Compile Data Set for Download or QSAR
maximum 50k data
Found 19 Enz. Inhib. hit(s) with all data for entry = 50009643
TargetCytosolic phospholipase A2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50085993((E)-N-(((2S,4R)-4-((biphenyl-2-ylmethyl)(isobutyl)...)
Affinity DataIC50:  1.80nMAssay Description:Inhibition of Human cPLA2 alpha using Enzyme assay(PC/DOG assay)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosolic phospholipase A2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50085984(CHEMBL9161 | N-[1-[2-(2,4-Difluoro-benzoyl)-benzoy...)
Affinity DataIC50:  2.10nMAssay Description:Inhibition of Human cPLA2 alpha using Enzyme assay(PC/DOG assay)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosolic phospholipase A2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50085986(CHEMBL267258 | N-{4-(Biphenyl-2-ylmethyl-isobutyl-...)
Affinity DataIC50:  3.10nMAssay Description:Inhibition of Human cPLA2 alpha using Enzyme assay(PC/DOG assay)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosolic phospholipase A2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50085987(4-(2,4-Dioxo-thiazolidin-5-ylidenemethyl)-N-[1-[2-...)
Affinity DataIC50:  5.30nMAssay Description:Inhibition of Human cPLA2 alpha using Enzyme assay(PC/DOG assay)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosolic phospholipase A2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50085994(CHEMBL8970 | N-{4-(Biphenyl-2-ylmethyl-isobutyl-am...)
Affinity DataIC50:  6.20nMAssay Description:Inhibition of Human cPLA2 alpha using Enzyme assay(PC/DOG assay)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosolic phospholipase A2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50085980(CHEMBL428996 | N-{4-(Biphenyl-2-ylmethyl-isobutyl-...)
Affinity DataIC50:  21nMAssay Description:Inhibition of Human cPLA2 alpha using Enzyme assay(PC/DOG assay)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosolic phospholipase A2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50085997(CHEMBL266374 | N-{4-(2-Bromo-6-isobutyl-phenoxy)-1...)
Affinity DataIC50:  22nMAssay Description:Inhibition of Human cPLA2 alpha using Enzyme assay(PC/DOG assay)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosolic phospholipase A2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50085990(CHEMBL268434 | N-{4-(Biphenyl-2-ylmethylsulfanyl)-...)
Affinity DataIC50:  34nMAssay Description:Inhibition of Human cPLA2 alpha using Enzyme assay(PC/DOG assay)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosolic phospholipase A2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50085991(CHEMBL268896 | N-{4-(2-Bromo-6-isobutyl-phenoxy)-1...)
Affinity DataIC50:  38nMAssay Description:Inhibition of Human cPLA2 alpha using Enzyme assay(PC/DOG assay)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosolic phospholipase A2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50085983(CHEMBL267697 | N-{4-(Biphenyl-2-ylmethoxy)-1-[2-(2...)
Affinity DataIC50:  49nMAssay Description:Inhibition of Human cPLA2 alpha using Enzyme assay(PC/DOG assay)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosolic phospholipase A2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50085988(CHEMBL416517 | N-{4-(Biphenyl-2-yloxy)-1-[2-(4-flu...)
Affinity DataIC50:  69nMAssay Description:Inhibition of Human cPLA2 alpha using Enzyme assay(PC/DOG assay)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosolic phospholipase A2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50085981(CHEMBL268419 | N-{4-(Biphenyl-2-ylmethylsulfanyl)-...)
Affinity DataIC50:  72nMAssay Description:Inhibition of Human cPLA2 alpha using Enzyme assay(PC/DOG assay)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosolic phospholipase A2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50085982(CHEMBL9277 | N-{4-(Biphenyl-2-ylmethoxy)-1-[2-(4-f...)
Affinity DataIC50:  78nMAssay Description:Inhibition of Human cPLA2 alpha using Enzyme assay(PC/DOG assay)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosolic phospholipase A2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50085989(CHEMBL428827 | N-{4-(Biphenyl-2-yloxy)-1-[2-(4-flu...)
Affinity DataIC50:  83nMAssay Description:Inhibition of Human cPLA2 alpha using Enzyme assay(PC/DOG assay)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosolic phospholipase A2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50085985(CHEMBL428653 | N-{4-(Biphenyl-2-ylmethoxy)-1-[2-(4...)
Affinity DataIC50:  90nMAssay Description:Inhibition of Human cPLA2 alpha using Enzyme assay(PC/DOG assay)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosolic phospholipase A2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50085992(CHEMBL268905 | N-[(2S,4R)-1-(2-Benzoyl-benzoyl)-4-...)
Affinity DataIC50:  165nMAssay Description:Inhibition of Human cPLA2 alpha using Enzyme assay(PC/DOG assay)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosolic phospholipase A2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50085998(1,1,1-Trifluoro-docosa-7,10,13,16-tetraen-3-one | ...)
Affinity DataIC50:  420nMAssay Description:Inhibition of Human cPLA2 alpha using Enzyme assay(PC/DOG assay)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosolic phospholipase A2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50085999(CHEMBL268904 | N-[1-(3-Benzoyl-benzoyl)-4-(bipheny...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Human cPLA2 alpha using Enzyme assay(PC/DOG assay)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosolic phospholipase A2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50085996(CHEMBL266580 | N-[1-(4-Benzoyl-benzoyl)-4-(bipheny...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Human cPLA2 alpha using Enzyme assay(PC/DOG assay)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed