Compile Data Set for Download or QSAR
maximum 50k data
Found 87 of ec50 data for polymerid = 50001092
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50332462(2-(2-methyl-4-((4-methyl-2-(4-(trifluoromethyl)phe...)
Affinity DataEC50:  2.30nMAssay Description:Agonist activity at mouse PPAR-delta expressed in african green monkey CV-1 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50312479(2-(4-((4-(6-Morpholinopyridin-3-yl)-5-(4-(trifluor...)
Affinity DataEC50:  5nMAssay Description:Agonist activity at mouse PPARdelta by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50312476(CHEMBL1080699 | {4-[4-(6-Isopropoxypyridin-3-yl)-5...)
Affinity DataEC50:  7nMAssay Description:Agonist activity at mouse PPARdelta by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50539514(CHEMBL4649683)
Affinity DataEC50:  7.90nMAssay Description:Modulator activity at mouse PPARdeltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50312421(2-(4-((4-(4-Isopropoxyphenyl)-5-(4-(trifluorometho...)
Affinity DataEC50:  9nMAssay Description:Agonist activity at mouse PPARdelta by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50312422(2-(4-((4-(4-(Cyclopentyloxy)phenyl)-5-(4-(trifluor...)
Affinity DataEC50:  9nMAssay Description:Agonist activity at mouse PPARdelta by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50312478(2-(4-((4-(2-Isopropoxypyrimidin-5-yl)-5-(4-(triflu...)
Affinity DataEC50:  10nMAssay Description:Agonist activity at mouse PPARdelta by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50312475(2-(4-((4-(6-Isopropoxypyridin-3-yl)-5-(4-(trifluor...)
Affinity DataEC50:  13nMAssay Description:Agonist activity at mouse PPARdelta by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50312469(2-(4-((4-(4-Isopropoxyphenyl)-5-(4-propylphenyl)th...)
Affinity DataEC50:  17nMAssay Description:Agonist activity at mouse PPARdelta by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50106105(2-[3-(3-{(2,4-Bis-trifluoromethyl-benzyl)-[2-(4-tr...)
Affinity DataEC50:  19nMAssay Description:Agonist activity against PPAR deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50584465(CHEMBL5084377)
Affinity DataEC50:  20nMAssay Description:Agonist activity at mouse PPARdelta in Cos7 cells transfected with pBIND and pGL4.35 Gal4 UAS Luc reporter plasmid by measuring luciferase activity i...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM28661(2-{2-methyl-4-[({4-methyl-2-[4-(trifluoromethyl)ph...)
Affinity DataEC50:  20nMAssay Description:Activity against murine PPAR delta receptorMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50312467(2-(4-((5-(4-(Trifluoromethyl)phenyl)-4-(4-isopropo...)
Affinity DataEC50:  20nMAssay Description:Agonist activity at mouse PPARdelta by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50085040(CHEMBL278994 | L-796449 | {3-Chloro-4-[3-(3-phenyl...)
Affinity DataEC50:  23nMAssay Description:Agonist activity for murine PPAR delta receptor in transcriptional activation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50312424(CHEMBL1080349 | {4-[4-(4-Isopropoxyphenyl)-5-(4-tr...)
Affinity DataEC50:  26nMAssay Description:Agonist activity at mouse PPARdelta by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50312470(2-(4-((4-(4-Isopropoxyphenyl)-5-(4-biphenyl)thiazo...)
Affinity DataEC50:  29nMAssay Description:Agonist activity at mouse PPARdelta by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50127222(CHEMBL38508 | GW-0742 | {4-[2-(3-Fluoro-4-trifluor...)
Affinity DataEC50:  30nMAssay Description:Activity against murine PPAR delta receptorMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50312472(2-(4-((5-(4-Biphenyl)-4-(pyridin-3-yl)oxazol-2-yl)...)
Affinity DataEC50:  30nMAssay Description:Agonist activity at mouse PPARdelta by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50312477(2-(4-((4-(2-Methoxypyrimidin-5-yl)-5-(4-propylphen...)
Affinity DataEC50:  30nMAssay Description:Agonist activity at mouse PPARdelta by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50312425(2-(4-((4-(4-(Cyclopentyloxy)phenyl)-5-(4-(trifluor...)
Affinity DataEC50:  31nMAssay Description:Agonist activity at mouse PPARdelta by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50312468(2-(4-((4-(4-Isopropoxyphenyl)-5-(3-(trifluorometho...)
Affinity DataEC50:  46nMAssay Description:Agonist activity at mouse PPARdelta by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50596502(CHEMBL5180328)
Affinity DataEC50:  49nMAssay Description:Transactivation of Gal4-fused mouse PPARdelta expressed in CHO cells co expressing pG5-Luc reporterMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM28661(2-{2-methyl-4-[({4-methyl-2-[4-(trifluoromethyl)ph...)
Affinity DataEC50:  54nMAssay Description:Agonist activity at mouse PPAR delta expressed in HEK293 cells by PPAR-GAL4 transactivation assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM28661(2-{2-methyl-4-[({4-methyl-2-[4-(trifluoromethyl)ph...)
Affinity DataEC50:  70nMAssay Description:Transactivation of mouse PPARdelta by cell-based luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50596500(CHEMBL5180073)
Affinity DataEC50:  71nMAssay Description:Transactivation of Gal4-fused mouse PPARdelta expressed in CHO cells co expressing pG5-Luc reporterMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50312471(2-(4-((4-(4-Morpholinophenyl)-5-(4-biphenyl)thiazo...)
Affinity DataEC50:  72nMAssay Description:Agonist activity at mouse PPARdelta by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM28661(2-{2-methyl-4-[({4-methyl-2-[4-(trifluoromethyl)ph...)
Affinity DataEC50:  76nMAssay Description:Transactivation of Gal4-fused mouse PPARdelta expressed in CHO cells co expressing pG5-Luc reporterMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM28661(2-{2-methyl-4-[({4-methyl-2-[4-(trifluoromethyl)ph...)
Affinity DataEC50:  77nMAssay Description:Agonist activity at mouse PPARdelta by FRET assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50312473(CHEMBL1079983 | {4-[4-(6-Methoxypyridin-3-yl)-5-(4...)
Affinity DataEC50:  90nMAssay Description:Agonist activity at mouse PPARdelta by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50312474(2-(4-((4-(6-Methoxypyridin-3-yl)-5-(4-(trifluorome...)
Affinity DataEC50:  97nMAssay Description:Agonist activity at mouse PPARdelta by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50176605((S)-2-(3-((3-fluoro-4-(trifluoromethyl)benzamido)m...)
Affinity DataEC50:  130nMAssay Description:Agonist activity at mouse PPARdelta transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50596501(CHEMBL5193666)
Affinity DataEC50:  151nMAssay Description:Transactivation of Gal4-fused mouse PPARdelta expressed in CHO cells co expressing pG5-Luc reporterMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50192829(CHEMBL3958704 | US10188627, Compound 8a)
Affinity DataEC50:  270nMAssay Description:Transactivation of mouse PPARdelta by cell-based luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50229206(CHEMBL253310 | N-(4-(trifluoromethylsulfonamido)be...)
Affinity DataEC50:  300nMAssay Description:Agonist activity at mouse PPARdelta assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50207469(CHEMBL222880 | {4-[3,3-bis-(4-bromo-phenyl)-allyls...)
Affinity DataEC50:  300nMAssay Description:Agonist activity at mouse PPAR delta expressed in HEK293 cells by PPAR-GAL4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50596503(CHEMBL5183133)
Affinity DataEC50:  330nMAssay Description:Transactivation of Gal4-fused mouse PPARdelta expressed in CHO cells co expressing pG5-Luc reporterMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM28662(2-[4-(3-{[2-(2-chloro-6-fluorophenyl)ethyl][(2,3-d...)
Affinity DataEC50:  410nMAssay Description:Agonist activity for murine PPAR delta receptor in transcriptional activation assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50596504(CHEMBL5178616)
Affinity DataEC50:  830nMAssay Description:Transactivation of Gal4-fused mouse PPARdelta expressed in CHO cells co expressing pG5-Luc reporterMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50596499(CHEMBL5185420)
Affinity DataEC50:  1.06E+3nMAssay Description:Transactivation of Gal4-fused mouse PPARdelta expressed in CHO cells co expressing pG5-Luc reporterMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50081222(2-(4-{2-[1-Cycloheptyl-3-(2,4-difluoro-phenyl)-ure...)
Affinity DataEC50:  1.40E+3nMAssay Description:Compound was tested for its agonist activity against murine Peroxisome proliferator activated receptor delta-GAL4 chimeric receptor in transfected CV...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50244350(CHEMBL4091374)
Affinity DataEC50:  1.56E+3nMAssay Description:Transactivation of mouse GAL4-fused PPARdelta LBD expressed in African green monkey COS7 cells co-expressing 5Gal4 pGL3 TK Luc after overnight incuba...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM28706(2-methyl-2-phenoxypropanoic acid, 25a | 2-methyl-2...)
Affinity DataEC50:  1.70E+3nMAssay Description:Agonist activity at mouse PPARdelta assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50319262(2-(4-(((2-(2,4-dimethylphenylamino)-2-oxoethyl)(fu...)
Affinity DataEC50:  2.00E+3nMAssay Description:Agonist activity at Gal4-fused mouse PPARdeltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM28799(2-{[4-(2-{[(2,4-difluorophenyl)carbamoyl](heptyl)a...)
Affinity DataEC50:  2.00E+3nMAssay Description:Agonist activity at Gal4-fused mouse PPARdeltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM28799(2-{[4-(2-{[(2,4-difluorophenyl)carbamoyl](heptyl)a...)
Affinity DataEC50:  2.60E+3nMAssay Description:Agonist activity for murine PPAR delta receptor in transcriptional activation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM28799(2-{[4-(2-{[(2,4-difluorophenyl)carbamoyl](heptyl)a...)
Affinity DataEC50:  2.60E+3nMAssay Description:Compound was tested for its agonist activity against murine Peroxisome proliferator activated receptor delta-GAL4 chimeric receptor in transfected CV...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50099491(2-(4-(2-(3-cyclohexyl-1-(4-cyclohexylbutyl)ureido)...)
Affinity DataEC50:  2.90E+3nMAssay Description:Activation of murine PPAR delta ligand binding domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50081223(2-(4-{2-[3-(2,4-Difluoro-phenyl)-1-heptyl-ureido]-...)
Affinity DataEC50:  3.20E+3nMAssay Description:Compound was tested for its agonist activity against murine Peroxisome proliferator activated receptor delta-GAL4 chimeric receptor in transfected CV...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50085041(2-(4-(3-(4-acetyl-3-hydroxy-2-propylphenoxy)propox...)
Affinity DataEC50:  3.80E+3nMAssay Description:Agonist activity for murine PPAR delta receptor in transcriptional activation assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50081225(2-(4-{2-[3-(4-Fluoro-phenyl)-1-heptyl-ureido]-ethy...)
Affinity DataEC50:  5.50E+3nMAssay Description:Compound was tested for its agonist activity against murine Peroxisome proliferator activated receptor delta-GAL4 chimeric receptor in transfected CV...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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