Affinity DataKi: 0.100nMAssay Description:Binding affinity by displacement of radiolabeled GR-100679 from Tachykinin receptor 2 from homogenized rat colonMore data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Inhibition of [125I]-NKA binding to neurokinin NK2 receptor from rat duodenum membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Inhibition of [125I]-NKA binding to neurokinin NK2 receptor from rat duodenum membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Inhibition of [125I]-NKA binding to neurokinin NK2 receptor from rat duodenum membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Binding affinity against bovine Tachykinin receptor 2More data for this Ligand-Target Pair
Affinity DataKi: 0.510nMAssay Description:Ability to displace [125I]NKA from Tachykinin receptor 2 in rat deodenum membraneMore data for this Ligand-Target Pair
Affinity DataKi: 0.900nMAssay Description:Inhibition of [125I]-NKA binding to neurokinin NK2 receptor from rat duodenum membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Binding affinity against bovine Tachykinin receptor 2More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Inhibition of [125I]-NKA binding to neurokinin NK2 receptor from rat duodenum membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Inhibition of [125I]-NKA binding to neurokinin NK2 receptor from rat duodenum membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:The compound was evaluated for the inhibition of [125I]-NKA binding to neurokinin NK2 receptor from hamster urinary bladder membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Inhibition of [125I]-NKA binding to neurokinin NK2 receptor from rat duodenum membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Inhibition of [125I]-NKA binding to neurokinin NK2 receptor from rat duodenum membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
Affinity DataKi: 3.98nMAssay Description:Binding affinity by displacement of radiolabeled GR-100679 from Tachykinin receptor 2 from homogenized rat colonMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Binding affinity by displacement of radiolabeled GR-100679 from Tachykinin receptor 2 from homogenized rat colonMore data for this Ligand-Target Pair
Affinity DataKi: 4.5nMAssay Description:Displacement of [3H]substance P frome rat NK2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
Affinity DataKi: 6.30nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
Affinity DataKi: 6.30nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
Affinity DataKi: 7.30nMAssay Description:Displacement of [3H]substance P frome rat NK2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 7.90nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
Affinity DataKi: 7.90nMAssay Description:Binding affinity by displacement of radiolabeled GR-100679 from Tachykinin receptor 2 from homogenized rat colonMore data for this Ligand-Target Pair
Affinity DataKi: 7.94nMAssay Description:Binding affinity by displacement of radiolabeled GR-100679 from Tachykinin receptor 2 from homogenized rat colonMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Displacement of [3H]substance P frome rat NK2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Inhibition constant for displacement of [3H]-NKA from Tachykinin receptor 2 found in hamster urinary bladder membrane (HUBM)More data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair