Compile Data Set for Download or QSAR
maximum 50k data
Found 67 Enz. Inhib. hit(s) with all data for entry = 50033304
TargetCollagenase 3(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50343062(CHEMBL1770709 | N-hydroxy-4-(4-(4-oxo-4-(4-(triflu...)
Affinity DataIC50:  0.200nMAssay Description:Inhibition of human MMP13More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50343059(4-(4-(4-(4-(dimethylamino)phenyl)-4-oxobutoxy)phen...)
Affinity DataIC50:  0.200nMAssay Description:Inhibition of human MMP13More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50343061(CHEMBL1770157 | N-hydroxy-4-(4-(4-(4-methoxyphenyl...)
Affinity DataIC50:  0.300nMAssay Description:Inhibition of human MMP13More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM11885(CHEMBL1082381 | N-Hydroxy-4-{[4-(phenylthio)phenyl...)
Affinity DataIC50:  0.330nMAssay Description:Inhibition of human MMP2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50343051(4-(4-(5-(4-(dimethylamino)phenyl)-5-oxopentyloxy)p...)
Affinity DataIC50:  0.400nMAssay Description:Inhibition of human MMP13More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50343054(CHEMBL1770702 | N-hydroxy-4-(4-(3-(4-(trifluoromet...)
Affinity DataIC50:  0.660nMAssay Description:Inhibition of human MMP13More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50343058(4-(4-(3-(4-(dimethylamino)phenyl)-3-oxopropoxy)phe...)
Affinity DataIC50:  0.900nMAssay Description:Inhibition of human MMP13More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50343066(CHEMBL1770712 | N-hydroxy-4-(4-(4-(4-methoxyphenox...)
Affinity DataIC50:  0.900nMAssay Description:Inhibition of human MMP13More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM11885(CHEMBL1082381 | N-Hydroxy-4-{[4-(phenylthio)phenyl...)
Affinity DataIC50: <1nMAssay Description:Inhibition of human MMP13More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50343064(CHEMBL1770710 | N-hydroxy-4-(4-(4-oxo-4-(piperidin...)
Affinity DataIC50:  1.20nMAssay Description:Inhibition of human MMP13More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM11885(CHEMBL1082381 | N-Hydroxy-4-{[4-(phenylthio)phenyl...)
Affinity DataIC50:  1.5nMAssay Description:Inhibition of human MMP9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50343052(CHEMBL1770700 | N-hydroxy-4-(4-(3-(4-methoxybenzam...)
Affinity DataIC50:  1.60nMAssay Description:Inhibition of human MMP13More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50343053(4-(4-(3-(4-(dimethylamino)benzamido)propoxy)phenyl...)
Affinity DataIC50:  1.60nMAssay Description:Inhibition of human MMP13More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50343060(4-(4-(4-(4-(dimethylamino)phenylamino)-4-oxobutoxy...)
Affinity DataIC50:  1.70nMAssay Description:Inhibition of human MMP13More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil collagenase(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM11885(CHEMBL1082381 | N-Hydroxy-4-{[4-(phenylthio)phenyl...)
Affinity DataIC50:  1.80nMAssay Description:Inhibition of human MMP8More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50343065(4-(4-(5-(4-(dimethylamino)phenylamino)-5-oxopentyl...)
Affinity DataIC50:  1.80nMAssay Description:Inhibition of human MMP2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50343065(4-(4-(5-(4-(dimethylamino)phenylamino)-5-oxopentyl...)
Affinity DataIC50:  1.80nMAssay Description:Inhibition of human MMP13More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50343061(CHEMBL1770157 | N-hydroxy-4-(4-(4-(4-methoxyphenyl...)
Affinity DataIC50:  2.5nMAssay Description:Inhibition of human MMP2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil collagenase(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50343065(4-(4-(5-(4-(dimethylamino)phenylamino)-5-oxopentyl...)
Affinity DataIC50:  2.60nMAssay Description:Inhibition of human MMP8More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50343063(CHEMBL1770697 | N-hydroxy-4-(4-(4-(methyl(4-(trifl...)
Affinity DataIC50:  3.30nMAssay Description:Inhibition of human MMP13More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50343066(CHEMBL1770712 | N-hydroxy-4-(4-(4-(4-methoxyphenox...)
Affinity DataIC50:  6.60nMAssay Description:Inhibition of human MMP2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil collagenase(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50343062(CHEMBL1770709 | N-hydroxy-4-(4-(4-oxo-4-(4-(triflu...)
Affinity DataIC50:  6.70nMAssay Description:Inhibition of human MMP8More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50343050(4-(4-(4-(4-(dimethylamino)benzoyl)piperidin-1-yl)p...)
Affinity DataIC50:  8nMAssay Description:Inhibition of human MMP13More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-14(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM11885(CHEMBL1082381 | N-Hydroxy-4-{[4-(phenylthio)phenyl...)
Affinity DataIC50:  8nMAssay Description:Inhibition of human MMP14More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50343055(4-(4-(3-(2,4-dimethylbenzamido)propoxy)phenylsulfo...)
Affinity DataIC50:  8nMAssay Description:Inhibition of human MMP13More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50343057(4-(4-(3-(2,2-dimethylpentanamido)propoxy)phenylsul...)
Affinity DataIC50:  8.20nMAssay Description:Inhibition of human MMP13More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50343056(4-(4-(3-(cyclohexanecarboxamido)propoxy)phenylsulf...)
Affinity DataIC50:  8.20nMAssay Description:Inhibition of human MMP13More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50343060(4-(4-(4-(4-(dimethylamino)phenylamino)-4-oxobutoxy...)
Affinity DataIC50:  10nMAssay Description:Inhibition of human MMP2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50343062(CHEMBL1770709 | N-hydroxy-4-(4-(4-oxo-4-(4-(triflu...)
Affinity DataIC50:  11nMAssay Description:Inhibition of human MMP2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50343058(4-(4-(3-(4-(dimethylamino)phenyl)-3-oxopropoxy)phe...)
Affinity DataIC50:  16nMAssay Description:Inhibition of human MMP2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50343059(4-(4-(4-(4-(dimethylamino)phenyl)-4-oxobutoxy)phen...)
Affinity DataIC50:  18nMAssay Description:Inhibition of human MMP2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50343061(CHEMBL1770157 | N-hydroxy-4-(4-(4-(4-methoxyphenyl...)
Affinity DataIC50:  23nMAssay Description:Inhibition of human MMP9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil collagenase(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50343061(CHEMBL1770157 | N-hydroxy-4-(4-(4-(4-methoxyphenyl...)
Affinity DataIC50:  31nMAssay Description:Inhibition of human MMP8More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50343051(4-(4-(5-(4-(dimethylamino)phenyl)-5-oxopentyloxy)p...)
Affinity DataIC50:  35nMAssay Description:Inhibition of human MMP2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil collagenase(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50343063(CHEMBL1770697 | N-hydroxy-4-(4-(4-(methyl(4-(trifl...)
Affinity DataIC50:  49nMAssay Description:Inhibition of human MMP8More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil collagenase(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50343066(CHEMBL1770712 | N-hydroxy-4-(4-(4-(4-methoxyphenox...)
Affinity DataIC50:  67nMAssay Description:Inhibition of human MMP8More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil collagenase(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50343060(4-(4-(4-(4-(dimethylamino)phenylamino)-4-oxobutoxy...)
Affinity DataIC50:  100nMAssay Description:Inhibition of human MMP8More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil collagenase(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50343058(4-(4-(3-(4-(dimethylamino)phenyl)-3-oxopropoxy)phe...)
Affinity DataIC50:  120nMAssay Description:Inhibition of human MMP8More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil collagenase(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50343051(4-(4-(5-(4-(dimethylamino)phenyl)-5-oxopentyloxy)p...)
Affinity DataIC50:  140nMAssay Description:Inhibition of human MMP8More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil collagenase(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50343054(CHEMBL1770702 | N-hydroxy-4-(4-(3-(4-(trifluoromet...)
Affinity DataIC50:  140nMAssay Description:Inhibition of human MMP8More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil collagenase(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50343059(4-(4-(4-(4-(dimethylamino)phenyl)-4-oxobutoxy)phen...)
Affinity DataIC50:  170nMAssay Description:Inhibition of human MMP8More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50343064(CHEMBL1770710 | N-hydroxy-4-(4-(4-oxo-4-(piperidin...)
Affinity DataIC50:  170nMAssay Description:Inhibition of human MMP2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50343062(CHEMBL1770709 | N-hydroxy-4-(4-(4-oxo-4-(4-(triflu...)
Affinity DataIC50:  180nMAssay Description:Inhibition of human MMP9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50343063(CHEMBL1770697 | N-hydroxy-4-(4-(4-(methyl(4-(trifl...)
Affinity DataIC50:  270nMAssay Description:Inhibition of human MMP2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50343054(CHEMBL1770702 | N-hydroxy-4-(4-(3-(4-(trifluoromet...)
Affinity DataIC50:  360nMAssay Description:Inhibition of human MMP2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50343063(CHEMBL1770697 | N-hydroxy-4-(4-(4-(methyl(4-(trifl...)
Affinity DataIC50:  380nMAssay Description:Inhibition of human MMP9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50343057(4-(4-(3-(2,2-dimethylpentanamido)propoxy)phenylsul...)
Affinity DataIC50:  450nMAssay Description:Inhibition of human MMP2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50343065(4-(4-(5-(4-(dimethylamino)phenylamino)-5-oxopentyl...)
Affinity DataIC50:  500nMAssay Description:Inhibition of human MMP9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50343052(CHEMBL1770700 | N-hydroxy-4-(4-(3-(4-methoxybenzam...)
Affinity DataIC50:  550nMAssay Description:Inhibition of human MMP2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50343056(4-(4-(3-(cyclohexanecarboxamido)propoxy)phenylsulf...)
Affinity DataIC50:  650nMAssay Description:Inhibition of human MMP2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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