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Found 202 Enz. Inhib. hit(s) with all data for entry = 6930
TargetMelanocortin receptor 4(Homo sapiens (Human))
Astrazeneca

US Patent
LigandPNGBDBM160158(US9040663, 4)
Affinity DataKi:  0.0550nM ΔG°:  -60.9kJ/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay was performed for exemplified peptides according to the invention using membrane homogenates prepared from HEK...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Astrazeneca

US Patent
LigandPNGBDBM160159(US9040663, 5)
Affinity DataKi:  0.0550nM ΔG°:  -60.9kJ/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay was performed for exemplified peptides according to the invention using membrane homogenates prepared from HEK...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Astrazeneca

US Patent
LigandPNGBDBM160174(US9040663, 20)
Affinity DataKi:  0.0600nM ΔG°:  -60.7kJ/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay was performed for exemplified peptides according to the invention using membrane homogenates prepared from HEK...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Astrazeneca

US Patent
LigandPNGBDBM160157(US9040663, 3)
Affinity DataKi:  0.0800nM ΔG°:  -59.9kJ/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay was performed for exemplified peptides according to the invention using membrane homogenates prepared from HEK...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Astrazeneca

US Patent
LigandPNGBDBM160175(US9040663, 21)
Affinity DataKi:  0.0850nM ΔG°:  -59.8kJ/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay was performed for exemplified peptides according to the invention using membrane homogenates prepared from HEK...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Astrazeneca

US Patent
LigandPNGBDBM160169(US9040663, 15)
Affinity DataKi:  0.145nM ΔG°:  -58.4kJ/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay was performed for exemplified peptides according to the invention using membrane homogenates prepared from HEK...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Astrazeneca

US Patent
LigandPNGBDBM160170(US9040663, 16)
Affinity DataKi:  0.150nM ΔG°:  -58.3kJ/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay was performed for exemplified peptides according to the invention using membrane homogenates prepared from HEK...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Astrazeneca

US Patent
LigandPNGBDBM160159(US9040663, 5)
Affinity DataKi:  0.200nM ΔG°:  -57.6kJ/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay was performed for exemplified peptides according to the invention using membrane homogenates prepared from HEK...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Astrazeneca

US Patent
LigandPNGBDBM160165(US9040663, 11)
Affinity DataKi:  0.25nM ΔG°:  -57.0kJ/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay was performed for exemplified peptides according to the invention using membrane homogenates prepared from HEK...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Astrazeneca

US Patent
LigandPNGBDBM160208(US9040663, 54)
Affinity DataKi:  0.25nM ΔG°:  -57.0kJ/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay was performed for exemplified peptides according to the invention using membrane homogenates prepared from HEK...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Astrazeneca

US Patent
LigandPNGBDBM160170(US9040663, 16)
Affinity DataKi:  0.25nM ΔG°:  -57.0kJ/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay was performed for exemplified peptides according to the invention using membrane homogenates prepared from HEK...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Astrazeneca

US Patent
LigandPNGBDBM160180(US9040663, 26)
Affinity DataKi:  0.300nM ΔG°:  -56.5kJ/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay was performed for exemplified peptides according to the invention using membrane homogenates prepared from HEK...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Astrazeneca

US Patent
LigandPNGBDBM160201(US9040663, 47)
Affinity DataKi:  0.300nM ΔG°:  -56.5kJ/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay was performed for exemplified peptides according to the invention using membrane homogenates prepared from HEK...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Astrazeneca

US Patent
LigandPNGBDBM160157(US9040663, 3)
Affinity DataKi:  0.300nM ΔG°:  -56.5kJ/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay was performed for exemplified peptides according to the invention using membrane homogenates prepared from HEK...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Astrazeneca

US Patent
LigandPNGBDBM160217(US9040663, 63)
Affinity DataKi:  0.350nM ΔG°:  -56.1kJ/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay was performed for exemplified peptides according to the invention using membrane homogenates prepared from HEK...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Astrazeneca

US Patent
LigandPNGBDBM160173(US9040663, 19)
Affinity DataKi:  0.400nM ΔG°:  -55.8kJ/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay was performed for exemplified peptides according to the invention using membrane homogenates prepared from HEK...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Astrazeneca

US Patent
LigandPNGBDBM160178(US9040663, 24)
Affinity DataKi:  0.450nM ΔG°:  -55.5kJ/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay was performed for exemplified peptides according to the invention using membrane homogenates prepared from HEK...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Astrazeneca

US Patent
LigandPNGBDBM160165(US9040663, 11)
Affinity DataKi:  0.5nM ΔG°:  -55.2kJ/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay was performed for exemplified peptides according to the invention using membrane homogenates prepared from HEK...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Astrazeneca

US Patent
LigandPNGBDBM160158(US9040663, 4)
Affinity DataKi:  0.5nM ΔG°:  -55.2kJ/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay was performed for exemplified peptides according to the invention using membrane homogenates prepared from HEK...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Astrazeneca

US Patent
LigandPNGBDBM160183(US9040663, 29)
Affinity DataKi:  0.5nM ΔG°:  -55.2kJ/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay was performed for exemplified peptides according to the invention using membrane homogenates prepared from HEK...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Astrazeneca

US Patent
LigandPNGBDBM160172(US9040663, 18)
Affinity DataKi:  0.5nM ΔG°:  -55.2kJ/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay was performed for exemplified peptides according to the invention using membrane homogenates prepared from HEK...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Astrazeneca

US Patent
LigandPNGBDBM160253(US9040663, 99)
Affinity DataKi:  0.5nM ΔG°:  -55.2kJ/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay was performed for exemplified peptides according to the invention using membrane homogenates prepared from HEK...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Astrazeneca

US Patent
LigandPNGBDBM160167(US9040663, 13)
Affinity DataKi:  0.600nM ΔG°:  -54.8kJ/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay was performed for exemplified peptides according to the invention using membrane homogenates prepared from HEK...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Astrazeneca

US Patent
LigandPNGBDBM160206(US9040663, 52)
Affinity DataKi:  0.600nM ΔG°:  -54.8kJ/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay was performed for exemplified peptides according to the invention using membrane homogenates prepared from HEK...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Astrazeneca

US Patent
LigandPNGBDBM160205(US9040663, 51)
Affinity DataKi:  0.600nM ΔG°:  -54.8kJ/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay was performed for exemplified peptides according to the invention using membrane homogenates prepared from HEK...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Astrazeneca

US Patent
LigandPNGBDBM160211(US9040663, 57)
Affinity DataKi:  0.650nM ΔG°:  -54.5kJ/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay was performed for exemplified peptides according to the invention using membrane homogenates prepared from HEK...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Astrazeneca

US Patent
LigandPNGBDBM160181(US9040663, 27)
Affinity DataKi:  0.667nM ΔG°:  -54.5kJ/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay was performed for exemplified peptides according to the invention using membrane homogenates prepared from HEK...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Astrazeneca

US Patent
LigandPNGBDBM160177(US9040663, 23)
Affinity DataKi:  0.700nM ΔG°:  -54.4kJ/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay was performed for exemplified peptides according to the invention using membrane homogenates prepared from HEK...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Astrazeneca

US Patent
LigandPNGBDBM160208(US9040663, 54)
Affinity DataKi:  0.700nM ΔG°:  -54.4kJ/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay was performed for exemplified peptides according to the invention using membrane homogenates prepared from HEK...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Astrazeneca

US Patent
LigandPNGBDBM160163(US9040663, 9)
Affinity DataKi:  0.700nM ΔG°:  -54.4kJ/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay was performed for exemplified peptides according to the invention using membrane homogenates prepared from HEK...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Astrazeneca

US Patent
LigandPNGBDBM160252(US9040663, 98)
Affinity DataKi:  0.75nM ΔG°:  -54.2kJ/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay was performed for exemplified peptides according to the invention using membrane homogenates prepared from HEK...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Astrazeneca

US Patent
LigandPNGBDBM160169(US9040663, 15)
Affinity DataKi:  0.75nM ΔG°:  -54.2kJ/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay was performed for exemplified peptides according to the invention using membrane homogenates prepared from HEK...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Astrazeneca

US Patent
LigandPNGBDBM160156(US9040663, 2)
Affinity DataKi:  0.75nM ΔG°:  -54.2kJ/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay was performed for exemplified peptides according to the invention using membrane homogenates prepared from HEK...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Astrazeneca

US Patent
LigandPNGBDBM160251(US9040663, 97)
Affinity DataKi:  0.75nM ΔG°:  -54.2kJ/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay was performed for exemplified peptides according to the invention using membrane homogenates prepared from HEK...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Astrazeneca

US Patent
LigandPNGBDBM160207(US9040663, 53)
Affinity DataKi:  0.75nM ΔG°:  -54.2kJ/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay was performed for exemplified peptides according to the invention using membrane homogenates prepared from HEK...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Astrazeneca

US Patent
LigandPNGBDBM160163(US9040663, 9)
Affinity DataKi:  0.800nM ΔG°:  -54.0kJ/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay was performed for exemplified peptides according to the invention using membrane homogenates prepared from HEK...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Astrazeneca

US Patent
LigandPNGBDBM160161(US9040663, 7)
Affinity DataKi:  0.833nM ΔG°:  -53.9kJ/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay was performed for exemplified peptides according to the invention using membrane homogenates prepared from HEK...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Astrazeneca

US Patent
LigandPNGBDBM160248(US9040663, 94)
Affinity DataKi:  0.900nM ΔG°:  -53.7kJ/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay was performed for exemplified peptides according to the invention using membrane homogenates prepared from HEK...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Astrazeneca

US Patent
LigandPNGBDBM160168(US9040663, 14)
Affinity DataKi:  0.950nM ΔG°:  -53.6kJ/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay was performed for exemplified peptides according to the invention using membrane homogenates prepared from HEK...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Astrazeneca

US Patent
LigandPNGBDBM160207(US9040663, 53)
Affinity DataKi:  0.950nM ΔG°:  -53.6kJ/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay was performed for exemplified peptides according to the invention using membrane homogenates prepared from HEK...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Astrazeneca

US Patent
LigandPNGBDBM160156(US9040663, 2)
Affinity DataKi:  1nM ΔG°:  -53.4kJ/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay was performed for exemplified peptides according to the invention using membrane homogenates prepared from HEK...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Astrazeneca

US Patent
LigandPNGBDBM160155(US9040663, 1)
Affinity DataKi:  1nM ΔG°:  -53.4kJ/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay was performed for exemplified peptides according to the invention using membrane homogenates prepared from HEK...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Astrazeneca

US Patent
LigandPNGBDBM160255(US9040663, 101)
Affinity DataKi:  1nM ΔG°:  -53.4kJ/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay was performed for exemplified peptides according to the invention using membrane homogenates prepared from HEK...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Astrazeneca

US Patent
LigandPNGBDBM160247(US9040663, 93)
Affinity DataKi:  1nM ΔG°:  -53.4kJ/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay was performed for exemplified peptides according to the invention using membrane homogenates prepared from HEK...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Astrazeneca

US Patent
LigandPNGBDBM160214(US9040663, 60)
Affinity DataKi:  1nM ΔG°:  -53.4kJ/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay was performed for exemplified peptides according to the invention using membrane homogenates prepared from HEK...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Astrazeneca

US Patent
LigandPNGBDBM160211(US9040663, 57)
Affinity DataKi:  1nM ΔG°:  -53.4kJ/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay was performed for exemplified peptides according to the invention using membrane homogenates prepared from HEK...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Astrazeneca

US Patent
LigandPNGBDBM160187(US9040663, 33)
Affinity DataKi:  1nM ΔG°:  -53.4kJ/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay was performed for exemplified peptides according to the invention using membrane homogenates prepared from HEK...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Astrazeneca

US Patent
LigandPNGBDBM160204(US9040663, 50)
Affinity DataKi:  1nM ΔG°:  -53.4kJ/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay was performed for exemplified peptides according to the invention using membrane homogenates prepared from HEK...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Astrazeneca

US Patent
LigandPNGBDBM160171(US9040663, 17)
Affinity DataKi:  2nM ΔG°:  -51.6kJ/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay was performed for exemplified peptides according to the invention using membrane homogenates prepared from HEK...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Astrazeneca

US Patent
LigandPNGBDBM160164(US9040663, 10)
Affinity DataKi:  2nM ΔG°:  -51.6kJ/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay was performed for exemplified peptides according to the invention using membrane homogenates prepared from HEK...More data for this Ligand-Target Pair
In DepthDetails US Patent
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