Affinity DataEC50: 258nMAssay Description:Agonist activity at recombinant GluA1 receptor flip isoform expressed in Xenopus oocytesMore data for this Ligand-Target Pair
Affinity DataEC50: 260nMAssay Description:Agonist activity at recombinant GluA1 receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
Affinity DataEC50: 270nMAssay Description:Agonist activity at recombinant GluA1 receptor flop isoform expressed in Xenopus oocytesMore data for this Ligand-Target Pair
Affinity DataEC50: 380nMAssay Description:Agonist activity at recombinant GluA1 receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
Affinity DataEC50: 382nMAssay Description:Agonist activity at recombinant GluA1 receptor flip isoform expressed in Xenopus oocytesMore data for this Ligand-Target Pair
Affinity DataEC50: 660nMAssay Description:Inhibition of GluR1 expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 910nMAssay Description:Inhibition of GluR1 expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 1.00E+3nMAssay Description:Agonist activity at recombinant GluA1 receptor flip isoform expressed in Xenopus oocytesMore data for this Ligand-Target Pair
Affinity DataEC50: 2.00E+3nMAssay Description:Activity at recombinant GluA1 receptor flip isoform expressed in Xenopus oocytes co-expressing gamma2-TARP assessed as effect on 10 uM glutamate-indu...More data for this Ligand-Target Pair
Affinity DataEC50: 2.26E+3nMAssay Description:Agonist activity at recombinant GluA1 receptor flip isoform expressed in Xenopus oocytes co-expressing gamma2-TARPMore data for this Ligand-Target Pair
Affinity DataEC50: 2.88E+3nMAssay Description:Inhibition of GluR1 expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 4.10E+3nMAssay Description:Agonist activity at GluA1 receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 4.10E+3nMAssay Description:Agonist activity at cyclothiazide-desensitized human flip iGluR1 expressed in CHO-K1 cells by whole cell patch-clamp methodMore data for this Ligand-Target Pair
Affinity DataEC50: 4.50E+3nMAssay Description:Electrophysiological data on Xenopus oocytes, expressing homomeric Ionotropic glutamate receptor AMPA 1 (GluR1o)More data for this Ligand-Target Pair
Affinity DataEC50: 4.70E+3nMAssay Description:Agonist activity at recombinant GluA1 receptor flip isoform expressed in Xenopus oocytesMore data for this Ligand-Target Pair
Affinity DataEC50: 5.20E+3nMAssay Description:Electrophysiological data on Xenopus oocytes, expressing homomeric Ionotropic glutamate receptor AMPA 1 (GluR1o)More data for this Ligand-Target Pair
Affinity DataEC50: 5.20E+3nMAssay Description:Agonist activity at GluA1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 5.65E+3nMAssay Description:Activity at human recombinant GluA1 receptor flip isoform expressed in HEK293 cells assessed as effect on glutamate-induced calcium flux by Fluo-4/AM...More data for this Ligand-Target Pair
Affinity DataEC50: 5.65E+3nMAssay Description:Inhibition of GluR1 expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 7.51E+3nMAssay Description:Agonist activity at recombinant GluA1 receptor flip isoform expressed in Xenopus oocytes co-expressing gamma2-TARPMore data for this Ligand-Target Pair
Affinity DataEC50: 1.00E+4nMAssay Description:Activity at recombinant GluA1 receptor flop isoform expressed in Xenopus oocytes co-expressing gamma2-TARP assessed as effect on 10 uM glutamate-indu...More data for this Ligand-Target Pair
Affinity DataEC50: 1.40E+4nMAssay Description:Agonist activity at recombinant GluA1 receptor flop isoform expressed in Xenopus oocytesMore data for this Ligand-Target Pair
Affinity DataEC50: 1.40E+4nMAssay Description:Agonist activity at recombinant GluA1 receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
Affinity DataEC50: 1.85E+4nMAssay Description:Agonist activity at cyclothiazide-desensitized human flip iGluR1 expressed in CHO-K1 cells by whole cell patch-clamp methodMore data for this Ligand-Target Pair
Affinity DataEC50: 1.98E+4nMAssay Description:Activity at human recombinant GluA1 receptor flip isoform expressed in HEK293 cells assessed as effect on glutamate-induced calcium flux by Fluo-4/AM...More data for this Ligand-Target Pair
Affinity DataEC50: 2.10E+4nMAssay Description:Inhibition of GluR1 expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 2.20E+4nMAssay Description:Agonist activity at recombinant GluA1 receptor flop isoform expressed in Xenopus oocytesMore data for this Ligand-Target Pair
Affinity DataEC50: 2.20E+4nMAssay Description:Electrophysiological data on Xenopus oocytes, expressing homomeric Ionotropic glutamate receptor AMPA 1 (GluR1o)More data for this Ligand-Target Pair
Affinity DataEC50: 2.80E+4nMAssay Description:Activity at recombinant GluA1 receptor flip isoform expressed in Xenopus oocytes co-expressing gamma2-TARP assessed as effect on glutamate/trichlorom...More data for this Ligand-Target Pair
Affinity DataEC50: 3.30E+4nMAssay Description:Agonist activity at GluA1 receptor (unknown origin) expressed in HEK293 cells assessed induction of S-glutamate-induced calcium flux measured after 9...More data for this Ligand-Target Pair
Affinity DataEC50: 3.31E+4nMAssay Description:Agonist activity at GluA1 receptor (unknown origin) expressed in HEK293 cells assessed induction of S-glutamate-induced calcium flux measured after 9...More data for this Ligand-Target Pair
Affinity DataEC50: 4.20E+4nMAssay Description:Agonist activity at GluR1 expressed in HEK293 cells by Fluo-4/Ca2+ assayMore data for this Ligand-Target Pair
Affinity DataEC50: 6.00E+4nMAssay Description:Agonist activity at recombinant GluA1 receptor flop isoform expressed in Xenopus oocytesMore data for this Ligand-Target Pair
Affinity DataEC50: 7.10E+4nMAssay Description:Agonist activity at GluR1 expressed in HEK293 cells by Fluo-4/Ca2+ assayMore data for this Ligand-Target Pair
Affinity DataEC50: 7.30E+4nMAssay Description:Agonist activity at recombinant GluA1 receptor flip isoform expressed in Xenopus oocytesMore data for this Ligand-Target Pair
Affinity DataEC50: >3.00E+5nMAssay Description:Agonist activity at GluA1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 4.80E+5nMAssay Description:Agonist activity at GluR1 expressed in HEK293 cells by Fluo-4/Ca2+ assayMore data for this Ligand-Target Pair
Affinity DataEC50: 5.50E+5nMAssay Description:Agonist activity at GluR1 expressed in HEK293 cells by Fluo-4/Ca2+ assayMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at GluA1 receptor (unknown origin) expressed in HEK293 cells assessed induction of S-glutamate-induced calcium flux measured after 9...More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at GluA1 receptor (unknown origin) expressed in HEK293 cells assessed induction of S-glutamate-induced calcium flux measured after 9...More data for this Ligand-Target Pair
Affinity DataEC50: >3.00E+6nMAssay Description:Agonist activity at GluR1 expressed in HEK293 cells by Fluo-4/Ca2+ assayMore data for this Ligand-Target Pair
Affinity DataEC50: 3.00E+6nMAssay Description:Agonist activity at GluR1 expressed in HEK293 cells by Fluo-4/Ca2+ assayMore data for this Ligand-Target Pair