Affinity DataIC50: 0.300nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.60nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 7.5nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 8.60nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 10.1nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 12.2nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 17.9nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 19.5nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 37.7nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 46.1nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 47.7nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 49nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 49.2nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 97nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 117nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB2 receptor expressed in CHO cellMore data for this Ligand-Target Pair
Affinity DataIC50: 132nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 136nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 186nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 203nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 234nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB2 receptor expressed in CHO cellMore data for this Ligand-Target Pair
Affinity DataIC50: 254nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB2 receptor expressed in CHO cellMore data for this Ligand-Target Pair
Affinity DataIC50: 285nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB2 receptor expressed in CHO cellMore data for this Ligand-Target Pair
Affinity DataIC50: 301nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 322nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB2 receptor expressed in CHO cellMore data for this Ligand-Target Pair
Affinity DataIC50: 353nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB2 receptor expressed in CHO cellMore data for this Ligand-Target Pair
Affinity DataIC50: 419nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB2 receptor expressed in CHO cellMore data for this Ligand-Target Pair
Affinity DataIC50: 547nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB2 receptor expressed in CHO cellMore data for this Ligand-Target Pair
Affinity DataIC50: 699nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB2 receptor expressed in CHO cellMore data for this Ligand-Target Pair
Affinity DataIC50: 1.41E+3nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB2 receptor expressed in CHO cellMore data for this Ligand-Target Pair
Affinity DataIC50: 1.72E+3nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB2 receptor expressed in CHO cellMore data for this Ligand-Target Pair
Affinity DataIC50: 1.83E+3nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB2 receptor expressed in CHO cellMore data for this Ligand-Target Pair
Affinity DataIC50: 2.03E+3nMAssay Description:Inhibition of CYP3A4More data for this Ligand-Target Pair
Affinity DataIC50: 2.31E+3nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB2 receptor expressed in CHO cellMore data for this Ligand-Target Pair
Affinity DataIC50: 2.98E+3nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 3.21E+3nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB2 receptor expressed in CHO cellMore data for this Ligand-Target Pair
Affinity DataIC50: 3.86E+3nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB2 receptor expressed in CHO cellMore data for this Ligand-Target Pair
Affinity DataIC50: 5.16E+3nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB2 receptor expressed in CHO cellMore data for this Ligand-Target Pair
Affinity DataIC50: 6.11E+3nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB2 receptor expressed in CHO cellMore data for this Ligand-Target Pair
Affinity DataIC50: 1.33E+4nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB2 receptor expressed in CHO cellMore data for this Ligand-Target Pair
Affinity DataIC50: 1.40E+4nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB2 receptor expressed in CHO cellMore data for this Ligand-Target Pair
Affinity DataIC50: 2.59E+4nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB2 receptor expressed in CHO cellMore data for this Ligand-Target Pair
Affinity DataIC50: >3.50E+4nMAssay Description:Inhibition of CYP3A4More data for this Ligand-Target Pair
Affinity DataEC50: 1.90nMAssay Description:Inverse agonist activity at human CB1 receptor assessed as forskolin-induced cAMP level by adenylyl cyclase activation flash plate assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.900nMAssay Description:Inverse agonist activity at human CB1 receptor assessed as forskolin-induced cAMP level by adenylyl cyclase activation flash plate assayMore data for this Ligand-Target Pair
Affinity DataEC50: 3.20nMAssay Description:Inverse agonist activity at human CB1 receptor assessed as forskolin-induced cAMP level by adenylyl cyclase activation flash plate assayMore data for this Ligand-Target Pair
Affinity DataEC50: 2.40nMAssay Description:Inverse agonist activity at human CB1 receptor assessed as forskolin-induced cAMP level by adenylyl cyclase activation flash plate assayMore data for this Ligand-Target Pair
Affinity DataEC50: 3.5nMAssay Description:Inverse agonist activity at human CB1 receptor assessed as forskolin-induced cAMP level by adenylyl cyclase activation flash plate assayMore data for this Ligand-Target Pair