Compile Data Set for Download or QSAR
maximum 50k data
Found 3 Enz. Inhib. hit(s) with all data for entry = 50031650
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50316633((S)-N-((4-(3-(dimethylamino)propyl)isoquinolin-3-y...)
Affinity DataIC50:  3.40nMAssay Description:Binding affinity to human CXCR4 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50316634((S)-2-(dimethylamino)-N-((3-((methyl(5,6,7,8-tetra...)
Affinity DataIC50:  16nMAssay Description:Binding affinity to human CXCR4 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50315287((R)-N1-((1H-benzo[d]imidazol-2-yl)methyl)-N1-(5,6,...)
Affinity DataIC50:  36nMAssay Description:Binding affinity to human CXCR4 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed