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Found 25 of ic50 data for polymerid = 50006118
TargetSolute carrier family 22 member 8(Homo sapiens (Human))
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50537500(CHEMBL4562825)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of OAT3 (unknown origin) expressed in HEK293 cells assessed as reduction in 6-CF uptake measured after 5 mins by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 8(Homo sapiens (Human))
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50537497(CHEMBL4519013)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of OAT3 (unknown origin) expressed in HEK293 cells assessed as reduction in 6-CF uptake measured after 5 mins by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 8(Homo sapiens (Human))
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50537498(CHEMBL4584575)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of OAT3 (unknown origin) expressed in HEK293 cells assessed as reduction in 6-CF uptake measured after 5 mins by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 8(Homo sapiens (Human))
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50537496(CHEMBL4527448)
Affinity DataIC50:  2.30E+3nMAssay Description:Inhibition of OAT3 (unknown origin) expressed in HEK293 cells assessed as reduction in 6-CF uptake measured after 5 mins by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 8(Homo sapiens (Human))
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50537501(CHEMBL4582456)
Affinity DataIC50:  2.80E+3nMAssay Description:Inhibition of OAT3 (unknown origin) expressed in HEK293 cells assessed as reduction in 6-CF uptake measured after 5 mins by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 8(Homo sapiens (Human))
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50206509(4-Dipropylsulfamoyl-benzoic acid | 4-Dipropylsulfa...)
Affinity DataIC50:  4.93E+3nMAssay Description:TP_TRANSPORTER: inhibition of ES uptake (ES: 50nM) in hOAT3-expressing S2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetSolute carrier family 22 member 8(Homo sapiens (Human))
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50305842(CHEMBL603656 | trans-4-((5-(2-(4-fluorobenzylcarba...)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibition of human OAT3 expressed in HEK cells assessed as reduction of [3H]-estrone sulfate uptake by radioactivity counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 8(Homo sapiens (Human))
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50537502(CHEMBL38650 | NSC-220968)
Affinity DataIC50:  6.50E+3nMAssay Description:Inhibition of OAT3 (unknown origin) expressed in HEK293 cells assessed as reduction in 6-CF uptake measured after 5 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 8(Homo sapiens (Human))
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50133599((7-Imidazol-1-yl-6-nitro-2,3-dioxo-3,4-dihydro-2H-...)
Affinity DataIC50:  6.60E+3nMAssay Description:Inhibition of human OAT3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 8(Homo sapiens (Human))
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50537499(CHEMBL4525573)
Affinity DataIC50:  8.30E+3nMAssay Description:Inhibition of OAT3 (unknown origin) expressed in HEK293 cells assessed as reduction in 6-CF uptake measured after 5 mins by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 8(Homo sapiens (Human))
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50206509(4-Dipropylsulfamoyl-benzoic acid | 4-Dipropylsulfa...)
Affinity DataIC50:  9.00E+3nMAssay Description:Inhibition of OAT3 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetSolute carrier family 22 member 8(Homo sapiens (Human))
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50344964(Betamipron | CHEMBL1231530 | N-(phenylcarbonyl)-be...)
Affinity DataIC50:  9.92E+3nMAssay Description:TP_TRANSPORTER: inhibition of ES uptake (ES: 50nM) in hOAT3-expressing S2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 8(Homo sapiens (Human))
Tianjin University

Curated by ChEMBL
LigandPNGBDBM20688((3R,5R)-7-[(1S,2S,6S,8S,8aR)-6-hydroxy-2-methyl-8-...)
Affinity DataIC50:  1.37E+4nMAssay Description:TP_TRANSPORTER: inhibition of ES uptake (ES: 50nM) in hOAT3-expressing S2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetSolute carrier family 22 member 8(Homo sapiens (Human))
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50265079((4-[1-methyl-2,4-dioxo-6-(3-phenyl-prop-1-ynyl)-1,...)
Affinity DataIC50:  1.80E+4nMAssay Description:Inhibition of human OAT3 expressed in HEK cells assessed as reduction of [3H]-estrone sulfate uptake by radioactivity counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 8(Homo sapiens (Human))
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50180512(1-methyl-5-vinyl-9,10-dihydrophenanthrene-2,7-diol...)
Affinity DataIC50:  2.27E+4nMAssay Description:Inhibition of OAT3 (unknown origin) expressed in HEK293 cells assessed as reduction in 6-CF uptake measured after 5 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 8(Homo sapiens (Human))
Tianjin University

Curated by ChEMBL
LigandPNGBDBM207624(US10501467, Example 69 | US9260440, 69 | US9617273...)
Affinity DataIC50:  2.39E+4nMAssay Description:Inhibition of OAT3 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 8(Homo sapiens (Human))
Tianjin University

Curated by ChEMBL
LigandPNGBDBM311267((S)-1-((2′,6-bis(difluoromethyl)-[2,4′...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of OAT3 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 8(Homo sapiens (Human))
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50511112(CHEMBL4567446)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human SLC22A8 expressed in HEK293 cells in presence of para-aminohippuric acid/metforminMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSolute carrier family 22 member 8(Homo sapiens (Human))
Tianjin University

Curated by ChEMBL
LigandPNGBDBM311268((S)-1-((2′,4-bis(difluoromethyl)-[2,4′...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of OAT3 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSolute carrier family 22 member 8(Homo sapiens (Human))
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50234348(4-((6-(4-methoxybenzylcarbamoyl)-4-oxopyrido[3,4-d...)
Affinity DataIC50:  5.90E+4nMAssay Description:Inhibition of human OAT3 expressed in HEK cells assessed as reduction of [3H]-estrone sulfate uptake by radioactivity counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 8(Homo sapiens (Human))
Tianjin University

Curated by ChEMBL
LigandPNGBDBM22889((Cimetidine) N-Methyl-N''''-[2-(5-methyl-1H-imidaz...)
Affinity DataIC50:  9.24E+4nMAssay Description:TP_TRANSPORTER: inhibition of ES uptake (ES: 50nM) in hOAT3-expressing S2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 8(Homo sapiens (Human))
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50228403((R)-8-(3-aminopiperidin-1-yl)-7-(but-2-ynyl)-3-met...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of OAT3 (unknown origin) expressed in HEK293 cells assessed as reduction of [3H]E-sul substrate uptake by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 8(Homo sapiens (Human))
Tianjin University

Curated by ChEMBL
LigandPNGBDBM42131(CEFACLOR | MLS000069617 | SMR000058250 | cid_51039)
Affinity DataIC50:  1.20E+5nMAssay Description:Inhibition of human OAT3 using estrone-3-sulfate as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 8(Homo sapiens (Human))
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50367502(CILASTATIN)
Affinity DataIC50:  2.49E+5nMAssay Description:TP_TRANSPORTER: inhibition of ES uptake (ES: 50nM) in hOAT3-expressing S2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetSolute carrier family 22 member 8(Homo sapiens (Human))
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50566497(2,2-DIMETHYLBUTYRATE | 2,2-Dimethyl-Butyric Acid |...)
Affinity DataIC50:  3.51E+6nMAssay Description:Inhibition of human OAT3 assessed as reduction in OAT3-mediated tenofovir transportMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed