Compile Data Set for Download or QSAR
maximum 50k data
Found 66 Enz. Inhib. hit(s) with all data for entry = 50011954
TargetCoagulation factor X(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112506(3-(3-{4-[1-(1-Imino-ethyl)-piperidin-4-yloxy]-3-ni...)
Affinity DataKi:  0.0700nMAssay Description:Competitive inhibition of coagulation factor XaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112502(CHEMBL26299 | N-[3-(5-Carbamimidoyl-2-hydroxy-phen...)
Affinity DataKi:  0.0700nMAssay Description:Competitive inhibition of coagulation factor XaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112503(7-({4-[1-(1-Imino-ethyl)-piperidin-4-yloxy]-3-nitr...)
Affinity DataKi:  0.0800nMAssay Description:Competitive inhibition of coagulation factor XaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112497(CHEMBL26240 | N-[3-(5-Carbamimidoyl-2-hydroxy-phen...)
Affinity DataKi:  0.100nMAssay Description:Competitive inhibition of coagulation factor XaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112491(4-Hydroxy-3-(3-{4-[1-(1-imino-ethyl)-piperidin-4-y...)
Affinity DataKi:  0.100nMAssay Description:Competitive inhibition of coagulation factor XaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112500(3'-({4-[1-(1-Imino-ethyl)-piperidin-4-yloxy]-3-nit...)
Affinity DataKi:  0.170nMAssay Description:Competitive inhibition of coagulation factor XaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112488(3-(3-{4-[1-(1-Imino-ethyl)-piperidin-4-yloxy]-3-ni...)
Affinity DataKi:  0.270nMAssay Description:Competitive inhibition of coagulation factor XaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112490(CHEMBL424589 | N-[3-(3-Carbamimidoyl-phenyl)-allyl...)
Affinity DataKi:  0.280nMAssay Description:Competitive inhibition of coagulation factor XaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112489(CHEMBL277424 | N-[3-(5-Carbamimidoyl-2-hydroxy-phe...)
Affinity DataKi:  0.280nMAssay Description:Competitive inhibition of coagulation factor XaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112494(7-{5-[1-(1-Imino-ethyl)-piperidin-4-yloxy]-2-methy...)
Affinity DataKi:  0.300nMAssay Description:Competitive inhibition of coagulation factor XaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112496(CHEMBL26709 | N-[3-(5-Carbamimidoyl-2-hydroxy-phen...)
Affinity DataKi:  0.340nMAssay Description:Competitive inhibition of coagulation factor XaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112492(CHEMBL26287 | N-[3-(3-Carbamimidoyl-phenyl)-allyl]...)
Affinity DataKi:  0.550nMAssay Description:Competitive inhibition of coagulation factor XaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112486(4-([3-(3-Carbamimidoyl-phenyl)-allyl]-{4-[1-(1-imi...)
Affinity DataKi:  0.560nMAssay Description:Competitive inhibition of coagulation factor XaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112505(4-Hydroxy-3-{3-[4-(1-methyl-piperidin-4-yloxy)-3-t...)
Affinity DataKi:  0.580nMAssay Description:Competitive inhibition of coagulation factor XaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112495(3-(3-{4-[1-(1-Imino-ethyl)-piperidin-4-yloxy]-3-tr...)
Affinity DataKi:  0.880nMAssay Description:Competitive inhibition of coagulation factor XaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112498(CHEMBL25170 | N-[4-(1-Acetyl-piperidin-4-yloxy)-3-...)
Affinity DataKi:  3nMAssay Description:Competitive inhibition of coagulation factor XaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112494(7-{5-[1-(1-Imino-ethyl)-piperidin-4-yloxy]-2-methy...)
Affinity DataKi:  3nMAssay Description:Competitive inhibition of trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112499(3-(3-{3-Fluoro-4-[1-(1-imino-ethyl)-piperidin-4-yl...)
Affinity DataKi:  4.10nMAssay Description:Competitive inhibition of coagulation factor XaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112506(3-(3-{4-[1-(1-Imino-ethyl)-piperidin-4-yloxy]-3-ni...)
Affinity DataKi:  5nMAssay Description:Competitive inhibition of trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112507(5-[3-(3-Carbamimidoyl-phenyl)-allylamino]-2-[1-(1-...)
Affinity DataKi:  6.80nMAssay Description:Competitive inhibition of coagulation factor XaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112503(7-({4-[1-(1-Imino-ethyl)-piperidin-4-yloxy]-3-nitr...)
Affinity DataKi:  7nMAssay Description:Competitive inhibition of trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112501(4-{4-[3-(5-Carbamimidoyl-2-hydroxy-phenyl)-allylam...)
Affinity DataKi:  7.30nMAssay Description:Competitive inhibition of coagulation factor XaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112493(3-(3-{4-[1-(1-Imino-ethyl)-piperidin-4-yloxy]-phen...)
Affinity DataKi:  7.5nMAssay Description:Competitive inhibition of coagulation factor XaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112486(4-([3-(3-Carbamimidoyl-phenyl)-allyl]-{4-[1-(1-imi...)
Affinity DataKi:  10nMAssay Description:Competitive inhibition of trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112487(3-{3-[4-(1-Acetyl-piperidin-4-yloxy)-3-trifluorome...)
Affinity DataKi:  19nMAssay Description:Competitive inhibition of coagulation factor XaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112488(3-(3-{4-[1-(1-Imino-ethyl)-piperidin-4-yloxy]-3-ni...)
Affinity DataKi:  27nMAssay Description:Competitive inhibition of trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112507(5-[3-(3-Carbamimidoyl-phenyl)-allylamino]-2-[1-(1-...)
Affinity DataKi:  40nMAssay Description:Competitive inhibition of trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112500(3'-({4-[1-(1-Imino-ethyl)-piperidin-4-yloxy]-3-nit...)
Affinity DataKi:  42nMAssay Description:Competitive inhibition of trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112504(4-Hydroxy-3-{3-[4-(1-methanesulfonyl-piperidin-4-y...)
Affinity DataKi:  44nMAssay Description:Competitive inhibition of coagulation factor XaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112495(3-(3-{4-[1-(1-Imino-ethyl)-piperidin-4-yloxy]-3-tr...)
Affinity DataKi:  50nMAssay Description:Competitive inhibition of trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112499(3-(3-{3-Fluoro-4-[1-(1-imino-ethyl)-piperidin-4-yl...)
Affinity DataKi:  70nMAssay Description:Competitive inhibition of trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112492(CHEMBL26287 | N-[3-(3-Carbamimidoyl-phenyl)-allyl]...)
Affinity DataKi:  76nMAssay Description:Competitive inhibition of trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112493(3-(3-{4-[1-(1-Imino-ethyl)-piperidin-4-yloxy]-phen...)
Affinity DataKi:  80nMAssay Description:Competitive inhibition of trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112490(CHEMBL424589 | N-[3-(3-Carbamimidoyl-phenyl)-allyl...)
Affinity DataKi:  110nMAssay Description:Competitive inhibition of trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112491(4-Hydroxy-3-(3-{4-[1-(1-imino-ethyl)-piperidin-4-y...)
Affinity DataKi:  200nMAssay Description:Competitive inhibition of trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112502(CHEMBL26299 | N-[3-(5-Carbamimidoyl-2-hydroxy-phen...)
Affinity DataKi:  230nMAssay Description:Competitive inhibition of trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112501(4-{4-[3-(5-Carbamimidoyl-2-hydroxy-phenyl)-allylam...)
Affinity DataKi:  250nMAssay Description:Competitive inhibition of coagulation factor IIaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112497(CHEMBL26240 | N-[3-(5-Carbamimidoyl-2-hydroxy-phen...)
Affinity DataKi:  280nMAssay Description:Competitive inhibition of trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112500(3'-({4-[1-(1-Imino-ethyl)-piperidin-4-yloxy]-3-nit...)
Affinity DataKi:  400nMAssay Description:Competitive inhibition of coagulation factor IIaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112507(5-[3-(3-Carbamimidoyl-phenyl)-allylamino]-2-[1-(1-...)
Affinity DataKi:  480nMAssay Description:Competitive inhibition of coagulation factor IIaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112487(3-{3-[4-(1-Acetyl-piperidin-4-yloxy)-3-trifluorome...)
Affinity DataKi:  480nMAssay Description:Competitive inhibition of coagulation factor IIaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112501(4-{4-[3-(5-Carbamimidoyl-2-hydroxy-phenyl)-allylam...)
Affinity DataKi:  520nMAssay Description:Competitive inhibition of trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112505(4-Hydroxy-3-{3-[4-(1-methyl-piperidin-4-yloxy)-3-t...)
Affinity DataKi:  630nMAssay Description:Competitive inhibition of trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112489(CHEMBL277424 | N-[3-(5-Carbamimidoyl-2-hydroxy-phe...)
Affinity DataKi:  765nMAssay Description:Competitive inhibition of trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112487(3-{3-[4-(1-Acetyl-piperidin-4-yloxy)-3-trifluorome...)
Affinity DataKi:  830nMAssay Description:Competitive inhibition of trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112496(CHEMBL26709 | N-[3-(5-Carbamimidoyl-2-hydroxy-phen...)
Affinity DataKi:  870nMAssay Description:Competitive inhibition of trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112504(4-Hydroxy-3-{3-[4-(1-methanesulfonyl-piperidin-4-y...)
Affinity DataKi:  890nMAssay Description:Competitive inhibition of coagulation factor IIaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112498(CHEMBL25170 | N-[4-(1-Acetyl-piperidin-4-yloxy)-3-...)
Affinity DataKi:  891nMAssay Description:Competitive inhibition of trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112492(CHEMBL26287 | N-[3-(3-Carbamimidoyl-phenyl)-allyl]...)
Affinity DataKi:  1.00E+3nMAssay Description:Competitive inhibition of coagulation factor IIaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112491(4-Hydroxy-3-(3-{4-[1-(1-imino-ethyl)-piperidin-4-y...)
Affinity DataKi:  1.10E+3nMAssay Description:Competitive inhibition of coagulation factor IIaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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