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Found 25 of ic50 data for polymerid = 50006438,5449
TargetOrexin receptor type 2(Rattus norvegicus (Rat))
TBA

US Patent
LigandPNGBDBM97406(Orexin receptor antagonist 1 | US20130102619, 1)
Affinity DataIC50:  12nMT: 2°CAssay Description:FLIPR assay using orexin receptor.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetOrexin receptor type 2(Rattus norvegicus (Rat))
TBA

US Patent
LigandPNGBDBM97397(Orexin receptor antagonist 29 | Orexin receptor an...)
Affinity DataIC50:  12nMT: 2°CAssay Description:FLIPR assay using orexin receptor.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetOrexin receptor type 2(Rattus norvegicus (Rat))
TBA

US Patent
LigandPNGBDBM97397(Orexin receptor antagonist 29 | Orexin receptor an...)
Affinity DataIC50:  17nMT: 2°CAssay Description:FLIPR assay using orexin receptor.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetOrexin receptor type 2(Rattus norvegicus (Rat))
TBA

US Patent
LigandPNGBDBM97373(Orexin receptor antagonist 5 | US20130102619, 5)
Affinity DataIC50:  17nMT: 2°CAssay Description:FLIPR assay using orexin receptor.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetOrexin receptor type 2(Rattus norvegicus (Rat))
TBA

US Patent
LigandPNGBDBM97408(Orexin receptor antagonist 3 | US20130102619, 3)
Affinity DataIC50:  18nMT: 2°CAssay Description:FLIPR assay using orexin receptor.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetOrexin receptor type 2(Rattus norvegicus (Rat))
TBA

US Patent
LigandPNGBDBM97375(Orexin receptor antagonist 6 | US20130102619, 6)
Affinity DataIC50:  18nMT: 2°CAssay Description:FLIPR assay using orexin receptor.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetOrexin receptor type 2(Rattus norvegicus (Rat))
TBA

US Patent
LigandPNGBDBM97378(Orexin receptor antagonist 9 | US20130102619, 9)
Affinity DataIC50:  22nMT: 2°CAssay Description:FLIPR assay using orexin receptor.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetOrexin receptor type 2(Rattus norvegicus (Rat))
TBA

US Patent
LigandPNGBDBM97390(Orexin receptor antagonist 22 | US20130102619, 22)
Affinity DataIC50:  23nMT: 2°CAssay Description:FLIPR assay using orexin receptor.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetOrexin receptor type 2(Rattus norvegicus (Rat))
TBA

US Patent
LigandPNGBDBM97407(Orexin receptor antagonist 2 | US20130102619, 2)
Affinity DataIC50:  28nMT: 2°CAssay Description:FLIPR assay using orexin receptor.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetOrexin receptor type 2(Rattus norvegicus (Rat))
TBA

US Patent
LigandPNGBDBM97377(Orexin receptor antagonist 8 | US20130102619, 8)
Affinity DataIC50:  29nMT: 2°CAssay Description:FLIPR assay using orexin receptor.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetOrexin receptor type 2(Rattus norvegicus (Rat))
TBA

US Patent
LigandPNGBDBM97379(Orexin receptor antagonist 10 | US20130102619, 10)
Affinity DataIC50:  29nMT: 2°CAssay Description:FLIPR assay using orexin receptor.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetOrexin receptor type 2(Rattus norvegicus (Rat))
TBA

US Patent
LigandPNGBDBM97374(Orexin receptor antagonist 4 | US20130102619, 4)
Affinity DataIC50:  29nMT: 2°CAssay Description:FLIPR assay using orexin receptor.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetOrexin receptor type 2(Rattus norvegicus (Rat))
TBA

US Patent
LigandPNGBDBM97403(Orexin receptor antagonist 35 | US20130102619, 35)
Affinity DataIC50:  31nMT: 2°CAssay Description:FLIPR assay using orexin receptor.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetOrexin receptor type 2(Rattus norvegicus (Rat))
TBA

US Patent
LigandPNGBDBM97399(Orexin receptor antagonist 31 | US20130102619, 31)
Affinity DataIC50:  38nMT: 2°CAssay Description:FLIPR assay using orexin receptor.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetOrexin receptor type 2(Rattus norvegicus (Rat))
TBA

US Patent
LigandPNGBDBM97400(Orexin receptor antagonist 32 | US20130102619, 32)
Affinity DataIC50:  44nMT: 2°CAssay Description:FLIPR assay using orexin receptor.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetOrexin receptor type 2(Rattus norvegicus (Rat))
TBA

US Patent
LigandPNGBDBM97404(Orexin receptor antagonist 36 | US20130102619, 36)
Affinity DataIC50:  47nMT: 2°CAssay Description:FLIPR assay using orexin receptor.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetOrexin receptor type 2(Rattus norvegicus (Rat))
TBA

US Patent
LigandPNGBDBM97402(Orexin receptor antagonist 34 | US20130102619, 34)
Affinity DataIC50:  48nMT: 2°CAssay Description:FLIPR assay using orexin receptor.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetOrexin receptor type 2(Rattus norvegicus (Rat))
TBA

US Patent
LigandPNGBDBM97401(Orexin receptor antagonist 33 | US20130102619, 33)
Affinity DataIC50:  52nMT: 2°CAssay Description:FLIPR assay using orexin receptor.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetOrexin receptor type 2(Rattus norvegicus (Rat))
TBA

US Patent
LigandPNGBDBM97384(Orexin receptor antagonist 15 | US20130102619, 15)
Affinity DataIC50:  62nMT: 2°CAssay Description:FLIPR assay using orexin receptor.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetOrexin receptor type 2(Rattus norvegicus (Rat))
TBA

US Patent
LigandPNGBDBM97383(Orexin receptor antagonist 14 | US20130102619, 14)
Affinity DataIC50:  65nMT: 2°CAssay Description:FLIPR assay using orexin receptor.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetOrexin receptor type 2(Rattus norvegicus (Rat))
TBA

US Patent
LigandPNGBDBM97388(Orexin receptor antagonist 20 | US20130102619, 20)
Affinity DataIC50:  67nMT: 2°CAssay Description:FLIPR assay using orexin receptor.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetOrexin receptor type 2(Rattus norvegicus (Rat))
TBA

US Patent
LigandPNGBDBM97385(Orexin receptor antagonist 17 | US20130102619, 17)
Affinity DataIC50:  82nMT: 2°CAssay Description:FLIPR assay using orexin receptor.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetOrexin receptor type 2(Rattus norvegicus (Rat))
TBA

US Patent
LigandPNGBDBM97398(Orexin receptor antagonist 30 | US20130102619, 30)
Affinity DataIC50:  110nMT: 2°CAssay Description:FLIPR assay using orexin receptor.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetOrexin receptor type 2(Rattus norvegicus (Rat))
TBA

US Patent
LigandPNGBDBM50060937(CHEMBL3394848)
Affinity DataIC50:  1.31E+3nMAssay Description:Antagonist activity at rat OX2 receptor assessed as inhibition of Ala-6,12 orexin-A-induced calcium increase preincubated for 5 mins prior to Ala-6,1...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin receptor type 2(Rattus norvegicus (Rat))
TBA

US Patent
LigandPNGBDBM50203731(CHEMBL3973097)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at rat OX2 receptor assessed as inhibition of Ala-6,12 orexin-A-induced calcium increase preincubated for 5 mins prior to Ala-6,1...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed