Compile Data Set for Download or QSAR
maximum 50k data
Found 173 Enz. Inhib. hit(s) with all data for entry = 50041178
TargetNeutrophil elastase(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50288098(2-Ethoxy-5-ethyl-benzo[d][1,3]oxazin-4-one | CHEMB...)
Affinity DataKi:  0.0430nM Kon:  0.0000145M-1s-1 Koff:  3.39E+5s-1Assay Description:Component deacylation rate constant for interaction with human leukocyte elastaseChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50406288(CHEMBL344066)
Affinity DataKi:  0.0680nM Kon:  0.0000759M-1s-1 Koff:  1.12E+6s-1Assay Description:Component deacylation rate constant for interaction with human leukocyte elastaseChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50406293(CHEMBL356120)
Affinity DataKi:  0.0710nM Kon:  0.0000550M-1s-1 Koff:  7.76E+5s-1Assay Description:Component deacylation rate constant for interaction with human leukocyte elastaseChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50406217(CHEMBL145002)
Affinity DataKi:  0.100nM Kon:  0.00000617M-1s-1 Koff:  6.46E+4s-1Assay Description:Component deacylation rate constant for interaction with human leukocyte elastaseChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50288087(2-Ethoxy-5-methyl-benzo[d][1,3]oxazin-4-one | CHEM...)
Affinity DataKi:  0.126nM Kon:  0.0000117M-1s-1 Koff:  1.02E+5s-1Assay Description:Component deacylation rate constant for interaction with human leukocyte elastaseChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50406234(CHEMBL145774)
Affinity DataKi:  0.200nM Kon:  0.0000661M-1s-1 Koff:  3.47E+5s-1Assay Description:Component deacylation rate constant for interaction with human leukocyte elastaseChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50406239(CHEMBL357464)
Affinity DataKi:  0.251nM Kon:  0.0000708M-1s-1 Koff:  3.09E+5s-1Assay Description:Component deacylation rate constant for interaction with human leukocyte elastaseChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50406240(CHEMBL347760)
Affinity DataKi:  0.398nM Kon:  0.0000182M-1s-1 Koff:  4.57E+4s-1Assay Description:Component deacylation rate constant for interaction with human leukocyte elastaseChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50406245(CHEMBL145592)
Affinity DataKi:  0.501nM Kon:  0.00468M-1s-1 Koff:  1.00E+7s-1Assay Description:Component deacylation rate constant for interaction with human leukocyte elastaseChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50406185(CHEMBL144906)
Affinity DataKi:  1nM Kon:  0.00141M-1s-1 Koff:  1.51E+6s-1Assay Description:Component deacylation rate constant for interaction with human leukocyte elastaseChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50291760(5-Ethyl-2-isopropylamino-benzo[d][1,3]oxazin-4-one...)
Affinity DataKi:  1nM Kon:  0.0000661M-1s-1 Koff:  7.08E+4s-1Assay Description:Component deacylation rate constant for interaction with human leukocyte elastaseChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50406260(CHEMBL143793)
Affinity DataKi:  1.41nM Kon:  0.000355M-1s-1 Koff:  2.51E+5s-1Assay Description:Component deacylation rate constant for interaction with human leukocyte elastaseChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50406221(CHEMBL145729)
Affinity DataKi:  1.58nM Kon:  0.0000112M-1s-1 Koff:  7.08E+3s-1Assay Description:Component deacylation rate constant for interaction with human leukocyte elastaseChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50063719(2-Isopropylamino-5-methyl-benzo[d][1,3]oxazin-4-on...)
Affinity DataKi:  1.58nM Kon:  0.0000178M-1s-1 Koff:  1.18E+4s-1Assay Description:Component deacylation rate constant for interaction with human leukocyte elastaseChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50406198(CHEMBL145035)
Affinity DataKi:  2.51nM Kon:  0.000813M-1s-1 Koff:  3.02E+5s-1Assay Description:Component deacylation rate constant for interaction with human leukocyte elastaseChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50291763(2-Butylamino-5-ethyl-benzo[d][1,3]oxazin-4-one | C...)
Affinity DataKi:  3.98nM Kon:  0.000537M-1s-1 Koff:  1.29E+5s-1Assay Description:Component deacylation rate constant for interaction with human leukocyte elastaseChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50406226(CHEMBL342522)
Affinity DataKi:  5.01nM Kon:  0.0000141M-1s-1 Koff:  2.88E+3s-1Assay Description:Component deacylation rate constant for interaction with human leukocyte elastaseChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50406271(CHEMBL141553)
Affinity DataKi:  6.31nM Kon:  0.00631M-1s-1 Koff:  1.10E+6s-1Assay Description:Component deacylation rate constant for interaction with human leukocyte elastaseChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50406208(CHEMBL146004)
Affinity DataKi:  6.31nM Kon:  0.0000151M-1s-1 Koff:  2.57E+3s-1Assay Description:Component deacylation rate constant for interaction with human leukocyte elastaseChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50406216(CHEMBL146003)
Affinity DataKi:  6.31nM Kon:  0.00000871M-1s-1 Koff:  1.32E+3s-1Assay Description:Component deacylation rate constant for interaction with human leukocyte elastaseChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50291758(5-Methyl-2-propylamino-benzo[d][1,3]oxazin-4-one |...)
Affinity DataKi:  6.31nM Kon:  0.000339M-1s-1 Koff:  5.62E+4s-1Assay Description:Component deacylation rate constant for interaction with human leukocyte elastaseChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50288095(2-Ethoxy-benzo[d][1,3]oxazin-4-one | CHEMBL450273)
Affinity DataKi:  6.31nM Kon:  0.00102M-1s-1 Koff:  1.59E+5s-1Assay Description:Component deacylation rate constant for interaction with human leukocyte elastaseChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50406290(CHEMBL141707)
Affinity DataKi:  6.31nM Kon:  0.0000436M-1s-1 Koff:  7.59E+3s-1Assay Description:Component deacylation rate constant for interaction with human leukocyte elastaseChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50406313(CHEMBL143792)
Affinity DataKi:  7.94nM Koff:  2.00E+6s-1Assay Description:Component deacylation rate constant for interaction with human leukocyte elastaseChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50406266(CHEMBL358112)
Affinity DataKi:  7.94nM Kon:  0.0224M-1s-1 Koff:  2.88E+6s-1Assay Description:Component deacylation rate constant for interaction with human leukocyte elastaseChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50406319(CHEMBL145492)
Affinity DataKi:  10nM Koff:  6.46E+3s-1Assay Description:Component deacylation rate constant for interaction with human leukocyte elastaseChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50406257(CHEMBL145252)
Affinity DataKi:  10nM Koff:  3.47E+4s-1Assay Description:Component deacylation rate constant for interaction with human leukocyte elastaseChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50406307(CHEMBL146010)
Affinity DataKi:  10nM Kon:  0.00246M-1s-1 Koff:  2.24E+5s-1Assay Description:Component deacylation rate constant for interaction with human leukocyte elastaseChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50449417(CHEMBL356307)
Affinity DataKi:  10nMAssay Description:Component deacylation rate constant for interaction with human leukocyte elastaseChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50406186(CHEMBL142970)
Affinity DataKi:  12.6nM Kon:  0.000562M-1s-1 Koff:  4.90E+4s-1Assay Description:Component deacylation rate constant for interaction with human leukocyte elastaseChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50406285(CHEMBL145583)
Affinity DataKi:  12.6nM Kon:  0.0000562M-1s-1 Koff:  4.68E+3s-1Assay Description:Component deacylation rate constant for interaction with human leukocyte elastaseChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50406273(CHEMBL145471)
Affinity DataKi:  15.8nM Kon:  0.0000282M-1s-1 Koff:  1.66E+3s-1Assay Description:Component deacylation rate constant for interaction with human leukocyte elastaseChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50406202(CHEMBL343675)
Affinity DataKi:  17.8nM Kon:  0.00107M-1s-1 Koff:  6.03E+4s-1Assay Description:Component deacylation rate constant for interaction with human leukocyte elastaseChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50406215(CHEMBL145718)
Affinity DataKi:  19.9nM Kon:  0.000229M-1s-1 Koff:  1.10E+4s-1Assay Description:Component deacylation rate constant for interaction with human leukocyte elastaseChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50406237(CHEMBL343003)
Affinity DataKi:  19.9nM Koff:  2.00E+6s-1Assay Description:Component deacylation rate constant for interaction with human leukocyte elastaseChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50406223(CHEMBL143922)
Affinity DataKi:  19.9nM Kon:  0.00724M-1s-1 Koff:  3.47E+5s-1Assay Description:Component deacylation rate constant for interaction with human leukocyte elastaseChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50406201(CHEMBL145694)
Affinity DataKi:  19.9nM Kon:  0.000324M-1s-1 Koff:  1.51E+4s-1Assay Description:Component deacylation rate constant for interaction with human leukocyte elastaseChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50406203(CHEMBL145214)
Affinity DataKi:  19.9nM Kon:  0.000912M-1s-1 Koff:  4.27E+4s-1Assay Description:Component deacylation rate constant for interaction with human leukocyte elastaseChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50291761(2-Butylamino-5-methyl-benzo[d][1,3]oxazin-4-one | ...)
Affinity DataKi:  25.1nM Kon:  0.000174M-1s-1 Koff:  7.59E+3s-1Assay Description:Component deacylation rate constant for interaction with human leukocyte elastaseChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50406281(CHEMBL145601)
Affinity DataKi:  25.1nM Kon:  0.000417M-1s-1 Koff:  1.51E+4s-1Assay Description:Component deacylation rate constant for interaction with human leukocyte elastaseChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50406238(CHEMBL144915)
Affinity DataKi:  28.2nM Koff:  2.00E+6s-1Assay Description:Component deacylation rate constant for interaction with human leukocyte elastaseChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50406224(CHEMBL145565)
Affinity DataKi:  31.6nM Kon:  0.00371M-1s-1 Koff:  1.29E+5s-1Assay Description:Component deacylation rate constant for interaction with human leukocyte elastaseChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50291753(2-Ethylamino-5-methyl-benzo[d][1,3]oxazin-4-one | ...)
Affinity DataKi:  31.6nM Kon:  0.00178M-1s-1 Koff:  5.25E+4s-1Assay Description:Component deacylation rate constant for interaction with human leukocyte elastaseChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50406189(CHEMBL146381)
Affinity DataKi:  31.6nM Kon:  0.0000977M-1s-1 Koff:  2.57E+3s-1Assay Description:Component deacylation rate constant for interaction with human leukocyte elastaseChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50406190(CHEMBL356045)
Affinity DataKi:  39.8nM Kon:  0.00138M-1s-1 Koff:  3.98E+4s-1Assay Description:Component deacylation rate constant for interaction with human leukocyte elastaseChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50406295(CHEMBL424495)
Affinity DataKi:  39.8nM Koff:  1.26E+3s-1Assay Description:Component deacylation rate constant for interaction with human leukocyte elastaseChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50406197(CHEMBL358949)
Affinity DataKi:  39.8nM Kon:  0.00209M-1s-1 Koff:  5.25E+4s-1Assay Description:Component deacylation rate constant for interaction with human leukocyte elastaseChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50291762(2-sec-Butylamino-benzo[d][1,3]oxazin-4-one | CHEMB...)
Affinity DataKi:  39.8nM Kon:  0.0105M-1s-1 Koff:  2.40E+5s-1Assay Description:Component deacylation rate constant for interaction with human leukocyte elastaseChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50406256(CHEMBL144900)
Affinity DataKi:  39.8nM Kon:  0.000537M-1s-1 Koff:  1.45E+4s-1Assay Description:Component deacylation rate constant for interaction with human leukocyte elastaseChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50406200(CHEMBL145055)
Affinity DataKi:  39.8nM Kon:  0.000794M-1s-1 Koff:  2.09E+4s-1Assay Description:Component deacylation rate constant for interaction with human leukocyte elastaseChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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