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Compile Data Set for Download or QSAR

Found 60 hits Enz. Inhib. hit(s) with all data for entry = 50033930   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Corticotropin releasing factor receptor 1


(Homo sapiens (Human))
BDBM50354028
PNG
(CHEMBL1830524)
Show SMILES CCC(CC)n1ccc2c(Nc3ccc(OC)cc3CC)nc3ccnn3c12
Show InChI InChI=1S/C22H27N5O/c1-5-15-14-17(28-4)8-9-19(15)24-21-18-11-13-26(16(6-2)7-3)22(18)27-20(25-21)10-12-23-27/h8-14,16H,5-7H2,1-4H3,(H,24,25)
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n/an/a 2.40n/an/an/an/an/an/a



Minase Research Institute

Curated by ChEMBL


Assay Description
Displacement of [125I]-CRF from human CRF1 receptor expressed in CHO-K1 cells after 2 hrs by gamma counting


Bioorg Med Chem 19: 5955-66 (2011)


Article DOI: 10.1016/j.bmc.2011.08.055
BindingDB Entry DOI: 10.7270/Q24X5862
More data for this
Ligand-Target Pair
Corticotropin releasing factor receptor 1


(Homo sapiens (Human))
BDBM50354027
PNG
(CHEMBL1830523)
Show SMILES CCC(CC)n1ccc2c(Nc3ccc(OC)cc3Cl)nc3ccnn3c12
Show InChI InChI=1S/C20H22ClN5O/c1-4-13(5-2)25-11-9-15-19(24-18-8-10-22-26(18)20(15)25)23-17-7-6-14(27-3)12-16(17)21/h6-13H,4-5H2,1-3H3,(H,23,24)
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n/an/a 3.20n/an/an/an/an/an/a



Minase Research Institute

Curated by ChEMBL


Assay Description
Displacement of [125I]-CRF from human CRF1 receptor expressed in CHO-K1 cells after 2 hrs by gamma counting


Bioorg Med Chem 19: 5955-66 (2011)


Article DOI: 10.1016/j.bmc.2011.08.055
BindingDB Entry DOI: 10.7270/Q24X5862
More data for this
Ligand-Target Pair
Corticotropin releasing factor receptor 1


(Homo sapiens (Human))
BDBM50354036
PNG
(CHEMBL1828890)
Show SMILES CCCN(CCC)c1c(CC)c(Nc2ccc(OC)cc2Cl)nc2ccnn12
Show InChI InChI=1S/C21H28ClN5O/c1-5-12-26(13-6-2)21-16(7-3)20(25-19-10-11-23-27(19)21)24-18-9-8-15(28-4)14-17(18)22/h8-11,14H,5-7,12-13H2,1-4H3,(H,24,25)
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n/an/a 4.20n/an/an/an/an/an/a



Minase Research Institute

Curated by ChEMBL


Assay Description
Displacement of [125I]-CRF from human CRF1 receptor expressed in CHO-K1 cells after 2 hrs by gamma counting


Bioorg Med Chem 19: 5955-66 (2011)


Article DOI: 10.1016/j.bmc.2011.08.055
BindingDB Entry DOI: 10.7270/Q24X5862
More data for this
Ligand-Target Pair
Corticotropin releasing factor receptor 1


(Homo sapiens (Human))
BDBM50354015
PNG
(CHEMBL1828900)
Show SMILES CCCN(CCC)c1cc(nc2ccnn12)N(CC=C)c1ccc(OC)cc1Cl
Show InChI InChI=1S/C22H28ClN5O/c1-5-12-26(13-6-2)22-16-21(25-20-10-11-24-28(20)22)27(14-7-3)19-9-8-17(29-4)15-18(19)23/h7-11,15-16H,3,5-6,12-14H2,1-2,4H3
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n/an/a 4.40n/an/an/an/an/an/a



Minase Research Institute

Curated by ChEMBL


Assay Description
Displacement of [125I]-CRF from human CRF1 receptor expressed in CHO-K1 cells after 2 hrs by gamma counting


Bioorg Med Chem 19: 5955-66 (2011)


Article DOI: 10.1016/j.bmc.2011.08.055
BindingDB Entry DOI: 10.7270/Q24X5862
More data for this
Ligand-Target Pair
Corticotropin releasing factor receptor 1


(Homo sapiens (Human))
BDBM50354029
PNG
(CHEMBL1830525)
Show SMILES CCC(CC)n1ccc2c(Nc3ccc(Cl)cc3CC)nc3ccnn3c12
Show InChI InChI=1S/C21H24ClN5/c1-4-14-13-15(22)7-8-18(14)24-20-17-10-12-26(16(5-2)6-3)21(17)27-19(25-20)9-11-23-27/h7-13,16H,4-6H2,1-3H3,(H,24,25)
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n/an/a 4.70n/an/an/an/an/an/a



Minase Research Institute

Curated by ChEMBL


Assay Description
Displacement of [125I]-CRF from human CRF1 receptor expressed in CHO-K1 cells after 2 hrs by gamma counting


Bioorg Med Chem 19: 5955-66 (2011)


Article DOI: 10.1016/j.bmc.2011.08.055
BindingDB Entry DOI: 10.7270/Q24X5862
More data for this
Ligand-Target Pair
Corticotropin releasing factor receptor 1


(Homo sapiens (Human))
BDBM50354038
PNG
(CHEMBL1830527)
Show SMILES CCC(CC)n1ccc2c(Nc3c(C)cc(C)cc3C)nc3ccnn3c12
Show InChI InChI=1S/C22H27N5/c1-6-17(7-2)26-11-9-18-21(24-19-8-10-23-27(19)22(18)26)25-20-15(4)12-14(3)13-16(20)5/h8-13,17H,6-7H2,1-5H3,(H,24,25)
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n/an/a 6.10n/an/an/an/an/an/a



Minase Research Institute

Curated by ChEMBL


Assay Description
Displacement of [125I]-CRF from human CRF1 receptor expressed in CHO-K1 cells after 2 hrs by gamma counting


Bioorg Med Chem 19: 5955-66 (2011)


Article DOI: 10.1016/j.bmc.2011.08.055
BindingDB Entry DOI: 10.7270/Q24X5862
More data for this
Ligand-Target Pair
Corticotropin releasing factor receptor 1


(Homo sapiens (Human))
BDBM50354031
PNG
(CHEMBL1830528)
Show SMILES CCC(CC)n1ccc2c(Oc3ccc(CC)cc3OC)nc3ccnn3c12
Show InChI InChI=1S/C22H26N4O2/c1-5-15-8-9-18(19(14-15)27-4)28-21-17-11-13-25(16(6-2)7-3)22(17)26-20(24-21)10-12-23-26/h8-14,16H,5-7H2,1-4H3
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n/an/a 7n/an/an/an/an/an/a



Minase Research Institute

Curated by ChEMBL


Assay Description
Displacement of [125I]-CRF from human CRF1 receptor expressed in CHO-K1 cells after 2 hrs by gamma counting


Bioorg Med Chem 19: 5955-66 (2011)


Article DOI: 10.1016/j.bmc.2011.08.055
BindingDB Entry DOI: 10.7270/Q24X5862
More data for this
Ligand-Target Pair
Corticotropin releasing factor receptor 1


(Homo sapiens (Human))
BDBM50354030
PNG
(CHEMBL1830526)
Show SMILES CCC(CC)n1ccc2c(Cc3c(C)cc(C)cc3C)nc3ccnn3c12
Show InChI InChI=1S/C23H28N4/c1-6-18(7-2)26-11-9-19-21(25-22-8-10-24-27(22)23(19)26)14-20-16(4)12-15(3)13-17(20)5/h8-13,18H,6-7,14H2,1-5H3
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n/an/a 7.10n/an/an/an/an/an/a



Minase Research Institute

Curated by ChEMBL


Assay Description
Displacement of [125I]-CRF from human CRF1 receptor expressed in CHO-K1 cells after 2 hrs by gamma counting


Bioorg Med Chem 19: 5955-66 (2011)


Article DOI: 10.1016/j.bmc.2011.08.055
BindingDB Entry DOI: 10.7270/Q24X5862
More data for this
Ligand-Target Pair
Corticotropin releasing factor receptor 1


(Homo sapiens (Human))
BDBM50354033
PNG
(CHEMBL1828887)
Show SMILES CCC(CC)Nc1c(C)c(Nc2ccc(OC)cc2Cl)nc2ccnn12
Show InChI InChI=1S/C19H24ClN5O/c1-5-13(6-2)22-19-12(3)18(24-17-9-10-21-25(17)19)23-16-8-7-14(26-4)11-15(16)20/h7-11,13,22H,5-6H2,1-4H3,(H,23,24)
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n/an/a 7.40n/an/an/an/an/an/a



Minase Research Institute

Curated by ChEMBL


Assay Description
Displacement of [125I]-CRF from human CRF1 receptor expressed in CHO-K1 cells after 2 hrs by gamma counting


Bioorg Med Chem 19: 5955-66 (2011)


Article DOI: 10.1016/j.bmc.2011.08.055
BindingDB Entry DOI: 10.7270/Q24X5862
More data for this
Ligand-Target Pair
Corticotropin releasing factor receptor 1


(Homo sapiens (Human))
BDBM50354021
PNG
(CHEMBL1830517)
Show SMILES CCCN(CCC)c1c(C)c(Nc2ccc(OC)cc2Cl)nc2ncnn12
Show InChI InChI=1S/C19H25ClN6O/c1-5-9-25(10-6-2)18-13(3)17(24-19-21-12-22-26(18)19)23-16-8-7-14(27-4)11-15(16)20/h7-8,11-12H,5-6,9-10H2,1-4H3,(H,21,22,23,24)
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n/an/a 8n/an/an/an/an/an/a



Minase Research Institute

Curated by ChEMBL


Assay Description
Displacement of [125I]-CRF from human CRF1 receptor expressed in CHO-K1 cells after 2 hrs by gamma counting


Bioorg Med Chem 19: 5955-66 (2011)


Article DOI: 10.1016/j.bmc.2011.08.055
BindingDB Entry DOI: 10.7270/Q24X5862
More data for this
Ligand-Target Pair
Corticotropin releasing factor receptor 1


(Homo sapiens (Human))
BDBM50354035
PNG
(CHEMBL1828889)
Show SMILES CCCN(CCC)c1c(C)c(Nc2ccc(OC)cc2Cl)nc2ccnn12
Show InChI InChI=1S/C20H26ClN5O/c1-5-11-25(12-6-2)20-14(3)19(24-18-9-10-22-26(18)20)23-17-8-7-15(27-4)13-16(17)21/h7-10,13H,5-6,11-12H2,1-4H3,(H,23,24)
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n/an/a 8n/an/an/an/an/an/a



Minase Research Institute

Curated by ChEMBL


Assay Description
Displacement of [125I]-CRF from human CRF1 receptor expressed in CHO-K1 cells after 2 hrs by gamma counting


Bioorg Med Chem 19: 5955-66 (2011)


Article DOI: 10.1016/j.bmc.2011.08.055
BindingDB Entry DOI: 10.7270/Q24X5862
More data for this
Ligand-Target Pair
Corticotropin releasing factor receptor 1


(Homo sapiens (Human))
BDBM50354023
PNG
(CHEMBL1830519)
Show SMILES CCCN(CCC)c1c(C)c(Nc2ccc(OC)cc2Cl)nc2nccn12
Show InChI InChI=1S/C20H26ClN5O/c1-5-10-25(11-6-2)19-14(3)18(24-20-22-9-12-26(19)20)23-17-8-7-15(27-4)13-16(17)21/h7-9,12-13H,5-6,10-11H2,1-4H3,(H,22,23,24)
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n/an/a 12n/an/an/an/an/an/a



Minase Research Institute

Curated by ChEMBL


Assay Description
Displacement of [125I]-CRF from human CRF1 receptor expressed in CHO-K1 cells after 2 hrs by gamma counting


Bioorg Med Chem 19: 5955-66 (2011)


Article DOI: 10.1016/j.bmc.2011.08.055
BindingDB Entry DOI: 10.7270/Q24X5862
More data for this
Ligand-Target Pair
Corticotropin releasing factor receptor 1


(Homo sapiens (Human))
BDBM50354010
PNG
(CHEMBL1828895)
Show SMILES CCCN(CCC)c1c(OC)c(Nc2ccc(OC)cc2Cl)nc2ccnn12
Show InChI InChI=1S/C20H26ClN5O2/c1-5-11-25(12-6-2)20-18(28-4)19(24-17-9-10-22-26(17)20)23-16-8-7-14(27-3)13-15(16)21/h7-10,13H,5-6,11-12H2,1-4H3,(H,23,24)
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n/an/a 13n/an/an/an/an/an/a



Minase Research Institute

Curated by ChEMBL


Assay Description
Displacement of [125I]-CRF from human CRF1 receptor expressed in CHO-K1 cells after 2 hrs by gamma counting


Bioorg Med Chem 19: 5955-66 (2011)


Article DOI: 10.1016/j.bmc.2011.08.055
BindingDB Entry DOI: 10.7270/Q24X5862
More data for this
Ligand-Target Pair
Corticotropin releasing factor receptor 1


(Homo sapiens (Human))
BDBM50354032
PNG
(CHEMBL1828886)
Show SMILES CCC(CC)Nc1cc(Nc2ccc(OC)cc2Cl)nc2ccnn12
Show InChI InChI=1S/C18H22ClN5O/c1-4-12(5-2)21-18-11-16(23-17-8-9-20-24(17)18)22-15-7-6-13(25-3)10-14(15)19/h6-12,21H,4-5H2,1-3H3,(H,22,23)
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n/an/a 14n/an/an/an/an/an/a



Minase Research Institute

Curated by ChEMBL


Assay Description
Displacement of [125I]-CRF from human CRF1 receptor expressed in CHO-K1 cells after 2 hrs by gamma counting


Bioorg Med Chem 19: 5955-66 (2011)


Article DOI: 10.1016/j.bmc.2011.08.055
BindingDB Entry DOI: 10.7270/Q24X5862
More data for this
Ligand-Target Pair
Corticotropin releasing factor receptor 1


(Homo sapiens (Human))
BDBM50354018
PNG
(CHEMBL1830514)
Show SMILES CCCN(CCC)c1cc(nc2ccnn12)N(COC)c1ccc(OC)cc1Cl
Show InChI InChI=1S/C21H28ClN5O2/c1-5-11-25(12-6-2)21-14-20(24-19-9-10-23-27(19)21)26(15-28-3)18-8-7-16(29-4)13-17(18)22/h7-10,13-14H,5-6,11-12,15H2,1-4H3
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n/an/a 15n/an/an/an/an/an/a



Minase Research Institute

Curated by ChEMBL


Assay Description
Displacement of [125I]-CRF from human CRF1 receptor expressed in CHO-K1 cells after 2 hrs by gamma counting


Bioorg Med Chem 19: 5955-66 (2011)


Article DOI: 10.1016/j.bmc.2011.08.055
BindingDB Entry DOI: 10.7270/Q24X5862
More data for this
Ligand-Target Pair
Corticotropin releasing factor receptor 1


(Homo sapiens (Human))
BDBM50354019
PNG
(CHEMBL1830515)
Show SMILES CCC(CC)Nc1c(C)c(Nc2ccc(OC)cc2Cl)nc2ncnn12
Show InChI InChI=1S/C18H23ClN6O/c1-5-12(6-2)22-17-11(3)16(24-18-20-10-21-25(17)18)23-15-8-7-13(26-4)9-14(15)19/h7-10,12,22H,5-6H2,1-4H3,(H,20,21,23,24)
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n/an/a 16n/an/an/an/an/an/a



Minase Research Institute

Curated by ChEMBL


Assay Description
Displacement of [125I]-CRF from human CRF1 receptor expressed in CHO-K1 cells after 2 hrs by gamma counting


Bioorg Med Chem 19: 5955-66 (2011)


Article DOI: 10.1016/j.bmc.2011.08.055
BindingDB Entry DOI: 10.7270/Q24X5862
More data for this
Ligand-Target Pair
Corticotropin releasing factor receptor 1


(Homo sapiens (Human))
BDBM50354026
PNG
(CHEMBL1830522)
Show SMILES CCCN(CCC)c1nc(nc2ccnn12)N(C)c1ccc(OC)cc1Cl
Show InChI InChI=1S/C19H25ClN6O/c1-5-11-25(12-6-2)19-23-18(22-17-9-10-21-26(17)19)24(3)16-8-7-14(27-4)13-15(16)20/h7-10,13H,5-6,11-12H2,1-4H3
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n/an/a 20n/an/an/an/an/an/a



Minase Research Institute

Curated by ChEMBL


Assay Description
Displacement of [125I]-CRF from human CRF1 receptor expressed in CHO-K1 cells after 2 hrs by gamma counting


Bioorg Med Chem 19: 5955-66 (2011)


Article DOI: 10.1016/j.bmc.2011.08.055
BindingDB Entry DOI: 10.7270/Q24X5862
More data for this
Ligand-Target Pair
Corticotropin releasing factor receptor 1


(Homo sapiens (Human))
BDBM50354011
PNG
(CHEMBL1828896)
Show SMILES CCCN(CCC)c1cc(nc2ccnn12)N(C)c1ccc(OC)cc1Cl
Show InChI InChI=1S/C20H26ClN5O/c1-5-11-25(12-6-2)20-14-19(23-18-9-10-22-26(18)20)24(3)17-8-7-15(27-4)13-16(17)21/h7-10,13-14H,5-6,11-12H2,1-4H3
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Minase Research Institute

Curated by ChEMBL


Assay Description
Displacement of [125I]-CRF from human CRF1 receptor expressed in CHO-K1 cells after 2 hrs by gamma counting


Bioorg Med Chem 19: 5955-66 (2011)


Article DOI: 10.1016/j.bmc.2011.08.055
BindingDB Entry DOI: 10.7270/Q24X5862
More data for this
Ligand-Target Pair
Corticotropin releasing factor receptor 1


(Homo sapiens (Human))
BDBM50354012
PNG
(CHEMBL1828897)
Show SMILES CCCN(CCC)c1cc(nc2ccnn12)N(CC)c1ccc(OC)cc1Cl
Show InChI InChI=1S/C21H28ClN5O/c1-5-12-25(13-6-2)21-15-20(24-19-10-11-23-27(19)21)26(7-3)18-9-8-16(28-4)14-17(18)22/h8-11,14-15H,5-7,12-13H2,1-4H3
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n/an/a 31.6n/an/an/an/an/an/a



Minase Research Institute

Curated by ChEMBL


Assay Description
Displacement of [125I]-CRF from human CRF1 receptor expressed in CHO-K1 cells after 2 hrs by gamma counting


Bioorg Med Chem 19: 5955-66 (2011)


Article DOI: 10.1016/j.bmc.2011.08.055
BindingDB Entry DOI: 10.7270/Q24X5862
More data for this
Ligand-Target Pair
Corticotropin releasing factor receptor 1


(Homo sapiens (Human))
BDBM50354037
PNG
(CHEMBL1828891)
Show SMILES CCCN(CCC)c1c(CCC)c(Nc2ccc(OC)cc2Cl)nc2ccnn12
Show InChI InChI=1S/C22H30ClN5O/c1-5-8-17-21(25-19-10-9-16(29-4)15-18(19)23)26-20-11-12-24-28(20)22(17)27(13-6-2)14-7-3/h9-12,15H,5-8,13-14H2,1-4H3,(H,25,26)
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n/an/a 32n/an/an/an/an/an/a



Minase Research Institute

Curated by ChEMBL


Assay Description
Displacement of [125I]-CRF from human CRF1 receptor expressed in CHO-K1 cells after 2 hrs by gamma counting


Bioorg Med Chem 19: 5955-66 (2011)


Article DOI: 10.1016/j.bmc.2011.08.055
BindingDB Entry DOI: 10.7270/Q24X5862
More data for this
Ligand-Target Pair
Corticotropin releasing factor receptor 1


(Homo sapiens (Human))
BDBM50354022
PNG
(CHEMBL1830518)
Show SMILES CCCN(CCC)c1cc(nc2ncnn12)N(C)c1ccc(OC)cc1Cl
Show InChI InChI=1S/C19H25ClN6O/c1-5-9-25(10-6-2)18-12-17(23-19-21-13-22-26(18)19)24(3)16-8-7-14(27-4)11-15(16)20/h7-8,11-13H,5-6,9-10H2,1-4H3
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n/an/a 33n/an/an/an/an/an/a



Minase Research Institute

Curated by ChEMBL


Assay Description
Displacement of [125I]-CRF from human CRF1 receptor expressed in CHO-K1 cells after 2 hrs by gamma counting


Bioorg Med Chem 19: 5955-66 (2011)


Article DOI: 10.1016/j.bmc.2011.08.055
BindingDB Entry DOI: 10.7270/Q24X5862
More data for this
Ligand-Target Pair
Corticotropin releasing factor receptor 1


(Homo sapiens (Human))
BDBM50354025
PNG
(CHEMBL1830521)
Show SMILES CCCN(CCC)c1cc(nc2nccn12)N(CC)c1ccc(OC)cc1Cl
Show InChI InChI=1S/C21H28ClN5O/c1-5-11-25(12-6-2)20-15-19(24-21-23-10-13-27(20)21)26(7-3)18-9-8-16(28-4)14-17(18)22/h8-10,13-15H,5-7,11-12H2,1-4H3
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n/an/a 42n/an/an/an/an/an/a



Minase Research Institute

Curated by ChEMBL


Assay Description
Displacement of [125I]-CRF from human CRF1 receptor expressed in CHO-K1 cells after 2 hrs by gamma counting


Bioorg Med Chem 19: 5955-66 (2011)


Article DOI: 10.1016/j.bmc.2011.08.055
BindingDB Entry DOI: 10.7270/Q24X5862
More data for this
Ligand-Target Pair
Corticotropin releasing factor receptor 1


(Homo sapiens (Human))
BDBM50354020
PNG
(CHEMBL1830516)
Show SMILES CCC(CC)Nc1cc(nc2ncnn12)N(C)c1ccc(OC)cc1Cl
Show InChI InChI=1S/C18H23ClN6O/c1-5-12(6-2)22-17-10-16(23-18-20-11-21-25(17)18)24(3)15-8-7-13(26-4)9-14(15)19/h7-12,22H,5-6H2,1-4H3
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n/an/a 42n/an/an/an/an/an/a



Minase Research Institute

Curated by ChEMBL


Assay Description
Displacement of [125I]-CRF from human CRF1 receptor expressed in CHO-K1 cells after 2 hrs by gamma counting


Bioorg Med Chem 19: 5955-66 (2011)


Article DOI: 10.1016/j.bmc.2011.08.055
BindingDB Entry DOI: 10.7270/Q24X5862
More data for this
Ligand-Target Pair
Corticotropin releasing factor receptor 1


(Homo sapiens (Human))
BDBM50354034
PNG
(CHEMBL1828888)
Show SMILES CCCN(CCC)c1cc(Nc2ccc(OC)cc2Cl)nc2ccnn12
Show InChI InChI=1S/C19H24ClN5O/c1-4-10-24(11-5-2)19-13-17(23-18-8-9-21-25(18)19)22-16-7-6-14(26-3)12-15(16)20/h6-9,12-13H,4-5,10-11H2,1-3H3,(H,22,23)
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n/an/a 61n/an/an/an/an/an/a



Minase Research Institute

Curated by ChEMBL


Assay Description
Displacement of [125I]-CRF from human CRF1 receptor expressed in CHO-K1 cells after 2 hrs by gamma counting


Bioorg Med Chem 19: 5955-66 (2011)


Article DOI: 10.1016/j.bmc.2011.08.055
BindingDB Entry DOI: 10.7270/Q24X5862
More data for this
Ligand-Target Pair
Corticotropin releasing factor receptor 1


(Homo sapiens (Human))
BDBM50354024
PNG
(CHEMBL1830520)
Show SMILES CCCN(CCC)c1cc(nc2nccn12)N(C)c1ccc(OC)cc1Cl
Show InChI InChI=1S/C20H26ClN5O/c1-5-10-25(11-6-2)19-14-18(23-20-22-9-12-26(19)20)24(3)17-8-7-15(27-4)13-16(17)21/h7-9,12-14H,5-6,10-11H2,1-4H3
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n/an/a 67n/an/an/an/an/an/a



Minase Research Institute

Curated by ChEMBL


Assay Description
Displacement of [125I]-CRF from human CRF1 receptor expressed in CHO-K1 cells after 2 hrs by gamma counting


Bioorg Med Chem 19: 5955-66 (2011)


Article DOI: 10.1016/j.bmc.2011.08.055
BindingDB Entry DOI: 10.7270/Q24X5862
More data for this
Ligand-Target Pair
Corticotropin releasing factor receptor 1


(Homo sapiens (Human))
BDBM50354014
PNG
(CHEMBL1828899)
Show SMILES CCCN(CCC)c1cc(nc2ccnn12)N(CC(C)=C)c1ccc(OC)cc1Cl
Show InChI InChI=1S/C23H30ClN5O/c1-6-12-27(13-7-2)23-15-22(26-21-10-11-25-29(21)23)28(16-17(3)4)20-9-8-18(30-5)14-19(20)24/h8-11,14-15H,3,6-7,12-13,16H2,1-2,4-5H3
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n/an/a 76.7n/an/an/an/an/an/a



Minase Research Institute

Curated by ChEMBL


Assay Description
Displacement of [125I]-CRF from human CRF1 receptor expressed in CHO-K1 cells after 2 hrs by gamma counting


Bioorg Med Chem 19: 5955-66 (2011)


Article DOI: 10.1016/j.bmc.2011.08.055
BindingDB Entry DOI: 10.7270/Q24X5862
More data for this
Ligand-Target Pair
Corticotropin releasing factor receptor 1


(Homo sapiens (Human))
BDBM50354007
PNG
(CHEMBL1828892)
Show SMILES CCCN(CCC)c1c(C(C)C)c(Nc2ccc(OC)cc2Cl)nc2ccnn12
Show InChI InChI=1S/C22H30ClN5O/c1-6-12-27(13-7-2)22-20(15(3)4)21(26-19-10-11-24-28(19)22)25-18-9-8-16(29-5)14-17(18)23/h8-11,14-15H,6-7,12-13H2,1-5H3,(H,25,26)
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n/an/a 113n/an/an/an/an/an/a



Minase Research Institute

Curated by ChEMBL


Assay Description
Displacement of [125I]-CRF from human CRF1 receptor expressed in CHO-K1 cells after 2 hrs by gamma counting


Bioorg Med Chem 19: 5955-66 (2011)


Article DOI: 10.1016/j.bmc.2011.08.055
BindingDB Entry DOI: 10.7270/Q24X5862
More data for this
Ligand-Target Pair
Corticotropin releasing factor receptor 1


(Homo sapiens (Human))
BDBM50354016
PNG
(CHEMBL1828901)
Show SMILES CCCN(CCC)c1cc(nc2ccnn12)N(CC1CC1)c1ccc(OC)cc1Cl
Show InChI InChI=1S/C23H30ClN5O/c1-4-12-27(13-5-2)23-15-22(26-21-10-11-25-29(21)23)28(16-17-6-7-17)20-9-8-18(30-3)14-19(20)24/h8-11,14-15,17H,4-7,12-13,16H2,1-3H3
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n/an/a 213n/an/an/an/an/an/a



Minase Research Institute

Curated by ChEMBL


Assay Description
Displacement of [125I]-CRF from human CRF1 receptor expressed in CHO-K1 cells after 2 hrs by gamma counting


Bioorg Med Chem 19: 5955-66 (2011)


Article DOI: 10.1016/j.bmc.2011.08.055
BindingDB Entry DOI: 10.7270/Q24X5862
More data for this
Ligand-Target Pair
Corticotropin releasing factor receptor 1


(Homo sapiens (Human))
BDBM50354009
PNG
(CHEMBL1828894)
Show SMILES CCCN(CCC)c1c(C2CCCC2)c(Nc2ccc(OC)cc2Cl)nc2ccnn12
Show InChI InChI=1S/C24H32ClN5O/c1-4-14-29(15-5-2)24-22(17-8-6-7-9-17)23(28-21-12-13-26-30(21)24)27-20-11-10-18(31-3)16-19(20)25/h10-13,16-17H,4-9,14-15H2,1-3H3,(H,27,28)
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n/an/a 308n/an/an/an/an/an/a



Minase Research Institute

Curated by ChEMBL


Assay Description
Displacement of [125I]-CRF from human CRF1 receptor expressed in CHO-K1 cells after 2 hrs by gamma counting


Bioorg Med Chem 19: 5955-66 (2011)


Article DOI: 10.1016/j.bmc.2011.08.055
BindingDB Entry DOI: 10.7270/Q24X5862
More data for this
Ligand-Target Pair
Corticotropin releasing factor receptor 1


(Homo sapiens (Human))
BDBM50354008
PNG
(CHEMBL1828893)
Show SMILES CCCCc1c(Nc2ccc(OC)cc2Cl)nc2ccnn2c1N(CCC)CCC
Show InChI InChI=1S/C23H32ClN5O/c1-5-8-9-18-22(26-20-11-10-17(30-4)16-19(20)24)27-21-12-13-25-29(21)23(18)28(14-6-2)15-7-3/h10-13,16H,5-9,14-15H2,1-4H3,(H,26,27)
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n/an/a 340n/an/an/an/an/an/a



Minase Research Institute

Curated by ChEMBL


Assay Description
Displacement of [125I]-CRF from human CRF1 receptor expressed in CHO-K1 cells after 2 hrs by gamma counting


Bioorg Med Chem 19: 5955-66 (2011)


Article DOI: 10.1016/j.bmc.2011.08.055
BindingDB Entry DOI: 10.7270/Q24X5862
More data for this
Ligand-Target Pair
Corticotropin releasing factor receptor 1


(Homo sapiens (Human))
BDBM50354013
PNG
(CHEMBL1828898)
Show SMILES CCCN(CCC)c1cc(nc2ccnn12)N(CCC)c1ccc(OC)cc1Cl
Show InChI InChI=1S/C22H30ClN5O/c1-5-12-26(13-6-2)22-16-21(25-20-10-11-24-28(20)22)27(14-7-3)19-9-8-17(29-4)15-18(19)23/h8-11,15-16H,5-7,12-14H2,1-4H3
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n/an/a 418n/an/an/an/an/an/a



Minase Research Institute

Curated by ChEMBL


Assay Description
Displacement of [125I]-CRF from human CRF1 receptor expressed in CHO-K1 cells after 2 hrs by gamma counting


Bioorg Med Chem 19: 5955-66 (2011)


Article DOI: 10.1016/j.bmc.2011.08.055
BindingDB Entry DOI: 10.7270/Q24X5862
More data for this
Ligand-Target Pair
Corticotropin releasing factor receptor 1


(Homo sapiens (Human))
BDBM50354017
PNG
(CHEMBL1830513)
Show SMILES CCCN(CCC)c1cc(nc2ccnn12)N(CCOC)c1ccc(OC)cc1Cl
Show InChI InChI=1S/C22H30ClN5O2/c1-5-11-26(12-6-2)22-16-21(25-20-9-10-24-28(20)22)27(13-14-29-3)19-8-7-17(30-4)15-18(19)23/h7-10,15-16H,5-6,11-14H2,1-4H3
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Minase Research Institute

Curated by ChEMBL


Assay Description
Displacement of [125I]-CRF from human CRF1 receptor expressed in CHO-K1 cells after 2 hrs by gamma counting


Bioorg Med Chem 19: 5955-66 (2011)


Article DOI: 10.1016/j.bmc.2011.08.055
BindingDB Entry DOI: 10.7270/Q24X5862
More data for this
Ligand-Target Pair
Corticotropin releasing factor receptor 1


(Homo sapiens (Human))
BDBM50354010
PNG
(CHEMBL1828895)
Show SMILES CCCN(CCC)c1c(OC)c(Nc2ccc(OC)cc2Cl)nc2ccnn12
Show InChI InChI=1S/C20H26ClN5O2/c1-5-11-25(12-6-2)20-18(28-4)19(24-17-9-10-22-26(17)20)23-16-8-7-14(27-3)13-15(16)21/h7-10,13H,5-6,11-12H2,1-4H3,(H,23,24)
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n/an/an/an/a 883n/an/an/an/a



Minase Research Institute

Curated by ChEMBL


Assay Description
Antagonist activity at human CRF1 receptor expressed in CHO-K1 cells assessed as inhibition of CRF-induced cAMP accumulation after 15 mins by cAMP en...


Bioorg Med Chem 19: 5955-66 (2011)


Article DOI: 10.1016/j.bmc.2011.08.055
BindingDB Entry DOI: 10.7270/Q24X5862
More data for this
Ligand-Target Pair
Corticotropin releasing factor receptor 1


(Homo sapiens (Human))
BDBM50354011
PNG
(CHEMBL1828896)
Show SMILES CCCN(CCC)c1cc(nc2ccnn12)N(C)c1ccc(OC)cc1Cl
Show InChI InChI=1S/C20H26ClN5O/c1-5-11-25(12-6-2)20-14-19(23-18-9-10-22-26(18)20)24(3)17-8-7-15(27-4)13-16(17)21/h7-10,13-14H,5-6,11-12H2,1-4H3
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n/an/an/an/a 97n/an/an/an/a



Minase Research Institute

Curated by ChEMBL


Assay Description
Antagonist activity at human CRF1 receptor expressed in CHO-K1 cells assessed as inhibition of CRF-induced cAMP accumulation after 15 mins by cAMP en...


Bioorg Med Chem 19: 5955-66 (2011)


Article DOI: 10.1016/j.bmc.2011.08.055
BindingDB Entry DOI: 10.7270/Q24X5862
More data for this
Ligand-Target Pair
Corticotropin releasing factor receptor 1


(Homo sapiens (Human))
BDBM50354013
PNG
(CHEMBL1828898)
Show SMILES CCCN(CCC)c1cc(nc2ccnn12)N(CCC)c1ccc(OC)cc1Cl
Show InChI InChI=1S/C22H30ClN5O/c1-5-12-26(13-6-2)22-16-21(25-20-10-11-24-28(20)22)27(14-7-3)19-9-8-17(29-4)15-18(19)23/h8-11,15-16H,5-7,12-14H2,1-4H3
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n/an/an/an/a 75.7n/an/an/an/a



Minase Research Institute

Curated by ChEMBL


Assay Description
Antagonist activity at human CRF1 receptor expressed in CHO-K1 cells assessed as inhibition of CRF-induced cAMP accumulation after 15 mins by cAMP en...


Bioorg Med Chem 19: 5955-66 (2011)


Article DOI: 10.1016/j.bmc.2011.08.055
BindingDB Entry DOI: 10.7270/Q24X5862
More data for this
Ligand-Target Pair
Corticotropin releasing factor receptor 1


(Homo sapiens (Human))
BDBM50354014
PNG
(CHEMBL1828899)
Show SMILES CCCN(CCC)c1cc(nc2ccnn12)N(CC(C)=C)c1ccc(OC)cc1Cl
Show InChI InChI=1S/C23H30ClN5O/c1-6-12-27(13-7-2)23-15-22(26-21-10-11-25-29(21)23)28(16-17(3)4)20-9-8-18(30-5)14-19(20)24/h8-11,14-15H,3,6-7,12-13,16H2,1-2,4-5H3
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Minase Research Institute

Curated by ChEMBL


Assay Description
Antagonist activity at human CRF1 receptor expressed in CHO-K1 cells assessed as inhibition of CRF-induced cAMP accumulation after 15 mins by cAMP en...


Bioorg Med Chem 19: 5955-66 (2011)


Article DOI: 10.1016/j.bmc.2011.08.055
BindingDB Entry DOI: 10.7270/Q24X5862
More data for this
Ligand-Target Pair
Corticotropin releasing factor receptor 1


(Homo sapiens (Human))
BDBM50354015
PNG
(CHEMBL1828900)
Show SMILES CCCN(CCC)c1cc(nc2ccnn12)N(CC=C)c1ccc(OC)cc1Cl
Show InChI InChI=1S/C22H28ClN5O/c1-5-12-26(13-6-2)22-16-21(25-20-10-11-24-28(20)22)27(14-7-3)19-9-8-17(29-4)15-18(19)23/h7-11,15-16H,3,5-6,12-14H2,1-2,4H3
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n/an/an/an/a 28.9n/an/an/an/a



Minase Research Institute

Curated by ChEMBL


Assay Description
Antagonist activity at human CRF1 receptor expressed in CHO-K1 cells assessed as inhibition of CRF-induced cAMP accumulation after 15 mins by cAMP en...


Bioorg Med Chem 19: 5955-66 (2011)


Article DOI: 10.1016/j.bmc.2011.08.055
BindingDB Entry DOI: 10.7270/Q24X5862
More data for this
Ligand-Target Pair
Corticotropin releasing factor receptor 1


(Homo sapiens (Human))
BDBM50354019
PNG
(CHEMBL1830515)
Show SMILES CCC(CC)Nc1c(C)c(Nc2ccc(OC)cc2Cl)nc2ncnn12
Show InChI InChI=1S/C18H23ClN6O/c1-5-12(6-2)22-17-11(3)16(24-18-20-10-21-25(17)18)23-15-8-7-13(26-4)9-14(15)19/h7-10,12,22H,5-6H2,1-4H3,(H,20,21,23,24)
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Minase Research Institute

Curated by ChEMBL


Assay Description
Antagonist activity at human CRF1 receptor expressed in CHO-K1 cells assessed as inhibition of CRF-induced cAMP accumulation after 15 mins by cAMP en...


Bioorg Med Chem 19: 5955-66 (2011)


Article DOI: 10.1016/j.bmc.2011.08.055
BindingDB Entry DOI: 10.7270/Q24X5862
More data for this
Ligand-Target Pair
Corticotropin releasing factor receptor 1


(Homo sapiens (Human))
BDBM50354020
PNG
(CHEMBL1830516)
Show SMILES CCC(CC)Nc1cc(nc2ncnn12)N(C)c1ccc(OC)cc1Cl
Show InChI InChI=1S/C18H23ClN6O/c1-5-12(6-2)22-17-10-16(23-18-20-11-21-25(17)18)24(3)15-8-7-13(26-4)9-14(15)19/h7-12,22H,5-6H2,1-4H3
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Minase Research Institute

Curated by ChEMBL


Assay Description
Antagonist activity at human CRF1 receptor expressed in CHO-K1 cells assessed as inhibition of CRF-induced cAMP accumulation after 15 mins by cAMP en...


Bioorg Med Chem 19: 5955-66 (2011)


Article DOI: 10.1016/j.bmc.2011.08.055
BindingDB Entry DOI: 10.7270/Q24X5862
More data for this
Ligand-Target Pair
Corticotropin releasing factor receptor 1


(Homo sapiens (Human))
BDBM50354021
PNG
(CHEMBL1830517)
Show SMILES CCCN(CCC)c1c(C)c(Nc2ccc(OC)cc2Cl)nc2ncnn12
Show InChI InChI=1S/C19H25ClN6O/c1-5-9-25(10-6-2)18-13(3)17(24-19-21-12-22-26(18)19)23-16-8-7-14(27-4)11-15(16)20/h7-8,11-12H,5-6,9-10H2,1-4H3,(H,21,22,23,24)
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Minase Research Institute

Curated by ChEMBL


Assay Description
Antagonist activity at human CRF1 receptor expressed in CHO-K1 cells assessed as inhibition of CRF-induced cAMP accumulation after 15 mins by cAMP en...


Bioorg Med Chem 19: 5955-66 (2011)


Article DOI: 10.1016/j.bmc.2011.08.055
BindingDB Entry DOI: 10.7270/Q24X5862
More data for this
Ligand-Target Pair
Corticotropin releasing factor receptor 1


(Homo sapiens (Human))
BDBM50354022
PNG
(CHEMBL1830518)
Show SMILES CCCN(CCC)c1cc(nc2ncnn12)N(C)c1ccc(OC)cc1Cl
Show InChI InChI=1S/C19H25ClN6O/c1-5-9-25(10-6-2)18-12-17(23-19-21-13-22-26(18)19)24(3)16-8-7-14(27-4)11-15(16)20/h7-8,11-13H,5-6,9-10H2,1-4H3
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n/an/an/an/a 889n/an/an/an/a



Minase Research Institute

Curated by ChEMBL


Assay Description
Antagonist activity at human CRF1 receptor expressed in CHO-K1 cells assessed as inhibition of CRF-induced cAMP accumulation after 15 mins by cAMP en...


Bioorg Med Chem 19: 5955-66 (2011)


Article DOI: 10.1016/j.bmc.2011.08.055
BindingDB Entry DOI: 10.7270/Q24X5862
More data for this
Ligand-Target Pair
Corticotropin releasing factor receptor 1


(Homo sapiens (Human))
BDBM50354023
PNG
(CHEMBL1830519)
Show SMILES CCCN(CCC)c1c(C)c(Nc2ccc(OC)cc2Cl)nc2nccn12
Show InChI InChI=1S/C20H26ClN5O/c1-5-10-25(11-6-2)19-14(3)18(24-20-22-9-12-26(19)20)23-17-8-7-15(27-4)13-16(17)21/h7-9,12-13H,5-6,10-11H2,1-4H3,(H,22,23,24)
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n/an/an/an/a 46n/an/an/an/a



Minase Research Institute

Curated by ChEMBL


Assay Description
Antagonist activity at human CRF1 receptor expressed in CHO-K1 cells assessed as inhibition of CRF-induced cAMP accumulation after 15 mins by cAMP en...


Bioorg Med Chem 19: 5955-66 (2011)


Article DOI: 10.1016/j.bmc.2011.08.055
BindingDB Entry DOI: 10.7270/Q24X5862
More data for this
Ligand-Target Pair
Corticotropin releasing factor receptor 1


(Homo sapiens (Human))
BDBM50354025
PNG
(CHEMBL1830521)
Show SMILES CCCN(CCC)c1cc(nc2nccn12)N(CC)c1ccc(OC)cc1Cl
Show InChI InChI=1S/C21H28ClN5O/c1-5-11-25(12-6-2)20-15-19(24-21-23-10-13-27(20)21)26(7-3)18-9-8-16(28-4)14-17(18)22/h8-10,13-15H,5-7,11-12H2,1-4H3
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n/an/an/an/a 76n/an/an/an/a



Minase Research Institute

Curated by ChEMBL


Assay Description
Antagonist activity at human CRF1 receptor expressed in CHO-K1 cells assessed as inhibition of CRF-induced cAMP accumulation after 15 mins by cAMP en...


Bioorg Med Chem 19: 5955-66 (2011)


Article DOI: 10.1016/j.bmc.2011.08.055
BindingDB Entry DOI: 10.7270/Q24X5862
More data for this
Ligand-Target Pair
Corticotropin releasing factor receptor 1


(Homo sapiens (Human))
BDBM50354027
PNG
(CHEMBL1830523)
Show SMILES CCC(CC)n1ccc2c(Nc3ccc(OC)cc3Cl)nc3ccnn3c12
Show InChI InChI=1S/C20H22ClN5O/c1-4-13(5-2)25-11-9-15-19(24-18-8-10-22-26(18)20(15)25)23-17-7-6-14(27-3)12-16(17)21/h6-13H,4-5H2,1-3H3,(H,23,24)
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n/an/an/an/a 0.700n/an/an/an/a



Minase Research Institute

Curated by ChEMBL


Assay Description
Antagonist activity at human CRF1 receptor expressed in CHO-K1 cells assessed as inhibition of CRF-induced cAMP accumulation after 15 mins by cAMP en...


Bioorg Med Chem 19: 5955-66 (2011)


Article DOI: 10.1016/j.bmc.2011.08.055
BindingDB Entry DOI: 10.7270/Q24X5862
More data for this
Ligand-Target Pair
Corticotropin releasing factor receptor 1


(Homo sapiens (Human))
BDBM50354028
PNG
(CHEMBL1830524)
Show SMILES CCC(CC)n1ccc2c(Nc3ccc(OC)cc3CC)nc3ccnn3c12
Show InChI InChI=1S/C22H27N5O/c1-5-15-14-17(28-4)8-9-19(15)24-21-18-11-13-26(16(6-2)7-3)22(18)27-20(25-21)10-12-23-27/h8-14,16H,5-7H2,1-4H3,(H,24,25)
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n/an/an/an/a 3.5n/an/an/an/a



Minase Research Institute

Curated by ChEMBL


Assay Description
Antagonist activity at human CRF1 receptor expressed in CHO-K1 cells assessed as inhibition of CRF-induced cAMP accumulation after 15 mins by cAMP en...


Bioorg Med Chem 19: 5955-66 (2011)


Article DOI: 10.1016/j.bmc.2011.08.055
BindingDB Entry DOI: 10.7270/Q24X5862
More data for this
Ligand-Target Pair
Corticotropin releasing factor receptor 1


(Homo sapiens (Human))
BDBM50354029
PNG
(CHEMBL1830525)
Show SMILES CCC(CC)n1ccc2c(Nc3ccc(Cl)cc3CC)nc3ccnn3c12
Show InChI InChI=1S/C21H24ClN5/c1-4-14-13-15(22)7-8-18(14)24-20-17-10-12-26(16(5-2)6-3)21(17)27-19(25-20)9-11-23-27/h7-13,16H,4-6H2,1-3H3,(H,24,25)
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n/an/an/an/a 3.90n/an/an/an/a



Minase Research Institute

Curated by ChEMBL


Assay Description
Antagonist activity at human CRF1 receptor expressed in CHO-K1 cells assessed as inhibition of CRF-induced cAMP accumulation after 15 mins by cAMP en...


Bioorg Med Chem 19: 5955-66 (2011)


Article DOI: 10.1016/j.bmc.2011.08.055
BindingDB Entry DOI: 10.7270/Q24X5862
More data for this
Ligand-Target Pair
Corticotropin releasing factor receptor 1


(Homo sapiens (Human))
BDBM50354030
PNG
(CHEMBL1830526)
Show SMILES CCC(CC)n1ccc2c(Cc3c(C)cc(C)cc3C)nc3ccnn3c12
Show InChI InChI=1S/C23H28N4/c1-6-18(7-2)26-11-9-19-21(25-22-8-10-24-27(22)23(19)26)14-20-16(4)12-15(3)13-17(20)5/h8-13,18H,6-7,14H2,1-5H3
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n/an/an/an/a 32.2n/an/an/an/a



Minase Research Institute

Curated by ChEMBL


Assay Description
Antagonist activity at human CRF1 receptor expressed in CHO-K1 cells assessed as inhibition of CRF-induced cAMP accumulation after 15 mins by cAMP en...


Bioorg Med Chem 19: 5955-66 (2011)


Article DOI: 10.1016/j.bmc.2011.08.055
BindingDB Entry DOI: 10.7270/Q24X5862
More data for this
Ligand-Target Pair
Corticotropin releasing factor receptor 1


(Homo sapiens (Human))
BDBM50354038
PNG
(CHEMBL1830527)
Show SMILES CCC(CC)n1ccc2c(Nc3c(C)cc(C)cc3C)nc3ccnn3c12
Show InChI InChI=1S/C22H27N5/c1-6-17(7-2)26-11-9-18-21(24-19-8-10-23-27(19)22(18)26)25-20-15(4)12-14(3)13-16(20)5/h8-13,17H,6-7H2,1-5H3,(H,24,25)
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n/an/an/an/a 4.10n/an/an/an/a



Minase Research Institute

Curated by ChEMBL


Assay Description
Antagonist activity at human CRF1 receptor expressed in CHO-K1 cells assessed as inhibition of CRF-induced cAMP accumulation after 15 mins by cAMP en...


Bioorg Med Chem 19: 5955-66 (2011)


Article DOI: 10.1016/j.bmc.2011.08.055
BindingDB Entry DOI: 10.7270/Q24X5862
More data for this
Ligand-Target Pair
Corticotropin releasing factor receptor 1


(Homo sapiens (Human))
BDBM50354031
PNG
(CHEMBL1830528)
Show SMILES CCC(CC)n1ccc2c(Oc3ccc(CC)cc3OC)nc3ccnn3c12
Show InChI InChI=1S/C22H26N4O2/c1-5-15-8-9-18(19(14-15)27-4)28-21-17-11-13-25(16(6-2)7-3)22(17)26-20(24-21)10-12-23-26/h8-14,16H,5-7H2,1-4H3
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n/an/an/an/a 5.60n/an/an/an/a



Minase Research Institute

Curated by ChEMBL


Assay Description
Antagonist activity at human CRF1 receptor expressed in CHO-K1 cells assessed as inhibition of CRF-induced cAMP accumulation after 15 mins by cAMP en...


Bioorg Med Chem 19: 5955-66 (2011)


Article DOI: 10.1016/j.bmc.2011.08.055
BindingDB Entry DOI: 10.7270/Q24X5862
More data for this
Ligand-Target Pair
Corticotropin releasing factor receptor


(Rattus norvegicus (rat))
BDBM50354035
PNG
(CHEMBL1828889)
Show SMILES CCCN(CCC)c1c(C)c(Nc2ccc(OC)cc2Cl)nc2ccnn12
Show InChI InChI=1S/C20H26ClN5O/c1-5-11-25(12-6-2)20-14(3)19(24-18-9-10-22-26(18)20)23-17-8-7-15(27-4)13-16(17)21/h7-10,13H,5-6,11-12H2,1-4H3,(H,23,24)
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n/an/an/an/a 81n/an/an/an/a



Minase Research Institute

Curated by ChEMBL


Assay Description
Antagonist activity at rat CRF1 receptor expressed in CHO-K1 cells assessed as inhibition of CRF-induced cAMP accumulation after 15 mins by cAMP enzy...


Bioorg Med Chem 19: 5955-66 (2011)


Article DOI: 10.1016/j.bmc.2011.08.055
BindingDB Entry DOI: 10.7270/Q24X5862
More data for this
Ligand-Target Pair
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