TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Tohoku University
Curated by ChEMBL
Tohoku University
Curated by ChEMBL
Affinity DataEC50: 1.90nMAssay Description:Inhibition of NaV1.5 (unknown origin)More data for this Ligand-Target Pair
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Tohoku University
Curated by ChEMBL
Tohoku University
Curated by ChEMBL
Affinity DataEC50: 28nMAssay Description:Modulator activity at human Nav1.5 expressed in Xenopus laevis oocytes assessed as elicitation in sodium current measured after 1 to 4 days by two-el...More data for this Ligand-Target Pair
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Tohoku University
Curated by ChEMBL
Tohoku University
Curated by ChEMBL
Affinity DataEC50: 108nMAssay Description:Modulator activity at human Nav1.5 expressed in Xenopus laevis oocytes assessed as elicitation in sodium current measured after 1 to 4 days by two-el...More data for this Ligand-Target Pair
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Tohoku University
Curated by ChEMBL
Tohoku University
Curated by ChEMBL
Affinity DataEC50: 133nMAssay Description:Modulator activity at human Nav1.5 expressed in Xenopus laevis oocytes assessed as elicitation in sodium current measured after 1 to 4 days by two-el...More data for this Ligand-Target Pair
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Tohoku University
Curated by ChEMBL
Tohoku University
Curated by ChEMBL
Affinity DataEC50: 138nMAssay Description:Modulator activity at human Nav1.5 expressed in Xenopus laevis oocytes assessed as elicitation in sodium current measured after 1 to 4 days by two-el...More data for this Ligand-Target Pair
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Tohoku University
Curated by ChEMBL
Tohoku University
Curated by ChEMBL
Affinity DataEC50: 149nMAssay Description:Modulator activity at human Nav1.5 expressed in Xenopus laevis oocytes assessed as elicitation in sodium current measured after 1 to 4 days by two-el...More data for this Ligand-Target Pair
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Tohoku University
Curated by ChEMBL
Tohoku University
Curated by ChEMBL
Affinity DataEC50: 156nMAssay Description:Modulator activity at human Nav1.5 expressed in Xenopus laevis oocytes assessed as elicitation in sodium current measured after 1 to 4 days by two-el...More data for this Ligand-Target Pair
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Tohoku University
Curated by ChEMBL
Tohoku University
Curated by ChEMBL
Affinity DataEC50: 215nMAssay Description:Modulator activity at human Nav1.5 expressed in Xenopus laevis oocytes assessed as elicitation in sodium current measured after 1 to 4 days by two-el...More data for this Ligand-Target Pair
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Tohoku University
Curated by ChEMBL
Tohoku University
Curated by ChEMBL
Affinity DataEC50: 5.80E+3nMpH: 7.35 T: 2°CAssay Description:All experiments were conducted at room temperature (22-24° C.) with an EPC-10 amplifier and Pulse software (HEKA, Lambrecht/Pfalz, Germany) in the wh...More data for this Ligand-Target Pair
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Tohoku University
Curated by ChEMBL
Tohoku University
Curated by ChEMBL
Affinity DataEC50: >3.30E+4nMAssay Description:Inhibition of human Nav1.5 expressed in HEK293 cells by IonWorks patch clamp electrophysiology assayMore data for this Ligand-Target Pair