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Found 95 of ic50 data for polymerid = 50006733
TargetPhosphatidylinositol 4-kinase type 2-alpha(Homo sapiens (Human))TBA
LigandPNGBDBM50215065(CHEMBL171366)
Affinity DataIC50:  75.7nMAssay Description:Inhibition of Phosphatidylinositol 4-kinase of human epidermoid carcinoma A431 cellsMore data for this Ligand-Target Pair
In DepthDetails
TargetPhosphatidylinositol 4-kinase type 2-alpha(Homo sapiens (Human))TBA
LigandPNGBDBM50214291(ECHIGUANINE A)
Affinity DataIC50:  113nMAssay Description:Inhibition of Phosphatidylinositol 4-kinase of human epidermoid carcinoma A431 cellsMore data for this Ligand-Target Pair
In DepthDetails
TargetPhosphatidylinositol 4-kinase type 2-alpha(Homo sapiens (Human))TBA
LigandPNGBDBM50214291(ECHIGUANINE A)
Affinity DataIC50:  113nMAssay Description:Inhibition of phosphatidylinositol 4-kinaseMore data for this Ligand-Target Pair
In DepthDetails
TargetPhosphatidylinositol 4-kinase type 2-alpha(Homo sapiens (Human))TBA
LigandPNGBDBM50215064(CHEMBL170865)
Affinity DataIC50:  513nMAssay Description:Inhibition of Phosphatidylinositol 4-kinase of human epidermoid carcinoma A431 cellsMore data for this Ligand-Target Pair
In DepthDetails
TargetPhosphatidylinositol 4-kinase type 2-alpha(Homo sapiens (Human))TBA
LigandPNGBDBM50215084(Echiguanine B)
Affinity DataIC50:  719nMAssay Description:Inhibition of Phosphatidylinositol 4-kinase of human epidermoid carcinoma A431 cellsMore data for this Ligand-Target Pair
In DepthDetails
TargetPhosphatidylinositol 4-kinase type 2-alpha(Homo sapiens (Human))TBA
LigandPNGBDBM50215080(CHEMBL369443)
Affinity DataIC50:  1.07E+3nMAssay Description:Inhibition of Phosphatidylinositol 4-kinase of human epidermoid carcinoma A431 cellsMore data for this Ligand-Target Pair
In DepthDetails
TargetPhosphatidylinositol 4-kinase type 2-alpha(Homo sapiens (Human))TBA
LigandPNGBDBM50607059(CHEMBL5220205)
Affinity DataIC50:  1.46E+3nMAssay Description:Inhibition of PI4K2A catalytic domain (unknown origin) assessed as enzyme residual activity incubated for 60 mins using ATP as substrate by ATP-Glo l...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPhosphatidylinositol 4-kinase type 2-alpha(Homo sapiens (Human))TBA
LigandPNGBDBM50215067(CHEMBL169505)
Affinity DataIC50:  1.82E+3nMAssay Description:Inhibition of Phosphatidylinositol 4-kinase of human epidermoid carcinoma A431 cellsMore data for this Ligand-Target Pair
In DepthDetails
TargetPhosphatidylinositol 4-kinase type 2-alpha(Homo sapiens (Human))TBA
LigandPNGBDBM50215063(CHEMBL608216)
Affinity DataIC50:  2.35E+3nMAssay Description:Inhibition of Phosphatidylinositol 4-kinase of human epidermoid carcinoma A431 cellsMore data for this Ligand-Target Pair
In DepthDetails
TargetPhosphatidylinositol 4-kinase type 2-alpha(Homo sapiens (Human))TBA
LigandPNGBDBM50013711(9-Cyclohexyl-9H-adenine | 9-Cyclohexyl-9H-purin-6-...)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibitory activity (IC50) against human phosphatidylinositol 4-kinase at the ATP binding siteMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4-kinase type 2-alpha(Homo sapiens (Human))TBA
LigandPNGBDBM50228349(CHEMBL293027)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibitory activity (IC50) against human phosphatidylinositol 4-kinase at the ATP binding siteMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4-kinase type 2-alpha(Homo sapiens (Human))TBA
LigandPNGBDBM50215082(CHEMBL607667)
Affinity DataIC50:  6.05E+3nMAssay Description:Inhibition of Phosphatidylinositol 4-kinase of human epidermoid carcinoma A431 cellsMore data for this Ligand-Target Pair
In DepthDetails
TargetPhosphatidylinositol 4-kinase type 2-alpha(Homo sapiens (Human))TBA
LigandPNGBDBM50013712(2-aminopyridin | 2-aminopyridine | CHEMBL21619 | P...)
Affinity DataIC50:  7.10E+3nMAssay Description:Inhibitory activity (IC50) against human phosphatidylinositol 4-kinase at the ATP binding siteMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4-kinase type 2-alpha(Homo sapiens (Human))TBA
LigandPNGBDBM50013702(9-Cycloheptyl-9H-adenine | 9-Cycloheptyl-9H-purin-...)
Affinity DataIC50:  7.20E+3nMAssay Description:Inhibitory activity (IC50) against human phosphatidylinositol 4-kinase at the ATP binding siteMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4-kinase type 2-alpha(Homo sapiens (Human))TBA
LigandPNGBDBM50228342(CHEMBL413106)
Affinity DataIC50:  7.20E+3nMAssay Description:Inhibitory activity (IC50) against human phosphatidylinositol 4-kinase at the ATP binding siteMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4-kinase type 2-alpha(Homo sapiens (Human))TBA
LigandPNGBDBM50009680(6-Amino-9-cyclopentyl-9H-purine | 9-Cyclopentyl-9H...)
Affinity DataIC50:  8.70E+3nMAssay Description:Inhibitory activity (IC50) against human phosphatidylinositol 4-kinase at the ATP binding siteMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4-kinase type 2-alpha(Homo sapiens (Human))TBA
LigandPNGBDBM50536410(CHEMBL4561692)
Affinity DataIC50: <1.00E+4nMAssay Description:Inhibition of PI4K2A (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4-kinase type 2-alpha(Homo sapiens (Human))TBA
LigandPNGBDBM50199888(CHEMBL3976651)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of PI4K2A (unknown origin) by ADP-Glo kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4-kinase type 2-alpha(Homo sapiens (Human))TBA
LigandPNGBDBM50228481(CHEMBL306444)
Affinity DataIC50:  1.02E+4nMAssay Description:Inhibitory activity (IC50) against human phosphatidylinositol 4-kinase at the ATP binding siteMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4-kinase type 2-alpha(Homo sapiens (Human))TBA
LigandPNGBDBM50228483(CHEMBL291377)
Affinity DataIC50:  1.19E+4nMAssay Description:Inhibitory activity (IC50) against human phosphatidylinositol 4-kinase at the ATP binding siteMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4-kinase type 2-alpha(Homo sapiens (Human))TBA
LigandPNGBDBM50228351(CHEMBL1321883)
Affinity DataIC50:  1.21E+4nMAssay Description:Inhibitory activity (IC50) against human phosphatidylinositol 4-kinase at the ATP binding siteMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4-kinase type 2-alpha(Homo sapiens (Human))TBA
LigandPNGBDBM50607056(CHEMBL5218945)
Affinity DataIC50:  1.22E+4nMAssay Description:Inhibition of PI4K2A catalytic domain (unknown origin) assessed as enzyme residual activity incubated for 60 mins using ATP as substrate by ATP-Glo l...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPhosphatidylinositol 4-kinase type 2-alpha(Homo sapiens (Human))TBA
LigandPNGBDBM50228343(CHEMBL304265)
Affinity DataIC50:  1.28E+4nMAssay Description:Inhibitory activity (IC50) against human phosphatidylinositol 4-kinase at the ATP binding siteMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4-kinase type 2-alpha(Homo sapiens (Human))TBA
LigandPNGBDBM50013685(9-Isopropyl-9H-adenine | 9-Isopropyl-9H-purin-6-yl...)
Affinity DataIC50:  1.49E+4nMAssay Description:Inhibitory activity (IC50) against human phosphatidylinositol 4-kinase at the ATP binding siteMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4-kinase type 2-alpha(Homo sapiens (Human))TBA
LigandPNGBDBM50009689(9-Phenyl-9H-purin-6-ylamine | CHEMBL62756)
Affinity DataIC50:  1.54E+4nMAssay Description:Inhibitory activity (IC50) against human phosphatidylinositol 4-kinase at the ATP binding siteMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4-kinase type 2-alpha(Homo sapiens (Human))TBA
LigandPNGBDBM50013720(1-Phenyl-1H-pyrazolo[3,4-d]pyrimidin-4-ylamine | C...)
Affinity DataIC50:  1.61E+4nMAssay Description:Inhibitory activity (IC50) against human phosphatidylinositol 4-kinase at the ATP binding siteMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4-kinase type 2-alpha(Homo sapiens (Human))TBA
LigandPNGBDBM50228346(CHEMBL65685)
Affinity DataIC50:  1.64E+4nMAssay Description:Inhibitory activity (IC50) against human phosphatidylinositol 4-kinase at the ATP binding siteMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4-kinase type 2-alpha(Homo sapiens (Human))TBA
LigandPNGBDBM50228348(CHEMBL64565)
Affinity DataIC50:  1.64E+4nMAssay Description:Inhibitory activity (IC50) against human phosphatidylinositol 4-kinase at the ATP binding siteMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4-kinase type 2-alpha(Homo sapiens (Human))TBA
LigandPNGBDBM50215083(CHEMBL608492)
Affinity DataIC50:  1.76E+4nMAssay Description:Inhibition of Phosphatidylinositol 4-kinase of human epidermoid carcinoma A431 cellsMore data for this Ligand-Target Pair
In DepthDetails
TargetPhosphatidylinositol 4-kinase type 2-alpha(Homo sapiens (Human))TBA
LigandPNGBDBM50607058(CHEMBL5220999)
Affinity DataIC50:  2.08E+4nMAssay Description:Inhibition of PI4K2A catalytic domain (unknown origin) assessed as enzyme residual activity incubated for 60 mins using ATP as substrate by ATP-Glo l...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPhosphatidylinositol 4-kinase type 2-alpha(Homo sapiens (Human))TBA
LigandPNGBDBM50228499(CHEMBL305102)
Affinity DataIC50:  2.19E+4nMAssay Description:Inhibitory activity (IC50) against human phosphatidylinositol 4-kinase at the ATP binding siteMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4-kinase type 2-alpha(Homo sapiens (Human))TBA
LigandPNGBDBM50228486(CHEMBL63815)
Affinity DataIC50:  2.29E+4nMAssay Description:Inhibitory activity (IC50) against human phosphatidylinositol 4-kinase at the ATP binding siteMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4-kinase type 2-alpha(Homo sapiens (Human))TBA
LigandPNGBDBM50228559(CHEMBL603180)
Affinity DataIC50:  2.31E+4nMAssay Description:Inhibitory activity (IC50) against human phosphatidylinositol 4-kinase at the ATP binding siteMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4-kinase type 2-alpha(Homo sapiens (Human))TBA
LigandPNGBDBM50228492(CHEMBL61397)
Affinity DataIC50:  2.36E+4nMAssay Description:Inhibitory activity (IC50) against human phosphatidylinositol 4-kinase at the ATP binding siteMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4-kinase type 2-alpha(Homo sapiens (Human))TBA
LigandPNGBDBM50607053(CHEMBL5218823)
Affinity DataIC50:  2.48E+4nMAssay Description:Inhibition of PI4K2A catalytic domain (unknown origin) assessed as enzyme residual activity incubated for 60 mins using ATP as substrate by ATP-Glo l...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails PubMed
TargetPhosphatidylinositol 4-kinase type 2-alpha(Homo sapiens (Human))TBA
LigandPNGBDBM50228350(CHEMBL292498)
Affinity DataIC50:  2.56E+4nMAssay Description:Inhibitory activity (IC50) against human phosphatidylinositol 4-kinase at the ATP binding siteMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4-kinase type 2-alpha(Homo sapiens (Human))TBA
LigandPNGBDBM50009687(9-(Tetrahydro-furan-2-yl)-9H-purin-6-ylamine | 9-(...)
Affinity DataIC50:  2.82E+4nMAssay Description:Inhibitory activity (IC50) against human phosphatidylinositol 4-kinase at the ATP binding siteMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4-kinase type 2-alpha(Homo sapiens (Human))TBA
LigandPNGBDBM50607057(CHEMBL5219275)
Affinity DataIC50:  2.84E+4nMAssay Description:Inhibition of PI4K2A catalytic domain (unknown origin) assessed as enzyme residual activity incubated for 60 mins using ATP as substrate by ATP-Glo l...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPhosphatidylinositol 4-kinase type 2-alpha(Homo sapiens (Human))TBA
LigandPNGBDBM15234((1R,3R,5S,9R,18S)-18-(methoxymethyl)-1,5-dimethyl-...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of PI4K2A catalytic domain (unknown origin) assessed as enzyme residual activity incubated for 60 mins using ATP as substrate by ATP-Glo l...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetPhosphatidylinositol 4-kinase type 2-alpha(Homo sapiens (Human))TBA
LigandPNGBDBM14487((2R,3R,4S,5R)-2-(6-amino-9H-purin-9-yl)-5-(hydroxy...)
Affinity DataIC50:  3.03E+4nMAssay Description:Inhibitory activity (IC50) against human phosphatidylinositol 4-kinase at the ATP binding siteMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4-kinase type 2-alpha(Homo sapiens (Human))TBA
LigandPNGBDBM50009681(9-Ethyl-9H-adenine | 9-Ethyl-9H-purin-6-ylamine | ...)
Affinity DataIC50:  3.24E+4nMAssay Description:Inhibitory activity (IC50) against human phosphatidylinositol 4-kinase at the ATP binding siteMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4-kinase type 2-alpha(Homo sapiens (Human))TBA
LigandPNGBDBM50228490(Benzo[G]Quinazolin-4-Ylamine | CHEMBL62648)
Affinity DataIC50:  3.30E+4nMAssay Description:Inhibitory activity (IC50) against human phosphatidylinositol 4-kinase at the ATP binding siteMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4-kinase type 2-alpha(Homo sapiens (Human))TBA
LigandPNGBDBM50228500(CHEMBL424597)
Affinity DataIC50:  3.49E+4nMAssay Description:Inhibitory activity (IC50) against human phosphatidylinositol 4-kinase at the ATP binding siteMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4-kinase type 2-alpha(Homo sapiens (Human))TBA
LigandPNGBDBM50034808(CHEMBL3353011)
Affinity DataIC50:  3.77E+4nMAssay Description:Inhibition of PI4K2A catalytic domain (unknown origin) assessed as enzyme residual activity incubated for 60 mins using ATP as substrate by ATP-Glo l...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetPhosphatidylinositol 4-kinase type 2-alpha(Homo sapiens (Human))TBA
LigandPNGBDBM50607055(CHEMBL5218631)
Affinity DataIC50:  4.09E+4nMAssay Description:Inhibition of PI4K2A catalytic domain (unknown origin) assessed as enzyme residual activity incubated for 60 mins using ATP as substrate by ATP-Glo l...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPhosphatidylinositol 4-kinase type 2-alpha(Homo sapiens (Human))TBA
LigandPNGBDBM50228501(CHEMBL65379)
Affinity DataIC50:  4.11E+4nMAssay Description:Inhibitory activity (IC50) against human phosphatidylinositol 4-kinase at the ATP binding siteMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4-kinase type 2-alpha(Homo sapiens (Human))TBA
LigandPNGBDBM50607052(CHEMBL5220036)
Affinity DataIC50:  4.42E+4nMAssay Description:Inhibition of PI4K2A catalytic domain (unknown origin) assessed as enzyme residual activity incubated for 60 mins using ATP as substrate by ATP-Glo l...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPhosphatidylinositol 4-kinase type 2-alpha(Homo sapiens (Human))TBA
LigandPNGBDBM50607054(CHEMBL5220692)
Affinity DataIC50:  4.54E+4nMAssay Description:Inhibition of PI4K2A catalytic domain (unknown origin) assessed as enzyme residual activity incubated for 60 mins using ATP as substrate by ATP-Glo l...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPhosphatidylinositol 4-kinase type 2-alpha(Homo sapiens (Human))TBA
LigandPNGBDBM50228493(CHEMBL291843)
Affinity DataIC50:  4.61E+4nMAssay Description:Inhibitory activity (IC50) against human phosphatidylinositol 4-kinase at the ATP binding siteMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4-kinase type 2-alpha(Homo sapiens (Human))TBA
LigandPNGBDBM50228480(CHEMBL62757)
Affinity DataIC50:  4.62E+4nMAssay Description:Inhibitory activity (IC50) against human phosphatidylinositol 4-kinase at the ATP binding siteMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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