
Phenex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50358655(CHEMBL1921996)
Affinity DataIC50:  770nMAssay Description:Displacement of [125I]galanin from GalR2 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 2(Homo sapiens (Human))
Phenex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50358678(CHEMBL1922008)
Affinity DataIC50:  780nMAssay Description:Displacement of [125I]galanin from GalR2 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 2(Homo sapiens (Human))
Phenex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50358653(CHEMBL1921993)
Affinity DataIC50:  930nMAssay Description:Displacement of [125I]galanin from GalR2 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 2(Homo sapiens (Human))
Phenex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50358682(CHEMBL1922012)
Affinity DataIC50:  980nMAssay Description:Displacement of [125I]galanin from GalR2 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 2(Homo sapiens (Human))
Phenex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50358656(CHEMBL1921997)
Affinity DataIC50:  1.06E+3nMAssay Description:Displacement of [125I]galanin from GalR2 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 2(Homo sapiens (Human))
Phenex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50358648(CHEMBL1921902)
Affinity DataIC50:  1.09E+3nMAssay Description:Displacement of [125I]galanin from GalR2 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 2(Homo sapiens (Human))
Phenex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50358674(CHEMBL1922004)
Affinity DataIC50:  1.18E+3nMAssay Description:Displacement of [125I]galanin from GalR2 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 2(Homo sapiens (Human))
Phenex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM42052(2-N,3-N-dimethyl-6,7-dinitroquinoxaline-2,3-diamin...)
Affinity DataIC50:  1.29E+3nMAssay Description:Source (MLSCN Center Name): The Scripps Research Institute Molecular Screening Center Affiliation: The Scripps Florida Research Institute, TSRI Assay...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PCBioAssay
TargetGalanin receptor type 2(Homo sapiens (Human))
Phenex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50358668(CHEMBL1922019)
Affinity DataIC50:  1.34E+3nMAssay Description:Displacement of [125I]galanin from GalR2 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 2(Homo sapiens (Human))
Phenex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50358657(CHEMBL1921998)
Affinity DataIC50:  1.75E+3nMAssay Description:Displacement of [125I]galanin from GalR2 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 2(Homo sapiens (Human))
Phenex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50358659(CHEMBL1922000)
Affinity DataIC50:  1.92E+3nMAssay Description:Displacement of [125I]galanin from GalR2 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 2(Homo sapiens (Human))
Phenex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50358681(CHEMBL1922011)
Affinity DataIC50:  1.93E+3nMAssay Description:Displacement of [125I]galanin from GalR2 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 2(Homo sapiens (Human))
Phenex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50358661(CHEMBL1922002)
Affinity DataIC50:  2.03E+3nMAssay Description:Displacement of [125I]galanin from GalR2 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 2(Homo sapiens (Human))
Phenex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50358660(CHEMBL1922001)
Affinity DataIC50:  2.08E+3nMAssay Description:Displacement of [125I]galanin from GalR2 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 2(RAT)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50256664((S)-2-((2S,5S,8S,11S)-5-benzyl-8,11-di-sec-butyl-3...)
Affinity DataIC50:  2.26E+3nMAssay Description:Inhibition of [3H]glycine uptake at rat glycine transporter 2 expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 2(Homo sapiens (Human))
Phenex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50358685(CHEMBL1922017)
Affinity DataIC50:  2.85E+3nMAssay Description:Displacement of [125I]galanin from GalR2 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 2(Homo sapiens (Human))
Phenex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50358664(CHEMBL1921988)
Affinity DataIC50:  3.38E+3nMAssay Description:Displacement of [125I]galanin from GalR2 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 2(Homo sapiens (Human))
Phenex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50358652(CHEMBL1921992)
Affinity DataIC50:  3.40E+3nMAssay Description:Displacement of [125I]galanin from GalR2 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 2(Homo sapiens (Human))
Phenex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50358665(CHEMBL1921990)
Affinity DataIC50:  3.69E+3nMAssay Description:Displacement of [125I]galanin from GalR2 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 2(Homo sapiens (Human))
Phenex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50358650(CHEMBL1921989)
Affinity DataIC50:  4.15E+3nMAssay Description:Displacement of [125I]galanin from GalR2 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 2(Homo sapiens (Human))
Phenex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50358684(CHEMBL1922014)
Affinity DataIC50:  4.18E+3nMAssay Description:Displacement of [125I]galanin from GalR2 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 2(Homo sapiens (Human))
Phenex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50358663(CHEMBL1921901)
Affinity DataIC50:  4.57E+3nMAssay Description:Displacement of [125I]galanin from GalR2 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 2(Homo sapiens (Human))
Phenex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50007082((E)-2-methoxy-4-(2-nitrovinyl)phenol | 2-Methoxy-4...)
Affinity DataIC50: >4.60E+3nMAssay Description:Source (MLSCN Center Name): The Scripps Research Institute Molecular Screening Center Affiliation: The Scripps Florida Research Institute, TSRI Assay...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetGalanin receptor type 2(Homo sapiens (Human))
Phenex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM42060(4,5-bis(chloranyl)-2-[2-(4-naphthalen-2-ylsulfonyl...)
Affinity DataIC50:  5.37E+3nMAssay Description:Source (MLSCN Center Name): The Scripps Research Institute Molecular Screening Center Affiliation: The Scripps Florida Research Institute, TSRI Assay...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetGalanin receptor type 2(Homo sapiens (Human))
Phenex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50358649(CHEMBL1921903)
Affinity DataIC50:  6.62E+3nMAssay Description:Displacement of [125I]galanin from GalR2 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 2(Homo sapiens (Human))
Phenex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM42053(MLS000573994 | N-[4-[[(E)-3-(4-chlorophenyl)acrylo...)
Affinity DataIC50:  6.77E+3nMAssay Description:Source (MLSCN Center Name): The Scripps Research Institute Molecular Screening Center Affiliation: The Scripps Florida Research Institute, TSRI Assay...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetGalanin receptor type 2(Homo sapiens (Human))
Phenex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM42069(2-acetamido-4,5-dinitro-benzoic acid ethyl ester |...)
Affinity DataIC50:  7.53E+3nMAssay Description:Source (MLSCN Center Name): The Scripps Research Institute Molecular Screening Center Affiliation: The Scripps Research Institute (TSRI) Assay Provid...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PCBioAssay
TargetGalanin receptor type 2(Homo sapiens (Human))
Phenex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM42061(2-(4,5-dichloro-6-keto-pyridazin-1-yl)-N-[2-(2-eth...)
Affinity DataIC50:  7.62E+3nMAssay Description:Source (MLSCN Center Name): The Scripps Research Institute Molecular Screening Center Affiliation: The Scripps Florida Research Institute, TSRI Assay...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetGalanin receptor type 2(Homo sapiens (Human))
Phenex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50358666(CHEMBL1921994)
Affinity DataIC50:  8.04E+3nMAssay Description:Displacement of [125I]galanin from GalR2 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 2(Homo sapiens (Human))
Phenex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50358651(CHEMBL1921991)
Affinity DataIC50:  8.65E+3nMAssay Description:Displacement of [125I]galanin from GalR2 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 142 total ) | Next | Last >>
Jump to: