Compile Data Set for Download or QSAR
maximum 50k data
Found 7 of ki data for polymerid = 50001398,50006609
TargetHistamine N-methyltransferase(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50041457(4-[(7-chloroquinolin-4-yl)amino]-2-[(diethylamino)...)
Affinity DataKi:  19nMAssay Description:Inhibition of histamine N-methyltransferase by radiochemical assayMore data for this Ligand-Target Pair
TargetHistamine N-methyltransferase(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50026331(2-Amino-4-[4-(6-amino-purin-9-yl)-2,3-dihydroxy-cy...)
Affinity DataKi:  1.04E+4nMAssay Description:Inhibition constant was evaluated against Histamine N-methyl-transferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine N-methyltransferase(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50026331(2-Amino-4-[4-(6-amino-purin-9-yl)-2,3-dihydroxy-cy...)
Affinity DataKi:  1.04E+4nMAssay Description:Inhibition constant was evaluated against Histamine N-methyl-transferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine N-methyltransferase(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50009672(AdoHcy | CHEMBL418052 | S-(5'-adenosyl)-L-homocyst...)
Affinity DataKi:  1.81E+4nMAssay Description:Inhibition constant was evaluated against Histamine N-methyl-transferaseMore data for this Ligand-Target Pair
TargetHistamine N-methyltransferase(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50009672(AdoHcy | CHEMBL418052 | S-(5'-adenosyl)-L-homocyst...)
Affinity DataKi:  1.81E+4nMAssay Description:Inhibition constant was evaluated against Histamine N-methyl-transferaseMore data for this Ligand-Target Pair
TargetHistamine N-methyltransferase(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50016564(CHEMBL3272448)
Affinity DataKi:  3.16E+4nMAssay Description:Inhibition of histamine N-methyltransferase in guinea pig brain using S-adenosyl-L-methionine-14C as substrate by scintillation spectrophotometerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine N-methyltransferase(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50016547(CHEMBL3272447)
Affinity DataKi:  2.47E+5nMAssay Description:Inhibition of histamine N-methyltransferase in guinea pig brain using S-adenosyl-L-methionine-14C as substrate by scintillation spectrophotometerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed