TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
Roche Innovation Center Basel
Curated by ChEMBL
Roche Innovation Center Basel
Curated by ChEMBL
Affinity DataEC50: 0.600nMAssay Description:Agonist activity at rat TAAR1 expressed in recombinant HEK293 cells assessed as cAMP accumulation after 30 mins by luminometerMore data for this Ligand-Target Pair
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
Roche Innovation Center Basel
Curated by ChEMBL
Roche Innovation Center Basel
Curated by ChEMBL
Affinity DataEC50: 1nMAssay Description:Agonist activity at rat TAAR1 expressed in recombinant HEK293 cells assessed as cAMP accumulation after 30 mins by luminometerMore data for this Ligand-Target Pair
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
Roche Innovation Center Basel
Curated by ChEMBL
Roche Innovation Center Basel
Curated by ChEMBL
Affinity DataEC50: 1nMAssay Description:Agonist activity at rat TAAR1 expressed in recombinant HEK293 cells assessed as cAMP accumulation after 30 mins by luminometerMore data for this Ligand-Target Pair
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
Roche Innovation Center Basel
Curated by ChEMBL
Roche Innovation Center Basel
Curated by ChEMBL
Affinity DataEC50: 2.40nMAssay Description:Activity at rat TAAR1 by measuring cAMP accumulation in HEK293 cellsMore data for this Ligand-Target Pair
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
Roche Innovation Center Basel
Curated by ChEMBL
Roche Innovation Center Basel
Curated by ChEMBL
Affinity DataEC50: 2.70nMAssay Description:Activity at rat TAAR1 by measuring cAMP accumulation in HEK293 cellsMore data for this Ligand-Target Pair
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
Roche Innovation Center Basel
Curated by ChEMBL
Roche Innovation Center Basel
Curated by ChEMBL
Affinity DataEC50: 7.30nMAssay Description:Agonist activity at rat TAAR1 receptor expressed in HEK293 cells after 30 minsMore data for this Ligand-Target Pair
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
Roche Innovation Center Basel
Curated by ChEMBL
Roche Innovation Center Basel
Curated by ChEMBL
Affinity DataEC50: 8nMAssay Description:Agonist activity at rat TAAR1 expressed in recombinant HEK293 cells assessed as cAMP accumulation after 30 mins by luminometerMore data for this Ligand-Target Pair
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
Roche Innovation Center Basel
Curated by ChEMBL
Roche Innovation Center Basel
Curated by ChEMBL
Affinity DataEC50: 14nMAssay Description:Activation of rat TAAR1 transmembrane domain 7 Asn287(7.39)Tyr mutant expressed in HEK293 cells assessed as stimulation of cAMP production after 1 hr...More data for this Ligand-Target Pair
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
Roche Innovation Center Basel
Curated by ChEMBL
Roche Innovation Center Basel
Curated by ChEMBL
Affinity DataEC50: 14nMAssay Description:Agonist activity at rat TAAR1 expressed in recombinant HEK293 cells assessed as cAMP accumulation after 30 mins by luminometerMore data for this Ligand-Target Pair
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
Roche Innovation Center Basel
Curated by ChEMBL
Roche Innovation Center Basel
Curated by ChEMBL
Affinity DataEC50: 18nMAssay Description:Agonist activity at rat TAAR1 expressed in recombinant HEK293 cells assessed as cAMP accumulation after 30 mins by luminometerMore data for this Ligand-Target Pair
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
Roche Innovation Center Basel
Curated by ChEMBL
Roche Innovation Center Basel
Curated by ChEMBL
Affinity DataEC50: 18nMAssay Description:Activity at rat TAAR1 by measuring cAMP accumulation in HEK293 cellsMore data for this Ligand-Target Pair
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
Roche Innovation Center Basel
Curated by ChEMBL
Roche Innovation Center Basel
Curated by ChEMBL
Affinity DataEC50: 19nMAssay Description:Activity at rat TAAR1 expressed in HEK293 cells assessed as cAMP productionMore data for this Ligand-Target Pair
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
Roche Innovation Center Basel
Curated by ChEMBL
Roche Innovation Center Basel
Curated by ChEMBL
Affinity DataEC50: 22.4nMAssay Description:Activation of rat TAAR1 expressed in Syrian hamster AV12-664 cells assessed as accumulation of cAMP after 30 mins using cAMP XS EA/CL as substrate by...More data for this Ligand-Target Pair
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
Roche Innovation Center Basel
Curated by ChEMBL
Roche Innovation Center Basel
Curated by ChEMBL
Affinity DataEC50: 25nMAssay Description:Agonist activity at rat TAAR1 receptor expressed in HEK293 cells after 30 minsMore data for this Ligand-Target Pair
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
Roche Innovation Center Basel
Curated by ChEMBL
Roche Innovation Center Basel
Curated by ChEMBL
Affinity DataEC50: 25nMAssay Description:Agonist activity at rat TAAR1 receptor expressed in HEK293 cells after 30 minsMore data for this Ligand-Target Pair
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
Roche Innovation Center Basel
Curated by ChEMBL
Roche Innovation Center Basel
Curated by ChEMBL
Affinity DataEC50: 26nMAssay Description:Activity at rat TAAR1 expressed in HEK293 cells assessed as cAMP productionMore data for this Ligand-Target Pair
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
Roche Innovation Center Basel
Curated by ChEMBL
Roche Innovation Center Basel
Curated by ChEMBL
Affinity DataEC50: 27nMAssay Description:Agonist activity at rat TAAR1 receptor expressed in HEK293 cells after 30 minsMore data for this Ligand-Target Pair
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
Roche Innovation Center Basel
Curated by ChEMBL
Roche Innovation Center Basel
Curated by ChEMBL
Affinity DataEC50: 28nMAssay Description:Activity at rat TAAR1 expressed in HEK293 cells assessed as cAMP productionMore data for this Ligand-Target Pair
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
Roche Innovation Center Basel
Curated by ChEMBL
Roche Innovation Center Basel
Curated by ChEMBL
Affinity DataEC50: 29nMAssay Description:Agonist activity at rat TAAR1 expressed in recombinant HEK293 cells assessed as cAMP accumulation after 30 mins by luminometerMore data for this Ligand-Target Pair
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
Roche Innovation Center Basel
Curated by ChEMBL
Roche Innovation Center Basel
Curated by ChEMBL
Affinity DataEC50: 30nMAssay Description:Agonist activity at rat TAAR1 stably expressed in HEK293 cells incubated for 30 mins by cAMP assayMore data for this Ligand-Target Pair
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
Roche Innovation Center Basel
Curated by ChEMBL
Roche Innovation Center Basel
Curated by ChEMBL
Affinity DataEC50: 33nMAssay Description:Antagonist activity at rat TAAR1 expressed in HEK293 cells assessed as intracellular cAMP levelMore data for this Ligand-Target Pair
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
Roche Innovation Center Basel
Curated by ChEMBL
Roche Innovation Center Basel
Curated by ChEMBL
Affinity DataEC50: 33nMAssay Description:Antagonist activity at rat TAAR1 expressed in HEK293 cells assessed as intracellular cAMP levelMore data for this Ligand-Target Pair
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
Roche Innovation Center Basel
Curated by ChEMBL
Roche Innovation Center Basel
Curated by ChEMBL
Affinity DataEC50: 33nMAssay Description:Antagonist activity at rat TAAR1 expressed in HEK293 cells assessed as intracellular cAMP levelMore data for this Ligand-Target Pair
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
Roche Innovation Center Basel
Curated by ChEMBL
Roche Innovation Center Basel
Curated by ChEMBL
Affinity DataEC50: 33nMAssay Description:Antagonist activity at rat TAAR1 expressed in HEK293 cells assessed as intracellular cAMP levelMore data for this Ligand-Target Pair
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
Roche Innovation Center Basel
Curated by ChEMBL
Roche Innovation Center Basel
Curated by ChEMBL
Affinity DataEC50: 33nMAssay Description:Activity at rat TAAR1 expressed in HEK293 cells assessed as cAMP productionMore data for this Ligand-Target Pair
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
Roche Innovation Center Basel
Curated by ChEMBL
Roche Innovation Center Basel
Curated by ChEMBL
Affinity DataEC50: 33nMAssay Description:Activity at rat TAAR1 by measuring cAMP accumulation in HEK293 cellsMore data for this Ligand-Target Pair
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
Roche Innovation Center Basel
Curated by ChEMBL
Roche Innovation Center Basel
Curated by ChEMBL
Affinity DataEC50: 33nMAssay Description:Antagonist activity at rat TAAR1 expressed in HEK293 cells assessed as intracellular cAMP levelMore data for this Ligand-Target Pair
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
Roche Innovation Center Basel
Curated by ChEMBL
Roche Innovation Center Basel
Curated by ChEMBL
Affinity DataEC50: 34nMAssay Description:Activation of rat wild type TAAR1 expressed in HEK293 cells assessed as stimulation of cAMP production after 1 hr by chemiluminescent assayMore data for this Ligand-Target Pair
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
Roche Innovation Center Basel
Curated by ChEMBL
Roche Innovation Center Basel
Curated by ChEMBL
Affinity DataEC50: 35nMAssay Description:Agonist activity at rat TAAR1 expressed in recombinant HEK293 cells assessed as cAMP accumulation after 30 mins by luminometerMore data for this Ligand-Target Pair
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
Roche Innovation Center Basel
Curated by ChEMBL
Roche Innovation Center Basel
Curated by ChEMBL
Affinity DataEC50: 38nMAssay Description:Activity at rat TAAR1 by measuring cAMP accumulation in HEK293 cellsMore data for this Ligand-Target Pair
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
Roche Innovation Center Basel
Curated by ChEMBL
Roche Innovation Center Basel
Curated by ChEMBL
Affinity DataEC50: 40nMAssay Description:Activation of rat wild type TAAR1 expressed in HEK293 cells assessed as stimulation of cAMP production after 1 hr by chemiluminescent assayMore data for this Ligand-Target Pair
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
Roche Innovation Center Basel
Curated by ChEMBL
Roche Innovation Center Basel
Curated by ChEMBL
Affinity DataEC50: 41nMAssay Description:Activity at rat TAAR1 by measuring cAMP accumulation in HEK293 cellsMore data for this Ligand-Target Pair
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
Roche Innovation Center Basel
Curated by ChEMBL
Roche Innovation Center Basel
Curated by ChEMBL
Affinity DataEC50: 41nMAssay Description:Activity at rat TAAR1 expressed in HEK293 cells assessed as cAMP productionMore data for this Ligand-Target Pair
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
Roche Innovation Center Basel
Curated by ChEMBL
Roche Innovation Center Basel
Curated by ChEMBL
Affinity DataEC50: 43nMAssay Description:Activity at rat TAAR1 by measuring cAMP accumulation in HEK293 cellsMore data for this Ligand-Target Pair
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
Roche Innovation Center Basel
Curated by ChEMBL
Roche Innovation Center Basel
Curated by ChEMBL
Affinity DataEC50: 50nMAssay Description:Activation of rat TAAR1 expressed in HEK293 cells assessed as accumulation of [3H]cAMP after 1 hr by competitive binding assayMore data for this Ligand-Target Pair
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
Roche Innovation Center Basel
Curated by ChEMBL
Roche Innovation Center Basel
Curated by ChEMBL
Affinity DataEC50: 51nMAssay Description:Compound was evaluated for the binding affinity of Opioid receptor mu 1 by displacing the radioligand [3H]DAMGO from rat brain membraneMore data for this Ligand-Target Pair
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
Roche Innovation Center Basel
Curated by ChEMBL
Roche Innovation Center Basel
Curated by ChEMBL
Affinity DataEC50: 52nMAssay Description:Agonist activity at rat TAAR1 expressed in recombinant HEK293 cells assessed as cAMP accumulation after 30 mins by luminometerMore data for this Ligand-Target Pair
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
Roche Innovation Center Basel
Curated by ChEMBL
Roche Innovation Center Basel
Curated by ChEMBL
Affinity DataEC50: 52nMAssay Description:Activity at rat TAAR1 expressed in HEK293 cells assessed as cAMP productionMore data for this Ligand-Target Pair
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
Roche Innovation Center Basel
Curated by ChEMBL
Roche Innovation Center Basel
Curated by ChEMBL
Affinity DataEC50: 55nMAssay Description:Activity at rat TAAR1 by measuring cAMP accumulation in HEK293 cellsMore data for this Ligand-Target Pair
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
Roche Innovation Center Basel
Curated by ChEMBL
Roche Innovation Center Basel
Curated by ChEMBL
Affinity DataEC50: 56nMAssay Description:Activation of rat wild type TAAR1 expressed in HEK293 cells assessed as stimulation of cAMP production after 1 hr by chemiluminescent assayMore data for this Ligand-Target Pair
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
Roche Innovation Center Basel
Curated by ChEMBL
Roche Innovation Center Basel
Curated by ChEMBL
Affinity DataEC50: 56nMAssay Description:Activity at rat TAAR1 by measuring cAMP accumulation in HEK293 cellsMore data for this Ligand-Target Pair
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
Roche Innovation Center Basel
Curated by ChEMBL
Roche Innovation Center Basel
Curated by ChEMBL
Affinity DataEC50: 60nMAssay Description:Activation of rat TAAR1 expressed in HEK293 cells assessed as accumulation of [3H]cAMP after 1 hr by liquid scintillation countingMore data for this Ligand-Target Pair
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
Roche Innovation Center Basel
Curated by ChEMBL
Roche Innovation Center Basel
Curated by ChEMBL
Affinity DataEC50: 61nMAssay Description:Activity at rat TAAR1 by measuring cAMP accumulation in HEK293 cellsMore data for this Ligand-Target Pair
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
Roche Innovation Center Basel
Curated by ChEMBL
Roche Innovation Center Basel
Curated by ChEMBL
Affinity DataEC50: 61nMAssay Description:Agonist activity at rat TAAR1 receptor expressed in HEK293 cells after 30 minsMore data for this Ligand-Target Pair
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
Roche Innovation Center Basel
Curated by ChEMBL
Roche Innovation Center Basel
Curated by ChEMBL
Affinity DataEC50: 62nMAssay Description:Activity at rat TAAR1 expressed in HEK293 cells assessed as cAMP productionMore data for this Ligand-Target Pair
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
Roche Innovation Center Basel
Curated by ChEMBL
Roche Innovation Center Basel
Curated by ChEMBL
Affinity DataEC50: 63nMAssay Description:Agonist activity at rat TAAR1 expressed in recombinant HEK293 cells assessed as cAMP accumulation after 30 mins by luminometerMore data for this Ligand-Target Pair
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
Roche Innovation Center Basel
Curated by ChEMBL
Roche Innovation Center Basel
Curated by ChEMBL
Affinity DataEC50: 63nMAssay Description:Activity at rat TAAR1 expressed in HEK293 cells assessed as cAMP productionMore data for this Ligand-Target Pair
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
Roche Innovation Center Basel
Curated by ChEMBL
Roche Innovation Center Basel
Curated by ChEMBL
Affinity DataEC50: 64nMAssay Description:Activity at rat TAAR1 by measuring cAMP accumulation in HEK293 cellsMore data for this Ligand-Target Pair
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
Roche Innovation Center Basel
Curated by ChEMBL
Roche Innovation Center Basel
Curated by ChEMBL
Affinity DataEC50: 68nMAssay Description:Activity at rat TAAR1 by measuring cAMP accumulation in HEK293 cellsMore data for this Ligand-Target Pair
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
Roche Innovation Center Basel
Curated by ChEMBL
Roche Innovation Center Basel
Curated by ChEMBL
Affinity DataEC50: 69nMAssay Description:Agonist activity at rat N-terminal FLAG-tagged TAAR1 expressed in HEK293 cells assessed as [3H]cAMP accumulation measured after 1 hrMore data for this Ligand-Target Pair