TargetTelomeric repeat-binding factor 2(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 90nMAssay Description:Binding affinity to TRFH domain of TRF2 (residues 42 to 245) (unknown origin) by FP based assayMore data for this Ligand-Target Pair
TargetTelomeric repeat-binding factor 2(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 90nMAssay Description:Displacement of 5-((2R,6S,9S,12S,15S,18S,21S,24S)-3-((S)-2-((S)-1-amino-3-methyl-1-oxobutan-2-ylcarbamoyl)pyrrolidine-1-carbonyl)-15-(4-aminobutyl)-2...More data for this Ligand-Target Pair
TargetTelomeric repeat-binding factor 2(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 210nMAssay Description:Displacement of 5-((2R,6S,9S,12S,15S,18S,21S,24S)-3-((S)-2-((S)-1-amino-3-methyl-1-oxobutan-2-ylcarbamoyl)pyrrolidine-1-carbonyl)-15-(4-aminobutyl)-2...More data for this Ligand-Target Pair
TargetTelomeric repeat-binding factor 2(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 240nMAssay Description:Displacement of 5-((2R,6S,9S,12S,15S,18S,21S,24S)-3-((S)-2-((S)-1-amino-3-methyl-1-oxobutan-2-ylcarbamoyl)pyrrolidine-1-carbonyl)-15-(4-aminobutyl)-2...More data for this Ligand-Target Pair
TargetTelomeric repeat-binding factor 2(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 330nMAssay Description:Binding affinity to TRFH domain of TRF2 (residues 42 to 245) (unknown origin) by FP based assayMore data for this Ligand-Target Pair
TargetTelomeric repeat-binding factor 2(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 340nMAssay Description:Displacement of 5-((2R,6S,9S,12S,15S,18S,21S,24S)-3-((S)-2-((S)-1-amino-3-methyl-1-oxobutan-2-ylcarbamoyl)pyrrolidine-1-carbonyl)-15-(4-aminobutyl)-2...More data for this Ligand-Target Pair
TargetTelomeric repeat-binding factor 2(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 380nMAssay Description:Displacement of 5-((2R,6S,9S,12S,15S,18S,21S,24S)-3-((S)-2-((S)-1-amino-3-methyl-1-oxobutan-2-ylcarbamoyl)pyrrolidine-1-carbonyl)-15-(4-aminobutyl)-2...More data for this Ligand-Target Pair
TargetTelomeric repeat-binding factor 2(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 510nMAssay Description:Displacement of 5-((2R,6S,9S,12S,15S,18S,21S,24S)-3-((S)-2-((S)-1-amino-3-methyl-1-oxobutan-2-ylcarbamoyl)pyrrolidine-1-carbonyl)-15-(4-aminobutyl)-2...More data for this Ligand-Target Pair
TargetTelomeric repeat-binding factor 2(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 720nMAssay Description:Displacement of 5-((2R,6S,9S,12S,15S,18S,21S,24S)-3-((S)-2-((S)-1-amino-3-methyl-1-oxobutan-2-ylcarbamoyl)pyrrolidine-1-carbonyl)-15-(4-aminobutyl)-2...More data for this Ligand-Target Pair
TargetTelomeric repeat-binding factor 2(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 1.40E+3nMAssay Description:Displacement of 5-((2R,6S,9S,12S,15S,18S,21S,24S)-3-((S)-2-((S)-1-amino-3-methyl-1-oxobutan-2-ylcarbamoyl)pyrrolidine-1-carbonyl)-15-(4-aminobutyl)-2...More data for this Ligand-Target Pair
TargetTelomeric repeat-binding factor 2(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 1.89E+3nMAssay Description:Displacement of 5-((2R,6S,9S,12S,15S,18S,21S,24S)-3-((S)-2-((S)-1-amino-3-methyl-1-oxobutan-2-ylcarbamoyl)pyrrolidine-1-carbonyl)-15-(4-aminobutyl)-2...More data for this Ligand-Target Pair
TargetTelomeric repeat-binding factor 2(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 2.20E+3nMAssay Description:Displacement of 5-((2R,6S,9S,12S,15S,18S,21S,24S)-3-((S)-2-((S)-1-amino-3-methyl-1-oxobutan-2-ylcarbamoyl)pyrrolidine-1-carbonyl)-15-(4-aminobutyl)-2...More data for this Ligand-Target Pair
TargetTelomeric repeat-binding factor 2(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 3.20E+3nMAssay Description:Displacement of 5-((2R,6S,9S,12S,15S,18S,21S,24S)-3-((S)-2-((S)-1-amino-3-methyl-1-oxobutan-2-ylcarbamoyl)pyrrolidine-1-carbonyl)-15-(4-aminobutyl)-2...More data for this Ligand-Target Pair
TargetTelomeric repeat-binding factor 2(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 3.40E+3nMAssay Description:Displacement of 5-((2R,6S,9S,12S,15S,18S,21S,24S)-3-((S)-2-((S)-1-amino-3-methyl-1-oxobutan-2-ylcarbamoyl)pyrrolidine-1-carbonyl)-15-(4-aminobutyl)-2...More data for this Ligand-Target Pair
TargetTelomeric repeat-binding factor 2(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 4.20E+3nMAssay Description:Binding affinity to TRFH domain of TRF2 (residues 42 to 245) (unknown origin) by FP based assayMore data for this Ligand-Target Pair
TargetTelomeric repeat-binding factor 2(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 4.30E+3nMAssay Description:Binding affinity to TRFH domain of TRF2 (residues 42 to 245) (unknown origin) by FP based assayMore data for this Ligand-Target Pair
TargetTelomeric repeat-binding factor 2(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 4.70E+3nMAssay Description:Displacement of 5-((2R,6S,9S,12S,15S,18S,21S,24S)-3-((S)-2-((S)-1-amino-3-methyl-1-oxobutan-2-ylcarbamoyl)pyrrolidine-1-carbonyl)-15-(4-aminobutyl)-2...More data for this Ligand-Target Pair
TargetTelomeric repeat-binding factor 2(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 4.90E+3nMAssay Description:Binding affinity to TRFH domain of TRF2 (residues 42 to 245) (unknown origin) by FP based assayMore data for this Ligand-Target Pair
TargetTelomeric repeat-binding factor 2(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 5.10E+3nMAssay Description:Binding affinity to TRFH domain of TRF2 (residues 42 to 245) (unknown origin) by FP based assayMore data for this Ligand-Target Pair
TargetTelomeric repeat-binding factor 2(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 5.20E+3nMAssay Description:Binding affinity to TRFH domain of TRF2 (residues 42 to 245) (unknown origin) by FP based assayMore data for this Ligand-Target Pair
TargetTelomeric repeat-binding factor 2(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 6.10E+3nMAssay Description:Displacement of 5-((2R,6S,9S,12S,15S,18S,21S,24S)-3-((S)-2-((S)-1-amino-3-methyl-1-oxobutan-2-ylcarbamoyl)pyrrolidine-1-carbonyl)-15-(4-aminobutyl)-2...More data for this Ligand-Target Pair
TargetTelomeric repeat-binding factor 2(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 6.90E+3nMAssay Description:Binding affinity to TRFH domain of TRF2 (residues 42 to 245) (unknown origin) by FP based assayMore data for this Ligand-Target Pair
TargetTelomeric repeat-binding factor 2(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 8.50E+3nMAssay Description:Displacement of 5-((2R,6S,9S,12S,15S,18S,21S,24S)-3-((S)-2-((S)-1-amino-3-methyl-1-oxobutan-2-ylcarbamoyl)pyrrolidine-1-carbonyl)-15-(4-aminobutyl)-2...More data for this Ligand-Target Pair
TargetTelomeric repeat-binding factor 2(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 8.80E+3nMAssay Description:Binding affinity to TRFH domain of TRF2 (residues 42 to 245) (unknown origin) by FP based assayMore data for this Ligand-Target Pair
TargetTelomeric repeat-binding factor 2(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 1.10E+4nMAssay Description:Binding affinity to TRFH domain of TRF2 (residues 42 to 245) (unknown origin) by FP based assayMore data for this Ligand-Target Pair
TargetTelomeric repeat-binding factor 2(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 1.12E+4nMAssay Description:Displacement of 5-((2R,6S,9S,12S,15S,18S,21S,24S)-3-((S)-2-((S)-1-amino-3-methyl-1-oxobutan-2-ylcarbamoyl)pyrrolidine-1-carbonyl)-15-(4-aminobutyl)-2...More data for this Ligand-Target Pair
TargetTelomeric repeat-binding factor 2(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 1.13E+4nMAssay Description:Displacement of 5-((2R,6S,9S,12S,15S,18S,21S,24S)-3-((S)-2-((S)-1-amino-3-methyl-1-oxobutan-2-ylcarbamoyl)pyrrolidine-1-carbonyl)-15-(4-aminobutyl)-2...More data for this Ligand-Target Pair
TargetTelomeric repeat-binding factor 2(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 1.30E+4nMAssay Description:Binding affinity to TRFH domain of TRF2 (residues 42 to 245) (unknown origin) by FP based assayMore data for this Ligand-Target Pair
TargetTelomeric repeat-binding factor 2(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 1.30E+4nMAssay Description:Binding affinity to TRFH domain of TRF2 (residues 42 to 245) (unknown origin) by FP based assayMore data for this Ligand-Target Pair
TargetTelomeric repeat-binding factor 2(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 1.40E+4nMAssay Description:Binding affinity to TRFH domain of TRF2 (residues 42 to 245) (unknown origin) by FP based assayMore data for this Ligand-Target Pair
TargetTelomeric repeat-binding factor 2(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 1.40E+4nMAssay Description:Binding affinity to TRFH domain of TRF2 (residues 42 to 245) (unknown origin) by FP based assayMore data for this Ligand-Target Pair
TargetTelomeric repeat-binding factor 2(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 1.43E+4nMAssay Description:Displacement of 5-((2R,6S,9S,12S,15S,18S,21S,24S)-3-((S)-2-((S)-1-amino-3-methyl-1-oxobutan-2-ylcarbamoyl)pyrrolidine-1-carbonyl)-15-(4-aminobutyl)-2...More data for this Ligand-Target Pair
TargetTelomeric repeat-binding factor 2(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 1.84E+4nMAssay Description:Displacement of 5-((2R,6S,9S,12S,15S,18S,21S,24S)-3-((S)-2-((S)-1-amino-3-methyl-1-oxobutan-2-ylcarbamoyl)pyrrolidine-1-carbonyl)-15-(4-aminobutyl)-2...More data for this Ligand-Target Pair
TargetTelomeric repeat-binding factor 2(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 2.00E+4nMAssay Description:Binding affinity to TRFH domain of TRF2 (residues 42 to 245) (unknown origin) by FP based assayMore data for this Ligand-Target Pair
TargetTelomeric repeat-binding factor 2(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 2.10E+4nMAssay Description:Binding affinity to TRFH domain of TRF2 (residues 42 to 245) (unknown origin) by FP based assayMore data for this Ligand-Target Pair
TargetTelomeric repeat-binding factor 2(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 2.28E+4nMAssay Description:Displacement of 5-((2R,6S,9S,12S,15S,18S,21S,24S)-3-((S)-2-((S)-1-amino-3-methyl-1-oxobutan-2-ylcarbamoyl)pyrrolidine-1-carbonyl)-15-(4-aminobutyl)-2...More data for this Ligand-Target Pair
TargetTelomeric repeat-binding factor 2(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 2.63E+4nMAssay Description:Displacement of 5-((2R,6S,9S,12S,15S,18S,21S,24S)-3-((S)-2-((S)-1-amino-3-methyl-1-oxobutan-2-ylcarbamoyl)pyrrolidine-1-carbonyl)-15-(4-aminobutyl)-2...More data for this Ligand-Target Pair
TargetTelomeric repeat-binding factor 2(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 2.68E+4nMAssay Description:Displacement of 5-((2R,6S,9S,12S,15S,18S,21S,24S)-3-((S)-2-((S)-1-amino-3-methyl-1-oxobutan-2-ylcarbamoyl)pyrrolidine-1-carbonyl)-15-(4-aminobutyl)-2...More data for this Ligand-Target Pair
TargetTelomeric repeat-binding factor 2(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 2.90E+4nMAssay Description:Binding affinity to TRFH domain of TRF2 (residues 42 to 245) (unknown origin) by FP based assayMore data for this Ligand-Target Pair
TargetTelomeric repeat-binding factor 2(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 3.00E+4nMAssay Description:Binding affinity to TRFH domain of TRF2 (residues 42 to 245) (unknown origin) by FP based assayMore data for this Ligand-Target Pair
TargetTelomeric repeat-binding factor 2(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 3.00E+4nMAssay Description:Binding affinity to TRFH domain of TRF2 (residues 42 to 245) (unknown origin) by FP based assayMore data for this Ligand-Target Pair
TargetTelomeric repeat-binding factor 2(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 3.20E+4nMAssay Description:Binding affinity to TRFH domain of TRF2 (residues 42 to 245) (unknown origin) by FP based assayMore data for this Ligand-Target Pair
TargetTelomeric repeat-binding factor 2(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 3.50E+4nMAssay Description:Binding affinity to TRFH domain of TRF2 (residues 42 to 245) (unknown origin) by FP based assayMore data for this Ligand-Target Pair
TargetTelomeric repeat-binding factor 2(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 3.90E+4nMAssay Description:Binding affinity to TRFH domain of TRF2 (residues 42 to 245) (unknown origin) by FP based assayMore data for this Ligand-Target Pair
TargetTelomeric repeat-binding factor 2(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 3.90E+4nMAssay Description:Binding affinity to TRFH domain of TRF2 (residues 42 to 245) (unknown origin) by FP based assayMore data for this Ligand-Target Pair
TargetTelomeric repeat-binding factor 2(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 3.90E+4nMAssay Description:Binding affinity to TRFH domain of TRF2 (residues 42 to 245) (unknown origin) by FP based assayMore data for this Ligand-Target Pair
TargetTelomeric repeat-binding factor 2(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 4.14E+4nMAssay Description:Displacement of 5-((2R,6S,9S,12S,15S,18S,21S,24S)-3-((S)-2-((S)-1-amino-3-methyl-1-oxobutan-2-ylcarbamoyl)pyrrolidine-1-carbonyl)-15-(4-aminobutyl)-2...More data for this Ligand-Target Pair
TargetTelomeric repeat-binding factor 2(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 4.32E+4nMAssay Description:Displacement of 5-((2R,6S,9S,12S,15S,18S,21S,24S)-3-((S)-2-((S)-1-amino-3-methyl-1-oxobutan-2-ylcarbamoyl)pyrrolidine-1-carbonyl)-15-(4-aminobutyl)-2...More data for this Ligand-Target Pair
TargetTelomeric repeat-binding factor 2(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 4.60E+4nMAssay Description:Binding affinity to TRFH domain of TRF2 (residues 42 to 245) (unknown origin) by FP based assayMore data for this Ligand-Target Pair
TargetTelomeric repeat-binding factor 2(Homo sapiens)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 5.82E+4nMAssay Description:Displacement of 5-((2R,6S,9S,12S,15S,18S,21S,24S)-3-((S)-2-((S)-1-amino-3-methyl-1-oxobutan-2-ylcarbamoyl)pyrrolidine-1-carbonyl)-15-(4-aminobutyl)-2...More data for this Ligand-Target Pair