Compile Data Set for Download or QSAR
maximum 50k data
Found 348 Enz. Inhib. hit(s) with all data for entry = 5880
TargetActivated CDC42 kinase 1(Homo sapiens (Human))
Osi Pharmaceuticals

US Patent
LigandPNGBDBM98411(US8481733, 223)
Affinity DataIC50:  30nMAssay Description:AlphaScreen (amplified luminescent proximity homogeneous assay) assay was used to test for ACK1 inhibitory activity.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetActivated CDC42 kinase 1(Homo sapiens (Human))
Osi Pharmaceuticals

US Patent
LigandPNGBDBM98237(US8481733, 49)
Affinity DataIC50:  35.2nMAssay Description:AlphaScreen (amplified luminescent proximity homogeneous assay) assay was used to test for ACK1 inhibitory activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetActivated CDC42 kinase 1(Homo sapiens (Human))
Osi Pharmaceuticals

US Patent
LigandPNGBDBM98449(US8481733, 261)
Affinity DataIC50:  36.9nMAssay Description:AlphaScreen (amplified luminescent proximity homogeneous assay) assay was used to test for ACK1 inhibitory activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetActivated CDC42 kinase 1(Homo sapiens (Human))
Osi Pharmaceuticals

US Patent
LigandPNGBDBM98341(US8481733, 219)
Affinity DataIC50:  43.9nMAssay Description:AlphaScreen (amplified luminescent proximity homogeneous assay) assay was used to test for ACK1 inhibitory activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetActivated CDC42 kinase 1(Homo sapiens (Human))
Osi Pharmaceuticals

US Patent
LigandPNGBDBM98208(US8481733, 20)
Affinity DataIC50:  48.7nMAssay Description:AlphaScreen (amplified luminescent proximity homogeneous assay) assay was used to test for ACK1 inhibitory activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetActivated CDC42 kinase 1(Homo sapiens (Human))
Osi Pharmaceuticals

US Patent
LigandPNGBDBM98450(US8481733, 262)
Affinity DataIC50:  50nMAssay Description:AlphaScreen (amplified luminescent proximity homogeneous assay) assay was used to test for ACK1 inhibitory activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetActivated CDC42 kinase 1(Homo sapiens (Human))
Osi Pharmaceuticals

US Patent
LigandPNGBDBM98200(US8481733, 11)
Affinity DataIC50:  50nMAssay Description:AlphaScreen (amplified luminescent proximity homogeneous assay) assay was used to test for ACK1 inhibitory activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetActivated CDC42 kinase 1(Homo sapiens (Human))
Osi Pharmaceuticals

US Patent
LigandPNGBDBM98274(US8481733, 86)
Affinity DataIC50:  58.9nMAssay Description:AlphaScreen (amplified luminescent proximity homogeneous assay) assay was used to test for ACK1 inhibitory activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetActivated CDC42 kinase 1(Homo sapiens (Human))
Osi Pharmaceuticals

US Patent
LigandPNGBDBM98238(US8481733, 50)
Affinity DataIC50:  60.4nMAssay Description:AlphaScreen (amplified luminescent proximity homogeneous assay) assay was used to test for ACK1 inhibitory activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetActivated CDC42 kinase 1(Homo sapiens (Human))
Osi Pharmaceuticals

US Patent
LigandPNGBDBM98343(US8481733, 155)
Affinity DataIC50:  66.7nMAssay Description:AlphaScreen (amplified luminescent proximity homogeneous assay) assay was used to test for ACK1 inhibitory activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetActivated CDC42 kinase 1(Homo sapiens (Human))
Osi Pharmaceuticals

US Patent
LigandPNGBDBM98260(US8481733, 72)
Affinity DataIC50:  75nMAssay Description:AlphaScreen (amplified luminescent proximity homogeneous assay) assay was used to test for ACK1 inhibitory activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetActivated CDC42 kinase 1(Homo sapiens (Human))
Osi Pharmaceuticals

US Patent
LigandPNGBDBM98426(US8481733, 238)
Affinity DataIC50:  75.1nMAssay Description:AlphaScreen (amplified luminescent proximity homogeneous assay) assay was used to test for ACK1 inhibitory activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetActivated CDC42 kinase 1(Homo sapiens (Human))
Osi Pharmaceuticals

US Patent
LigandPNGBDBM98226(US8481733, 38)
Affinity DataIC50:  86.5nMAssay Description:AlphaScreen (amplified luminescent proximity homogeneous assay) assay was used to test for ACK1 inhibitory activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetActivated CDC42 kinase 1(Homo sapiens (Human))
Osi Pharmaceuticals

US Patent
LigandPNGBDBM98209(US8481733, 21)
Affinity DataIC50:  88nMAssay Description:AlphaScreen (amplified luminescent proximity homogeneous assay) assay was used to test for ACK1 inhibitory activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetActivated CDC42 kinase 1(Homo sapiens (Human))
Osi Pharmaceuticals

US Patent
LigandPNGBDBM98297(US8481733, 109)
Affinity DataIC50:  88.6nMAssay Description:AlphaScreen (amplified luminescent proximity homogeneous assay) assay was used to test for ACK1 inhibitory activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetActivated CDC42 kinase 1(Homo sapiens (Human))
Osi Pharmaceuticals

US Patent
LigandPNGBDBM98236(US8481733, 48)
Affinity DataIC50:  90nMAssay Description:AlphaScreen (amplified luminescent proximity homogeneous assay) assay was used to test for ACK1 inhibitory activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetActivated CDC42 kinase 1(Homo sapiens (Human))
Osi Pharmaceuticals

US Patent
LigandPNGBDBM98376(US8481733, 188)
Affinity DataIC50:  95.2nMAssay Description:AlphaScreen (amplified luminescent proximity homogeneous assay) assay was used to test for ACK1 inhibitory activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetActivated CDC42 kinase 1(Homo sapiens (Human))
Osi Pharmaceuticals

US Patent
LigandPNGBDBM98195(US8481733, 6)
Affinity DataIC50:  95.8nMAssay Description:AlphaScreen (amplified luminescent proximity homogeneous assay) assay was used to test for ACK1 inhibitory activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetActivated CDC42 kinase 1(Homo sapiens (Human))
Osi Pharmaceuticals

US Patent
LigandPNGBDBM98259(US8481733, 71)
Affinity DataIC50:  100nMAssay Description:AlphaScreen (amplified luminescent proximity homogeneous assay) assay was used to test for ACK1 inhibitory activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetActivated CDC42 kinase 1(Homo sapiens (Human))
Osi Pharmaceuticals

US Patent
LigandPNGBDBM98370(US8481733, 182)
Affinity DataIC50:  109nMAssay Description:AlphaScreen (amplified luminescent proximity homogeneous assay) assay was used to test for ACK1 inhibitory activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetActivated CDC42 kinase 1(Homo sapiens (Human))
Osi Pharmaceuticals

US Patent
LigandPNGBDBM98446(US8481733, 258)
Affinity DataIC50:  110nMAssay Description:AlphaScreen (amplified luminescent proximity homogeneous assay) assay was used to test for ACK1 inhibitory activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetActivated CDC42 kinase 1(Homo sapiens (Human))
Osi Pharmaceuticals

US Patent
LigandPNGBDBM98440(US8481733, 252)
Affinity DataIC50:  112nMAssay Description:AlphaScreen (amplified luminescent proximity homogeneous assay) assay was used to test for ACK1 inhibitory activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetActivated CDC42 kinase 1(Homo sapiens (Human))
Osi Pharmaceuticals

US Patent
LigandPNGBDBM98280(US8481733, 92)
Affinity DataIC50:  115nMAssay Description:AlphaScreen (amplified luminescent proximity homogeneous assay) assay was used to test for ACK1 inhibitory activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetActivated CDC42 kinase 1(Homo sapiens (Human))
Osi Pharmaceuticals

US Patent
LigandPNGBDBM98295(US8481733, 107)
Affinity DataIC50:  117nMAssay Description:AlphaScreen (amplified luminescent proximity homogeneous assay) assay was used to test for ACK1 inhibitory activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetActivated CDC42 kinase 1(Homo sapiens (Human))
Osi Pharmaceuticals

US Patent
LigandPNGBDBM98282(US8481733, 94)
Affinity DataIC50:  119nMAssay Description:AlphaScreen (amplified luminescent proximity homogeneous assay) assay was used to test for ACK1 inhibitory activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetActivated CDC42 kinase 1(Homo sapiens (Human))
Osi Pharmaceuticals

US Patent
LigandPNGBDBM98347(US8481733, 159)
Affinity DataIC50:  122nMAssay Description:AlphaScreen (amplified luminescent proximity homogeneous assay) assay was used to test for ACK1 inhibitory activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetActivated CDC42 kinase 1(Homo sapiens (Human))
Osi Pharmaceuticals

US Patent
LigandPNGBDBM98474(US8481733, 286)
Affinity DataIC50:  136nMAssay Description:AlphaScreen (amplified luminescent proximity homogeneous assay) assay was used to test for ACK1 inhibitory activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetActivated CDC42 kinase 1(Homo sapiens (Human))
Osi Pharmaceuticals

US Patent
LigandPNGBDBM98296(US8481733, 108)
Affinity DataIC50:  137nMAssay Description:AlphaScreen (amplified luminescent proximity homogeneous assay) assay was used to test for ACK1 inhibitory activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetActivated CDC42 kinase 1(Homo sapiens (Human))
Osi Pharmaceuticals

US Patent
LigandPNGBDBM98428(US8481733, 240)
Affinity DataIC50:  139nMAssay Description:AlphaScreen (amplified luminescent proximity homogeneous assay) assay was used to test for ACK1 inhibitory activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetActivated CDC42 kinase 1(Homo sapiens (Human))
Osi Pharmaceuticals

US Patent
LigandPNGBDBM98293(US8481733, 105)
Affinity DataIC50:  140nMAssay Description:AlphaScreen (amplified luminescent proximity homogeneous assay) assay was used to test for ACK1 inhibitory activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetActivated CDC42 kinase 1(Homo sapiens (Human))
Osi Pharmaceuticals

US Patent
LigandPNGBDBM98336(US8481733, 148)
Affinity DataIC50:  145nMAssay Description:AlphaScreen (amplified luminescent proximity homogeneous assay) assay was used to test for ACK1 inhibitory activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetActivated CDC42 kinase 1(Homo sapiens (Human))
Osi Pharmaceuticals

US Patent
LigandPNGBDBM50199622(3-cyclobutyl-1-(4-phenoxyphenyl)imidazo[1,5-a]pyra...)
Affinity DataIC50:  148nMAssay Description:AlphaScreen (amplified luminescent proximity homogeneous assay) assay was used to test for ACK1 inhibitory activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetActivated CDC42 kinase 1(Homo sapiens (Human))
Osi Pharmaceuticals

US Patent
LigandPNGBDBM98199(US8481733, 10)
Affinity DataIC50:  153nMAssay Description:AlphaScreen (amplified luminescent proximity homogeneous assay) assay was used to test for ACK1 inhibitory activity.More data for this Ligand-Target Pair
TargetActivated CDC42 kinase 1(Homo sapiens (Human))
Osi Pharmaceuticals

US Patent
LigandPNGBDBM98424(US8481733, 236)
Affinity DataIC50:  154nMAssay Description:AlphaScreen (amplified luminescent proximity homogeneous assay) assay was used to test for ACK1 inhibitory activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetActivated CDC42 kinase 1(Homo sapiens (Human))
Osi Pharmaceuticals

US Patent
LigandPNGBDBM98459(US8481733, 271)
Affinity DataIC50:  176nMAssay Description:AlphaScreen (amplified luminescent proximity homogeneous assay) assay was used to test for ACK1 inhibitory activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetActivated CDC42 kinase 1(Homo sapiens (Human))
Osi Pharmaceuticals

US Patent
LigandPNGBDBM98279(US8481733, 91)
Affinity DataIC50:  178nMAssay Description:AlphaScreen (amplified luminescent proximity homogeneous assay) assay was used to test for ACK1 inhibitory activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetActivated CDC42 kinase 1(Homo sapiens (Human))
Osi Pharmaceuticals

US Patent
LigandPNGBDBM98257(US8481733, 69)
Affinity DataIC50:  181nMAssay Description:AlphaScreen (amplified luminescent proximity homogeneous assay) assay was used to test for ACK1 inhibitory activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetActivated CDC42 kinase 1(Homo sapiens (Human))
Osi Pharmaceuticals

US Patent
LigandPNGBDBM98235(US8481733, 47)
Affinity DataIC50:  181nMAssay Description:AlphaScreen (amplified luminescent proximity homogeneous assay) assay was used to test for ACK1 inhibitory activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetActivated CDC42 kinase 1(Homo sapiens (Human))
Osi Pharmaceuticals

US Patent
LigandPNGBDBM98276(US8481733, 88)
Affinity DataIC50:  183nMAssay Description:AlphaScreen (amplified luminescent proximity homogeneous assay) assay was used to test for ACK1 inhibitory activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetActivated CDC42 kinase 1(Homo sapiens (Human))
Osi Pharmaceuticals

US Patent
LigandPNGBDBM98329(US8481733, 141)
Affinity DataIC50:  183nMAssay Description:AlphaScreen (amplified luminescent proximity homogeneous assay) assay was used to test for ACK1 inhibitory activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetActivated CDC42 kinase 1(Homo sapiens (Human))
Osi Pharmaceuticals

US Patent
LigandPNGBDBM98351(US8481733, 163)
Affinity DataIC50:  188nMAssay Description:AlphaScreen (amplified luminescent proximity homogeneous assay) assay was used to test for ACK1 inhibitory activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetActivated CDC42 kinase 1(Homo sapiens (Human))
Osi Pharmaceuticals

US Patent
LigandPNGBDBM98253(US8481733, 65)
Affinity DataIC50:  188nMAssay Description:AlphaScreen (amplified luminescent proximity homogeneous assay) assay was used to test for ACK1 inhibitory activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetActivated CDC42 kinase 1(Homo sapiens (Human))
Osi Pharmaceuticals

US Patent
LigandPNGBDBM98465(US8481733, 277)
Affinity DataIC50:  197nMAssay Description:AlphaScreen (amplified luminescent proximity homogeneous assay) assay was used to test for ACK1 inhibitory activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetActivated CDC42 kinase 1(Homo sapiens (Human))
Osi Pharmaceuticals

US Patent
LigandPNGBDBM98460(US8481733, 272)
Affinity DataIC50:  199nMAssay Description:AlphaScreen (amplified luminescent proximity homogeneous assay) assay was used to test for ACK1 inhibitory activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetActivated CDC42 kinase 1(Homo sapiens (Human))
Osi Pharmaceuticals

US Patent
LigandPNGBDBM98464(US8481733, 276)
Affinity DataIC50:  201nMAssay Description:AlphaScreen (amplified luminescent proximity homogeneous assay) assay was used to test for ACK1 inhibitory activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetActivated CDC42 kinase 1(Homo sapiens (Human))
Osi Pharmaceuticals

US Patent
LigandPNGBDBM98255(US8481733, 67)
Affinity DataIC50:  203nMAssay Description:AlphaScreen (amplified luminescent proximity homogeneous assay) assay was used to test for ACK1 inhibitory activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetActivated CDC42 kinase 1(Homo sapiens (Human))
Osi Pharmaceuticals

US Patent
LigandPNGBDBM98234(US8481733, 46)
Affinity DataIC50:  205nMAssay Description:AlphaScreen (amplified luminescent proximity homogeneous assay) assay was used to test for ACK1 inhibitory activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetActivated CDC42 kinase 1(Homo sapiens (Human))
Osi Pharmaceuticals

US Patent
LigandPNGBDBM98192(US8481733, 3)
Affinity DataIC50:  212nMAssay Description:AlphaScreen (amplified luminescent proximity homogeneous assay) assay was used to test for ACK1 inhibitory activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetActivated CDC42 kinase 1(Homo sapiens (Human))
Osi Pharmaceuticals

US Patent
LigandPNGBDBM98294(US8481733, 106)
Affinity DataIC50:  216nMAssay Description:AlphaScreen (amplified luminescent proximity homogeneous assay) assay was used to test for ACK1 inhibitory activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetActivated CDC42 kinase 1(Homo sapiens (Human))
Osi Pharmaceuticals

US Patent
LigandPNGBDBM98461(US8481733, 273)
Affinity DataIC50:  216nMAssay Description:AlphaScreen (amplified luminescent proximity homogeneous assay) assay was used to test for ACK1 inhibitory activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
Displayed 1 to 50 (of 348 total ) | Next | Last >>
Jump to: