Compile Data Set for Download or QSAR
maximum 50k data
Found 57 of ki data for polymerid = 5030
TargetXanthine dehydrogenase/oxidase(Homo sapiens (Human))
National Institute Of Pharmaceutical Education And Research

LigandPNGBDBM85771(6-(N-benzoylamino)purine, 2)
Affinity DataKi:  0.0475nM IC50:  450nMAssay Description:Inhibition assay of the xanthine oxidase reaction by various purine based inhibitors was measured in terms of the decrease in uric acid formation at ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Homo sapiens (Human))
National Institute Of Pharmaceutical Education And Research

LigandPNGBDBM50320491(2-(3-CYANO-4-ISOBUTOXY-PHENYL)-4-METHYL-5-THIAZOLE...)
Affinity DataKi:  0.100nMAssay Description:Non-competitive inhibition of human xanthine oxidaseMore data for this Ligand-Target Pair
TargetXanthine dehydrogenase/oxidase(Homo sapiens (Human))
National Institute Of Pharmaceutical Education And Research

LigandPNGBDBM50320491(2-(3-CYANO-4-ISOBUTOXY-PHENYL)-4-METHYL-5-THIAZOLE...)
Affinity DataKi:  0.100nMAssay Description:Mixed-type inhibition of xanthine oxidase (unknown origin) assessed as inhibitory constant of enzyme-substrate complex using xanthine as substrate at...More data for this Ligand-Target Pair
TargetXanthine dehydrogenase/oxidase(Homo sapiens (Human))
National Institute Of Pharmaceutical Education And Research

LigandPNGBDBM50320491(2-(3-CYANO-4-ISOBUTOXY-PHENYL)-4-METHYL-5-THIAZOLE...)
Affinity DataKi:  0.600nMAssay Description:Inhibition of xanthine oxidase (unknown origin)More data for this Ligand-Target Pair
TargetXanthine dehydrogenase/oxidase(Homo sapiens (Human))
National Institute Of Pharmaceutical Education And Research

LigandPNGBDBM50320491(2-(3-CYANO-4-ISOBUTOXY-PHENYL)-4-METHYL-5-THIAZOLE...)
Affinity DataKi:  3.10nMAssay Description:Inhibition of xanthine dehydrogenase (unknown origin)More data for this Ligand-Target Pair
TargetXanthine dehydrogenase/oxidase(Homo sapiens (Human))
National Institute Of Pharmaceutical Education And Research

LigandPNGBDBM50603070(CHEMBL5197177)
Affinity DataKi:  3.70nMAssay Description:Mixed-type inhibition of xanthine oxidase (unknown origin) assessed as inhibitory constant of enzyme-substrate complex using xanthine as substrate at...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetXanthine dehydrogenase/oxidase(Homo sapiens (Human))
National Institute Of Pharmaceutical Education And Research

LigandPNGBDBM50517021(CHEMBL4445985)
Affinity DataKi:  4.20nMAssay Description:Mixed-type inhibition of xanthine oxidase (unknown origin) assessed as inhibitory constant of enzyme-substrate complex using xanthine as substrate at...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetXanthine dehydrogenase/oxidase(Homo sapiens (Human))
National Institute Of Pharmaceutical Education And Research

LigandPNGBDBM50267750(CHEMBL1078685)
Affinity DataKi:  5.70nMAssay Description:Inhibition of xanthine oxidase (unknown origin)More data for this Ligand-Target Pair
TargetXanthine dehydrogenase/oxidase(Homo sapiens (Human))
National Institute Of Pharmaceutical Education And Research

LigandPNGBDBM50051737(2-Hexylsulfanyl-1,9-dihydro-purin-6-one | CHEMBL86...)
Affinity DataKi:  9.80nMAssay Description:Inhibitory activity against Xanthine OxidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Homo sapiens (Human))
National Institute Of Pharmaceutical Education And Research

LigandPNGBDBM50603060(CHEMBL5186383)
Affinity DataKi:  24nMAssay Description:Mixed-type inhibition of xanthine oxidase (unknown origin) assessed as inhibitory constant of enzyme-substrate complex using xanthine as substrate at...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetXanthine dehydrogenase/oxidase(Homo sapiens (Human))
National Institute Of Pharmaceutical Education And Research

LigandPNGBDBM50603046(CHEMBL5189353)
Affinity DataKi:  33nMAssay Description:Mixed-type inhibition of xanthine oxidase (unknown origin) assessed as inhibitory constant of enzyme-substrate complex using xanthine as substrate at...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetXanthine dehydrogenase/oxidase(Homo sapiens (Human))
National Institute Of Pharmaceutical Education And Research

LigandPNGBDBM50423777(OXYPURINOL | Oxipurinol)
Affinity DataKi:  35nMAssay Description:Inhibition of human xanthine oxidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Homo sapiens (Human))
National Institute Of Pharmaceutical Education And Research

LigandPNGBDBM50135279(CHEMBL3747521)
Affinity DataKi:  55nMAssay Description:Non-competitive inhibition of xanthine oxidase (unknown origin) by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Homo sapiens (Human))
National Institute Of Pharmaceutical Education And Research

LigandPNGBDBM50140241(Allopurinol | Aloral | Aluline 100 | Aluline 300 |...)
Affinity DataKi:  100nMAssay Description:Inhibition of human xanthine oxidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Homo sapiens (Human))
National Institute Of Pharmaceutical Education And Research

LigandPNGBDBM50051727(2-Pentylsulfanyl-1,9-dihydro-purin-6-one | CHEMBL8...)
Affinity DataKi:  155nMAssay Description:Inhibitory activity against Xanthine OxidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Homo sapiens (Human))
National Institute Of Pharmaceutical Education And Research

LigandPNGBDBM50051734(2-Hexylsulfanyl-8-hydroxy-1,9-dihydro-purin-6-one ...)
Affinity DataKi:  160nMAssay Description:Inhibitory activity against Xanthine OxidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Homo sapiens (Human))
National Institute Of Pharmaceutical Education And Research

LigandPNGBDBM50051711(2-Butylsulfanyl-1,9-dihydro-purin-6-one | CHEMBL84...)
Affinity DataKi:  176nMAssay Description:Inhibitory activity against Xanthine OxidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Homo sapiens (Human))
National Institute Of Pharmaceutical Education And Research

LigandPNGBDBM50051714(CHEMBL85737 | N-(5-Carbamoyl-3H-imidazol-4-yl)-oxa...)
Affinity DataKi:  260nMAssay Description:Inhibitory activity against Xanthine OxidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Homo sapiens (Human))
National Institute Of Pharmaceutical Education And Research

LigandPNGBDBM7460(2-(3,4-dihydroxyphenyl)-3,5,7-trihydroxy-4H-chrome...)
Affinity DataKi:  280nMAssay Description:Inhibition of xanthine oxidase (unknown origin) at 37 degC at ph 7..8More data for this Ligand-Target Pair
TargetXanthine dehydrogenase/oxidase(Homo sapiens (Human))
National Institute Of Pharmaceutical Education And Research

LigandPNGBDBM50051732(2-Hydroxy-7,8-dihydro-3H,6H-9-thia-1,3,4,5a-tetraa...)
Affinity DataKi:  330nMAssay Description:Inhibitory activity against Xanthine OxidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Homo sapiens (Human))
National Institute Of Pharmaceutical Education And Research

LigandPNGBDBM50051739(2-Hexylsulfanyl-8-phenyl-1,9-dihydro-purin-6-one |...)
Affinity DataKi:  490nMAssay Description:Inhibitory activity against Xanthine OxidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Homo sapiens (Human))
National Institute Of Pharmaceutical Education And Research

LigandPNGBDBM7458(5,7-dihydroxy-2-(4-hydroxyphenyl)-4H-chromen-4-one...)
Affinity DataKi:  520nMAssay Description:Inhibition of xanthine oxidase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Homo sapiens (Human))
National Institute Of Pharmaceutical Education And Research

LigandPNGBDBM50140241(Allopurinol | Aloral | Aluline 100 | Aluline 300 |...)
Affinity DataKi:  700nMAssay Description:Competitive inhibition of xanthine oxidase (unknown origin) assessed as inhibitory constant of enzyme-substrate complex using xanthine as substrate a...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetXanthine dehydrogenase/oxidase(Homo sapiens (Human))
National Institute Of Pharmaceutical Education And Research

LigandPNGBDBM50140241(Allopurinol | Aloral | Aluline 100 | Aluline 300 |...)
Affinity DataKi:  700nMAssay Description:Inhibition of xanthine oxidase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Homo sapiens (Human))
National Institute Of Pharmaceutical Education And Research

LigandPNGBDBM50051722(2-Mercapto-7,8-dihydro-3H,6H-9-thia-1,3,4,5a-tetra...)
Affinity DataKi:  890nMAssay Description:Inhibitory activity against Xanthine OxidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Homo sapiens (Human))
National Institute Of Pharmaceutical Education And Research

LigandPNGBDBM50423777(OXYPURINOL | Oxipurinol)
Affinity DataKi:  1.00E+3nMAssay Description:Inhibition of oxidized form of human xanthine oxidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Homo sapiens (Human))
National Institute Of Pharmaceutical Education And Research

LigandPNGBDBM50051710(CHEMBL83530 | N-(5-Carbamoyl-3H-imidazol-4-yl)-oxa...)
Affinity DataKi:  1.04E+3nMAssay Description:Inhibitory activity against Xanthine OxidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Homo sapiens (Human))
National Institute Of Pharmaceutical Education And Research

LigandPNGBDBM50051716(CHEMBL84643 | N-(5-Carbamoyl-3H-imidazol-4-yl)-oxa...)
Affinity DataKi:  1.06E+3nMAssay Description:Inhibitory activity against Xanthine OxidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Homo sapiens (Human))
National Institute Of Pharmaceutical Education And Research

LigandPNGBDBM50051725(2-Hydroxy-7,8-dihydro-3H-thiazolo[2,3-i]purin-5-on...)
Affinity DataKi:  1.26E+3nMAssay Description:Inhibitory activity against Xanthine OxidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Homo sapiens (Human))
National Institute Of Pharmaceutical Education And Research

LigandPNGBDBM50016784(ALLOPURINOL | BW-56-158 | BW-56158 | CHEBI:40279 |...)
Affinity DataKi:  1.55E+3nMAssay Description:Non-competitive inhibition of xanthine oxidase (unknown origin) by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetXanthine dehydrogenase/oxidase(Homo sapiens (Human))
National Institute Of Pharmaceutical Education And Research

LigandPNGBDBM50051740(2-Mercapto-7,8-dihydro-3H-thiazolo[2,3-i]purin-5-o...)
Affinity DataKi:  1.86E+3nMAssay Description:Inhibitory activity against Xanthine OxidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Homo sapiens (Human))
National Institute Of Pharmaceutical Education And Research

LigandPNGBDBM50051712(2-Mercapto-8-phenyl-1,9-dihydro-purin-6-one | CHEM...)
Affinity DataKi:  2.07E+3nMAssay Description:Inhibitory activity against Xanthine OxidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Homo sapiens (Human))
National Institute Of Pharmaceutical Education And Research

LigandPNGBDBM50051738(5-Hexanoylamino-1H-imidazole-4-carboxylic acid ami...)
Affinity DataKi:  2.56E+3nMAssay Description:Inhibitory activity against Xanthine OxidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Homo sapiens (Human))
National Institute Of Pharmaceutical Education And Research

LigandPNGBDBM50460206(CHEMBL4228510)
Affinity DataKi:  2.89E+3nMAssay Description:Competitive inhibition of Xanthine oxidase (unknown origin) using xanthine as substrate preincubated for 1 to 5 mins followed by substrate addition b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Homo sapiens (Human))
National Institute Of Pharmaceutical Education And Research

LigandPNGBDBM7459(2-(3,4-dihydroxyphenyl)-5,7-dihydroxy-4H-chromen-4...)
Affinity DataKi:  2.90E+3nMAssay Description:Inhibition of xanthine oxidase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Homo sapiens (Human))
National Institute Of Pharmaceutical Education And Research

LigandPNGBDBM50233808(CHEMBL4086701 | US11021454, Compound 6e)
Affinity DataKi:  3.43E+3nMAssay Description:Mixed-type competitive inhibition of Xanthine oxidase (unknown origin) assessed as enzyme-inhibitor complex preincubated for 3 mins followed by xanth...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Homo sapiens (Human))
National Institute Of Pharmaceutical Education And Research

LigandPNGBDBM50051713(2-Benzylsulfanyl-8-hydroxy-1,9-dihydro-purin-6-one...)
Affinity DataKi:  4.49E+3nMAssay Description:Inhibitory activity against Xanthine OxidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Homo sapiens (Human))
National Institute Of Pharmaceutical Education And Research

LigandPNGBDBM50051731(2-Methylsulfanyl-8-phenyl-1,9-dihydro-purin-6-one ...)
Affinity DataKi:  5.70E+3nMAssay Description:Inhibitory activity against Xanthine OxidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Homo sapiens (Human))
National Institute Of Pharmaceutical Education And Research

LigandPNGBDBM35440(ALLOPURINOL | MLS000069453 | SMR000059083 | cid_20...)
Affinity DataKi:  7.00E+3nMAssay Description:Inhibitory activity against Xanthine OxidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Homo sapiens (Human))
National Institute Of Pharmaceutical Education And Research

LigandPNGBDBM50016784(ALLOPURINOL | BW-56-158 | BW-56158 | CHEBI:40279 |...)
Affinity DataKi:  7.30E+3nMAssay Description:Inhibition of xanthine oxidase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetXanthine dehydrogenase/oxidase(Homo sapiens (Human))
National Institute Of Pharmaceutical Education And Research

LigandPNGBDBM50269378(CHEMBL447311 | apigenin-4'-O-(2''-O-p-coumaroyl)-b...)
Affinity DataKi:  1.44E+4nMAssay Description:Inhibition of xanthine oxidase (unknown origin) by competitive Lineweaver-burk plotMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Homo sapiens (Human))
National Institute Of Pharmaceutical Education And Research

LigandPNGBDBM50013097(2-Butylamino-1,9-dihydro-purin-6-one | 2-Butylamin...)
Affinity DataKi:  1.77E+4nMAssay Description:Inhibitory activity against Xanthine OxidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Homo sapiens (Human))
National Institute Of Pharmaceutical Education And Research

LigandPNGBDBM50051726(2-Mercapto-6,7-dihydro-3H-thiazolo[3,2-a]purin-9-o...)
Affinity DataKi:  2.44E+4nMAssay Description:Inhibitory activity against Xanthine OxidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Homo sapiens (Human))
National Institute Of Pharmaceutical Education And Research

LigandPNGBDBM50051743(2-Pentylamino-1,9-dihydro-purin-6-one | CHEMBL8431...)
Affinity DataKi:  2.57E+4nMAssay Description:Inhibitory activity against Xanthine OxidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Homo sapiens (Human))
National Institute Of Pharmaceutical Education And Research

LigandPNGBDBM50330722(2-(2-chlorophenyl)-4-methyl-5-(pyridin-2-ylmethyl)...)
Affinity DataKi: >3.00E+4nMAssay Description:Inhibition of xanthine oxidase by invitro enzymatic assay in presence of xanthineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Homo sapiens (Human))
National Institute Of Pharmaceutical Education And Research

LigandPNGBDBM50359523(CHEMBL1927147)
Affinity DataKi: >3.00E+4nMAssay Description:Inhibition of xanthine oxidase assessed as inhibition of ROS production after 20 mins by cell-free amplex red assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Homo sapiens (Human))
National Institute Of Pharmaceutical Education And Research

LigandPNGBDBM50330688(4-methyl-2-phenyl-5-(pyridin-3-ylmethyl)-1H-pyrazo...)
Affinity DataKi: >3.00E+4nMAssay Description:Inhibition of xanthine oxidase by invitro enzymatic assay in presence of xanthineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Homo sapiens (Human))
National Institute Of Pharmaceutical Education And Research

LigandPNGBDBM50013077(2-Hexylamino-1,9-dihydro-purin-6-one | 2-Hexylamin...)
Affinity DataKi:  3.21E+4nMAssay Description:Inhibitory activity against Xanthine OxidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Homo sapiens (Human))
National Institute Of Pharmaceutical Education And Research

LigandPNGBDBM50051719(2-Hydroxy-6,7-dihydro-3H-thiazolo[3,2-a]purin-9-on...)
Affinity DataKi:  4.03E+4nMAssay Description:Inhibitory activity against Xanthine OxidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Homo sapiens (Human))
National Institute Of Pharmaceutical Education And Research

LigandPNGBDBM50051715(2-Hydroxy-7,8-dihydro-3H,6H-5-thia-1,3,4,8a-tetraa...)
Affinity DataKi:  6.68E+4nMAssay Description:Inhibitory activity against Xanthine OxidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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