Compile Data Set for Download or QSAR
maximum 50k data
Found 8 of ec50 for UniProtKB: O95665
TargetNeurotensin receptor type 2(Homo sapiens (Human))
Medical University Of South Carolina Campus

Curated by ChEMBL
LigandPNGBDBM50322368((S)-5-((S)-1-((S)-2-((S)-1-((S)-1-((S)-1-carboxy-3...)
Affinity DataEC50:  54nMAssay Description:Binding affinity to human NTR2 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 2(Homo sapiens (Human))
Medical University Of South Carolina Campus

Curated by ChEMBL
LigandPNGBDBM50130880(CHEMBL407196 | NT(1-13) | neurotensin | pGlu-Leu-T...)
Affinity DataEC50:  110nMAssay Description:Agonist activity at human NTS2 receptor expressed in HEK293 cells assessed as inhibition of constitutive activity on MAPK-mediated luciferase activit...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 2(Homo sapiens (Human))
Medical University Of South Carolina Campus

Curated by ChEMBL
LigandPNGBDBM50342251((S)-2-((2S,3S)-2-(2-((S)-1-((S)-2-((S)-2-amino-5-g...)
Affinity DataEC50:  480nMAssay Description:Agonist activity at human NTS2 receptor expressed in HEK293 cells assessed as inhibition of constitutive activity on MAPK-mediated luciferase activit...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 2(Homo sapiens (Human))
Medical University Of South Carolina Campus

Curated by ChEMBL
LigandPNGBDBM50342244((S)-2-((2S,3S)-2-(2-((S)-1-((S)-6-amino-2-((S)-2,6...)
Affinity DataEC50:  590nMAssay Description:Agonist activity at human NTS2 receptor expressed in HEK293 cells assessed as inhibition of constitutive activity on MAPK-mediated luciferase activit...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 2(Homo sapiens (Human))
Medical University Of South Carolina Campus

Curated by ChEMBL
LigandPNGBDBM50342245((S)-2-((2S,3S)-2-(2-((S)-1-((S)-2-((S)-2,6-diamino...)
Affinity DataEC50:  690nMAssay Description:Agonist activity at human NTS2 receptor expressed in HEK293 cells assessed as inhibition of constitutive activity on MAPK-mediated luciferase activit...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 2(Homo sapiens (Human))
Medical University Of South Carolina Campus

Curated by ChEMBL
LigandPNGBDBM50342248((S)-2-((2S,3S)-2-(2-((S)-1-((S)-6-amino-2-((S)-2-a...)
Affinity DataEC50:  840nMAssay Description:Agonist activity at human NTS2 receptor expressed in HEK293 cells assessed as inhibition of constitutive activity on MAPK-mediated luciferase activit...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 2(Homo sapiens (Human))
Medical University Of South Carolina Campus

Curated by ChEMBL
LigandPNGBDBM50444943(CHEMBL3099773)
Affinity DataEC50: >8.00E+4nMAssay Description:Agonist activity at NTR2 in human U2OS cells after 1 hr by beta-arrestin GFP reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 2(Homo sapiens (Human))
Medical University Of South Carolina Campus

Curated by ChEMBL
LigandPNGBDBM50248035((2S)-2-(1-(7-chloroquinolin-4-yl)-5-(2,6-dimethoxy...)
Affinity DataEC50: >8.00E+4nMAssay Description:Agonist activity at NTR2 in human U2OS cells after 1 hr by beta-arrestin GFP reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed