Compile Data Set for Download or QSAR
maximum 50k data
Found 62 Enz. Inhib. hit(s) with all data for entry = 50018067
TargetAdenosine receptor A1(Rattus norvegicus (rat))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50190710(8-[4-(phenylamidosulfonyl)phenyl]-1-propylxanthine...)
Affinity DataKi:  1.80nMAssay Description:Displacement of [3H]CCPA from adenosine A1 receptor in rat brain cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50190709(8-(4-(4-benzylpiperazin-1-ylsulfonyl)phenyl)-1-pro...)
Affinity DataKi:  3.60nMAssay Description:Displacement of [3H]PSB298 from human recombinant adenosine A2B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50190702(8-[4-(phenylethylamidosulfonyl)phenyl]-1-propylxan...)
Affinity DataKi:  3.62nMAssay Description:Displacement of [3H]PSB298 from human recombinant adenosine A2B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50190706(8-[4-(benzylamidosulfonyl)phenyl]-1-propylxanthine...)
Affinity DataKi:  4.20nMAssay Description:Displacement of [3H]PSB298 from human recombinant adenosine A2B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50190699(8-[4-(phenylethylamidosulfonyl)phenyl]-1,3-dimethy...)
Affinity DataKi:  4.48nMAssay Description:Displacement of [3H]PSB298 from human recombinant adenosine A2B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50190706(8-[4-(benzylamidosulfonyl)phenyl]-1-propylxanthine...)
Affinity DataKi:  4.60nMAssay Description:Displacement of [3H]CCPA from adenosine A1 receptor in rat brain cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50190703(8-[4-(dipropylamidosulfonyl)phenyl]-1-propylxanthi...)
Affinity DataKi:  5.5nMAssay Description:Displacement of [3H]CCPA from adenosine A1 receptor in rat brain cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50190702(8-[4-(phenylethylamidosulfonyl)phenyl]-1-propylxan...)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]CCPA from adenosine A1 receptor in rat brain cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50190699(8-[4-(phenylethylamidosulfonyl)phenyl]-1,3-dimethy...)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]CCPA from adenosine A1 receptor in rat brain cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50190710(8-[4-(phenylamidosulfonyl)phenyl]-1-propylxanthine...)
Affinity DataKi:  23nMAssay Description:Displacement of [3H]MSX2 from adenosine A2A receptor in rat brain striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50190706(8-[4-(benzylamidosulfonyl)phenyl]-1-propylxanthine...)
Affinity DataKi:  26.7nMAssay Description:Displacement of [3H]MSX2 from adenosine A2A receptor in rat brain striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50190707(8-[4-(butylamidosulfonyl)phenyl]-1,3-dimethylxanth...)
Affinity DataKi:  27nMAssay Description:Displacement of [3H]CCPA from adenosine A1 receptor in rat brain cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50190704(8-[4-(2-Hydroxyethylamidosulfonyl)phenyl]-1-propyl...)
Affinity DataKi:  27.1nMAssay Description:Displacement of [3H]PSB298 from human recombinant adenosine A2B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50190710(8-[4-(phenylamidosulfonyl)phenyl]-1-propylxanthine...)
Affinity DataKi:  31.4nMAssay Description:Displacement of [3H]PSB298 from human recombinant adenosine A2B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50190699(8-[4-(phenylethylamidosulfonyl)phenyl]-1,3-dimethy...)
Affinity DataKi:  32.6nMAssay Description:Displacement of [3H]MSX2 from human recombinant adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50190703(8-[4-(dipropylamidosulfonyl)phenyl]-1-propylxanthi...)
Affinity DataKi:  42nMAssay Description:Displacement of [3H]MSX2 from adenosine A2A receptor in rat brain striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50190704(8-[4-(2-Hydroxyethylamidosulfonyl)phenyl]-1-propyl...)
Affinity DataKi:  45nMAssay Description:Displacement of [3H]CCPA from adenosine A1 receptor in rat brain cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50042209(4-(2,6-Dioxo-1-propyl-2,3,6,7-tetrahydro-1H-purin-...)
Affinity DataKi:  53.4nMAssay Description:Displacement of [3H]ZM241385 from human recombinant adenosine A2B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50190703(8-[4-(dipropylamidosulfonyl)phenyl]-1-propylxanthi...)
Affinity DataKi:  53.8nMAssay Description:Displacement of [3H]PSB298 from human recombinant adenosine A2B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50190706(8-[4-(benzylamidosulfonyl)phenyl]-1-propylxanthine...)
Affinity DataKi:  54.8nMAssay Description:Displacement of [3H]CCPA from human recombinant adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50190708(2-(4-(1,3-dimethyl-2,6-dioxo-2,3,6,7-tetrahydro-1H...)
Affinity DataKi:  64nMAssay Description:Displacement of [3H]CCPA from adenosine A1 receptor in rat brain cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50190701(8-[4-(isopropylamidosulfonyl)phenyl]-1,3-dimethylx...)
Affinity DataKi:  75nMAssay Description:Displacement of [3H]CCPA from adenosine A1 receptor in rat brain cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50190709(8-(4-(4-benzylpiperazin-1-ylsulfonyl)phenyl)-1-pro...)
Affinity DataKi:  93.7nMAssay Description:Displacement of [3H]MSX2 from adenosine A2A receptor in rat brain striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50190700(8-[4-(2-hydroxyethylamidosulfonyl)phenyl]-1,3-dime...)
Affinity DataKi:  98nMAssay Description:Displacement of [3H]CCPA from adenosine A1 receptor in rat brain cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50190705(4-(1-propylxanthin-8-yl)phenylsulfonamidoacetic ac...)
Affinity DataKi:  100nMAssay Description:Displacement of [3H]CCPA from adenosine A1 receptor in rat brain cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50190705(4-(1-propylxanthin-8-yl)phenylsulfonamidoacetic ac...)
Affinity DataKi:  101nMAssay Description:Displacement of [3H]PSB298 from human recombinant adenosine A2B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50190701(8-[4-(isopropylamidosulfonyl)phenyl]-1,3-dimethylx...)
Affinity DataKi:  102nMAssay Description:Displacement of [3H]PSB298 from human recombinant adenosine A2B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50190699(8-[4-(phenylethylamidosulfonyl)phenyl]-1,3-dimethy...)
Affinity DataKi:  113nMAssay Description:Displacement of [3H]MSX2 from adenosine A2A receptor in rat brain striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50190707(8-[4-(butylamidosulfonyl)phenyl]-1,3-dimethylxanth...)
Affinity DataKi:  122nMAssay Description:Displacement of [3H]PSB298 from human recombinant adenosine A2B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50190708(2-(4-(1,3-dimethyl-2,6-dioxo-2,3,6,7-tetrahydro-1H...)
Affinity DataKi:  154nMAssay Description:Displacement of [3H]PSB298 from human recombinant adenosine A2B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50190706(8-[4-(benzylamidosulfonyl)phenyl]-1-propylxanthine...)
Affinity DataKi:  162nMAssay Description:Displacement of [3H]MSX2 from human recombinant adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50190707(8-[4-(butylamidosulfonyl)phenyl]-1,3-dimethylxanth...)
Affinity DataKi:  165nMAssay Description:Displacement of [3H]MSX2 from adenosine A2A receptor in rat brain striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50190708(2-(4-(1,3-dimethyl-2,6-dioxo-2,3,6,7-tetrahydro-1H...)
Affinity DataKi:  182nMAssay Description:Displacement of [3H]MSX2 from adenosine A2A receptor in rat brain striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50190702(8-[4-(phenylethylamidosulfonyl)phenyl]-1-propylxan...)
Affinity DataKi:  183nMAssay Description:Displacement of [3H]CCPA from human recombinant adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50018162(4-(2,6-Dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-pu...)
Affinity DataKi:  183nMAssay Description:Displacement of [125I]AB-MECA from sheep adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50190699(8-[4-(phenylethylamidosulfonyl)phenyl]-1,3-dimethy...)
Affinity DataKi:  185nMAssay Description:Displacement of [3H]CCPA from human recombinant adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50018162(4-(2,6-Dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-pu...)
Affinity DataKi:  210nMAssay Description:Displacement of [3H]R-PIA from adenosine A1 receptor in rat brain cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50018162(4-(2,6-Dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-pu...)
Affinity DataKi:  250nMAssay Description:Displacement of [125I]ABOPX from human recombinant adenosine A2B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50190700(8-[4-(2-hydroxyethylamidosulfonyl)phenyl]-1,3-dime...)
Affinity DataKi:  250nMAssay Description:Displacement of [3H]PSB298 from human recombinant adenosine A2B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50190709(8-(4-(4-benzylpiperazin-1-ylsulfonyl)phenyl)-1-pro...)
Affinity DataKi:  260nMAssay Description:Displacement of [3H]CCPA from adenosine A1 receptor in rat brain cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50190701(8-[4-(isopropylamidosulfonyl)phenyl]-1,3-dimethylx...)
Affinity DataKi:  283nMAssay Description:Displacement of [3H]MSX2 from adenosine A2A receptor in rat brain striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50190704(8-[4-(2-Hydroxyethylamidosulfonyl)phenyl]-1-propyl...)
Affinity DataKi:  287nMAssay Description:Displacement of [3H]MSX2 from adenosine A2A receptor in rat brain striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50190702(8-[4-(phenylethylamidosulfonyl)phenyl]-1-propylxan...)
Affinity DataKi:  297nMAssay Description:Displacement of [3H]MSX2 from adenosine A2A receptor in rat brain striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50190705(4-(1-propylxanthin-8-yl)phenylsulfonamidoacetic ac...)
Affinity DataKi:  320nMAssay Description:Displacement of [3H]MSX2 from adenosine A2A receptor in rat brain striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50190700(8-[4-(2-hydroxyethylamidosulfonyl)phenyl]-1,3-dime...)
Affinity DataKi:  347nMAssay Description:Displacement of [3H]MSX2 from adenosine A2A receptor in rat brain striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50190709(8-(4-(4-benzylpiperazin-1-ylsulfonyl)phenyl)-1-pro...)
Affinity DataKi:  484nMAssay Description:Displacement of [3H]MSX2 from human recombinant adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50190702(8-[4-(phenylethylamidosulfonyl)phenyl]-1-propylxan...)
Affinity DataKi:  769nMAssay Description:Displacement of [3H]MSX2 from human recombinant adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50190703(8-[4-(dipropylamidosulfonyl)phenyl]-1-propylxanthi...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]PSB11 from human recombinant adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50190709(8-(4-(4-benzylpiperazin-1-ylsulfonyl)phenyl)-1-pro...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]PSB11 from human recombinant adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50190699(8-[4-(phenylethylamidosulfonyl)phenyl]-1,3-dimethy...)
Affinity DataKi:  1.08E+3nMAssay Description:Displacement of [3H]PSB11 from human recombinant adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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