Compile Data Set for Download or QSAR
maximum 50k data
Found 116 Enz. Inhib. hit(s) with all data for entry = 50021147
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50221531(6-methoxy-7-(3-(4-methylpiperazin-1-yl)propoxy)-4-...)
Affinity DataKi:  3nMAssay Description:Inhibition of human recombinant EGFR by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50221516(6-methoxy-7-(3-morpholinopropoxy)-4-((1R,2S)-2-phe...)
Affinity DataKi:  8.40nMAssay Description:Inhibition of human recombinant EGFR by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50221518(6,7-dimethoxy-4-((1R,2S)-2-phenylcyclopropylamino)...)
Affinity DataKi:  24nMAssay Description:Inhibition of human recombinant EGFR by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50221531(6-methoxy-7-(3-(4-methylpiperazin-1-yl)propoxy)-4-...)
Affinity DataKi:  27nMAssay Description:Inhibition of SRCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50221535(4-((1R,2S)-2-(2-fluorophenyl)cyclopropylamino)-6,7...)
Affinity DataKi:  36nMAssay Description:Inhibition of human recombinant EGFR by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50221522(6-(4-(aminomethyl)phenyl)-4-((1R,2S)-2-phenylcyclo...)
Affinity DataKi:  40nMAssay Description:Inhibition of human recombinant EGFR by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50221531(6-methoxy-7-(3-(4-methylpiperazin-1-yl)propoxy)-4-...)
Affinity DataKi:  41nMAssay Description:Inhibition of SYKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50221530(6,7-diethyl-2-ethynyl-1-(((1S,2R)-2-p-tolylcyclopr...)
Affinity DataKi:  44nMAssay Description:Inhibition of human recombinant EGFR by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50221531(6-methoxy-7-(3-(4-methylpiperazin-1-yl)propoxy)-4-...)
Affinity DataKi:  44nMAssay Description:Inhibition of ABLMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50221516(6-methoxy-7-(3-morpholinopropoxy)-4-((1R,2S)-2-phe...)
Affinity DataKi:  45nMAssay Description:Inhibition of SRCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50221524(6-methoxy-4-((1R,2S)-2-phenylcyclopropylamino)-7-(...)
Affinity DataKi:  49nMAssay Description:Inhibition of SRCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50221527(7-methoxy-6-(3-morpholinopropoxy)-4-((1R,2S)-2-phe...)
Affinity DataKi:  52nMAssay Description:Inhibition of human recombinant EGFR by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50221533(4-((1R,2S)-2-(3-bromophenyl)cyclopropylamino)-6,7-...)
Affinity DataKi:  52nMAssay Description:Inhibition of human recombinant EGFR by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50221517(6-methoxy-7-(2-methoxyethoxy)-4-((1R,2S)-2-phenylc...)
Affinity DataKi:  60nMAssay Description:Inhibition of human recombinant EGFR by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50221521(7-methoxy-6-(2-morpholinoethoxy)-4-((1R,2S)-2-phen...)
Affinity DataKi:  64nMAssay Description:Inhibition of human recombinant EGFR by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50221528(7-methoxy-4-((1R,2S)-2-phenylcyclopropylamino)-6-(...)
Affinity DataKi:  68nMAssay Description:Inhibition of human recombinant EGFR by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50221532(6,7-dimethoxy-4-((1R,2S)-2-(4-phenoxyphenyl)cyclop...)
Affinity DataKi:  80nMAssay Description:Inhibition of human recombinant EGFR by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50221529(7-(4-(morpholinomethyl)phenyl)-4-((1R,2S)-2-phenyl...)
Affinity DataKi:  80nMAssay Description:Inhibition of human recombinant EGFR by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50221522(6-(4-(aminomethyl)phenyl)-4-((1R,2S)-2-phenylcyclo...)
Affinity DataKi:  86nMAssay Description:Inhibition of SRCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50221524(6-methoxy-4-((1R,2S)-2-phenylcyclopropylamino)-7-(...)
Affinity DataKi:  99nMAssay Description:Inhibition of KDRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50221517(6-methoxy-7-(2-methoxyethoxy)-4-((1R,2S)-2-phenylc...)
Affinity DataKi:  110nMAssay Description:Inhibition of SRCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 1(Homo sapiens (Human))
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50221531(6-methoxy-7-(3-(4-methylpiperazin-1-yl)propoxy)-4-...)
Affinity DataKi:  110nMAssay Description:Inhibition of Flt1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50221515(6-(benzyloxy)-7-methoxy-4-((1R,2S)-2-phenylcyclopr...)
Affinity DataKi:  120nMAssay Description:Inhibition of human recombinant EGFR by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50221517(6-methoxy-7-(2-methoxyethoxy)-4-((1R,2S)-2-phenylc...)
Affinity DataKi:  140nMAssay Description:Inhibition of KDRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50221524(6-methoxy-4-((1R,2S)-2-phenylcyclopropylamino)-7-(...)
Affinity DataKi:  140nMAssay Description:Inhibition of SYKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50221529(7-(4-(morpholinomethyl)phenyl)-4-((1R,2S)-2-phenyl...)
Affinity DataKi:  140nMAssay Description:Inhibition of SRCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50221518(6,7-dimethoxy-4-((1R,2S)-2-phenylcyclopropylamino)...)
Affinity DataKi:  150nMAssay Description:Inhibition of SRCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50221521(7-methoxy-6-(2-morpholinoethoxy)-4-((1R,2S)-2-phen...)
Affinity DataKi:  150nMAssay Description:Inhibition of KDRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50221517(6-methoxy-7-(2-methoxyethoxy)-4-((1R,2S)-2-phenylc...)
Affinity DataKi:  160nMAssay Description:Inhibition of SYKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50221529(7-(4-(morpholinomethyl)phenyl)-4-((1R,2S)-2-phenyl...)
Affinity DataKi:  170nMAssay Description:Inhibition of KDRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50221523(7-methoxy-4-((1R,2S)-2-phenylcyclopropylamino)quin...)
Affinity DataKi:  170nMAssay Description:Inhibition of SRCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50221523(7-methoxy-4-((1R,2S)-2-phenylcyclopropylamino)quin...)
Affinity DataKi:  180nMAssay Description:Inhibition of human recombinant EGFR by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50221516(6-methoxy-7-(3-morpholinopropoxy)-4-((1R,2S)-2-phe...)
Affinity DataKi:  200nMAssay Description:Inhibition of ABLMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50221526(6-methoxy-4-((1R,2S)-2-phenylcyclopropylamino)quin...)
Affinity DataKi:  210nMAssay Description:Inhibition of SRCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50221524(6-methoxy-4-((1R,2S)-2-phenylcyclopropylamino)-7-(...)
Affinity DataKi:  220nMAssay Description:Inhibition of human recombinant EGFR by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50221534(4-((1R,2S)-2-(4-bromophenyl)cyclopropylamino)-6,7-...)
Affinity DataKi:  220nMAssay Description:Inhibition of human recombinant EGFR by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50221518(6,7-dimethoxy-4-((1R,2S)-2-phenylcyclopropylamino)...)
Affinity DataKi:  250nMAssay Description:Inhibition of SYKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50221520(6-(3-(morpholinomethyl)phenyl)-4-((1R,2S)-2-phenyl...)
Affinity DataKi:  280nMAssay Description:Inhibition of SRCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50221529(7-(4-(morpholinomethyl)phenyl)-4-((1R,2S)-2-phenyl...)
Affinity DataKi:  300nMAssay Description:Inhibition of ABLMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50221529(7-(4-(morpholinomethyl)phenyl)-4-((1R,2S)-2-phenyl...)
Affinity DataKi:  300nMAssay Description:Inhibition of SYKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50221531(6-methoxy-7-(3-(4-methylpiperazin-1-yl)propoxy)-4-...)
Affinity DataKi:  300nMAssay Description:Inhibition of KDRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50221524(6-methoxy-4-((1R,2S)-2-phenylcyclopropylamino)-7-(...)
Affinity DataKi:  300nMAssay Description:Inhibition of ABLMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50221515(6-(benzyloxy)-7-methoxy-4-((1R,2S)-2-phenylcyclopr...)
Affinity DataKi:  330nMAssay Description:Inhibition of SRCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50221520(6-(3-(morpholinomethyl)phenyl)-4-((1R,2S)-2-phenyl...)
Affinity DataKi:  340nMAssay Description:Inhibition of human recombinant EGFR by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 1(Homo sapiens (Human))
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50221516(6-methoxy-7-(3-morpholinopropoxy)-4-((1R,2S)-2-phe...)
Affinity DataKi:  350nMAssay Description:Inhibition of Flt1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50221526(6-methoxy-4-((1R,2S)-2-phenylcyclopropylamino)quin...)
Affinity DataKi:  360nMAssay Description:Inhibition of human recombinant EGFR by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50221519(6-methoxy-7-(1-methylpiperidin-4-yloxy)-4-((1R,2S)...)
Affinity DataKi:  360nMAssay Description:Inhibition of human recombinant EGFR by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50221517(6-methoxy-7-(2-methoxyethoxy)-4-((1R,2S)-2-phenylc...)
Affinity DataKi:  390nMAssay Description:Inhibition of ABLMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50221525(6-(4-(morpholinomethyl)phenyl)-4-((1R,2S)-2-phenyl...)
Affinity DataKi:  400nMAssay Description:Inhibition of human recombinant EGFR by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Tanabe Research Laboratories Usa

Curated by ChEMBL
LigandPNGBDBM50221516(6-methoxy-7-(3-morpholinopropoxy)-4-((1R,2S)-2-phe...)
Affinity DataKi:  420nMAssay Description:Inhibition of KDRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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