Compile Data Set for Download or QSAR
maximum 50k data
Found 10 of ic50 data for polymerid = 50001092,50004899
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Philipps University

Curated by ChEMBL
LigandPNGBDBM50383371(CHEMBL2030550)
Affinity DataIC50:  9.5nMAssay Description:Inverse agonist activity at PPARbeta/delta in mouse C2C12 cells assessed as inhibition of Angptl4 expression after 24 hrs by RT-qPCR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Philipps University

Curated by ChEMBL
LigandPNGBDBM50383371(CHEMBL2030550)
Affinity DataIC50:  26.9nMAssay Description:Displacement of fluormone Pan-PPAR Green from mouse recombinant GST-tagged PPARbeta/delta LBD after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Philipps University

Curated by ChEMBL
LigandPNGBDBM50383373(CHEMBL592652 | GSK0660)
Affinity DataIC50:  48nMAssay Description:Inverse agonist activity at PPARbeta/delta in mouse C2C12 cells assessed as inhibition of Angptl4 expression after 24 hrs by RT-qPCR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Philipps University

Curated by ChEMBL
LigandPNGBDBM50383370(CHEMBL2030543)
Affinity DataIC50:  52nMAssay Description:Inverse agonist activity at PPARbeta/delta in mouse C2C12 cells assessed as inhibition of Angptl4 expression after 24 hrs by RT-qPCR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Philipps University

Curated by ChEMBL
LigandPNGBDBM50383370(CHEMBL2030543)
Affinity DataIC50:  180nMAssay Description:Displacement of fluormone Pan-PPAR Green from mouse recombinant GST-tagged PPARbeta/delta LBD after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Philipps University

Curated by ChEMBL
LigandPNGBDBM50200411((S)-2-(5-(3-((2-(4-ethylphenyl)-5-methylpyrimidin-...)
Affinity DataIC50:  370nMAssay Description:Activity at mouse PPARdelta expressed in CV1 cells by GAL4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Philipps University

Curated by ChEMBL
LigandPNGBDBM50383372(CHEMBL1998001)
Affinity DataIC50: >500nMAssay Description:Inverse agonist activity at PPARbeta/delta in mouse C2C12 cells assessed as inhibition of Angptl4 expression after 24 hrs by RT-qPCR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Philipps University

Curated by ChEMBL
LigandPNGBDBM50200403((S)-2-(5-(3-((2-(4-isopropylphenyl)-5-methylpyrimi...)
Affinity DataIC50:  610nMAssay Description:Activity at mouse PPARdelta expressed in CV1 cells by GAL4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Philipps University

Curated by ChEMBL
LigandPNGBDBM50508127(CHEMBL4449687)
Affinity DataIC50:  960nMAssay Description:Antagonist activity at mouse PPARdeltaMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Philipps University

Curated by ChEMBL
LigandPNGBDBM50200402(2-((S)-5-(3-(5-(5-acetyl-4-methylthiazol-2-yl)pyri...)
Affinity DataIC50:  1.39E+3nMAssay Description:Activity at mouse PPARdelta expressed in CV1 cells by GAL4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed