Compile Data Set for Download or QSAR
maximum 50k data
Found 8 of ki for UniProtKB: Q8RLA6
TargetOxa40(Acinetobacter baumannii)
Case Western Reserve University

LigandPNGBDBM227598(Penem 1)
Affinity DataKi:  30nM IC50:  150nMpH: 7.2Assay Description:Steady-state kinetics were performed on an Agilent 8453 diode array spectrophotometer (Palo Alto, CA) in 50 mM sodium phosphate buffer (pH 7.2) suppl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOxa40(Acinetobacter baumannii)
Case Western Reserve University

LigandPNGBDBM227599(Penem 3)
Affinity DataKi:  150nM IC50:  160nMpH: 7.2Assay Description:Steady-state kinetics were performed on an Agilent 8453 diode array spectrophotometer (Palo Alto, CA) in 50 mM sodium phosphate buffer (pH 7.2) suppl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOxa40(Acinetobacter baumannii)
Case Western Reserve University

LigandPNGBDBM92463(Imipenem)
Affinity DataKi:  3.20E+3nMAssay Description:Beta-lactam compounds were assessed as competitive inhibitors using nitrocefin as a reporter substrate.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOxa40(Acinetobacter baumannii)
Case Western Reserve University

LigandPNGBDBM50140672((2S,5R,6R)-6-Hydroxymethyl-3,3-dimethyl-7-oxo-4-th...)
Affinity DataKi:  3.00E+4nMAssay Description:Beta-lactam compounds were assessed as competitive inhibitors using nitrocefin as a reporter substrate.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxa40(Acinetobacter baumannii)
Case Western Reserve University

LigandPNGBDBM92461(Beta-lactam compound, 4)
Affinity DataKi:  4.20E+4nMAssay Description:Beta-lactam compounds were assessed as competitive inhibitors using nitrocefin as a reporter substrate.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxa40(Acinetobacter baumannii)
Case Western Reserve University

LigandPNGBDBM92464(Carbenicillin)
Affinity DataKi:  7.80E+4nMAssay Description:Beta-lactam compounds were assessed as competitive inhibitors using nitrocefin as a reporter substrate.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxa40(Acinetobacter baumannii)
Case Western Reserve University

LigandPNGBDBM50140671((2S,5R,6S)-6-Hydroxymethyl-3,3-dimethyl-7-oxo-4-th...)
Affinity DataKi:  8.30E+4nMAssay Description:Beta-lactam compounds were assessed as competitive inhibitors using nitrocefin as a reporter substrate.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxa40(Acinetobacter baumannii)
Case Western Reserve University

LigandPNGBDBM92462(Beta-lactam compound, 3)
Affinity DataKi:  4.04E+5nMAssay Description:Beta-lactam compounds were assessed as competitive inhibitors using nitrocefin as a reporter substrate.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed