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Found 10 of ki for UniProtKB: O75751
TargetSolute carrier family 22 member 3(Homo sapiens (Human))
University Of Heidelberg

Curated by ChEMBL
LigandPNGBDBM50420215(CHEMBL339858)
Affinity DataKi:  15nMAssay Description:TP_TRANSPORTER: inhibition of MPP+ uptake in OCT3-expressing HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 3(Homo sapiens (Human))
University Of Heidelberg

Curated by ChEMBL
LigandPNGBDBM50014846((S)-N-(5,6,7,9-tetrahydro-1,2,3,10-tetramethoxy-9-...)
Affinity DataKi:  120nMAssay Description:TP_TRANSPORTER: inhibition of MPP+ uptake in OCT3-expressing HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 3(Homo sapiens (Human))
University Of Heidelberg

Curated by ChEMBL
LigandPNGBDBM35229(3-(10,11-dihydro-5H-dibenzo[b,f]azepin-5-yl)-N-met...)
Affinity DataKi:  1.40E+4nMAssay Description:TP_TRANSPORTER: inhibition of MPP+ uptake in OCT3-expressing HRPE cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetSolute carrier family 22 member 3(Homo sapiens (Human))
University Of Heidelberg

Curated by ChEMBL
LigandPNGBDBM50010859(CHEMBL11 | IMIPRAMINE HYDROCHLORIDE | IMIPRAMINE P...)
Affinity DataKi:  4.20E+4nMAssay Description:TP_TRANSPORTER: inhibition of MPP+ uptake in OCT3-expressing HRPE cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetSolute carrier family 22 member 3(Homo sapiens (Human))
University Of Heidelberg

Curated by ChEMBL
LigandPNGBDBM81945(CAS_39484 | CHEMBL105891 | CHEMBL108926 | CHEMBL27...)
Affinity DataKi:  5.40E+4nMAssay Description:TP_TRANSPORTER: inhibition of MPP+ uptake in OCT3-expressing HRPE cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 3(Homo sapiens (Human))
University Of Heidelberg

Curated by ChEMBL
LigandPNGBDBM7966(2-(1H-imidazol-4-yl)ethan-1-amine | CHEMBL544208 |...)
Affinity DataKi:  1.40E+5nMAssay Description:TP_TRANSPORTER: inhibition of MPP+ uptake in OCT3-expressing HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetSolute carrier family 22 member 3(Homo sapiens (Human))
University Of Heidelberg

Curated by ChEMBL
LigandPNGBDBM50225285(CHEBI:3757 | Catapres | Catapres-Tts-1 | Catapres-...)
Affinity DataKi:  3.73E+5nMAssay Description:TP_TRANSPORTER: inhibition of MPP+ uptake in OCT3-expressing HRPE cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 3(Homo sapiens (Human))
University Of Heidelberg

Curated by ChEMBL
LigandPNGBDBM39344(4-amino-N-[2-(diethylamino)ethyl]benzamide;hydroch...)
Affinity DataKi:  7.38E+5nMAssay Description:TP_TRANSPORTER: inhibition of MPP+ uptake in OCT3-expressing HRPE cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetSolute carrier family 22 member 3(Homo sapiens (Human))
University Of Heidelberg

Curated by ChEMBL
LigandPNGBDBM50149890(CHEMBL9324 | tetraethylammonium)
Affinity DataKi:  1.37E+6nMAssay Description:TP_TRANSPORTER: inhibition of MPP+ uptake in OCT3-expressing HRPE cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 3(Homo sapiens (Human))
University Of Heidelberg

Curated by ChEMBL
LigandPNGBDBM50420178(GUANIDINE)
Affinity DataKi:  6.20E+6nMAssay Description:TP_TRANSPORTER: inhibition of MPP+ uptake in OCT3-expressing HRPE cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank