Compile Data Set for Download or QSAR
maximum 50k data
Found 20 Enz. Inhib. hit(s) with all data for entry = 7516
TargetMatrix metalloproteinase-9(Rattus norvegicus (Rat))
Zhejiang Hospital

LigandPNGBDBM199123(N-(4-(1-(4,6-bis((4-hydroxyphenyl)amino)-1,3,5-tri...)
Affinity DataIC50:  2.34nMpH: 7.5 T: 2°CAssay Description:where a pro-fluorescing peptide is used as substrate, and the fluorogenic activity of its cleavage product is measured after co-incubation with the a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Rattus norvegicus (Rat))
Zhejiang Hospital

LigandPNGBDBM199123(N-(4-(1-(4,6-bis((4-hydroxyphenyl)amino)-1,3,5-tri...)
Affinity DataIC50:  8.12nMpH: 7.5 T: 2°CAssay Description:where a pro-fluorescing peptide is used as substrate, and the fluorogenic activity of its cleavage product is measured after co-incubation with the a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Rattus norvegicus (Rat))
Zhejiang Hospital

LigandPNGBDBM199124(N-(4-(1-(4,6-bis((4-methoxyphenyl)amino)-1,3,5-tri...)
Affinity DataIC50:  10.2nMpH: 7.5 T: 2°CAssay Description:where a pro-fluorescing peptide is used as substrate, and the fluorogenic activity of its cleavage product is measured after co-incubation with the a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Rattus norvegicus (Rat))
Zhejiang Hospital

LigandPNGBDBM199124(N-(4-(1-(4,6-bis((4-methoxyphenyl)amino)-1,3,5-tri...)
Affinity DataIC50:  18.6nMpH: 7.5 T: 2°CAssay Description:where a pro-fluorescing peptide is used as substrate, and the fluorogenic activity of its cleavage product is measured after co-incubation with the a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Rattus norvegicus (Rat))
Zhejiang Hospital

LigandPNGBDBM199128(N-(4-(1-(4,6-dimorpholino-1,3,5-triazin-2-yl)-5-(4...)
Affinity DataIC50:  31.2nMpH: 7.5 T: 2°CAssay Description:where a pro-fluorescing peptide is used as substrate, and the fluorogenic activity of its cleavage product is measured after co-incubation with the a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Rattus norvegicus (Rat))
Zhejiang Hospital

LigandPNGBDBM199128(N-(4-(1-(4,6-dimorpholino-1,3,5-triazin-2-yl)-5-(4...)
Affinity DataIC50:  42.3nMpH: 7.5 T: 2°CAssay Description:where a pro-fluorescing peptide is used as substrate, and the fluorogenic activity of its cleavage product is measured after co-incubation with the a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Rattus norvegicus (Rat))
Zhejiang Hospital

LigandPNGBDBM199127(N-(4-(1-(4,6-di(piperazin-1-yl)-1,3,5-triazin-2-yl...)
Affinity DataIC50:  47.1nMpH: 7.5 T: 2°CAssay Description:where a pro-fluorescing peptide is used as substrate, and the fluorogenic activity of its cleavage product is measured after co-incubation with the a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Rattus norvegicus (Rat))
Zhejiang Hospital

LigandPNGBDBM199127(N-(4-(1-(4,6-di(piperazin-1-yl)-1,3,5-triazin-2-yl...)
Affinity DataIC50:  55.3nMpH: 7.5 T: 2°CAssay Description:where a pro-fluorescing peptide is used as substrate, and the fluorogenic activity of its cleavage product is measured after co-incubation with the a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Rattus norvegicus (Rat))
Zhejiang Hospital

LigandPNGBDBM199125(N-(4-(1-(4,6-bis(o-tolylamino)-1,3,5-triazin-2-yl)...)
Affinity DataIC50:  58.2nMpH: 7.5 T: 2°CAssay Description:where a pro-fluorescing peptide is used as substrate, and the fluorogenic activity of its cleavage product is measured after co-incubation with the a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Rattus norvegicus (Rat))
Zhejiang Hospital

LigandPNGBDBM199125(N-(4-(1-(4,6-bis(o-tolylamino)-1,3,5-triazin-2-yl)...)
Affinity DataIC50:  67.1nMpH: 7.5 T: 2°CAssay Description:where a pro-fluorescing peptide is used as substrate, and the fluorogenic activity of its cleavage product is measured after co-incubation with the a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Rattus norvegicus (Rat))
Zhejiang Hospital

LigandPNGBDBM199126(N-(4-(1-(4,6-bis((4-nitrophenyl)amino)-1,3,5-triaz...)
Affinity DataIC50:  68.5nMpH: 7.5 T: 2°CAssay Description:where a pro-fluorescing peptide is used as substrate, and the fluorogenic activity of its cleavage product is measured after co-incubation with the a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Rattus norvegicus (Rat))
Zhejiang Hospital

LigandPNGBDBM199126(N-(4-(1-(4,6-bis((4-nitrophenyl)amino)-1,3,5-triaz...)
Affinity DataIC50:  76.6nMpH: 7.5 T: 2°CAssay Description:where a pro-fluorescing peptide is used as substrate, and the fluorogenic activity of its cleavage product is measured after co-incubation with the a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Rattus norvegicus (Rat))
Zhejiang Hospital

LigandPNGBDBM199122(N-(4-(1-(4,6-bis(phenylamino)-1,3,5-triazin-2-yl)-...)
Affinity DataIC50:  105nMpH: 7.5 T: 2°CAssay Description:where a pro-fluorescing peptide is used as substrate, and the fluorogenic activity of its cleavage product is measured after co-incubation with the a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Rattus norvegicus (Rat))
Zhejiang Hospital

LigandPNGBDBM199122(N-(4-(1-(4,6-bis(phenylamino)-1,3,5-triazin-2-yl)-...)
Affinity DataIC50:  123nMpH: 7.5 T: 2°CAssay Description:where a pro-fluorescing peptide is used as substrate, and the fluorogenic activity of its cleavage product is measured after co-incubation with the a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Rattus norvegicus (Rat))
Zhejiang Hospital

LigandPNGBDBM199121(N-(4-(1-(4,6-bis((3-aminopropyl)amino)-1,3,5-triaz...)
Affinity DataIC50:  156nMpH: 7.5 T: 2°CAssay Description:where a pro-fluorescing peptide is used as substrate, and the fluorogenic activity of its cleavage product is measured after co-incubation with the a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Rattus norvegicus (Rat))
Zhejiang Hospital

LigandPNGBDBM199121(N-(4-(1-(4,6-bis((3-aminopropyl)amino)-1,3,5-triaz...)
Affinity DataIC50:  189nMpH: 7.5 T: 2°CAssay Description:where a pro-fluorescing peptide is used as substrate, and the fluorogenic activity of its cleavage product is measured after co-incubation with the a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Rattus norvegicus (Rat))
Zhejiang Hospital

LigandPNGBDBM199120(N-(4-(1-(4,6-bis(ethylamino)-1,3,5-triazin-2-yl)-5...)
Affinity DataIC50:  302nMpH: 7.5 T: 2°CAssay Description:where a pro-fluorescing peptide is used as substrate, and the fluorogenic activity of its cleavage product is measured after co-incubation with the a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Rattus norvegicus (Rat))
Zhejiang Hospital

LigandPNGBDBM199120(N-(4-(1-(4,6-bis(ethylamino)-1,3,5-triazin-2-yl)-5...)
Affinity DataIC50:  332nMpH: 7.5 T: 2°CAssay Description:where a pro-fluorescing peptide is used as substrate, and the fluorogenic activity of its cleavage product is measured after co-incubation with the a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Rattus norvegicus (Rat))
Zhejiang Hospital

LigandPNGBDBM199119(N-(4-(1-(4,6-bis(methylamino)-1,3,5-triazin-2-yl)-...)
Affinity DataIC50:  625nMpH: 7.5 T: 2°CAssay Description:where a pro-fluorescing peptide is used as substrate, and the fluorogenic activity of its cleavage product is measured after co-incubation with the a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Rattus norvegicus (Rat))
Zhejiang Hospital

LigandPNGBDBM199119(N-(4-(1-(4,6-bis(methylamino)-1,3,5-triazin-2-yl)-...)
Affinity DataIC50:  666nMpH: 7.5 T: 2°CAssay Description:where a pro-fluorescing peptide is used as substrate, and the fluorogenic activity of its cleavage product is measured after co-incubation with the a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed